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Casein Kinase

Casein Kinase

Casein kinases are a family of serine/threonine protein kinases that regulate various cellular processes, including DNA repair, circadian rhythms, and signal transduction. These kinases are involved in the phosphorylation of numerous proteins and are implicated in diseases such as cancer, neurodegenerative disorders, and metabolic syndromes. At CymitQuimica, we offer a selection of casein kinase inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.

Found 130 products of "Casein Kinase"

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  • HDAC/CK2-IN-1

    CAS:
    <p>HDAC/CK2-IN-1 (compound 38) acts as an inhibitor of HDAC1 (IC 50 = 1.46 μM), HDAC6 (IC 50 = 0.66 μM), and CK2 (IC 50 = 3.67 μM). It demonstrates promising antiproliferative effects on various cell lines, including Jurkat, MCF-7, HCT-116, and HL-60.</p>
    Formula:C15H18Br4N4O2
    Color and Shape:Solid
    Molecular weight:605.95
  • CK2-IN-4

    CAS:
    <p>CK2-IN-4 is a protein kinase (CK2) inhibitor with an IC50 value of 8.6 µM.</p>
    Formula:C18H11N3O4S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:365.36
  • CK2α-IN-1

    CAS:
    <p>CK2α-IN-1 is a selective non-ATP-competitive CK2α inhibitor with an IC50 of 7.0 µM and a Ki of 1.6 µM.CK2α-IN-1 exhibits potential anticancer activity and can</p>
    Formula:C16H11N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.34
  • CK1-IN-2

    CAS:
    <p>CK1-IN-2 (compound Nr.4) is a potent CK1 inhibitor p38a, and is used in DUX4 overexpression-associated diseases, such as muscular dystrophy.</p>
    Formula:C17H12FN3O2
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:309.29
  • PI-828

    CAS:
    <p>PI-828 (LY 294002), a PI3K inhibitor, researches PI3K function and aids stem cell differentiation into mesoderm.</p>
    Formula:C19H18N2O3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:322.36
  • XL413 xHCl

    CAS:
    <p>BMS-863233 HCl is an ATP-competitive Cdc7 inhibitor (IC50: 3.4 nM) that is potent and selective.BMS-863233 HCl inhibited CK2 and PIM1 with IC50 values of 215</p>
    Formula:C14H12ClN3O2·xHCl
    Purity:99.37% - 99.67%
    Color and Shape:Solid
    Molecular weight:326.18
  • BioE-1115

    CAS:
    <p>BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 nM). BioE-1115 is a potent inhibitor of CK2α (IC50 = 10 μM).</p>
    Formula:C19H18FN3O2
    Purity:97.54%
    Color and Shape:Solid
    Molecular weight:339.36
  • Casein kinase 1δ-IN-1

    CAS:
    <p>Casein kinase 1δ-IN-1 (WAY-643895) is an inhibitor of casein kinase 1δ (CK1δ), which inhibits CK1δ.</p>
    Formula:C11H7N3OS
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:229.26
  • Ac-VDVAD-CHO

    CAS:
    <p>Ac-VDVAD-CHO is an inhibitor of caspase-2 and caspase-3 (IC50: 46 nM for caspase-2 and 15 nM for caspase-3) [1].</p>
    Formula:C23H37N5O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:543.57
  • ON 108600

    CAS:
    <p>ON 108600 is a chemical inhibitor targeting CK2 (Casein Kinase 2), TNIK, and DYRK1, demonstrating IC50 values of 0.016 μM and 0.007 μM for DYRK1A and DYRK1B, 0.</p>
    Formula:C22H14Cl2N2O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:537.39
  • Casein kinase 1δ-IN-5

    CAS:
    <p>Casein kinase 1δ-IN-5 is a potent and selective CK-1δ inhibitor, exhibiting an IC50 of 47 nM, and demonstrates neuroprotective and anti-inflammatory effects in</p>
    Formula:C16H11F3N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:336.33
  • Casein kinase 1δ-IN-10

    CAS:
    <p>Casein kinase 1δ-IN-10 is an inhibitor of casein kinase 1δ (CK1δ).</p>
    Formula:C21H17N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.38
  • TID43

    CAS:
    <p>TID43, a CK2 inhibitor, exhibits potent inhibition with an IC50 value of 0.3 μM. It is applicable in anti-angiogenic research [1].</p>
    Formula:C10H3I4NO4
    Color and Shape:Solid
    Molecular weight:708.755
  • XL413 hydrochloride

    CAS:
    <p>XL413 hydrochloride (BMS-863233 Hydrochloride) is a potent, selective and ATP competitive inhibitor of Cdc7. XL413 hydrochloride also inhibits CK2 and PIM1.</p>
    Formula:C14H13Cl2N3O2
    Purity:98.81% - 99.8%
    Color and Shape:Solid
    Molecular weight:326.18
  • Casein kinase 1δ-IN-4

    CAS:
    <p>"Casein kinase 1δ-IN-4 (compound 567) is a potent inhibitor of casein kinase 1δ with potential application in Alzheimer's disease research [1]."</p>
    Formula:C16H12N6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:320.37
  • Casein Kinase II Inhibitor IV

    CAS:
    <p>Casein kinase II inhibitor IV is an effective small molecule inducer, which can be used to induce epidermal keratinocyte differentiation.</p>
    Formula:C24H23N5O3
    Purity:99.65% - 99.75%
    Color and Shape:Solid
    Molecular weight:429.47
  • Casein kinase 1δ-IN-13

    CAS:
    Casein kinase1δ-IN-13 (compound 401) is an inhibitor of Casein kinase1δ. It is utilized in the research of neurodegenerative diseases.
    Formula:C15H13N3O2S
    Color and Shape:Solid
    Molecular weight:299.35
  • Casein kinase 1δ-IN-28

    CAS:
    <p>Casein kinase1δ-IN-28 (Compound 4) is an inhibitor of CK1ε, with an IC50 of 0.0146 μM. The human liver microsome metabolism rate for Casein kinase1δ-IN-28 is 52%.</p>
    Formula:C23H23FN6
    Color and Shape:Solid
    Molecular weight:402.467
  • CK1δ-IN-6

    CAS:
    <p>CK1δ-IN-6 (Compound 303) is an inhibitor of Casein kinase 1δ, with potential applications in Alzheimer's disease research.</p>
    Formula:C23H17N3O4
    Color and Shape:Solid
    Molecular weight:399.399
  • WAY-606344

    CAS:
    <p>WAY-606344 (Compound 97) is an inhibitor of Casein kinase 1δ and shows potential for Alzheimer's disease research.</p>
    Formula:C14H8ClN3O2
    Color and Shape:Solid
    Molecular weight:285.685