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Casein Kinase

Casein Kinase

Casein kinases are a family of serine/threonine protein kinases that regulate various cellular processes, including DNA repair, circadian rhythms, and signal transduction. These kinases are involved in the phosphorylation of numerous proteins and are implicated in diseases such as cancer, neurodegenerative disorders, and metabolic syndromes. At CymitQuimica, we offer a selection of casein kinase inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.

Found 130 products of "Casein Kinase"

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  • Silmitasertib
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    Silmitasertib

    CAS:
    <p>Silmitasertib (CX-4945) is a potent, orally bioavailable inhibitor of casein kinase 2 (CK2; Ki: 0.38 nM).</p>
    Formula:C19H12ClN3O2
    Purity:98% - 99.90%
    Color and Shape:Solid
    Molecular weight:349.77

    Ref: TM-T2259

  • PF-670462
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    PF-670462

    CAS:
    <p>PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (&gt;30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.</p>
    Formula:C19H22Cl2FN5
    Purity:99.42% - 99.72%
    Color and Shape:Solid
    Molecular weight:410.32

    Ref: TM-T3073

  • XL413
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    XL413

    CAS:
    <p>XL-413 is an oral CDC7 kinase inhibitor, potentially blocking DNA replication, mitosis, and cancer cell growth.</p>
    Formula:C14H12ClN3O2
    Purity:98.40% - >99.99%
    Color and Shape:Solid
    Molecular weight:289.72

    Ref: TM-T3352

  • SSTC3
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    SSTC3

    CAS:
    <p>SSTC3 is a casein kinase 1α (CK1α) activator with potential antitumor activity that inhibits WNT signaling.</p>
    Formula:C23H17F3N4O3S2
    Purity:98.65% - 99.94%
    Color and Shape:Solid
    Molecular weight:518.53

    Ref: TM-T13004

  • AMG-548
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    AMG-548

    CAS:
    <p>AMG-548, oral p38α inhibitor (Ki=0.5 nM), &gt;1000x selectivity over p38γ/δ, blocks TNFα (IC50=3 nM), also inhibits Wnt/Casein kinase 1δ/ε.</p>
    Formula:C29H27N5O
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:461.56

    Ref: TM-T10298L

  • SR-1277
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    SR-1277

    CAS:
    <p>SR-1277 is a potent, highly selective and ATP-competitive CK1δ/ε inhibitor, regulating Wee1 activity at the G2/M cell-cycle interface, and antiproliferative.</p>
    Formula:C21H19N9O3S
    Color and Shape:Solid
    Molecular weight:477.5

    Ref: TM-T38927

  • CK2/PIM1-IN-1
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    CK2/PIM1-IN-1

    CAS:
    <p>CK2/PIM1-IN-1 inhibits CK2 &amp; PIM1 (IC50s: 3.787 &amp; 4.327 μM), aimed for cancer research.</p>
    Formula:C15H9NO4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.37

    Ref: TM-T10828

  • 4,5,6,7-Tetrabromobenzimidazole
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    4,5,6,7-Tetrabromobenzimidazole

    CAS:
    <p>4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].</p>
    Formula:C7H2Br4N2
    Color and Shape:Solid
    Molecular weight:433.72

    Ref: TM-T21642

  • CK2-IN-9
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    CK2-IN-9

    CAS:
    <p>CK2-IN-9, a potent and selective CK2 kinase inhibitor, exhibits an inhibitory concentration (IC50) of 3 nM against its target enzyme and hampers Wnt reporter</p>
    Formula:C23H29N9O
    Color and Shape:Solid
    Molecular weight:447.54

    Ref: TM-T78599

  • Quinalizarin
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    Quinalizarin

    CAS:
    <p>Quinalizarin, the most selective CK2 inhibitor, is superior to CX-4945 which is the first-in-class CK2 inhibitor.</p>
    Formula:C14H8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:272.21

    Ref: TM-T20791

  • Tyrphostin AG 1112
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    Tyrphostin AG 1112

    CAS:
    <p>Tyrphostin AG 1112 is a Bcr-Abl kinase blocker. It can activate the terminal differentiation of K562 cells and the purging of Ph+ cells.</p>
    Formula:C15H10N6
    Color and Shape:Solid
    Molecular weight:274.28

    Ref: TM-T24911

  • PF 4800567 hydrochloride
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    PF 4800567 hydrochloride

    CAS:
    <p>casein kinase 1ε inhibitor</p>
    Formula:C17H19Cl2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.27

    Ref: TM-T23138

  • IQA
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    IQA

    CAS:
    <p>IQA is a casein kinase 2 (CK2) inhibitor.</p>
    Formula:C17H12N2O3
    Color and Shape:Solid
    Molecular weight:292.29

    Ref: TM-T69307

  • (R)-DRF053 dihydrochloride
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    (R)-DRF053 dihydrochloride

    CAS:
    <p>cdk/CK1 inhibitor,potent and ATP-competitive</p>
    Formula:C23H29Cl2N7O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:490.43

    Ref: TM-T23224

  • TMCB
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    TMCB

    CAS:
    <p>CK2 and ERK8 inhibitor</p>
    Formula:C11H9Br4N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:534.82

    Ref: TM-T23461

  • CK2-IN-6
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    CK2-IN-6

    CAS:
    <p>CK2-IN-6: Potent CK2 inhibitor for cancer, inflammation, pain, and immune research.</p>
    Formula:C19H16ClN7O2
    Color and Shape:Solid
    Molecular weight:409.83

    Ref: TM-T73380

  • SRPIN-803
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    SRPIN-803

    CAS:
    <p>SRPIN-803 is a selective dual SRPK1 and CK2 inhibitor.</p>
    Formula:C14H9F3N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.31

    Ref: TM-T24832

  • Umbralisib sulfate
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    Umbralisib sulfate

    CAS:
    <p>Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.</p>
    Formula:C31H26F3N5O7S
    Color and Shape:Solid
    Molecular weight:669.63

    Ref: TM-T72527

  • Umbralisib tosylate
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    Umbralisib tosylate

    CAS:
    <p>Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.</p>
    Formula:C38H32F3N5O6S
    Color and Shape:Solid
    Molecular weight:743.75

    Ref: TM-T72465

  • BTX161
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    BTX161

    CAS:
    <p>BTX161: potent CKIα degrader, surpasses Lenalidomide in AML, triggers DDR + p53, stabilizes MDM2.</p>
    Formula:C15H16N2O3
    Color and Shape:Solid
    Molecular weight:272.3

    Ref: TM-T60478