Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
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Ralaniten
CAS:1203490-23-6
Ralaniten (EPI-002), a potent AR-NTD antagonist, inhibits AR with IC50 of 7.4 μM, for CRPC …
Formula:
C21H27ClO5
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
394.89
Ref: TM-T28502
| 1mg | 40.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 393.00 € | ||
| 100mg | 628.00 € | ||
| 200mg | 879.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 5 Jun 2025
MK-3984
CAS:871325-55-2
MK-3984 is a selective androgen receptor modulator, used in the study of conditions caused by …
Formula:
C17H12F7NO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
395.27
Ref: TM-T33433
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Thursday 5 Jun 2025
BMS-564929
CAS:627530-84-1
BMS-564929 is an AR agonist that upregulates the expression and activity of fat-producing enzymes, reducing …
Formula:
C14H12ClN3O3
Purity:
98.17%
Color and Shape:
Solid
Molecular weight:
305.72
Ref: TM-T14675
| 50mg | 1,941.00 € | ||
| 100mg | 2,745.00 € |
Estimated delivery in United States, on Thursday 5 Jun 2025
Prochloraz
CAS:67747-09-5
Prochloraz: broad-spectrum imidazole fungicide; blocks placental aromatase (IC50=40nM), estrogen/androgen receptors; activates aryl hydrocarbon receptors.
Formula:
C15H16Cl3N3O2
Purity:
99.4%
Color and Shape:
Colorless Solid
Molecular weight:
376.67
Ref: TM-T20625
| 200mg | 40.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 5 Jun 2025
Ralaniten triacetate
CAS:1637573-04-6
Ralaniten triacetate (EPI-506) is a precursor of Ralaniten, an AR-NTD inhibitor, which can be used …
Formula:
C27H33ClO8
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
521.00
Ref: TM-T36375
| 1mg | 162.00 € | ||
| 5mg | 393.00 € | ||
| 10mg | 655.00 € | ||
| 25mg | 1,415.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € | ||
| 1mL*10mM (DMSO) | 449.00 € |
Estimated delivery in United States, on Thursday 5 Jun 2025
ONC1-13B
CAS:1351185-54-0
ONC1-13B, an androgen receptor antagonist, is used potentially for the treatment of prostate cancer.
Formula:
C22H16F4N4O3S
Purity:
99.45% - 99.85%
Color and Shape:
Solid
Molecular weight:
492.45
Ref: TM-T28238
| 1mg | 279.00 € | ||
| 5mg | 683.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,415.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,612.00 € |
Estimated delivery in United States, on Thursday 5 Jun 2025
Androgen receptor degrader-1
CAS:2616553-35-4
Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in …
Formula:
C15H14ClN3O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
335.74
Ref: TM-T80633
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 20 Jun 2025
RU 59063
CAS:155180-53-3
RU 59063 is a prototype of a new class of high-affinity nonsteroidal androgen receptor (AR) …
Formula:
C17H18F3N3O2S
Purity:
98.21%
Color and Shape:
Solid
Molecular weight:
385.4
Ref: TM-T20761
| 1mg | 87.00 € | ||
| 5mg | 192.00 € | ||
| 10mg | 284.00 € | ||
| 25mg | 452.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 867.00 € | ||
| 200mg | 1,130.00 € | ||
| 1mL*10mM (DMSO) | 208.00 € |
Estimated delivery in United States, on Friday 20 Jun 2025
YXG-158
CAS:2952994-34-0
YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) …
Formula:
C30H36FN3O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
473.62
Ref: TM-T79519
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 20 Jun 2025
Androgen receptor degrader-3
CAS:2753650-84-7
Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the …
Formula:
C45H51ClN8O5
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
819.39
Ref: TM-T79891
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 20 Jun 2025
Androgen receptor-IN-5
CAS:1391944-16-3
Androgen receptor-IN-5 is a potent inhibitor of the androgen receptor with anticancer properties.
Formula:
C22H10Cl2F4N4OS
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
525.31
Ref: TM-T79024
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 20 Jun 2025
Androgen receptor degrader-2
CAS:2616553-33-2
Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application …
Formula:
C16H16ClN3O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
349.77
Ref: TM-T80647
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 20 Jun 2025
N-Nitrosodicyclohexylamine
CAS:947-92-2
N-Nitrosodicyclohexylamine (NDCHA), an N-nitrosocompound, exhibits anti-androgenic activity by competitively binding to the androgen receptor (AR) …
Formula:
C12H22N2O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
210.32
Ref: TM-T81662
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 20 Jun 2025
Celiprolol hydrochloride
CAS:57470-78-7
Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.
Formula:
C20H33N3O4·HCl
Color and Shape:
White Crystalline Solid
Molecular weight:
415.96
Ref: TM-T1244
| 2mg | 78.00 € | ||
| 1mL*10mM (DMSO) | 138.00 € |
Estimated delivery in United States, on Friday 20 Jun 2025
VPC-14228
CAS:19983-28-9
VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.
Formula:
C13H14N2OS
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
246.33
Ref: TM-T24943
| 1mg | 39.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 298.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 658.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Friday 20 Jun 2025
FL442
CAS:1431166-12-9
FL442 is an Androgen Receptor (AR) modulator. This compound exhibits potent inhibitory effects in AR-dependent …
Formula:
C15H13F3N2O
Color and Shape:
Liquid
Molecular weight:
294.27
Ref: TM-T200138
| 10mg | To inquire | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Thursday 17 Jul 2025
(+)-JJ-74-138
CAS:2135545-34-3
(+)-JJ-74-138 is a novel non-competitive androgen receptor (AR) antagonist capable of inhibiting enzalutamide-resistant castration-resistant prostate …
Formula:
C22H22F8N2OS
Color and Shape:
Liquid
Molecular weight:
514.48
Ref: TM-T200319
| 10mg | To inquire | ||
| 25mg | 2,470.00 € | ||
| 50mg | 3,019.00 € | ||
| 100mg | 3,725.00 € |
Estimated delivery in United States, on Thursday 17 Jul 2025
LX1
CAS:2647877-84-5
LX1, an anti-prostate cancer compound, specifically targets the androgen receptor (AR), AR variants, and the …
Formula:
C22H15F6NO2
Color and Shape:
Liquid
Molecular weight:
439.35
Ref: TM-T200147
| 10mg | To inquire | ||
| 25mg | 1,539.00 € | ||
| 50mg | 1,941.00 € | ||
| 100mg | 2,451.00 € |
Estimated delivery in United States, on Thursday 17 Jul 2025
Androgen receptor degrader-5
CAS:2902679-11-0
Androgen receptor degrader-5 (compound 14k) demonstrates superior capabilities, specifically in androgen receptor degradation and antiproliferative …
Formula:
C29H25F4N5O2
Color and Shape:
Liquid
Molecular weight:
551.53
Ref: TM-T200197
| 10mg | To inquire | ||
| 25mg | 1,539.00 € | ||
| 50mg | 1,941.00 € | ||
| 100mg | 2,451.00 € |
Estimated delivery in United States, on Thursday 17 Jul 2025
Pentomone
CAS:67102-87-8
Pentomone (LY-113935) is an anti-androgen compound that acts as a prostate growth inhibitor.
Formula:
C24H26O5
Color and Shape:
Liquid
Molecular weight:
394.46
Ref: TM-T201000
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 17 Jul 2025
