GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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2'MeO6MF
CAS:89112-85-6
2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers …
Formula:
C17H14O3
Purity:
99.28% - 99.63%
Color and Shape:
Solid
Molecular weight:
266.29
Ref: TM-T8887
| 1mg | 51.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 485.00 € | ||
| 200mg | 662.00 € | ||
| 1mL*10mM (DMSO) | 101.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Pikamilone
CAS:34562-97-5
Pikamilone (Picamilon) is an intelligent medicine.
Formula:
C10H12N2O3
Purity:
98.25%
Color and Shape:
White Crystalline Powder
Molecular weight:
208.21
Ref: TM-T3290
| 500mg | 81.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
(+)-Kavain
CAS:500-64-1
(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) …
Formula:
C14H14O3
Purity:
97% - ≥95%
Color and Shape:
White Fine Powder
Molecular weight:
230.26
Ref: TM-T4590
| 5mg | 47.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 131.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
(-)-Securinine
CAS:5610-40-2
(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.
Formula:
C13H15NO2
Purity:
99.58% - 99.87%
Color and Shape:
Solid
Molecular weight:
217.26
Ref: TM-T3S2100
| 5mg | 55.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 241.00 € | ||
| 100mg | 361.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Isonipecotic acid
CAS:498-94-2
Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA …
Formula:
C6H11NO2
Purity:
99.82%
Color and Shape:
White To Faint Pink-Beige Powder
Molecular weight:
129.16
Ref: TM-T22348
| 1g | 34.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
SKF89976A hydrochloride
CAS:85375-15-1
SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = …
Formula:
C22H26ClNO2
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
371.9
Ref: TM-T12930
| 5mg | 69.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 363.00 € | ||
| 100mg | 533.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Miltirone
CAS:27210-57-7
Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central …
Formula:
C19H22O2
Purity:
99.22% - 99.66%
Color and Shape:
Solid
Molecular weight:
282.38
Ref: TM-TN1023
| 1mg | 133.00 € | ||
| 5mg | 202.00 € | ||
| 10mg | 329.00 € | ||
| 25mg | 548.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,035.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Phenibut (hydrochloride)
CAS:3060-41-1
Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at …
Formula:
C10H14ClNO2
Purity:
99.93%
Color and Shape:
White Crystalline Powder
Molecular weight:
215.68
Ref: TM-T8639
| 50mg | 48.00 € | ||
| 100mg | 65.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
4-Acetamidobutanoic acid
CAS:3025-96-5
4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.
Formula:
C6H11NO3
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
145.16
Ref: TM-T4728
| 200mg | 67.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
CGP52432
CAS:139667-74-6
CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).
Formula:
C15H24Cl2NO4P
Purity:
99.16%
Color and Shape:
Solid
Molecular weight:
384.24
Ref: TM-T4363
| 1mg | 40.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 374.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
(E)-3,4,5-Trimethoxycinnamic acid
CAS:20329-98-0
(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium …
Formula:
C12H14O5
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
238.24
Ref: TM-TN2865
| 1g | 133.00 € | ||
| 100mg | 48.00 € | ||
| 500mg | 90.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Imidazenil
CAS:151271-08-8
Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion …
Formula:
C18H12BrFN4O
Purity:
98.4%
Color and Shape:
Solid
Molecular weight:
399.22
Ref: TM-T8971
| 1mg | 99.00 € | ||
| 5mg | 207.00 € | ||
| 10mg | 343.00 € | ||
| 25mg | 565.00 € | ||
| 50mg | 822.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
SSD114 HCl
CAS:2319790-02-6
SSD114 is a novel GABAB receptor positive allosteric modulator.
Formula:
C18H21ClF3N3O
Purity:
97.83% - 99.03%
Color and Shape:
Solid
Molecular weight:
387.83
Ref: TM-T4522
| 1mg | 38.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 300.00 € | ||
| 100mg | 512.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
p-Hydroxybenzaldehyde
CAS:123-08-0
1.
Formula:
C7H6O2
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
122.12
Ref: TM-T2S1814
| 5g | 51.00 € | ||
| 10g | 74.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Aminooxyacetic acid hemihydrochloride
CAS:2921-14-4
Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the …
Formula:
C2H5NO3·5HCl
Purity:
98.03%
Color and Shape:
Light Beige Crystalline Powder
Molecular weight:
109.3
Ref: TM-T5880
| 1g | 74.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Amentoflavone
CAS:1617-53-4
Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other …
Formula:
C30H18O10
Purity:
98.21% - 99.22%
Color and Shape:
Odourless Whitish Solid
Molecular weight:
538.46
Ref: TM-T3417
| 1mg | 35.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 163.00 € | ||
| 50mg | 278.00 € | ||
| 100mg | 424.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Tiagabine
CAS:115103-54-3
Tiagabine (NO050328) is an Anti-epileptic Agent.
Formula:
C20H25NO2S2
Purity:
99.24%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
375.55
Ref: TM-T2407
| 5mg | 44.00 € | ||
| 10mg | 55.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
Gabazine
CAS:104104-50-9
Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)
Formula:
C15H18BrN3O3
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
368.23
Ref: TM-T7622
| 5mg | 51.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 464.00 € | ||
| 200mg | 627.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
6-(4-Methoxyphenyl)-3-pyridazinamine
CAS:4776-87-8
6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist
Formula:
C11H11N3O
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
201.22
Ref: TM-T7793
| 10mg | 50.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 235.00 € | ||
| 200mg | 335.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
2'-O-Methylisoliquiritigenin
CAS:51828-10-5
2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, …
Formula:
C16H14O4
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
270.28
Ref: TM-TN1217
| 1mg | 153.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 540.00 € | ||
| 25mg | 868.00 € | ||
| 1mL*10mM (DMSO) | 434.00 € |
Estimated delivery in United States, on Monday 10 Mar 2025
