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5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 942 products of "5-HT Receptor"

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  • FG-5893
    Targetmol
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    FG-5893

    CAS:
    <p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>
    Formula:C27H29F2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:465.53

    Ref: TM-T27317

  • S 14063
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    S 14063

    CAS:
    <p>S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.</p>
    Formula:C22H29Cl2N3O2S
    Color and Shape:Solid
    Molecular weight:470.45

    Ref: TM-T70839

  • Tertatolol
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    Tertatolol

    CAS:
    <p>Tertatolol is an effective antagonist of beta-adrenoceptor and 5-HT receptors.</p>
    Formula:C16H25NO2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.44

    Ref: TM-T17041

  • Piclozotan
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    Piclozotan

    CAS:
    <p>Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)</p>
    Formula:C23H24ClN3O2
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:409.91

    Ref: TM-T28414

  • Alniditan
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    Alniditan

    CAS:
    <p>Alniditan is a receptors agonist of 5-HT1B/1D in HEK 293 cells (IC50: 1.7 and 1.3 nM). For 5-HT1B/1D receptors, the pKi values are 8.96 and 9.40, respectively.</p>
    Formula:C17H26N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.41

    Ref: TM-T14190

  • 5-HT2A receptor agonist-2
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    5-HT2A receptor agonist-2

    CAS:
    <p>Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.</p>
    Formula:C20H21ClN2O3
    Color and Shape:Solid
    Molecular weight:372.85

    Ref: TM-T61507

  • AP-521 (Free base)
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    AP-521 (Free base)

    CAS:
    <p>AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.</p>
    Formula:C20H18N2O3S
    Color and Shape:Solid
    Molecular weight:366.43

    Ref: TM-T26640

  • Bopindolol (malonate)
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    Bopindolol (malonate)

    CAS:
    <p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>
    Formula:C26H32N2O7
    Color and Shape:Solid
    Molecular weight:484.549

    Ref: TM-T35871

  • RS 39604
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    RS 39604

    CAS:
    <p>potent and selective 5-HT4 antagonist</p>
    Formula:C26H37Cl2N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:590.56

    Ref: TM-T23260

  • Naronapride
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    Naronapride

    CAS:
    <p>Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.</p>
    Formula:C27H41ClN4O5
    Color and Shape:Solid
    Molecular weight:537.09

    Ref: TM-T63785

  • Bifeprunox
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    Bifeprunox

    CAS:
    <p>Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.</p>
    Formula:C24H23N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.46

    Ref: TM-T10542

  • TMPPAA
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    TMPPAA

    CAS:
    <p>TMPPAA is an allosteric agonist of 5-HT3 receptor.</p>
    Formula:C15H21NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:247.33

    Ref: TM-T28986

  • Ziprasidone mesylate trihydrate
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    Ziprasidone mesylate trihydrate

    CAS:
    <p>Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.</p>
    Formula:C22H31ClN4O7S2
    Color and Shape:Solid
    Molecular weight:563.08

    Ref: TM-T63979

  • 5-HT7 agonist 1
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    5-HT7 agonist 1

    CAS:
    <p>5-HT7 agonist 1 (4-[4-[(2-chlorophenyl)methyl]piperazin-1-yl]-1H-indole) is a selective agonist of 5-HT7 (IC50 = 222.93 nM).</p>
    Formula:C19H20ClN3
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:325.84

    Ref: TM-T10170

  • Pruvanserin hydrochloride
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    Pruvanserin hydrochloride

    CAS:
    <p>Pruvanserin hydrochloride (EMD 281014 HCl) is a selective 5-HT2A receptor antagonist, inhibits GTP-gamma-S accumulation and alleviates tactile allodynia.</p>
    Formula:C22H22ClFN4O
    Purity:99.6%
    Color and Shape:Solid
    Molecular weight:412.89

    Ref: TM-T22762

  • Eplivanserin
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    Eplivanserin

    CAS:
    <p>Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.</p>
    Formula:C19H21FN2O2
    Purity:97.04%
    Color and Shape:Solid
    Molecular weight:328.38

    Ref: TM-T11217

  • SB-737050A
    Targetmol
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    SB-737050A

    CAS:
    <p>SB-737050A, a 5-HT antagonist, is used potentially for the treatment of schizophrenia.</p>
    Formula:C22H23ClN2O3S2
    Color and Shape:Solid
    Molecular weight:463.01

    Ref: TM-T28693

  • EMDT
    Targetmol
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    EMDT

    CAS:
    <p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>
    Formula:C15H22N2O
    Purity:97.66% - 99.78%
    Color and Shape:Solid
    Molecular weight:246.35

    Ref: TM-T11183

  • GR 113808
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    GR 113808

    CAS:
    <p>GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.</p>
    Formula:C19H27N3O4S
    Purity:98.16%
    Color and Shape:Solid
    Molecular weight:393.5

    Ref: TM-T15414

  • PNU-142633
    Targetmol
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    PNU-142633

    CAS:
    <p>PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; &gt;18,000 nM for 5-HT1B.</p>
    Formula:C24H30N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:422.52

    Ref: TM-T16556