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GABA Receptor

GABA Receptor

GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.

Found 336 products of "GABA Receptor"

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  • Pyrazolam

    CAS:
    <p>Pyrazolam is a psychoactive benzodiazepine compound serving as a central nervous system depressant. [Pyrazolam] can lead to psychomotor impairment.</p>
    Formula:C16H12BrN5
    Color and Shape:Solid
    Molecular weight:354.2
  • Rilmazolam

    CAS:
    <p>Rilmazolam is a triazolobenzodiazepine compound and serves as the active metabolite of Rilmazafone.</p>
    Formula:C19H15Cl2N5O
    Color and Shape:Solid
    Molecular weight:400.26
  • Imagabalin

    CAS:
    <p>Imagabalin is an active compound used in the study of neurological diseases.</p>
    Formula:C9H19NO2
    Color and Shape:Solid
    Molecular weight:173.25
  • FGIN-1-43

    CAS:
    <p>FGIN-1-43 is a potent and specific ligand for the mitochondrial DBI receptor.</p>
    Formula:C28H36Cl2N2O
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:487.5
  • (Iso)-Atagabalin HCl

    CAS:
    <p>(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) is an alpha -2- delta ligand that can be used to treat non-restorative sleep.</p>
    Formula:C10H20ClNO2
    Purity:99.26% - >99.99%
    Color and Shape:Soild
    Molecular weight:221.72
  • MIDD0301

    CAS:
    <p>MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of 17 nM.</p>
    Formula:C19H13BrFN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.23
  • 12,14-Dichlorodehydroabietic acid

    CAS:
    <p>12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.</p>
    Formula:C20H26Cl2O2
    Color and Shape:Solid
    Molecular weight:369.33
  • 3-Aminopropylphosphonic Acid

    CAS:
    <p>3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding</p>
    Formula:C3H10NO3P
    Purity:99.84%
    Color and Shape:Light Yellow Liquid
    Molecular weight:139.09
  • Cinazepam

    CAS:
    <p>Cinazepam is a GABAA receptor partial agonist and a benzodiazepine derivative with anxiolytic and sedative properties. Cinazepam can be utilized in research related to sleep disorders.</p>
    Formula:C19H14BrClN2O5
    Color and Shape:Solid
    Molecular weight:465.68
  • DAA-1106

    CAS:
    <p>DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.</p>
    Formula:C23H22FNO4
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:395.42
  • Atagabalin

    CAS:
    <p>Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.</p>
    Formula:C10H19NO2
    Color and Shape:Solid
    Molecular weight:185.26
  • 3-Aminopropylphosphinic acid

    CAS:
    <p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>
    Formula:C3H10NO2P
    Color and Shape:Solid
    Molecular weight:123.092
  • Fipronil sulfone

    CAS:
    <p>Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.</p>
    Formula:C12H4Cl2F6N4O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:453.14
  • Chrodrimanin B

    CAS:
    <p>Chrodrimanin B is a useful organic compound for research related to life sciences. The catalog number is T126052 and the CAS number is 132196-54-4.</p>
    Formula:C27H32O8
    Color and Shape:Solid
    Molecular weight:484.545
  • Emamectin B1a

    CAS:
    <p>Emamectin B1a can be used in relevant research in the life sciences. Its product number is T37663 and CAS number is 121124-29-6.</p>
    Formula:C49H75NO13
    Color and Shape:Solid
    Molecular weight:886.133
  • Flufiprole

    CAS:
    <p>Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.</p>
    Formula:C16H10Cl2F6N4OS
    Color and Shape:Solid
    Molecular weight:491.24
  • Anticonvulsant agent 9


    <p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>
    Formula:C22H24N4O2
    Color and Shape:Solid
    Molecular weight:376.45
  • AHN-683

    CAS:
    <p>AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.</p>
    Formula:C42H32FN3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:709.72
  • LU-32-176B

    CAS:
    <p>LU32-176B is a bioactive chemical.</p>
    Formula:C23H24F2N2O2
    Color and Shape:Solid
    Molecular weight:398.45
  • TET-13


    <p>TET-13 is a positive allosteric modulator of the GABAA receptor with an EC50 of 5.65 μM, which is more potent than Etomidate (EC50: 9.29 μM). It exhibits strong anesthetic effects in both mice and rats, with an ED50 of 0.48 mg/kg in mice and 0.69 mg/kg in rats.</p>
    Formula:C15H16N2O3S
    Color and Shape:Solid
    Molecular weight:304.36