Transporter
Transporter proteins are involved in the movement of molecules across cellular membranes, playing vital roles in nutrient uptake, waste removal, and drug resistance. Inhibitors of transporter proteins are used to study the function of these proteins in various physiological and pathological processes, including metabolic disorders, cancer, and drug delivery. By modulating transporter activity, researchers can gain insights into cellular transport mechanisms and develop novel therapeutic strategies. At CymitQuimica, we provide a range of transporter inhibitors to support your research in pharmacology, cell biology, and metabolic regulation.
Found 44 products of "Transporter"
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Hemicholinium 3
CAS:Hemicholinium 3 is a potent and selective choline uptake blocker.Formula:C24H34Br2N2O4Purity:98% - 99.95%Color and Shape:SolidMolecular weight:574.35Indican
CAS:Indican (Indoxyl-β-D-glucoside) is a natural protective compound that is used to protect the liver.Formula:C14H17NO6Purity:99.78% - 99.92%Color and Shape:White To Off-White Crystalline PowderMolecular weight:295.29EAAT2 activator 1
CAS:EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 proteinFormula:C16H11ClFN3SPurity:98.86%Color and Shape:SolidMolecular weight:331.8BPTES
CAS:BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.Formula:C24H24N6O2S3Purity:95.83% - 99.64%Color and Shape:SolidMolecular weight:524.68Ref: TM-T6791
1mg37.00€2mg52.00€5mg69.00€10mg88.00€25mg150.00€50mg217.00€100mg324.00€200mg472.00€500mg772.00€1mL*10mM (DMSO)88.00€Clodronate disodium tetrahydrate
CAS:Clodronate disodium tetrahydrate (Clastoban) inhibits bone resorption and soft tissue calcification.Formula:CH10Cl2Na2O10P2Purity:98%Color and Shape:SolidMolecular weight:360.92TCID
CAS:TCID (UCH-L3 Inhibitor)(IC50=0.6 μM) is a DUB inhibitor of ubiquitin C-terminal hydrolase L3. It has the 125-fold selectivity to L1.Formula:C9H2Cl4O2Purity:99.34%Color and Shape:SolidMolecular weight:283.92α-Cyano-4-hydroxycinnamic acid
CAS:α-Cyano-4-hydroxycinnamic acid (α-Cyano-4-hydroxycinnamic acid(α-CHCA)) (α-CHCA) is an inhibitor of monocarboxylate transporter 1 (MCT1) that blocks pyruvateFormula:C10H7NO3Purity:99.8% - 99.86%Color and Shape:PowderMolecular weight:189.17Tormentic acid
CAS:Tormentic acid is a natural product. It has anticancer, anti-inflammatory, anti-atherogenic , anti-allodynic, and hepatoprotective properties,Formula:C30H48O5Purity:97.02% - 99.86%Color and Shape:SolidMolecular weight:488.7UCPH-101
CAS:UCPH-101 is an inhibitor of excitatory amino acid transporter subtype 1 (EAAT1) with an IC50 of 0.66 μM.Formula:C27H22N2O3Purity:98.58%Color and Shape:SolidMolecular weight:422.48Ref: TM-T4138
1mg50.00€2mg75.00€5mg130.00€10mg203.00€25mg409.00€50mg655.00€100mg954.00€200mg1,288.00€1mL*10mM (DMSO)142.00€BAY-876
CAS:BAY-876 is a selective and orally GLUT1 inhibitor. BAY-876 inhibits glycolytic metabolism and exhibits antitumor activity. Cost-effective and quality-assured.Formula:C24H16F4N6O2Purity:98.61% - 99.78%Color and Shape:SolidMolecular weight:496.42Ref: TM-T3713
1mg55.00€2mg78.00€5mg95.00€10mg131.00€25mg221.00€50mg334.00€100mg533.00€200mg755.00€1mL*10mM (DMSO)96.00€Dotinurad
CAS:Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).Formula:C14H9Cl2NO4SPurity:97.43% - 98.04%Color and Shape:SolidMolecular weight:358.2Ref: TM-T15160
1mg123.00€5mg289.00€10mg447.00€25mg737.00€50mg982.00€100mg1,341.00€1mL*10mM (DMSO)226.00€CTPI-2
CAS:CTPI-2 inhibits SLC25A1 (KD: 3.5 μM), glycolysis, PPARγ, GLUT4, has anti-tumor effects, and combats NASH and diet-induced obesity.Formula:C13H9ClN2O6SPurity:97.23%Color and Shape:SolidMolecular weight:356.74Valbenazine
CAS:Valbenazine (NBI-98854), a highly selective vesicular monoamine transporter 2(VMAT2) inhibitor, is approved for the treatment of tardive dyskinesia.Formula:C24H38N2O4Purity:97.58%Color and Shape:SolidMolecular weight:418.57Ref: TM-T7147
1mg46.00€2mg58.00€5mg101.00€10mg167.00€25mg313.00€50mg485.00€100mg708.00€200mg964.00€1mL*10mM (DMSO)113.00€KL-11743
CAS:KL-11743 blocks glucose metabolism, collapses NADH, and increases aspartate, shifting cells to oxidative phosphorylation.Formula:C30H30N6O3Purity:98.46% - 99.57%Color and Shape:SolidMolecular weight:522.6Ref: TM-T9558
1mg113.00€5mg235.00€10mg378.00€25mg630.00€50mg898.00€100mg1,216.00€1mL*10mM (DMSO)269.00€Vorolanib
CAS:Vorolanib (X-82) is an orally active VEGFR/PDGFR dual inhibitor.Formula:C23H26FN5O3Purity:97.35%Color and Shape:SolidMolecular weight:439.48Ref: TM-T8491
1mg101.00€2mg142.00€5mg215.00€10mg340.00€25mg583.00€50mg842.00€100mg1,144.00€200mg1,521.00€1mL*10mM (DMSO)236.00€WZB117
CAS:WZB117 inhibits GLUT1; IC50 ~10μM slows A549 lung & MCF7 breast cancer cell growth.Formula:C20H13FO6Purity:99.03% - 99.18%Color and Shape:SolidMolecular weight:368.31Ref: TM-T7018
5mg50.00€10mg77.00€25mg140.00€50mg224.00€100mg330.00€200mg492.00€500mg790.00€1mL*10mM (DMSO)52.00€DA-023
CAS:DA-023 (Compound 4) acts as a selective positive allosteric modulator (PAM) of EAAT2, exhibiting an EC 50 value of 1 nM [1].Formula:C20H25N7Color and Shape:SolidMolecular weight:363.46WAY-213613
CAS:WAY-213613: Potent GLT-1/EAAT2 inhibitor (IC50: 85 nM), selective over EAAT1/EAAT3; inactive at glutamate receptors.Formula:C16H13BrF2N2O4Purity:98%Color and Shape:SolidMolecular weight:415.19GT 949
CAS:GT 949 is a selective excitatory positive allosteric modulator of amino acid transporter-2 (EAAT2) (EC50: 0.26 nM).Formula:C30H37N7O2Purity:99.95%Color and Shape:SolidMolecular weight:527.66V-9302
CAS:V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uMFormula:C34H38N2O4Purity:98% - 99.54%Color and Shape:SolidMolecular weight:538.68Ref: TM-T5345
2mg39.00€5mg58.00€10mg84.00€25mg137.00€50mg207.00€100mg334.00€200mg489.00€1mL*10mM (DMSO)96.00€
