Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
Found 207 products of "Androgen Receptor"
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Fenarimol
CAS:<p>Fenarimol, a pyrimidine-type fungicide, exhibits potent inhibitory activity against BR biosynthesis.</p>Formula:C17H12Cl2N2OColor and Shape:SolidMolecular weight:331.2MK-0773
CAS:<p>MK-0773 (PF-05314882) is a selective androgen receptor modulator that binds to AR (IC50: 6.6 nM) for the study of diseases caused by endocrine abnormalities.</p>Formula:C27H34FN5O2Purity:98.38% - 99.14%Color and Shape:SolidMolecular weight:479.59Dehydroepiandrosterone-d2
CAS:<p>Dehydroepiandrosterone-d2 is a deuterated compound of Dehydroepiandrosterone.</p>Formula:C19H26D2O2Color and Shape:SolidMolecular weight:290.44ARD-1676
CAS:<p>ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand with a cereblon ligand.</p>Formula:C44H46ClN7O5Purity:98%Color and Shape:SolidMolecular weight:788.33Leelamine hydrochloride
CAS:<p>Leelamine hydrochloride, a pine bark extract, inhibits androgen receptor and CB1, reducing lipid synthesis in prostate cancer.</p>Formula:C20H32ClNPurity:98%Color and Shape:SolidMolecular weight:321.93(Rac)-PF-998425
CAS:<p>(Rac)-PF-998425: nonsteroidal AR antagonist, potent & selective, IC50: 26 nM (binding), 90 nM (cellular), potential for androgenetic alopecia study.</p>Formula:C14H14F3NOColor and Shape:SolidMolecular weight:269.267Rezvilutamide
CAS:<p>Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and has antitumor activity.</p>Formula:C22H20F3N3O4SPurity:99.97%Color and Shape:SolidMolecular weight:479.47D4-abiraterone
CAS:<p>D4-abiraterone is the active metabolite of abiraterone.Δ4-Abiraterone is a inhibitor of CYP17A1, 3β-HSD and SRD5A, and an antagonist of the androgen receptor.</p>Formula:C24H29NOPurity:99.75% - 99.8%Color and Shape:SolidMolecular weight:347.49VPC-13566
CAS:<p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>Formula:C18H14N2Purity:99.55%Color and Shape:SolidMolecular weight:258.323-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:<p>3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.</p>Formula:C18H14N4OPurity:98.41%Color and Shape:SolidMolecular weight:302.33AH-3960
CAS:<p>AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。</p>Formula:C13H22N4O3Purity:98.44%Color and Shape:SolidMolecular weight:282.34Darolutamide
CAS:<p>Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).</p>Formula:C19H19ClN6O2Purity:97.36% - >99.99%Color and Shape:SolidMolecular weight:398.85Enzalutamide
CAS:<p>Enzalutamide (MDV3100) is an androgen receptor (AR) antagonist (IC50=36 nM in LNCaP).</p>Formula:C21H16F4N4O2SPurity:99% - 99.93%Color and Shape:SolidMolecular weight:464.44Nandrolone phenylpropionate
CAS:<p>Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosis</p>Formula:C27H34O3Purity:99.2% - 99.46%Color and Shape:White Or Milky Crystalline PowderMolecular weight:406.56CTK8A3536
CAS:<p>CTK8A3536 ((2-MORPHOLIN-4-YL-4-PHENYL-1,3-THIAZOL-5-YL)METHANOL) is an inhibitor of Androgen receptor.</p>Formula:C14H16N2O2SPurity:99.62%Color and Shape:SolidMolecular weight:276.35MI-136
CAS:<p>MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.</p>Formula:C23H21F3N6SPurity:98.63% - 99.12%Color and Shape:SolidMolecular weight:470.51Lupeol
CAS:<p>Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.</p>Formula:C30H50OPurity:98% - 99.96%Color and Shape:Needles From Alcohol Acetone White PowderMolecular weight:426.72ARD-2128
CAS:<p>ARD-2128: potent oral PROTAC that degrades AR, curbing prostate cancer growth with no toxicity.</p>Formula:C45H50ClN7O6Purity:98.8%Color and Shape:SolidMolecular weight:820.37Dimethylcurcumin
CAS:<p>Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.</p>Formula:C23H24O6Purity:97.36% - 98.96%Color and Shape:SolidMolecular weight:396.43Bavdegalutamide
CAS:<p>Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).</p>Formula:C41H43ClFN9O6Purity:97.17% - 99.04%Color and Shape:SolidMolecular weight:812.29
![3-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT9752.webp&w=3840&q=75)
