5-HT Receptor
5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.
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5-HT2 agonist-1 free base
CAS:2708279-77-8
Compound 24 (5-HT2 agonist-1 free base) is a potent agonist for 5-HT2A, 5-HT2B, and 5-HT2C …
Formula:
C19H22N2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
310.39
Ref: TM-T79805
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
5-HT2C agonist-3
CAS:2104810-18-4
5-HT2C agonist-3 ((+)-19), a selective 5-HT2C agonist (EC 50: 24 nM, Ki: 78 nM), exhibits …
Formula:
C19H23ClFNO2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
351.84
Ref: TM-T79802
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
SB 258719
CAS:195199-95-2
SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.
Formula:
C18H30N2O2S
Purity:
98.59%
Color and Shape:
Solid
Molecular weight:
338.51
Ref: TM-T12855
| 2mg | 35.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | 247.00 € | ||
| 100mg | 365.00 € | ||
| 200mg | 514.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
2-Methyl-5-HT
CAS:78263-90-8
2-Methyl-5-HT (2-Methyl-5-hydroxytryptamine) is a potent and selective 5-HT3 receptor agonist with anti-depressive-like effects.
Formula:
C11H14N2O
Purity:
95.64%
Color and Shape:
Solid
Molecular weight:
190.24
Ref: TM-T10075
| 5mg | 51.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 522.00 € | ||
| 500mg | 1,133.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Lumateperone
CAS:313368-91-1
Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).
Formula:
C24H28FN3O
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
393.5
Ref: TM-T21069
| 10mg | 39.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 83.00 € | ||
| 100mg | 115.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
SB-616234-A
CAS:908601-49-0
SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant …
Formula:
C32H36ClN5O3
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
574.11
Ref: TM-T12847
| 1mg | 103.00 € | ||
| 5mg | 248.00 € | ||
| 10mg | 358.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,007.00 € | ||
| 200mg | 1,358.00 € | ||
| 1mL*10mM (DMSO) | 313.00 € |
Estimated delivery in United States, on Wednesday 19 Feb 2025
SB-224289 hydrochloride
CAS:180084-26-8
SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.
Formula:
C32H33ClN4O3
Purity:
97.82% - 98.09%
Color and Shape:
Solid
Molecular weight:
557.08
Ref: TM-T12841
| 5mg | 52.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
5-HT2A/5-HT2C inverse agonist 1
CAS:2718990-76-0
5-HT2A/5-HT2C inverse agonist 1 serves as a dual and potent inverse agonist for the 5-HT2A …
Formula:
C24H35N5O2
Color and Shape:
Liquid
Molecular weight:
425.57
Ref: TM-T200089
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Mar 2025
SB 243213 dihydrochloride
CAS:1780372-25-9
SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi …
Formula:
C22H21Cl2F3N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
501.33
Ref: TM-T12859L
| 1mg | 108.00 € | ||
| 5mg | 313.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
SB 243213 hydrochloride
CAS:200940-23-4
SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi …
Formula:
C22H20ClF3N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
464.87
Ref: TM-T12859
| 25mg | 2,106.00 € | ||
| 50mg | 2,785.00 € | ||
| 100mg | 3,739.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
VA012
CAS:885898-58-8
VA012 (compound 11) acts as a positive allosteric modulator (PAM) of the serotonin 5-HT2C receptor. …
Formula:
C21H19N3
Color and Shape:
Liquid
Molecular weight:
313.4
Ref: TM-T200241
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Mar 2025
AM9405
AM9405: peripheral CB1/5-HT3 agonist, suppresses gut motility, relieves GI disorder symptoms in mice.
Formula:
C24H33BrN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
461.44
Ref: TM-T10294
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
F 14679
CAS:208109-38-0
F 14679 is a potent 5-HT1A agonist (pKi=10.23) with a maximum Ca2t response similar to …
Formula:
C21H25ClF2N4O
Purity:
99.09%
Color and Shape:
Liquid
Molecular weight:
422.9
Ref: TM-T62269
| 25mg | 1,234.00 € | ||
| 50mg | 1,604.00 € | ||
| 100mg | 2,419.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
Rodatristat ethyl
CAS:1673571-51-1
Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low …
Formula:
C29H31ClF3N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
590.04
Ref: TM-T16779
| 25mg | 2,233.00 € | ||
| 50mg | 3,615.00 € | ||
| 100mg | 5,781.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
Sulamserod
CAS:219757-90-1
Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study …
Formula:
C19H28ClN3O5S
Purity:
98.76%
Color and Shape:
Solid
Molecular weight:
445.96
Ref: TM-T13021
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
Befiradol hydrochloride
CAS:2436760-81-3
Befiradol HCl (NLX-112) is a selective 5-HT1A receptor agonist with anxiolytic effects and prevents ATXN3 …
Formula:
C20H23Cl2F2N3O
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
430.32
Ref: TM-T62385
| 1mg | 149.00 € | ||
| 2mg | 213.00 € | ||
| 5mg | 357.00 € | ||
| 10mg | 522.00 € | ||
| 25mg | 841.00 € | ||
| 50mg | 1,160.00 € | ||
| 100mg | 1,556.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
Cyclobenzaprine hydrochloride
CAS:6202-23-9
Cyclobenzaprine hydrochloride (MK130 hydrochloride) , a centrally acting muscle relaxant with antidepressant activity, leads to …
Formula:
C20H22ClN
Purity:
99.98%
Color and Shape:
Crystalline Solid
Molecular weight:
311.86
Ref: TM-T1509
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Bufotenidine
CAS:487-91-2
Bufotenidine is a natural alkaloid which also a neural tryptaminic receptor blocking agent blocks the …
Formula:
C13H18N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
218.29
Ref: TM-TN7062
| 5mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Clocapramine dihydrochloride hydrate
CAS:60789-62-0
Clocapramine dihydrochloride hydrate (3-Chlorocarpipramine hydrochloride hydrate) is an antagonist of the 5-HT2A and D2 receptors.
Formula:
C28H41Cl3N4O2
Purity:
97.68%
Color and Shape:
Solid
Molecular weight:
572.01
Ref: TM-T10837
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Granisetron
CAS:109889-09-0
Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for …
Formula:
C18H24N4O
Color and Shape:
Solid
Molecular weight:
312.41
Ref: TM-T22340
| 5mg | Discontinued | Request information |
