Retinoid Receptor
Retinoid Receptors are nuclear receptors that mediate the effects of retinoids (vitamin A derivatives) on gene expression. These receptors play a vital role in cell differentiation, proliferation, and apoptosis. Inhibitors of retinoid receptors are used to study their involvement in various diseases, including cancer, skin disorders, and metabolic conditions. By modulating retinoid receptor activity, these inhibitors can provide insights into the mechanisms of retinoid signaling and its therapeutic potential. At CymitQuimica, we provide retinoid receptor inhibitors to support your research in dermatology, oncology, and metabolic regulation.
Found 26 products of "Retinoid Receptor"
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LG-100064
CAS:LG-100064 is an agonist of retinoid-X-receptor (RXR)(EC50s of 330 nM, 200 nM, and 260 nM for RXRα, RXRβ and RXRγ)Formula:C23H26O3Purity:98.65%Color and Shape:SolidMolecular weight:350.45Ref: TM-T11844
2mg47.00€5mg70.00€10mg97.00€25mg167.00€50mg249.00€100mg369.00€200mg545.00€1mL*10mM (DMSO)77.00€BMS 195614
CAS:BMS 195614 (BMS614) is a selective RARα antagonist. BMS 195614 can bind to the RARα subunit.Formula:C29H24N2O3Purity:97.14%Color and Shape:SolidMolecular weight:448.51CD3254
CAS:CD3254 is a selective and potent retinoid X receptor-like (RXR) agonist that inhibits neuronal cell death with OGD/reoxygenation.Formula:C24H28O3Purity:98.71% - 98.71%Color and Shape:SolidMolecular weight:364.48CD437
CAS:CD437 (AHPN) is a specifc Retinoic Acid Receptor γ (RARγ) agonist.Formula:C27H26O3Purity:98.92% - 99.63%Color and Shape:SolidMolecular weight:398.49Tazarotene
CAS:Tazarotene (Zorac), a synthetic topical retinoid, treats psoriasis by normalizing keratinocytes and reducing growth.Formula:C21H21NO2SPurity:97.01% - 99.14%Color and Shape:White SolidMolecular weight:351.46Ref: TM-T6696
5mg38.00€10mg49.00€25mg88.00€50mg147.00€100mg256.00€200mg334.00€500mg563.00€1mL*10mM (DMSO)55.00€Fenretinide
CAS:Fenretinide (4-HPR) is an orally-active synthetic retinoid derivative with potential antineoplastic and chemopreventive activities.Formula:C26H33NO2Purity:98% - 99.68%Color and Shape:Yellow PowderMolecular weight:391.55UVI 3003
CAS:UVI 3003 blocks retinoid X receptor (RXRα) in Xenopus/human Cos7 cells; IC50: 0.22/0.24 μM.Formula:C28H36O4Purity:99.82%Color and Shape:SolidMolecular weight:436.58Ref: TM-T17209
1mg35.00€2mg52.00€5mg74.00€10mg119.00€25mg243.00€50mg406.00€100mg607.00€1mL*10mM (DMSO)86.00€AR7
CAS:AR7 is a retinoic acid receptor α (RARα) antagonist.Formula:C15H12ClNOPurity:98.12% - 99.86%Color and Shape:SolidMolecular weight:257.71Ref: TM-T3955
1mg37.00€5mg69.00€10mg96.00€25mg202.00€50mg329.00€100mg550.00€200mg758.00€500mg1,159.00€1mL*10mM (DMSO)74.00€palovarotene
CAS:<p>Palovarotene (Ro 3300074) is an agonist of nuclear retinoic acid receptor γ (RAR-γ).</p>Formula:C27H30N2O2Purity:97.88% - 98.05%Color and Shape:SolidMolecular weight:414.54trifarotene
CAS:<p>Trifarotene (CD5789) is a RARγ agonist, 65x more selective than RARα and 16x than RARβ, with EC50 of 7.7 nM.</p>Formula:C29H33NO4Purity:99.51%Color and Shape:SolidMolecular weight:459.58Bexarotene
CAS:Bexarotene (LGD1069) is a retinoid analogue that is used to treat the skin manifestations of cutaneous T cell lymphoma (CTCL).Formula:C24H28O2Purity:99% - 99.65%Color and Shape:White SolidMolecular weight:348.48BMS270394
CAS:BMS270394 is a RARγ agonist used in the study of breast cancer and skin diseases.Formula:C23H26FNO4Color and Shape:SolidMolecular weight:399.46CD2665
CAS:CD2665 is an orally active antagonist of retinoic acid receptor (RAR). For RARγ and RARβ, the Kis are 110 nM and 306 nM.Formula:C31H34O5Purity:99.71%Color and Shape:SolidMolecular weight:486.6MM 11253
CAS:MM 11253 is a RARγ antagonist with IC50 of 44nM.Formula:C28H30O2S2Purity:99.41%Color and Shape:SolidMolecular weight:462.67Ch55
CAS:Ch55, a potent HL60 cell differentiator (EC50=200nM), binds well to RAR-α/β, useful for cancer research.Formula:C24H28O3Purity:99.55%Color and Shape:SolidMolecular weight:364.48Ref: TM-T14946
1mg42.00€5mg87.00€10mg124.00€25mg254.00€50mg394.00€100mg612.00€200mg842.00€1mL*10mM (DMSO)94.00€Fluorobexarotene
CAS:Fluorobexarotene, a potent RXR agonist, has 75% higher affinity than Bexarotene with Ki of 12 nM and EC50 of 43 nM for RXRα.Formula:C24H27FO2Purity:99.08%Color and Shape:SolidMolecular weight:366.47Ref: TM-T11303
1mg170.00€5mg416.00€10mg615.00€25mg964.00€50mg1,305.00€100mg1,755.00€500mg3,501.00€1mL*10mM (DMSO)335.00€BMS 753
CAS:<p>BMS 753 is an agonist of isotype-selective retinoic acid receptor α (RARα, Ki= 2 nM).</p>Formula:C21H21NO4Purity:98.55%Color and Shape:SolidMolecular weight:351.4AGN 196996
CAS:AGN 196996: strong RARα inhibitor (Ki: 2 nM), weak for RARβ/γ (Ki: 1087/8523 nM).Formula:C24H20BrNO5Purity:99.94%Color and Shape:SolidMolecular weight:482.32Ref: TM-T10261
1mg59.00€5mg131.00€10mg190.00€25mg329.00€50mg477.00€100mg702.00€1mL*10mM (DMSO)138.00€AC-261066
CAS:AC-261066 is an orally available and isoform-selective agonist of RARβ2 with a pEC50 of 8.0.Formula:C17H20FNO4SPurity:99.64%Color and Shape:SolidMolecular weight:353.41KCL-286
CAS:KCL-286 is an available and potent retinoic acid receptor beta agonist for the amelioration of spinal cord injury (SCI).Formula:C19H14N2O4Purity:99.93%Color and Shape:SolidMolecular weight:334.33
