Casein Kinase
Casein kinases are a family of serine/threonine protein kinases that regulate various cellular processes, including DNA repair, circadian rhythms, and signal transduction. These kinases are involved in the phosphorylation of numerous proteins and are implicated in diseases such as cancer, neurodegenerative disorders, and metabolic syndromes. At CymitQuimica, we offer a selection of casein kinase inhibitors to support your research in signal transduction, cell cycle regulation, and therapeutic development.
Found 150 products for "Casein Kinase".
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CKI-7 free base
CAS:CKI-7 free base is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selective Cdc7 kinase inhibitor.Formula:C11H12ClN3O2SColor and Shape:SolidMolecular weight:285.75PF-4800567
CAS:PF-4800567 is a selective inhibitor of casein kinase 1ε (CK1ε; IC50 = 32 nM) with greater than 20-fold selectivity over CK1δ.Formula:C17H18ClN5O2Purity:99.74% - 99.76%Color and Shape:White SolidMolecular weight:359.81Longdaysin
CAS:Longdaysin is an inhibitor of CK1α and CK1δ (IC50s: 5.6/8.8 μM). It also can inhibit ERK2 (IC50: 52 μM).Formula:C16H16F3N5Purity:99.97%Color and Shape:SolidMolecular weight:335.33PF-670462
CAS:PF-670462 is a potent (IC50 = 7.7 ± 2.2 nM) and selective (>30-fold with respect to 42 additional kinases) inhibitor of CK1ε in isolated enzyme preparations.Formula:C19H22Cl2FN5Purity:99.42% - 99.72%Color and Shape:SolidMolecular weight:410.32LY294002
CAS:LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM).Formula:C19H17NO3Purity:98% - 99.96%Color and Shape:White SolidMolecular weight:307.34XL413
CAS:XL-413 is an oral CDC7 kinase inhibitor, potentially blocking DNA replication, mitosis, and cancer cell growth.Formula:C14H12ClN3O2Purity:98.40% - 99.94%Color and Shape:SolidMolecular weight:289.724,5,6,7-Tetrabromobenzimidazole
CAS:4,5,6,7-Tetrabromobenzimidazole is a selective and ATP-competitive inhibitor of protein kinase CK2 [1].Formula:C7H2Br4N2Color and Shape:SolidMolecular weight:433.72CK2-IN-9
CAS:CK2-IN-9, a potent and selective CK2 kinase inhibitor, exhibits an inhibitory concentration (IC50) of 3 nM against its target enzyme and hampers Wnt reporterFormula:C23H29N9OColor and Shape:SolidMolecular weight:447.54Tyrphostin AG 1112
CAS:Tyrphostin AG 1112 is a Bcr-Abl kinase blocker. It can activate the terminal differentiation of K562 cells and the purging of Ph+ cells.Formula:C15H10N6Color and Shape:SolidMolecular weight:274.28PF 4800567 hydrochloride
CAS:casein kinase 1ε inhibitorFormula:C17H19Cl2N5O2Purity:98%Color and Shape:SolidMolecular weight:396.27CK1-IN-2
CAS:CK1-IN-2 (compound Nr.4) is a potent CK1 inhibitor p38a, and is used in DUX4 overexpression-associated diseases, such as muscular dystrophy.Formula:C17H12FN3O2Purity:99.31%Color and Shape:SolidMolecular weight:309.29IQA
CAS:IQA is a casein kinase 2 (CK2) inhibitor.Formula:C17H12N2O3Color and Shape:SolidMolecular weight:292.29SSTC3
CAS:SSTC3 is a casein kinase 1α (CK1α) activator with potential antitumor activity that inhibits WNT signaling.Formula:C23H17F3N4O3S2Purity:98.65% - 99.94%Color and Shape:SolidMolecular weight:518.53Ref: TM-T13004
1mg94.00€5mg222.00€1mL*10mM (DMSO)225.00€10mg356.00€25mg583.00€50mg820.00€100mg1,099.00€(R)-DRF053 dihydrochloride
CAS:(R)-DRF053 dihydrochloride is a CK1 and CDK inhibitor, also inhibiting CDK1/cyclin B and CDK5/p25, used for studying cell cycle regulation.Formula:C23H29Cl2N7OPurity:98%Color and Shape:SolidMolecular weight:490.43SR-1277
CAS:SR-1277 is a potent, highly selective and ATP-competitive CK1δ/ε inhibitor, regulating Wee1 activity at the G2/M cell-cycle interface, and antiproliferative.Formula:C21H19N9O3SColor and Shape:SolidMolecular weight:477.5TMCB
CAS:CK2 and ERK8 inhibitorFormula:C11H9Br4N3O2Purity:98%Color and Shape:SolidMolecular weight:534.82CK2-IN-6
CAS:CK2-IN-6: Potent CK2 inhibitor for cancer, inflammation, pain, and immune research.Formula:C19H16ClN7O2Color and Shape:SolidMolecular weight:409.83SRPIN-803
CAS:SRPIN-803 is a selective dual SRPK1 and CK2 inhibitor.Formula:C14H9F3N4O3SPurity:98%Color and Shape:SolidMolecular weight:370.31Umbralisib sulfate
CAS:Umbralisib sulfate, an oral dual PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), targets CLL T cells for blood cancer research.Formula:C31H26F3N5O7SColor and Shape:SolidMolecular weight:669.63Umbralisib tosylate
CAS:Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.Formula:C38H32F3N5O6SColor and Shape:SolidMolecular weight:743.75
