GlyT
Glycine Transporter (GlyT) inhibitors are compounds that block the reuptake of glycine, an important inhibitory neurotransmitter in the spinal cord and brainstem. By inhibiting glycine transporters, these compounds increase the availability of glycine in the synaptic cleft, enhancing its inhibitory effects on neuronal activity. GlyT inhibitors are of interest for their potential therapeutic applications in conditions like chronic pain, spasticity, and schizophrenia. At CymitQuimica, we provide GlyT inhibitors to support your research in pain management, motor control, and neuropsychiatric disorders.
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LY2365109 hydrochloride
CAS:1779796-27-8
LY2365109 hydrochloride is a potent and selective GlyT1 inhibitor, with an IC50 of 15.8 nM …
Formula:
C22H28ClNO5
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
421.91
Ref: TM-T11908
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 500.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Amoxapine
CAS:14028-44-5
Amoxapine (CL-67772) exerts its antidepressant effect by inhibiting the re-uptake of norepinephrine and, to a …
Formula:
C17H16ClN3O
Purity:
98.25% - 98.84%
Color and Shape:
Solid
Molecular weight:
313.78
Ref: TM-T1568
| 500mg | 69.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Org 25543 hydrochloride
CAS:495076-64-7
Org 25543 hydrochloride is a potent and selective glycine transporter type 2 (GlyT2) inhibitor (IC50 …
Formula:
C24H33ClN2O4
Purity:
99.26%
Color and Shape:
Solid
Molecular weight:
448.983
Ref: TM-T22126
| 1mg | 81.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 252.00 € |
Estimated delivery in United States, on Monday 13 Jan 2025
Sarcosine
CAS:107-97-1
Sarcosine (Methylglycine) is a competitive inhibitor of the type I glycine transporter (GlyT1) and an …
Formula:
C3H7NO2
Purity:
99.34%
Color and Shape:
Deliquescent Water Soluble Physical Description Deliquescent Crystals Or Powder Has A Sweetish Taste (Ntp 1992)
Molecular weight:
89.09
Ref: TM-T6975
| 1g | 60.00 € | ||
| 5g | 129.00 € | ||
| 10g | 185.00 € | ||
| 500mg | 46.00 € |
Estimated delivery in United States, on Monday 13 Jan 2025
Opiranserin hydrochloride
CAS:1440796-75-7
Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin …
Formula:
C21H35ClN2O5
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
430.97
Ref: TM-T9833
| 1mg | 93.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 351.00 € | ||
| 25mg | 637.00 € | ||
| 50mg | 906.00 € | ||
| 100mg | 1,261.00 € | ||
| 500mg | 2,531.00 € | ||
| 1mL*10mM (DMSO) | 249.00 € |
Estimated delivery in United States, on Monday 13 Jan 2025
Bitopertin
CAS:845614-11-1
Bitopertin (Paliflutine) (RG1678, RO-4917838) is a potent inhibitor of glycine transporter 1 (GlyT1), with Ki …
Formula:
C21H20F7N3O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
543.46
Ref: TM-T6788
| 2mg | 41.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 423.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Monday 13 Jan 2025
Tilapertin
CAS:1000690-85-6
Tilapertin is an oral glycine transporter type-1 inhibitor.
Formula:
C20H21F3N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
378.39
Ref: TM-T17096
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Bitopertin (R enantiomer)
CAS:845614-12-2
Bitopertin R enantiomer (RG1678 R enantiomer) is the R-enantiomer of Bitopertin.
Formula:
C21H20F7N3O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
543.46
Ref: TM-T10552
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 24 Feb 2025
Opiranserin
CAS:1441000-45-8
Opiranserin is a development as an injectable agent for the treatment of postoperative pain.
Formula:
C21H34N2O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
394.51
Ref: TM-T16399
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
ASP2535
CAS:374886-51-8
ASP2535 is a potent, selective, orally bioavailable, brain permeable and centrally-active glycine transporter-1 (GlyT1) inhibitor.ASP2535 …
Formula:
C22H18N6O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
382.42
Ref: TM-T14334
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,321.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
ALX-1393
CAS:949164-09-4
ALX-1393 is a selective GlyT2 inhibitor that effectively reduces neuronal action potential activity in a …
Formula:
C23H22FNO4
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
395.42
Ref: TM-T14198
| 1mg | 1,290.00 € | ||
| 5mg | 2,616.00 € | ||
| 10mg | 3,521.00 € | ||
| 25mg | 5,250.00 € | ||
| 50mg | 7,046.00 € | ||
| 100mg | 9,200.00 € | ||
| 1mL*10mM (DMSO) | 2,718.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
PF-03463275
CAS:1173239-39-8
PF-03463275 is an orally active and selective reversible inhibitor of competitive glycine transporter protein-1 (GlyT1) …
Formula:
C19H22ClFN4O
Purity:
99.86%
Color and Shape:
Liquid
Molecular weight:
376.86
Ref: TM-T61564
| 1mg | 55.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 312.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 129.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Iclepertin
CAS:1421936-85-7
Iclepertin (BI-425809) is a GlyT1 inhibitor.Iclepertin is used for the treatment of Alzheimer;s disease and …
Formula:
C20H18F6N2O5S
Purity:
98.89% - 98.93%
Color and Shape:
Solid
Molecular weight:
512.42
Ref: TM-T37089
| 1mg | 211.00 € | ||
| 2mg | 314.00 € | ||
| 5mg | 524.00 € | ||
| 10mg | 831.00 € | ||
| 25mg | 1,854.00 € | ||
| 50mg | 3,046.00 € |
Estimated delivery in United States, on Monday 7 Apr 2025
