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Androgen Receptor

Androgen Receptor

The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.

Found 207 products of "Androgen Receptor"

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  • AR antagonist 2
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    AR antagonist 2

    CAS:
    <p>AR antagonist 2 (compound 58) is a potent inhibitor of the androgen receptor (AR) (IC50: 0.95 μM).</p>
    Formula:C22H17ClFN5O2S
    Color and Shape:Solid
    Molecular weight:469.92

    Ref: TM-T63030

  • AR antagonist 5
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    AR antagonist 5

    CAS:
    <p>Compound 30a, known as AR Antagonist 5, is a selective androgen receptor (AR) antagonist that demonstrates an IC 50 value of 134.8 nM. It exhibits favorable pharmacokinetic properties, characterized by high skin exposure and low plasma exposure [1].</p>
    Formula:C23H21F3N6O2
    Color and Shape:Solid
    Molecular weight:470.45

    Ref: TM-T85717

  • CSRM617
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    CSRM617

    CAS:
    <p>CSRM617: selective ONECUT2 inhibitor, Kd 7.43 uM, binds OC2-HOX, induces apoptosis, tolerable in mouse prostate cancer model.</p>
    Formula:C10H13N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.23

    Ref: TM-T10896

  • MK-4541
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    MK-4541

    CAS:
    <p>MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.</p>
    Formula:C22H31F3N2O3
    Color and Shape:Solid
    Molecular weight:428.49

    Ref: TM-T73410

  • (R)-UT-155
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    (R)-UT-155

    CAS:
    <p>(R)-UT-155 is a selective androgen receptor degrader (SARD) ligand.</p>
    Formula:C20H15F4N3O2
    Color and Shape:Solid
    Molecular weight:405.35

    Ref: TM-T13977

  • Carbazole derivative 1
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    Carbazole derivative 1

    CAS:
    <p>Carbazole derivative 1 is used to reduce androgen or oestrogen levels in mammals.</p>
    Formula:C18H13FN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:276.31

    Ref: TM-T19170

  • VPC-3033
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    VPC-3033

    CAS:
    <p>VPC-3033 is an antagonist of the androgen receptor. It acts by inhibiting the LNCaP cell line as well as cell lines with the wild-type androgen receptor.</p>
    Formula:C21H14O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:298.33

    Ref: TM-T26323

  • Androgen receptor antagonist 3
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    Androgen receptor antagonist 3

    CAS:
    <p>Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].</p>
    Formula:C22H18ClN
    Color and Shape:Solid
    Molecular weight:331.84

    Ref: TM-T60987

  • RU 58642
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    RU 58642

    CAS:
    <p>RU 58642 is an effective systemic antiandrogen for androgen-dependent disorders.</p>
    Formula:C15H11F3N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.27

    Ref: TM-T26156

  • VPC-13789
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    VPC-13789

    CAS:
    <p>VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.</p>
    Formula:C21H16F3N3O
    Color and Shape:Solid
    Molecular weight:383.37

    Ref: TM-T61653

  • Topterone
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    Topterone

    CAS:
    <p>Topterone (Win 17,665) is a potent topical antiandrogen that inhibits the stimulation of lumbar organ development by testosterone and dihydrotestosterone in</p>
    Formula:C22H34O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:330.5

    Ref: TM-T13187

  • Ar-V7-IN-1
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    Ar-V7-IN-1

    CAS:
    <p>Ar-V7-IN-1 (compound 47) is a potent inhibitor of Ar-V7,associated with resistance to AR-targeted therapy with desmoplasia-resistant prostate cancer (mCRPC).</p>
    Formula:C10H10Br2N4OS
    Color and Shape:Solid
    Molecular weight:394.09

    Ref: TM-T61820

  • Prochloraz
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    Prochloraz

    CAS:
    <p>Prochloraz: broad-spectrum imidazole fungicide; blocks placental aromatase (IC50=40nM), estrogen/androgen receptors; activates aryl hydrocarbon receptors.</p>
    Formula:C15H16Cl3N3O2
    Purity:99.75% - 99.79%
    Color and Shape:Colorless Solid
    Molecular weight:376.67

    Ref: TM-T20625

  • Androgen receptor antagonist 1
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    Androgen receptor antagonist 1

    CAS:
    <p>Androgen receptor antagonist 1, an oral full AR antagonist (IC50 59 nM), for PROTAC synthesis, reducing AR protein by 24–47% in LNCaP cells at 1–10 μM.</p>
    Formula:C21H25ClN4O3
    Purity:99.054%
    Color and Shape:Solid
    Molecular weight:416.9

    Ref: TM-T10320

  • Bromopropylate
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    Bromopropylate

    CAS:
    <p>Bromopropylate is an insecticide. Bromopropylate is the active substance in fumigant strips for mites.</p>
    Formula:C17H16Br2O3
    Purity:98%
    Color and Shape:White Crystalline Solid Yellowish Crystals
    Molecular weight:428.11

    Ref: TM-T19845

  • Dimethomorph
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    Dimethomorph

    CAS:
    <p>Dimethomorph is a fungicide and sterol biosynthesis inhibitor that inhibits fungal cell wall formation,. inhibits androgen receptor (AR) .</p>
    Formula:C21H22ClNO4
    Purity:99.2%
    Color and Shape:Solid Crystalline
    Molecular weight:387.86

    Ref: TM-T41322

  • MK-3984
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    MK-3984

    CAS:
    <p>MK-3984 is a selective androgen receptor modulator, used in the study of conditions caused by androgen deficiency.</p>
    Formula:C17H12F7NO2
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:395.27

    Ref: TM-T33433

  • Bifluranol
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    Bifluranol

    CAS:
    <p>Bifluranol (BX341) has anti-androgenic activity and has shown significant anti-prostatic activity in in vivo studies for the treatment of benign prostatic</p>
    Formula:C17H18F2O2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:292.32

    Ref: TM-T14843

  • VPC-14449
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    VPC-14449

    CAS:
    <p>VPC-14449 is a selective androgen receptor DNA-binding domain (AR-DBD) inhibitor, useful in prostate cancer research.</p>
    Formula:C10H10Br2N4OS
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:394.09

    Ref: TM-T24944

  • Ralaniten
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    Ralaniten

    CAS:
    <p>Ralaniten (EPI-002), a potent AR-NTD antagonist, inhibits AR with IC50 of 7.4 μM, for CRPC study.</p>
    Formula:C21H27ClO5
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:394.89

    Ref: TM-T28502