GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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JNJ16259685
CAS:409345-29-5
JNJ16259685 (TN.T 16259685) is a selective mGluR1 antagonist, and inhibits the synaptic activation of mGluR1 …
Formula:
C20H23NO3
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
325.4
Ref: TM-T5512
| 1mg | 48.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 289.00 € | ||
| 50mg | 443.00 € | ||
| 100mg | 647.00 € | ||
| 1mL*10mM (DMSO) | 99.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Farampator
CAS:211735-76-1
Farampator (CX-691) (CX-691;Org24448) is a positive modulator of AMPA receptor.
Formula:
C12H13N3O2
Purity:
99.76% - 99.83%
Color and Shape:
Solid
Molecular weight:
231.25
Ref: TM-T3957
| 2mg | 34.00 € | ||
| 5mg | 51.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 136.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 338.00 € | ||
| 200mg | 479.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
FTIDC
CAS:873551-53-2
FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 …
Formula:
C18H23FN6O
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
358.41
Ref: TM-T3483
| 1mg | 104.00 € | ||
| 2mg | 150.00 € | ||
| 5mg | 224.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 583.00 € | ||
| 50mg | 823.00 € | ||
| 100mg | 1,106.00 € | ||
| 1mL*10mM (DMSO) | 249.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(RS)-3-Hydroxyphenylglycine
CAS:31932-87-3
(RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.
Formula:
C8H9NO3
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
167.16
Ref: TM-T23259
| 1mg | 35.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 345.00 € | ||
| 100mg | 521.00 € | ||
| 500mg | 1,103.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
E4CPG
CAS:170846-89-6
E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.
Formula:
C11H13NO4
Purity:
99.96%
Color and Shape:
Solid
Molecular weight:
223.23
Ref: TM-T3477
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 244.00 € | ||
| 100mg | 368.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Chelidamic acid
CAS:138-60-3
Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors …
Formula:
C7H5NO5
Purity:
≥95%
Color and Shape:
Pale Yellow Powder
Molecular weight:
183.12
Ref: TM-T5884
| 1g | 82.00 € | ||
| 200mg | 39.00 € | ||
| 500mg | 56.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
VU-1545
CAS:890764-63-3
VU-1545 is mGlu5 positive allosteric modulator.
Formula:
C22H15FN4O3
Purity:
98.80%
Color and Shape:
Solid
Molecular weight:
402.38
Ref: TM-T23514
| 1mg | 41.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 364.00 € | ||
| 100mg | 524.00 € | ||
| 200mg | 704.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
IEM 1754 2HBr
CAS:162831-31-4
IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and …
Formula:
C16H30N2·2HBr
Purity:
99.71% - 99.72%
Color and Shape:
Solid
Molecular weight:
412.25
Ref: TM-T6134
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 154.00 € | ||
| 100mg | 221.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 13 Jan 2025
HexylHIBO
CAS:334887-43-3
HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values …
Formula:
C12H20N2O4
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
256.3
Ref: TM-T22840
| 1mg | 83.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 555.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 27 Jan 2025
NS 1209
CAS:205645-02-9
NS 1209 (SPD 502) is a AMPA receptor antagonist.
Formula:
C24H27N4NaO7S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
538.55
Ref: TM-T4009
| 25mg | 804.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Dipraglurant
CAS:872363-17-2
Dipraglurant: a blood-brain permeable mGluR5 NAM, orally active, selective, IC50 = 21 nM, treats PD-LID.
Formula:
C16H12FN3
Purity:
98.7%
Color and Shape:
Solid
Molecular weight:
265.29
Ref: TM-T15134
| 1mg | 95.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 707.00 € | ||
| 50mg | 1,057.00 € | ||
| 100mg | 1,406.00 € | ||
| 1mL*10mM (DMSO) | 273.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CMPDA
CAS:380607-77-2
CMPDA is a positive allosteric modulator of AMPA receptors [EC50s: 45.4 nM/63.4 nM for GluA2i/GluA2o …
Formula:
C16H28N2O4S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
376.53
Ref: TM-TQ0114
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 27 Jan 2025
MSOP
CAS:66515-29-5
MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM …
Formula:
C4H10NO6P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
199.1
Ref: TM-T12118
| 5mg | 342.00 € | ||
| 25mg | 1,262.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
(1R,2S)-VU0155041
CAS:1263273-14-8
(1R,2S)-VU0155041 is the cis regioisomer of VU0155041 and a partial agonist of mGluR4.
Formula:
C14H15Cl2NO3
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
316.18
Ref: TM-T13424
| 5mg | 38.00 € | ||
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
A-794282
CAS:869802-44-8
A-794282 is a selective antagonist of mGluR1.
Formula:
C19H18N4OS
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
350.44
Ref: TM-T26486
| 1mg | 273.00 € | ||
| 2mg | 406.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 919.00 € | ||
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
AZD 9272
CAS:327056-26-8
AZD 9272 is a brain-permeable mGluR5 antagonist for the study of gastroesophageal reflux.
Formula:
C14H6F2N4O
Purity:
97.53%
Color and Shape:
Solid
Molecular weight:
284.22
Ref: TM-T14389
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 330.00 € | ||
| 50mg | 495.00 € | ||
| 100mg | 727.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
VU0652835
CAS:1848252-81-2
VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 …
Formula:
C16H19N3O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
333.41
Ref: TM-T13319
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
LY-2300559
CAS:889115-58-6
LY-2300559 is an agonist of metabotropic glutamate receptor 2 (mGluR2) and can be used in …
Formula:
C26H26O6
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
434.48
Ref: TM-T27932
| 1mg | 327.00 € | ||
| 5mg | 772.00 € | ||
| 10mg | 1,054.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 4,568.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
ABP688
CAS:924298-51-1
ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used …
Formula:
C15H16N2O
Purity:
97.85%
Color and Shape:
Solid
Molecular weight:
240.3
Ref: TM-T26520
| 5mg | 57.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 275.00 € | ||
| 100mg | 401.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
VU 0469650
CAS:1443748-47-7
VU 0469650 is a potent and selective negative allosteric modulator of mGluR1 (IC50 = 99 …
Formula:
C22H28N4O
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
364.48
Ref: TM-T29118
| 1mg | 66.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 538.00 € | ||
| 100mg | 796.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
