P450
Cytochrome P450 enzymes are a large family of enzymes involved in the metabolism of various endogenous and exogenous compounds, including drugs, toxins, and hormones. P450 inhibitors are widely used to study drug metabolism, pharmacokinetics, and the role of these enzymes in disease states such as cancer and liver disorders. At CymitQuimica, we provide a broad selection of P450 inhibitors to support your research in pharmacology, toxicology, and metabolic regulation.
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Albaconazole
CAS:187949-02-6
Albaconazole, a small fungal CYP51A1 inhibitor, treats fungal infections and some musculoskeletal disorders.
Formula:
C20H16ClF2N5O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
431.82
Ref: TM-T7725
| 1mg | 327.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Cholesterol 24-hydroxylase-IN-1
CAS:1613480-70-8
Cholesterol 24-hydroxylase-IN-1 is a cholesterol 24-hydroxylase (CH24H or CYP46A1) inhibitor used in the study of …
Formula:
C17H23N5O
Purity:
98.40%
Color and Shape:
Liquid
Molecular weight:
313.40
Ref: TM-T60796
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 171.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
BMS-819881
CAS:1197420-05-5
BMS-819881 is a melaninconcentrating hormone receptor 1 (MCHR1) antagonist, which binds rat MCHR1 with a …
Formula:
C24H21ClN2O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
468.95
Ref: TM-T14678
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Vorozole
CAS:129731-10-8
Vorozole (R83842) is an orally active, potent, and selective nonsteroidal aromatase inhibitor.Vorozole exhibits antitumor activity …
Formula:
C16H13ClN6
Purity:
100% - 99%
Color and Shape:
Solid
Molecular weight:
324.77
Ref: TM-T26322
| 1mg | 178.00 € | ||
| 5mg | 446.00 € | ||
| 10mg | 638.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,375.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CYP1B1-IN-1
CAS:842122-33-2
CYP1B1-IN-1 is a selective and potent cytochrome P450 1B1 (CYP1B1) inhibitor with potential anticancer and …
Formula:
C19H11ClO2
Purity:
99.81%
Color and Shape:
Solid
Molecular weight:
306.74
Ref: TM-T60723
| 25mg | 1,967.00 € | ||
| 50mg | 2,559.00 € | ||
| 100mg | 3,235.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CYP4A11/CYP4F2-IN-1
CAS:502654-40-2
CYP4A11/CYP4F2-IN-1 is a cytochrome P450 (CYP) 4A11 and CYP4F2 inhibitor for the study of kidney …
Formula:
C15H15N3OS
Purity:
99.75%
Color and Shape:
Liquid
Molecular weight:
285.36
Ref: TM-T72501
| 1mg | 96.00 € | ||
| 2mg | 124.00 € | ||
| 5mg | 201.00 € | ||
| 10mg | 295.00 € | ||
| 25mg | 498.00 € | ||
| 50mg | 709.00 € | ||
| 100mg | 931.00 € | ||
| 500mg | 1,866.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Nampt activator-2
CAS:2237268-90-3
Nampt activator-2: Potent NAMPT activator (EC50: 0.023 μM), binds CYP2C9 (0.060 μM), 2D6 (0.41 μM), …
Formula:
C17H15ClN4O3S
Purity:
98.31% - 98.46%
Color and Shape:
Liquid
Molecular weight:
390.84
Ref: TM-T72617
| 1mg | 90.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 616.00 € | ||
| 50mg | 925.00 € | ||
| 100mg | 1,565.00 € | ||
| 500mg | 3,146.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Enerisant HCl
CAS:1152749-07-9
Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for …
Formula:
C22H31ClN4O3
Purity:
99.66%
Color and Shape:
Liquid
Molecular weight:
434.96
Ref: TM-T70489
| 1mg | 90.00 € | ||
| 5mg | 211.00 € | ||
| 10mg | 339.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 795.00 € | ||
| 100mg | 1,067.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CYP1B1-IN-5
CAS:176442-56-1
CYP1B1-IN-5: selective CYP1B1 inhibitor, IC50 = 4.7 nM, useful for metabolism disease research.
Formula:
C14H8INO2
Purity:
98.61%
Color and Shape:
Liquid
Molecular weight:
349.12
Ref: TM-T73042
| 1mg | 182.00 € | ||
| 5mg | 450.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,389.00 € | ||
| 100mg | 1,835.00 € | ||
| 500mg | 3,661.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
YM 511
CAS:148869-05-0
YM 511 is a specific non-steroidal aromatase inhibitor with IC50s of 0.4 and 0.12 nM, …
Formula:
C16H12BrN5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
354.2
Ref: TM-T23549
| 1mg | 37.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 253.00 € | ||
| 50mg | 404.00 € | ||
| 100mg | 547.00 € | ||
| 200mg | 724.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CYP11B2-IN-1
CAS:1356479-78-1
CYP11B2-IN-1 is an effective and selective inhibitor of CYP11B2 with IC50s of 2.3 nM and …
Formula:
C18H18FN3O
Purity:
97.89% - 98.39%
Color and Shape:
Solid
Molecular weight:
311.35
Ref: TM-T10922
| 1mg | 48.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 148.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 359.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Antihistamine-1
CAS:1186430-60-3
Antihistamine-1: H1 blocker, Ki 6.9 nM, crosses blood-brain barrier, inhibits CYP2D6 & hERG (IC50: 5.4 …
Formula:
C23H24FN5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
389.47
Ref: TM-T10335
| 5mg | 57.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 327.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CYP1B1-IN-4
CAS:2685779-55-7
CYP1B1-IN-4: 2,4-diarylthiazole, selective CYP1B1 inhibitor (IC50=0.2 nM), low cytotoxicity, stable in liver microsomes.
Formula:
C18H14N2O2S
Purity:
98.38%
Color and Shape:
Liquid
Molecular weight:
322.38
Ref: TM-T73040
| 5mg | 59.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 398.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Casopitant mesylate
CAS:414910-30-8
Casopitant mesylate (GW679769B): Selective, brain-permeable NK1 receptor blocker, oral antiemetic.
Formula:
C31H39F7N4O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
712.72
Ref: TM-T10688
| 25mg | 1,234.00 € | ||
| 50mg | 1,616.00 € | ||
| 100mg | 2,597.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
CRTH2-IN-1
CAS:926661-54-3
CRTH2-IN-1 is a selective prostaglandin D2 receptor DP2 (CRTH2) antagonist, a Ramatroban analog, with an …
Formula:
C21H21FN2O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
416.47
Ref: TM-T10891
| 25mg | 1,688.00 € | ||
| 50mg | 2,226.00 € | ||
| 100mg | 2,899.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
K777
CAS:233277-99-1
K777: Oral cysteine protease inhibitor, CYP3A4 blocker (IC50=60 nM), CCR4 antagonist, anti-Trypanosoma cruzi, antiviral, halts …
Formula:
C32H38N4O4S
Purity:
98.43% - 99.14%
Color and Shape:
Solid
Molecular weight:
574.73
Ref: TM-T15641
| 1mg | 84.00 € | ||
| 5mg | 176.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 461.00 € | ||
| 50mg | 676.00 € | ||
| 1mL*10mM (DMSO) | 405.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Bucolome
CAS:841-73-6
Bucolome (Paramidine) is a CYP2C9 inhibitor with uricosuric and anti-inflammatory activity.
Formula:
C14H22N2O3
Purity:
99.83%
Color and Shape:
Solid
Molecular weight:
266.34
Ref: TM-T10632
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 366.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | 1,049.00 € | ||
| 500mg | 2,098.00 € | ||
| 1mL*10mM (DMSO) | 225.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Inz-1
CAS:897776-15-7
Inz-1 is an effective and fungal-selective inhibitor of mitochondrial cytochrome bc1 with IC50s of 8.092 …
Formula:
C16H14N2O2
Purity:
98.57% - 99.89%
Color and Shape:
Solid
Molecular weight:
266.29
Ref: TM-T27617
| 1mg | 50.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 154.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 389.00 € | ||
| 100mg | 556.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
CYP17-IN-1
CAS:2093317-51-0
CYP17-IN-1 is an effective oral inhibitor of CYP17 that can inhibit CYP17 in rats and …
Formula:
C18H17FN2S
Purity:
98.82% - 99.17%
Color and Shape:
Solid
Molecular weight:
312.4
Ref: TM-T10923
| 1mg | 113.00 € | ||
| 2mg | 169.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 366.00 € | ||
| 25mg | 550.00 € | ||
| 50mg | 769.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
