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Retinoid Receptor

Retinoid Receptor

Retinoid Receptors are nuclear receptors that mediate the effects of retinoids (vitamin A derivatives) on gene expression. These receptors play a vital role in cell differentiation, proliferation, and apoptosis. Inhibitors of retinoid receptors are used to study their involvement in various diseases, including cancer, skin disorders, and metabolic conditions. By modulating retinoid receptor activity, these inhibitors can provide insights into the mechanisms of retinoid signaling and its therapeutic potential. At CymitQuimica, we provide retinoid receptor inhibitors to support your research in dermatology, oncology, and metabolic regulation.

Found 29 products of "Retinoid Receptor"

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  • LG-100064
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    LG-100064

    CAS:
    <p>LG-100064 is an agonist of retinoid-X-receptor (RXR)(EC50s of 330 nM, 200 nM, and 260 nM for RXRα, RXRβ and RXRγ)</p>
    Formula:C23H26O3
    Purity:98.65%
    Color and Shape:Solid
    Molecular weight:350.45

    Ref: TM-T11844

  • BMS 195614
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    BMS 195614

    CAS:
    <p>BMS 195614 (BMS614) is a selective RARα antagonist. BMS 195614 can bind to the RARα subunit.</p>
    Formula:C29H24N2O3
    Purity:97.7%
    Color and Shape:Solid
    Molecular weight:448.51

    Ref: TM-T22192

  • CD3254
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    CD3254

    CAS:
    <p>CD3254 is a selective and potent retinoid X receptor-like (RXR) agonist that inhibits neuronal cell death with OGD/reoxygenation.</p>
    Formula:C24H28O3
    Purity:98.71% - 98.71%
    Color and Shape:Solid
    Molecular weight:364.48

    Ref: TM-T14912

  • CD437
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    CD437

    CAS:
    <p>CD437 (AHPN) is a specifc Retinoic Acid Receptor γ (RARγ) agonist.</p>
    Formula:C27H26O3
    Purity:98.92% - 99.63%
    Color and Shape:Solid
    Molecular weight:398.49

    Ref: TM-T4371

  • Tazarotene
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    Tazarotene

    CAS:
    <p>Tazarotene (Zorac), a synthetic topical retinoid, treats psoriasis by normalizing keratinocytes and reducing growth.</p>
    Formula:C21H21NO2S
    Purity:97.01% - 99.14%
    Color and Shape:White Solid
    Molecular weight:351.46

    Ref: TM-T6696

  • Fenretinide
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    Fenretinide

    CAS:
    <p>Fenretinide (4-HPR) is an orally-active synthetic retinoid derivative with potential antineoplastic and chemopreventive activities.</p>
    Formula:C26H33NO2
    Purity:98% - 99.68%
    Color and Shape:Yellow Powder
    Molecular weight:391.55

    Ref: TM-T1872

  • AGN 193109
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    AGN 193109

    CAS:
    <p>AGN 193109, a retinoid analog, is a potent and specific antagonist of RARs (Kds: 2 nM, 2 nM, and 3 nM for RARα, RARβ, and RARγ).</p>
    Formula:C28H24O2
    Purity:99.87% - 99.89%
    Color and Shape:Solid
    Molecular weight:392.49

    Ref: TM-TQ0097

  • UVI 3003
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    UVI 3003

    CAS:
    <p>UVI 3003 blocks retinoid X receptor (RXRα) in Xenopus/human Cos7 cells; IC50: 0.22/0.24 μM.</p>
    Formula:C28H36O4
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:436.58

    Ref: TM-T17209

  • AR7
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    AR7

    CAS:
    <p>AR7 is a retinoic acid receptor α (RARα) antagonist.</p>
    Formula:C15H12ClNO
    Purity:98.12% - 99.86%
    Color and Shape:Solid
    Molecular weight:257.71

    Ref: TM-T3955

  • palovarotene
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    palovarotene

    CAS:
    <p>Palovarotene (Ro 3300074) is an agonist of nuclear retinoic acid receptor γ (RAR-γ).</p>
    Formula:C27H30N2O2
    Purity:97.88% - 98.05%
    Color and Shape:Solid
    Molecular weight:414.54

    Ref: TM-T4538

  • Tarenflurbil
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    Tarenflurbil

    CAS:
    <p>Tarenflurbil, the R-enantiomer of flurbiprofen, lacks COX inhibition and was tested for Alzheimer's treatment.</p>
    Formula:C15H13FO2
    Purity:98% - 99.9%
    Color and Shape:Solid
    Molecular weight:244.26

    Ref: TM-T5843

  • trifarotene
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    trifarotene

    CAS:
    <p>Trifarotene (CD5789) is a RARγ agonist, 65x more selective than RARα and 16x than RARβ, with EC50 of 7.7 nM.</p>
    Formula:C29H33NO4
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:459.58

    Ref: TM-T7586

  • Bexarotene
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    Bexarotene

    CAS:
    <p>Bexarotene (LGD1069) is a retinoid analogue that is used to treat the skin manifestations of cutaneous T cell lymphoma (CTCL).</p>
    Formula:C24H28O2
    Purity:99% - 99.65%
    Color and Shape:White Solid
    Molecular weight:348.48

    Ref: TM-T6410

  • BMS270394
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    BMS270394

    CAS:
    <p>BMS270394 is a RARγ agonist used in the study of breast cancer and skin diseases.</p>
    Formula:C23H26FNO4
    Color and Shape:Solid
    Molecular weight:399.46

    Ref: TM-T26846

  • CD 1530
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    CD 1530

    CAS:
    <p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>
    Formula:C27H26O3
    Purity:98.13%
    Color and Shape:Solid
    Molecular weight:398.49

    Ref: TM-T21686

  • CD2665
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    CD2665

    CAS:
    <p>CD2665 is an orally active antagonist of retinoic acid receptor (RAR). For RARγ and RARβ, the Kis are 110 nM and 306 nM.</p>
    Formula:C31H34O5
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:486.6

    Ref: TM-T14911

  • Ch55
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    Ch55

    CAS:
    <p>Ch55, a potent HL60 cell differentiator (EC50=200nM), binds well to RAR-α/β, useful for cancer research.</p>
    Formula:C24H28O3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:364.48

    Ref: TM-T14946

  • AGN 196996
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    AGN 196996

    CAS:
    <p>AGN 196996: strong RARα inhibitor (Ki: 2 nM), weak for RARβ/γ (Ki: 1087/8523 nM).</p>
    Formula:C24H20BrNO5
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:482.32

    Ref: TM-T10261

  • BMS 753
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    BMS 753

    CAS:
    <p>BMS 753 is an agonist of isotype-selective retinoic acid receptor α (RARα, Ki= 2 nM).</p>
    Formula:C21H21NO4
    Purity:98.55%
    Color and Shape:Solid
    Molecular weight:351.4

    Ref: TM-T22049

  • Fluorobexarotene
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    Fluorobexarotene

    CAS:
    <p>Fluorobexarotene, a potent RXR agonist, has 75% higher affinity than Bexarotene with Ki of 12 nM and EC50 of 43 nM for RXRα.</p>
    Formula:C24H27FO2
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:366.47

    Ref: TM-T11303