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5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 942 products of "5-HT Receptor"

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  • Piboserod

    CAS:
    <p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>
    Formula:C22H31N3O2
    Purity:97.21% - 99.49%
    Color and Shape:Solid
    Molecular weight:369.5
  • Tiprenolol

    CAS:
    <p>Tiprenolol is a beta adrenergic receptor antagonist.[1]</p>
    Formula:C13H21NO2S
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:255.38
  • Tandospirone hydrochloride

    CAS:
    <p>Tandospirone (SM-3997) HCl: potent 5-HT1A partial agonist; Ki: 27 nM; anxiolytic, antidepressant, for CNS disorder research.</p>
    Formula:C21H30ClN5O2
    Color and Shape:Solid
    Molecular weight:419.95
  • γ-Mangostin

    CAS:
    <p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>
    Formula:C23H24O6
    Purity:98.55% - 99.08%
    Color and Shape:Solid
    Molecular weight:396.43
  • Escitalopram Oxalate

    CAS:
    <p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>
    Formula:C22H23FN2O5
    Purity:97.39% - 99.73%
    Color and Shape:White Solid
    Molecular weight:414.43
  • Xanthotoxol

    CAS:
    <p>Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.</p>
    Formula:C11H6O4
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:202.16
  • Aripiprazole monohydrate

    CAS:
    <p>Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.</p>
    Formula:C23H29Cl2N3O3
    Color and Shape:Solid
    Molecular weight:466.4
  • MDL 100009

    CAS:
    <p>MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.</p>
    Formula:C22H28FNO3
    Purity:98.96%
    Color and Shape:Solid
    Molecular weight:373.46
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Formula:C21H32Cl2N4O
    Purity:99.68% - 99.87%
    Color and Shape:Solid
    Molecular weight:427.41
  • RS-127445

    CAS:
    <p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits &gt;1000-fold selectivity against other 5-HT receptors.</p>
    Formula:C17H16FN3
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:281.33
  • Relenopride hydrochloride

    CAS:
    <p>Relenopride, a 5-HT agonist, is used potentially for the treatment of chronic constipation.</p>
    Formula:C24H31Cl2FN4O4
    Color and Shape:Solid
    Molecular weight:529.43
  • 1-(1-Naphthyl) piperazine hydrochloride

    CAS:
    <p>1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple</p>
    Formula:C14H17ClN2
    Purity:98.27%
    Color and Shape:Solid
    Molecular weight:248.75
  • Clozapine HCl

    CAS:
    <p>Clozapine HCl, an atypical antipsychotic, binds CNS receptors, targets 5-HT2A/2C, has weaker D2 antagonism. Risk: Agranulocytosis.</p>
    Formula:C18H20Cl2N4
    Color and Shape:Solid
    Molecular weight:363.29
  • ARC-239

    CAS:
    <p>ARC-239 is an agonist of α2-adrenergic receptor.</p>
    Formula:C24H29N3O3
    Color and Shape:Solid
    Molecular weight:407.51
  • 7-Amino-4-(trifluoromethyl)coumarin

    CAS:
    7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.
    Formula:C10H6F3NO2
    Purity:97.31% - 97.84%
    Color and Shape:Yellow Powder
    Molecular weight:229.16
  • BMY 7378 dihydrochloride

    CAS:
    <p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>
    Formula:C22H33Cl2N3O3
    Purity:97.32% - 99.08%
    Color and Shape:Solid
    Molecular weight:458.42
  • Frovatriptan Succinate

    CAS:
    <p>Frovatriptan Succinate is a synthetic triptan with 5-HT1B/1D receptors agonist activity. It is indicated for the acute treatment of migraine.</p>
    Formula:C18H25N3O6
    Color and Shape:Solid
    Molecular weight:379.41
  • F-15599

    CAS:
    <p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>
    Formula:C19H21ClF2N4O
    Purity:98.72%
    Color and Shape:Solid
    Molecular weight:394.85
  • AVN-492

    CAS:
    AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).
    Formula:C17H21N5O2S
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:359.45
  • Intepirdine

    CAS:
    <p>Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.</p>
    Formula:C19H19N3O2S
    Purity:98% - 98.63%
    Color and Shape:Solid
    Molecular weight:353.44