P450
Cytochrome P450 enzymes are a large family of enzymes involved in the metabolism of various endogenous and exogenous compounds, including drugs, toxins, and hormones. P450 inhibitors are widely used to study drug metabolism, pharmacokinetics, and the role of these enzymes in disease states such as cancer and liver disorders. At CymitQuimica, we provide a broad selection of P450 inhibitors to support your research in pharmacology, toxicology, and metabolic regulation.
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EN3356
CAS:1429329-63-4
EN3356 is an orally available and selective inhibitor of steroidal 17-alpha-hydroxylase/C17,20 cleavage enzyme (CYP17A1 or …
Formula:
C16H13FN2OS
Purity:
97.47%
Color and Shape:
Soild
Molecular weight:
300.35
Ref: TM-T30161
| 1mg | 87.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 734.00 € | ||
| 100mg | 1,007.00 € | ||
| 500mg | 2,046.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
(S)-(+)-N-3-Benzylnirvanol
CAS:790676-40-3
(S)-(+)-N-3-Benzylnirvanol is a cytochrome P450 CYP2C19 inhibitor with a ki value of 82.5μM for CYP2C9 …
Formula:
C18H18N2O2
Purity:
98.76%
Color and Shape:
Soild
Molecular weight:
294.35
Ref: TM-T67926
| 1mg | 142.00 € | ||
| 5mg | 351.00 € | ||
| 10mg | 519.00 € | ||
| 25mg | 820.00 € | ||
| 50mg | 1,104.00 € | ||
| 100mg | 1,466.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Canadine
CAS:5096-57-1
Canadine has antioxidant activity with low-toxic effect.
Formula:
C20H21NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
339.39
Ref: TM-TN3574
| 1mg | 72.00 € | ||
| 5mg | 259.00 € | ||
| 10mg | 456.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
AG 045572
CAS:263847-55-8
AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans …
Formula:
C30H37NO5
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
491.62
Ref: TM-T22025
| 1mg | 119.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 323.00 € | ||
| 25mg | 522.00 € | ||
| 50mg | 730.00 € | ||
| 100mg | 993.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
MS-PPOH
CAS:206052-02-0
MS-PPOH is a potent and selective inhibitor of cytochrome P450 (CYP) epoxygenase. MS-PPOH inhibits CYP2C8 …
Formula:
C16H21NO4S
Purity:
98.42%
Color and Shape:
Liquid
Molecular weight:
323.41
Ref: TM-T41291
| 5mg | 51.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
CYP1B1-IN-7
CAS:52601-58-8
CYP1B1-IN-7 is a CYP1B1 inhibitor that can be used in synergy with anticancer compounds for …
Formula:
C19H13ClO
Purity:
99.49%
Color and Shape:
Soild
Molecular weight:
292.76
Ref: TM-T85344
| 1mg | 181.00 € | ||
| 5mg | 447.00 € | ||
| 10mg | 641.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,379.00 € | ||
| 100mg | 1,823.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
TP0472993
CAS:2126874-77-7
CYP4A11/CYP4F2-IN-2: Potent oral inhibitor of CYP4A11 & CYP4F2 (IC50: 140 & 40 nM), potential kidney …
Formula:
C16H20N4O2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
300.36
Ref: TM-T67916
| 1mg | 52.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 315.00 € | ||
| 50mg | 508.00 € | ||
| 100mg | 733.00 € | ||
| 500mg | 1,513.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
BI 653048 phosphate
CAS:1198784-97-2
BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : …
Formula:
C23H28F4N3O8PS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
613.52
Ref: TM-T10535L
| 25mg | 1,435.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
α-Viniferin
CAS:62218-13-7
α-Viniferin known as 2-arylbenzofuran flavonoids, that are inhibitors of prostaglandin H2 synthetase. α-Viniferin has anti-Alzheimer's …
Formula:
C42H30O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
678.68
Ref: TM-TN1378
| 5mg | To inquire | ||
| 1ml*10 (DMSO) | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
N-desmethyl Olanzapine
CAS:161696-76-0
N-desmethyl Olanzapine, a metabolite of Olanzapine, is created via CYP1A2 oxidative metabolism.
Formula:
C16H18N4S
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
298.41
Ref: TM-T35716
| 1mg | 41.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 498.00 € | ||
| 50mg | 714.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Dipterocarpol
CAS:471-69-2
Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng.
Formula:
C30H50O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
442.728
Ref: TM-TN3875
| 5mg | 586.00 € | ||
| 1mL*10mM (DMSO) | 595.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Humantenirine
CAS:82375-30-2
Humantenirine is a natural product of Gelsemium, Loganiaceae.
Formula:
C21H26N2O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
370.44
Ref: TM-TN1748
| 5mg | 618.00 € | ||
| 1mL*10mM (DMSO) | 627.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Pregnenolone Carbonitrile
CAS:1434-54-4
Pregnenolone Carbonitrile (5-Pregnen-3β-ol-20-one-16α-carbonitrile) is an activator of rodent-PXR and induces the expression of CYP3A.
Formula:
C22H31NO2
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
341.49
Ref: TM-T21818
| 5mg | 53.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
CAY10434
CAS:769917-29-5
CAY10434, a potent CYP4A hydroxylase inhibitor, has an IC50 of 8.8 nM and boosts angiotensin …
Formula:
C17H25N3O
Purity:
99.07%
Color and Shape:
Liquid
Molecular weight:
287.4
Ref: TM-T37825
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 136.00 € | ||
| 25mg | 280.00 € | ||
| 50mg | 409.00 € | ||
| 100mg | 555.00 € | ||
| 200mg | 734.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Opevesostat
CAS:2231294-96-3
Opevesostat (ODM-208) is an inhibitor of lyase (CYP11A1) (the enzyme cleavage cholesterol side chain).
Formula:
C21H26N2O5S
Purity:
99.25%
Color and Shape:
Soild
Molecular weight:
418.51
Ref: TM-T77627
| 1mg | 35.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 291.00 € | ||
| 100mg | 430.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
15-Hydroxydehydroabietic acid
CAS:54113-95-0
15-Hydroxydehydroabietic acid exhibits a promising alpha-glucosidase inhibitory activity, it also shows significant antibacterial activities.
Formula:
C20H28O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
316.441
Ref: TM-TMA0164
| 5mg | 453.00 € | ||
| 1mL*10mM (DMSO) | 463.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
CAY10462
CAS:502656-68-0
CAY10462 (CTK8E8405) is an effective and selective inhibitor of the 20-HETE synthase CYP4A11 with an …
Formula:
C17H27Cl2N3O
Purity:
99.49%
Color and Shape:
Liquid
Molecular weight:
360.32
Ref: TM-T37826
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 198.00 € | ||
| 50mg | 297.00 € | ||
| 100mg | 428.00 € | ||
| 200mg | 595.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
7-BFC
CAS:220001-53-6
7-BFC (7-Benzyloxy-4-(trifluoromethyl)coumarin) is a coumarin-like fluorescent substrate that is a cytochrome marker for the study …
Formula:
C17H11F3O3
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
320.26
Ref: TM-T117521
| 5mg | 47.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 322.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
6',7'-Dihydroxybergamottin
CAS:264234-05-1
6',7'-Dihydroxybergamottin (DHB) inhibits CYP3A4 and POR; affects nifedipine oxidation.
Formula:
C21H24O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.41
Ref: TM-TN3147
| 10mg | 2,837.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
BI 653048
CAS:1198784-72-3
BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). …
Formula:
C23H25F4N3O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
515.52
Ref: TM-T10535
| 25mg | 1,435.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
