Enzyme
Enzyme inhibitors are molecules that bind to enzymes and decrease their activity. These inhibitors are widely used in research to study enzyme kinetics, regulation, and the role of specific enzymes in metabolic pathways. Enzyme inhibitors are also crucial in drug development, as many therapeutic agents function by inhibiting enzymes involved in disease processes. By targeting enzymes, these inhibitors can modulate biochemical pathways and offer potential treatments for various diseases. At CymitQuimica, we provide a comprehensive selection of high-quality enzyme inhibitors to support your research in biochemistry, pharmacology, and drug discovery.
Subcategories of "Enzyme"
- Carbonic Anhydrase(196 products)
- Hydroxylase(36 products)
- MPO(2 products)
- Reductase(51 products)
- Tyrosinase(71 products)
Found 3619 products of "Enzyme"
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Pyrocatechol
CAS:Pyrocatechol, often known as catechol or benzene-1,2-diol, is a benzenediol, Pyrocatechol was produced at a large scale industrially, mainly as precursors to pesticides, flavors, and fragrances. Its sulfonic acid is often present in the urine of many mammals.Formula:C6H6O2Purity:99.96%Color and Shape:SolidMolecular weight:110.11Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2
CAS:Ac-[Nle4,D-Phe7]-α-MSH (4-10)-NH2, a melanotropin derivative and melanocyte-stimulating hormone, activates tyrosinase and demonstrates a thermoregulatory effectFormula:C47H64N14O10Color and Shape:SolidMolecular weight:985.1Carbonic anhydrase inhibitor 21
Compound 5h, known as Carbonic anhydrase inhibitor 21, is a specific inhibitor of carbonic anhydrase (hCA IX) with a K\(_i\) of 15.1 nM, demonstrating high selectivity compared to other isoforms studied. This compound is utilized in anticancer research.Formula:C32H48N4O10P2S2Molecular weight:774.22871TPT-004
TPT-004, a TPH inhibitor, exhibits superior pharmacokinetic and pharmacodynamic properties, and demonstrates efficacy in preclinical models for attenuatingColor and Shape:Odour SolidCAIX/CAXII-IN-4
CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.Formula:C23H21N5O3SColor and Shape:SolidMolecular weight:447.51Acesulfame
CAS:Acesulfame inhibits CA9/12 and can be used to study inflammation-related diseases.Formula:C4H5NO4SColor and Shape:SolidMolecular weight:163.15Proteinase K
CAS:Purity:≥ 30units/mg (pH 7.5, 37°C, dried basis)Color and Shape:White or almost white lyophilized powderMolecular weight:-Peroxidase, from horseradish, approx. 200 U/mg
CAS:Purity:≥ 150U/mgColor and Shape:Beige to light-brown, reddish brown or dark brown lyophilised powderMolecular weight:-Tyrosinase-IN-32
Tyrosinase-IN-32 (compound 11), a hydroxamate-based alkaloid extracted from black pepper (Piper nigrum L.), functions as an inhibitor of mushroom tyrosinase. In addition to its inhibitory properties, it exhibits antioxidant activity.Formula:C15H19NO3Color and Shape:SolidMolecular weight:261.32β-Glucosidase, from almonds
CAS:Purity:approx. 90% (biuret)Color and Shape:White to pale yellow or beige powderMolecular weight:-Carbonic anhydrase inhibitor 18
Carbonic anhydrase inhibitor18 (Compound 9) is an inhibitor of human carbonic anhydrase (hCA) isozymes, with Ki values of 604.8 nM for hCA I, 333.6 nM for hCA II, 1.9 nM for hCA IX, and 6.7 nM for hCA XII. Carbonic anhydrase inhibitor18 is applicable in cancer research.Formula:C26H28N4O6S2Molecular weight:556.14503P-Hydroxybenzoate Hydroxylase
CAS:Color and Shape:Yellowish lyophilised powderMolecular weight:55 ~ 60 kDaTyrosinase-IN-38
Tyrosinase-IN-38 (compound 6b) is a competitive inhibitor of tyrosinase, demonstrating an IC50 of 25.82 μM and exhibits antioxidant activity.Color and Shape:Odour SolidCalmodulin-dependent Protein Kinase II fragment 290-309
CAS:Formula:C103H185N31O24SMolecular weight:2273.83Xanthine Oxidase, ammonium sulfate suspension
CAS:Color and Shape:Faint brown to dark brown suspensionAnhydrotetracycline hydrochloride
CAS:Anhydrotetracycline (hydrochloride) is a potent competitive inhibitor of broad-spectrum tetracycline destructase enzymes.Formula:C22H23ClN2O7Purity:98% - 98.90%Color and Shape:SolidMolecular weight:462.88DPP IV/hCA II-IN-1
CAS:DPP IV/hCA II-IN-1: strong DPP IV & CA inhibitor, IC50=0.049μM (DPP IV), Ki=0.0361-3.034μM (CA II-IV).
Formula:C17H20N2O5SColor and Shape:SolidMolecular weight:364.42CA IX/VEGFR-2-IN-3
CAIX/VEGFR-2-IN-3 (Compound 6i) is an inhibitor of Carbonic Anhydrase IX and VEGFR-2, with IC50 values of 41 and 48 nM, respectively. It exhibits anticancer activity by inhibiting the growth of MCF-7 breast cancer cells (IC50 of 22.33 μM) and mouse fibroblast cell line 3T3, where cell viability is reduced to below 40% at a concentration of 100 μM. This compound is applicable for research in the field of cancer treatment.Formula:C19H16ClN3O5S2Color and Shape:SolidMolecular weight:465.93CAIX/CAXII-IN-3
CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.Color and Shape:Odour SolidTPH1-IN-1
TPH1-IN-1 (compound 40) is a xanthine derivative that serves as an inhibitor of tryptophan hydroxylase TPH1, with an IC50 of 110.1 nM.Formula:C21H18N6O4SColor and Shape:SolidMolecular weight:450.475,6-Dihydro-2H-pyran-2-one
CAS:5,6-Dihydro-2H-pyran-2-one is a carbonic anhydrase 1/9 inhibitor that inhibits KB cell viability.Formula:C5H6O2Color and Shape:SolidMolecular weight:98.1Tyrosinase-IN-36
Tyrosinase-IN-36 is a moderately potent inhibitor of tyrosine, exhibiting an inhibition percentage of 42.75% compared to kojic acid at a concentration of 100 μM and possesses antioxidant activity.Color and Shape:Odour SolidDOTA-XYIMSR-01
CAS:DOTA-XYIMSR-01 is a molecular probe targeting CAIX, capable of being labeled with 177Lu for the treatment and localization of malignant gliomas. The uptake of [177Lu]Lu-XYIMSR-01 in U87MG tumors is 6.19% injected dose per gram (% ID/g), with a tumor-to-muscle uptake ratio of 20.14. In an orthotopic glioma model, co-administration with temozolomide significantly enhances survival rates and inhibits tumor growth in mice. DOTA-XYIMSR-01 shows potential for research in the field of cancer treatment.Formula:C61H88N16O22S2Color and Shape:SolidMolecular weight:1461.57Bendroflumethiazide
CAS:Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)Formula:C15H14F3N3O4S2Purity:98% - >99.99%Color and Shape:Crystals From Dioxane SolidMolecular weight:421.41TrkA Protein, Canine, Recombinant (hFc)
TrkA Protein, Canine, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.Color and Shape:Lyophilized PowderMolecular weight:42.3 kDa (predicted); 55-61 kDa (reducing conditions)ErbB4 Protein, Human, Rhesus, Recombinant (hFc)
ErbB4 Protein, Human, Rhesus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag.Color and Shape:Lyophilized PowderMolecular weight:96.6 kDa (predicted); 117 kDa (reducing conditions)Ref: TM-TMPY-02814
1mg4,207.00€5µg77.00€10µg109.00€20µg174.00€50µg350.00€100µg668.00€200µg1,017.00€500µg2,071.00€FLT1 Protein, Human, Recombinant (aa 1-328, His)
FLT1 Protein, Human, Recombinant (aa 1-328, His) is expressed in HEK293 mammalian cells with His tag.Purity:97.5%Color and Shape:Lyophilized PowderMolecular weight:35.6 kDa (predicted)TrkB Protein, Human, Recombinant (His) V2
Expression System: HEK293 Cells
Length: 32-430, Extracellular Domain
Activity: ELISAColor and Shape:Lyophilized PowderMolecular weight:45.2 kDa (Predicted); 65-80 kDa (Due to glycosylation)HER3/ERBB3 Protein, Human, Recombinant (aa 20-643, His & Avi), Biotinylated
HER3/ERBB3 Protein, Human, Recombinant (aa 20-643, His & Avi), Biotinylated is expressed in HEK293 mammalian cells with C-6xHis-Avi tag.Color and Shape:Lyophilized PowderMolecular weight:90-120 KDa (reducing condition)Mer Protein, Mouse, Recombinant (His & GST)
Mer Protein, Mouse, Recombinant (His & GST) is expressed in Baculovirus insect cells with His and GST tag.Color and Shape:Lyophilized PowderMolecular weight:61.7 kDa (predicted); 58 kDa (reducing conditions)TrkB Protein, Human, Recombinant (His)
TrkB Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag.Purity:99.3%Color and Shape:Lyophilized PowderMolecular weight:45.7 kDa (predicted); 70-80 kDa (reducing condition, due to glycosylation)Thrombopoietin Protein, Mouse, Recombinant (C-His)
Expression System: HEK293 Cells
Length: 22-356, Full Length of Mature Protein
Activity: Cell ActivityColor and Shape:Lyophilized PowderMolecular weight:37.20 kDa (Predicted); 75-95 kDa (Due to glycosylation)
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