P450
Cytochrome P450 enzymes are a large family of enzymes involved in the metabolism of various endogenous and exogenous compounds, including drugs, toxins, and hormones. P450 inhibitors are widely used to study drug metabolism, pharmacokinetics, and the role of these enzymes in disease states such as cancer and liver disorders. At CymitQuimica, we provide a broad selection of P450 inhibitors to support your research in pharmacology, toxicology, and metabolic regulation.
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Harman hydrochloride
CAS:21655-84-5
Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.
Formula:
C12H11ClN2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
218.68
Ref: TM-T3158L
| 5mg | 42.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 133.00 € | ||
| 100mg | 182.00 € | ||
| 200mg | 287.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Choline Fenofibrate
CAS:856676-23-8
Choline Fenofibrate (Trilipix) is a choline formulation of fenofibrate, a synthetic phenoxy-isobutyric acid derivate and …
Formula:
C22H28ClNO5
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
421.91
Ref: TM-T3941
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 149.00 € | ||
| 100mg | 213.00 € | ||
| 200mg | 316.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Demethyleneberberine
CAS:25459-91-0
Demethyleneberberine, which is composed of a potential antioxidant structure, could penetrate the membrane of mitochondria …
Formula:
C19H18NO4
Purity:
98.08% - 99.18%
Color and Shape:
Solid
Molecular weight:
324.35
Ref: TM-T4S0800
| 1mg | 66.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 323.00 € | ||
| 50mg | 479.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
XL388
CAS:1251156-08-7
XL388 is a highly effective, specifc, ATP-competitive inhibitor of mTOR ( IC50: 9.9 nM), 1000-fold …
Formula:
C23H22FN3O4S
Purity:
99.39% - 99.53%
Color and Shape:
Solid
Molecular weight:
455.5
Ref: TM-T6030
| 1mg | 45.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 456.00 € | ||
| 100mg | 669.00 € | ||
| 1mL*10mM (DMSO) | 107.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Sulfaphenazole
CAS:526-08-9
Sulfaphenazole (Plisulfan) is an inhibitor of CYP2C9 (Ki: 0.3 μM) that demonstrates at least 100-fold …
Formula:
C15H14N4O2S
Purity:
97.53% - 99.67%
Color and Shape:
Solid
Molecular weight:
314.36
Ref: TM-T4567
| 100mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Cobicistat
CAS:1004316-88-4
Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for …
Formula:
C40H53N7O5S2
Purity:
97.36% - 99.62%
Color and Shape:
Solid
Molecular weight:
776.02
Ref: TM-T6246
| 1mg | 45.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 345.00 € | ||
| 100mg | 495.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Tebuconazole
CAS:107534-96-3
Tebuconazole: azole fungicide, inhibits CYP51 with IC50s 0.9 μM (C. albicans) and 1.3 μM (human).
Formula:
C16H22ClN3O
Purity:
99.21%
Color and Shape:
Solid
Molecular weight:
307.82
Ref: TM-T17022
| 500mg | 55.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
1-Ethynylpyrene
CAS:34993-56-1
1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and …
Formula:
C18H10
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
226.27
Ref: TM-T9704
| 200mg | 38.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Diflubenzuron
CAS:35367-38-5
Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis …
Formula:
C14H9ClF2N2O2
Purity:
98.53% - 99.83%
Color and Shape:
Colorless Crystals Diflubenzuron Is A Colorless To Yellow Crystals Used As A Selective Insecticide
Molecular weight:
310.68
Ref: TM-T7088
| 1g | 184.00 € | ||
| 25mg | 35.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 63.00 € | ||
| 500mg | 129.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Curdione
CAS:13657-68-6
Curdione hampers CYP3A4 and PGE2 synthesis, curbs MCF-7 cell growth by triggering apoptosis, and is …
Formula:
C15H24O2
Purity:
98% - 99.79%
Color and Shape:
Solid
Molecular weight:
236.35
Ref: TM-T3411
| 10mg | 48.00 € | ||
| 25mg | 76.00 € | ||
| 50mg | 111.00 € | ||
| 100mg | 171.00 € | ||
| 200mg | 242.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Dronedarone
CAS:141626-36-0
Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for …
Formula:
C31H44N2O5S
Purity:
98.85% - 99.58%
Color and Shape:
Solid
Molecular weight:
556.76
Ref: TM-T7056
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 134.00 € | ||
| 100mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
7-Hydroxyflavone
CAS:6665-86-7
7-Hydroxyflavone is a potent inhibitor of CYP1A1 with a Ki value of 0.015 μM and …
Formula:
C15H10O3
Purity:
99.79%
Color and Shape:
Off-White Crystals
Molecular weight:
238.24
Ref: TM-T7472
| 100mg | 54.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Norfluoxetine Hydrochloride
CAS:57226-68-3
Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.
Formula:
C16H17ClF3NO
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
331.76
Ref: TM-T21029
| 1mg | 48.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 224.00 € | ||
| 25mg | 371.00 € | ||
| 50mg | 492.00 € | ||
| 100mg | 716.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
SDZ285428
CAS:174262-13-6
SDZ285428 is a CYP24A1 inhibitor.
Formula:
C24H20ClN3O
Purity:
97.51%
Color and Shape:
Solid
Molecular weight:
401.89
Ref: TM-T4188
| 2mg | 36.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 362.00 € | ||
| 200mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
1-Ethynylnaphthalene
CAS:15727-65-8
1-Ethynylnaphthalene is a selective inhibitor of cytochrome P450 IB1
Formula:
C12H8
Purity:
99.27% - ≥95%
Color and Shape:
Yellow To Brown Liquid
Molecular weight:
152.19
Ref: TM-T7427
| 100mg | 53.00 € | ||
| 500mg | 92.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Miltirone
CAS:27210-57-7
Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central …
Formula:
C19H22O2
Purity:
99.22% - 99.66%
Color and Shape:
Solid
Molecular weight:
282.38
Ref: TM-TN1023
| 1mg | 131.00 € | ||
| 5mg | 200.00 € | ||
| 10mg | 326.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 772.00 € | ||
| 100mg | 1,023.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Rosavin
CAS:84954-92-7
Rosavin (Rosavidin) has antidepressant and anxiolytic actions, helps balance all the neurotransmitters.
Formula:
C20H28O10
Purity:
99.38% - 99.99%
Color and Shape:
Solid
Molecular weight:
428.43
Ref: TM-T3886
| 20mg | 112.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Acetylshikonin
CAS:24502-78-1
Acetylshikonin, an AChE inhibitor and a non-selective cytochrome P450 inhibitor, is derived from Comfrey and …
Formula:
C18H18O6
Purity:
92.45% - 97.56%
Color and Shape:
Solid
Molecular weight:
330.33
Ref: TM-T5S2343
| 1mg | 41.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 132.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 547.00 € | ||
| 500mg | 1,188.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Eupatorin
CAS:855-96-9
Eupatorin inhibits cancer cell growth, angiogenesis, and inflammation, inducing apoptosis via ROS.
Formula:
C18H16O7
Purity:
98.09% - 98.09%
Color and Shape:
Solid
Molecular weight:
344.32
Ref: TM-T7032
| 1mg | 48.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
Gentiopicroside
CAS:20831-76-9
Gentiopicroside, an iridoid from Gentiana manshurica, inhibits CYP2A6 (IC50=61μM, Ki=22.8μM), and has anti-inflammatory and antioxidant …
Formula:
C16H20O9
Purity:
98% - 99.8%
Color and Shape:
White Powder
Molecular weight:
356.32
Ref: TM-T2770
| 5mg | 45.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 313.00 € | ||
| 500mg | 730.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 12 Dec 2024
