Adrenergic Receptor
Adrenergic receptors are GPCRs that are activated by catecholamines, such as adrenaline and noradrenaline. These receptors are classified into alpha and beta subtypes, each of which plays a key role in the regulation of heart rate, blood pressure, and the fight-or-flight response. Adrenergic receptor modulators are essential in the treatment of cardiovascular diseases, asthma, and anxiety disorders. At CymitQuimica, we offer a wide range of high-quality adrenergic receptor modulators to support your research in endocrinology, cardiovascular pharmacology, and stress response.
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Subcategories of "Adrenergic Receptor"
Products of "Adrenergic Receptor"
Dibenamine hydrochloride
CAS:55-43-6
Dibenamine hydrochloride is a competitive and irreversible blocking agent of the β-adrenergic receptor.
Formula:
C16H19Cl2N
Purity:
96.43%
Color and Shape:
Oily Liquid Solid
Molecular weight:
296.23
Ref: TM-T37906
| 500mg | 34.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Vatinoxan hydrochloride
CAS:130466-38-5
Vatinoxan hydrochloride is an antagonist of the peripheral α2 adrenergic receptors.
Formula:
C20H27ClN4O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
454.97
Ref: TM-T13285
| 25mg | 1,967.00 € | ||
| 50mg | 2,598.00 € | ||
| 100mg | 3,458.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
RS 100329 hydrochloride
CAS:1215654-26-4
RS 100329 hydrochloride is an antagonist of α1A-adrenergic receptor.
Formula:
C20H26ClF3N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
462.89
Ref: TM-T23253
| 1mg | 36.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 103.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 461.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Bunazosin Hydrochloride
CAS:52712-76-2
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an …
Formula:
C19H28ClN5O3
Purity:
98.48%
Color and Shape:
Solid
Molecular weight:
409.91
Ref: TM-T26923
| 5mg | 40.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 144.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
(±)-N-Methylcoclaurine
CAS:1472-62-4
N-Methylcoclaurine (±) acts as a selective antagonist at the α2-adrenoceptor [1].
Formula:
C18H21NO3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
299.36
Ref: TM-T79641
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
(±)-Prenalterol
CAS:57526-81-5
(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to …
Formula:
C12H19NO3
Purity:
99.71%
Color and Shape:
Liquid
Molecular weight:
225.28
Ref: TM-T25984
| 1mg | 215.00 € | ||
| 2mg | 323.00 € | ||
| 5mg | 537.00 € | ||
| 10mg | 861.00 € | ||
| 25mg | 1,273.00 € | ||
| 50mg | 1,715.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
RS 17053 hydrochloride
CAS:169505-93-5
RS 17053 hydrochloride: selective α1A adrenoceptor antagonist, pKi 9.1, pA2 9.8.
Formula:
C24H30Cl2N2O2
Purity:
99.27%
Color and Shape:
Solid
Molecular weight:
449.41
Ref: TM-T16798
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Phentolamine Analogue 1
CAS:47142-51-8
Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.
Formula:
C17H19N3O
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
281.35
Ref: TM-T12444
| 1mg | 83.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € | ||
| 1mL*10mM (DMSO) | 166.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Todralazine hydrochloride
CAS:3778-76-5
Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.
Formula:
C11H13ClN4O2
Purity:
98.32%
Color and Shape:
Solid
Molecular weight:
268.7
Ref: TM-T17111
| 10mg | 46.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 87.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
CGP-20712
CAS:137888-49-4
CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.
Formula:
C23H25F3N4O5
Purity:
100% - 99.40%
Color and Shape:
Solid
Molecular weight:
494.46
Ref: TM-T30846
| 1mg | 327.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,481.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
OPC-28326
CAS:167626-17-7
OPC-28326: an α2-adrenergic blocker; dilates blood vessels; inhibits α2A/B/C receptors with Ki 2040/285/55 nM.
Formula:
C26H35N3O2
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
421.58
Ref: TM-T13804
| 1mg | 182.00 € | ||
| 5mg | 443.00 € | ||
| 10mg | 604.00 € | ||
| 25mg | 915.00 € | ||
| 50mg | 1,229.00 € | ||
| 100mg | 1,617.00 € | ||
| 200mg | 2,189.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Deriglidole
CAS:122830-14-2
Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.
Formula:
C16H21N3
Purity:
98.24% - 99.45%
Color and Shape:
Solid
Molecular weight:
255.36
Ref: TM-T10998
| 1mg | 427.00 € | ||
| 5mg | 991.00 € | ||
| 10mg | 1,327.00 € | ||
| 25mg | 1,950.00 € | ||
| 50mg | 2,396.00 € | ||
| 100mg | 3,158.00 € | ||
| 1mL*10mM (DMSO) | 748.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Bufuralol
CAS:54340-62-4
Bufuralol (Ro 3-4787) is a 尾-adrenergic receptor blocker with a certain degree of sympathomimetic effects …
Formula:
C16H23NO2
Purity:
98.26%
Color and Shape:
Solid
Molecular weight:
261.36
Ref: TM-T30611
| 2mg | 412.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
Fiduxosin
CAS:208993-54-8
Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and …
Formula:
C30H29N5O4S
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
555.65
Ref: TM-T11286
| 1mg | 650.00 € | ||
| 5mg | 1,678.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
TAAR1 agonist 3
CAS:1804129-70-1
TAAR1 agonist 3 is a potent agonist of Trace Amine-Associated Receptor 1 (TAAR1) with a …
Formula:
C10H13NO
Color and Shape:
Liquid
Molecular weight:
163.22
Ref: TM-T200046
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Mar 2025
(S)-Bucindolol
CAS:91548-61-7
(S)-Bucindolol is an enantiomer of bucindolol, specifically a β1-adrenergic receptor antagonist. It is primarily utilized …
Formula:
C22H25N3O2
Color and Shape:
Liquid
Molecular weight:
363.45
Ref: TM-T200285
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Mar 2025
Aclidinium
CAS:727649-81-2
Aclidinium, a dual-action compound, serves as a long-acting muscarinic antagonist and a β2-adrenoceptor (β2-AR) agonist, …
Formula:
C26H30NO4S2
Color and Shape:
Liquid
Molecular weight:
484.65
Ref: TM-T200043
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 5 Mar 2025
Xylazine hydrochloride
CAS:23076-35-9
Xylazine hydrochloride (BAY 1470 hydrochloride) is an adrenergic alpha-2 agonist used as a sedative, analgesic …
Formula:
C12H16N2S·HCl
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
256.79
Ref: TM-T1500
| 10mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Cimaterol
CAS:54239-37-1
Cimaterol is a potent β-adrenoceptor agonist. cimaterol binds to the L6β-receptor with a Kd value …
Formula:
C12H17N3O
Purity:
98.64%
Color and Shape:
Solid
Molecular weight:
219.28
Ref: TM-T19769
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Xylazine
CAS:7361-61-7
Xylazine (BAY 1470) is α2-adrenergic receptor agonist.
Formula:
C12H16N2S
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
220.33
Ref: TM-T7046
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
