Adrenergic Receptor
Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.
Subcategories of "Adrenergic Receptor"
Found 645 products of "Adrenergic Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Ivabradine-d3 hydrochloride
CAS:<p>Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.</p>Formula:C27H37ClN2O5Purity:98%Color and Shape:SolidMolecular weight:508.07YM 09538
CAS:<p>YM 09538 is a biochemical.</p>Formula:C18H25ClN2O5SColor and Shape:SolidMolecular weight:416.92Chir 2279
CAS:<p>CHIR 2279, a peptoid trimer, binds alpha 1-adrenoceptors, blocking epinephrine effects in dogs (pseudo pA2 6.86).</p>Formula:C34H36N4O4Color and Shape:SolidMolecular weight:564.67Tienoxolol FA
<p>Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.</p>Formula:C22H30N2O7SPurity:97.05% - 98.85%Color and Shape:SoildMolecular weight:466.55Bamosiran
CAS:<p>Bamosiran, a small interfering RNA (siRNA), specifically targets the β-adrenergic receptor 2 to reduce intraocular pressure.</p>Color and Shape:SolidSynephrine hemitartrate
CAS:<p>Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.</p>Formula:C9H13NO2C4H6O6Color and Shape:SolidMolecular weight:242.26Benzquinamide
CAS:<p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>Formula:C22H32N2O5Purity:94.86%Color and Shape:SolidMolecular weight:404.5Desglymidodrine
CAS:<p>Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.</p>Formula:C10H15NO3Purity:99.56%Color and Shape:SolidMolecular weight:197.23SB-206606
CAS:<p>SB-206606 is a novel, highly specific radioactive ligand for the β3-adrenergic receptor.</p>Formula:C19H22ClNO4Color and Shape:SolidMolecular weight:363.83CTP-amiodarone
<p>CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.</p>Formula:C97H131F3I2N20O25S2Color and Shape:SolidMolecular weight:2352.13Mapenterol hydrochloride
CAS:<p>Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.</p>Formula:C14H21Cl2F3N2OPurity:98.11% - 99.98%Color and Shape:SolidMolecular weight:361.23Metipranolol
CAS:<p>Metipranolol (Betamann) is a type of β- Adrenergic receptors（ β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta blocking potentials (pA2) of 8.3 and 8.4, respectively. It is also a potent substituent in the 3H DHA binding assay, with a ligand concentration of 0.7 nM and a Ki of 39 ± 24 nM.</p>Formula:C17H27NO4Purity:98.37%Color and Shape:SolidMolecular weight:309.4Formoterol O-β-D-Glucuronide
CAS:<p>Formoterol O-β-D-glucuronide is a metabolite of formoterol .</p>Formula:C25H32N2O10Color and Shape:SolidMolecular weight:520.535Sibenadet hydrochloride
CAS:<p>Sibenadet, a D2/beta2-agonist, is potential useful for the treatment of symptoms of chronic obstructive pulmonary disease.</p>Formula:C22H29ClN2O5S2Color and Shape:SolidMolecular weight:501.06(+)-ORM-10921
CAS:<p>(+)-ORM-10921 is a conformation of ORM-10921 and can be used in chemical synthesis studies.</p>Formula:C18H23NO2Purity:99.85%Color and Shape:SoildMolecular weight:285.38α1A-AR Degrader 9c
CAS:<p>α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.</p>Formula:C38H43N11O11Purity:98%Color and Shape:SolidMolecular weight:829.82Phenylethanolamine A
CAS:<p>Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.</p>Formula:C19H24N2O4Color and Shape:SolidMolecular weight:344.40L-770644
CAS:<p>L-770644 is an agonist of B3 adrenergic receptor.</p>Formula:C30H37N7O4SColor and Shape:SolidMolecular weight:591.72Bucindolol Formate
<p>Bucindolol is a β1-adrenergic blocker with sympathomimetic activity, used in heart failure research.</p>Formula:C23H27N3O4Purity:99.76% - 99.88%Color and Shape:SolidMolecular weight:409.48Nolomirole
CAS:<p>Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.</p>Formula:C19H27NO4Color and Shape:SolidMolecular weight:333.42Oxaprotiline hydrochloride
CAS:<p>Oxaprotiline hydrochloride is an antidepressant.</p>Formula:C20H24ClNOPurity:98%Color and Shape:SolidMolecular weight:329.86AG-825
CAS:<p>AG-825（Tyrphostin C15） is a selective and competitive ErbB2 inhibitor that inhibits tyrosine phosphorylation with an IC50 value of 0.35 μM.AG-825 (Tyrphostin</p>Formula:C19H15N3O3S2Purity:98.43%Color and Shape:Yellow SolidMolecular weight:397.47Carazolol-d7
CAS:<p>Carazolol-d7 is the deuterium-labeled isotope of Carazolol, commonly used in pharmacokinetic studies to investigate the metabolic pathways of Carazolol.</p>Formula:C18H22N2O2Color and Shape:SolidMolecular weight:305.42Prazobind
CAS:<p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>Formula:C23H27N5O3Color and Shape:SolidMolecular weight:421.501Benzoquinamide hydrochloride
CAS:<p>Benzoquinamide hydrochloride (3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride) is an antiemetic</p>Formula:C22H33ClN2O5Purity:97.13% - 99.56%Color and Shape:SolidMolecular weight:440.96YS-49 monohydrate
<p>YS-49, a PI3K/Akt activator, curbs RhoA/PTEN; inhibits VSMC growth by inducing HO-1; an isoquinoline alkaloid that stimulates cardiac β-adrenoceptors.</p>Formula:C20H22BrNO3Color and Shape:SolidMolecular weight:404.3Ethylnorepinephrine hydrochloride
CAS:<p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>Formula:C10H16ClNO3Purity:98%Color and Shape:SolidMolecular weight:233.69Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Color and Shape:Odour Solid5-hydroxy Propranolol
CAS:<p>5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.</p>Formula:C16H21NO3Color and Shape:SolidMolecular weight:275.348(R)-(+)-Atenolol
CAS:<p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>Formula:C14H22N2O3Purity:98.72%Color and Shape:SolidMolecular weight:266.34L-770644 dihydrochloride
CAS:<p>L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.</p>Formula:C30H38ClN7O4SColor and Shape:SolidMolecular weight:628.19Terazosin dimer impurity dihydrochloride
CAS:<p>Terazosin dimer impurity dihydrochloride is a chemical byproduct of the α1-antagonist Terazosin, derived from quinazoline.</p>Formula:C24H30Cl2N8O4Color and Shape:SolidMolecular weight:565.46Amitraz
CAS:<p>Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.</p>Formula:C19H23N3Purity:99.88%Color and Shape:White/Pale Yellow Crystalline SolidMolecular weight:293.41(±)5(6)-EET
CAS:<p>5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.</p>Formula:C20H32O3Color and Shape:SolidMolecular weight:320.473BMS-196085
CAS:<p>BMS-196085 is an effective and selective human β( 3) All agonists of adrenergic receptors, in β( 1) Partial agonist activity was 45%.</p>Formula:C24H26F2N2O5SColor and Shape:SolidMolecular weight:492.54Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS:<p>Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.</p>Formula:C25H26O13Color and Shape:SolidMolecular weight:534.47Mibenratide TFA
<p>Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].</p>Purity:98%Color and Shape:Odour SolidAbediterol napadisylate
CAS:<p>Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.</p>Formula:C60H68F4N4O14S2Purity:98%Color and Shape:SolidMolecular weight:1209.32Besipirdine hydrochloride
CAS:<p>Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.</p>Formula:C16H18ClN3Purity:98.45%Color and Shape:SoildMolecular weight:287.79AA 497 HCl
CAS:<p>AA 497, a beta-2 agonist, suppresses Ca spikes.</p>Formula:C14H22ClNO3Color and Shape:SolidMolecular weight:287.78Metaraminol
CAS:<p>Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>Formula:C9H13NO2Color and Shape:SolidMolecular weight:167.21Propranolol hydrochloride
CAS:<p>Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse</p>Formula:C16H22ClNO2Purity:99.94% - >99.99%Color and Shape:White Or Almost White Powder White PowderMolecular weight:295.80Meluadrine tartrate
CAS:<p>Meluadrine tartrate is an endogenous metabolite.</p>Formula:C16H24ClNO8Purity:98%Color and Shape:SolidMolecular weight:393.82Yohimbine
CAS:<p>Yohimbine is a nonselective alpha 2-adrenergic receptor (AR) antagonist(IC50 : 0.6 μM)</p>Formula:C21H26N2O3Purity:99.78% - 99.89%Color and Shape:SolidMolecular weight:354.4Acrinor
CAS:<p>Acrinor is a adrenergic beta receptor agonist.</p>Formula:C35H46Cl2N10O8Purity:98%Color and Shape:SolidMolecular weight:805.72AdTx1
<p>Selective non-competitive α1A adrenoceptor antagonist with Ki of 0.35 nM; inactive on other GPCRs; affects phenylephrine actions.</p>Formula:C310H481N87O100S8Purity:98%Color and Shape:SolidMolecular weight:7283.22Detomidine carboxylic acid
CAS:<p>Detomidine carboxylic acid, a urine metabolite of detomidine, is a synthetic α2-agonist, animal analgesic, with cardiac, respiratory, and diuretic effects.</p>Formula:C12H12N2O2Purity:98%Color and Shape:SolidMolecular weight:216.24O-Desmethyl Mebeverine alcohol
CAS:<p>Mebeverine metabolite O-desmethyl alcohol inhibits α1 receptors, relaxing the gut.</p>Formula:C15H25NO2Purity:98%Color and Shape:SolidMolecular weight:251.365-Bromoimidazo[1,2-A]Pyrazine
CAS:<p>5-Bromoimidazo[1,2-a]pyrazine inhibits phosphodiesterase and beta-adrenergic receptors.5-Bromoimidazo[1,2-a]pyrazine shows antibronchospastic activity in vitro.</p>Formula:C6H4BrN3Purity:97.04%Color and Shape:SolidMolecular weight:198.02ARC 239 dihydrochloride
CAS:<p>ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).</p>Formula:C24H31Cl2N3O3Purity:99.72%Color and Shape:SolidMolecular weight:480.43
![5-Bromoimidazo[1,2-A]Pyrazine](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT77641.webp&w=3840&q=75)
