GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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Cyclothiazide
CAS:2259-96-3
Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).
Formula:
C14H16ClN3O4S2
Purity:
98.23% - 99.49%
Color and Shape:
Crystals From Dilute Alcohol Solid
Molecular weight:
389.88
Ref: TM-T4573
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 349.00 € | ||
| 200mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Friday 16 May 2025
IDRA-21
CAS:22503-72-6
IDRA-21 is a positive AMPA receptor modulator.
Formula:
C8H9ClN2O2S
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
232.69
Ref: TM-T7823
| 50mg | 46.00 € | ||
| 100mg | 65.00 € | ||
| 500mg | 155.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 16 May 2025
HBT1
CAS:489408-02-8
HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and …
Formula:
C16H17F3N4O2S
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
386.39
Ref: TM-T8779
| 10mg | 48.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 116.00 € | ||
| 100mg | 188.00 € | ||
| 200mg | 281.00 € | ||
| 1mL*10mM (DMSO) | 48.00 € |
Estimated delivery in United States, on Friday 16 May 2025
ADX-47273
CAS:851881-60-2
ADX-47273 (BA 94673139) is a positive and selective allosteric modulator for the metabotropic glutamate receptor …
Formula:
C20H17F2N3O2
Purity:
97% - 99.18%
Color and Shape:
Solid
Molecular weight:
369.36
Ref: TM-T2053
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 166.00 € | ||
| 50mg | 300.00 € | ||
| 100mg | 540.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Caroverine hydrochloride
CAS:55750-05-5
Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.
Formula:
C22H28ClN3O2
Purity:
98.37% - 98.75%
Color and Shape:
Solid
Molecular weight:
401.9
Ref: TM-T9133
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 216.00 € | ||
| 100mg | 378.00 € | ||
| 200mg | 552.00 € | ||
| 500mg | 868.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 16 May 2025
AMN082 free base
CAS:83027-13-8
AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.
Formula:
C28H28N2
Purity:
97.75% - 97.79%
Color and Shape:
Solid
Molecular weight:
392.54
Ref: TM-T21935L
| 1mg | 39.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 567.00 € | ||
| 200mg | 793.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Friday 16 May 2025
ADX88178
CAS:1235318-89-4
ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 …
Formula:
C12H12N6S
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
272.33
Ref: TM-T4500
| 2mg | 38.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 243.00 € | ||
| 100mg | 354.00 € | ||
| 200mg | 505.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Friday 16 May 2025
VU0155041
CAS:1093757-42-6
VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, …
Formula:
C14H15Cl2NO3
Purity:
99.52% - 99.56%
Color and Shape:
Solid
Molecular weight:
316.18
Ref: TM-T3565
| 2mg | 40.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 188.00 € | ||
| 100mg | 301.00 € | ||
| 200mg | 435.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Friday 16 May 2025
JNJ-40411813
CAS:1127498-03-6
JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor …
Formula:
C20H25ClN2O
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
344.88
Ref: TM-TQ0094
| 1mg | 55.00 € | ||
| 5mg | 117.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 306.00 € | ||
| 50mg | 437.00 € | ||
| 100mg | 562.00 € | ||
| 200mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 131.00 € |
Estimated delivery in United States, on Friday 16 May 2025
IEM 1754 2HBr
CAS:162831-31-4
IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and …
Formula:
C16H30N2·2HBr
Purity:
99.71% - 99.72%
Color and Shape:
Solid
Molecular weight:
412.25
Ref: TM-T6134
| 25mg | 64.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 139.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Friday 13 Jun 2025
AZD 9272
CAS:327056-26-8
AZD 9272 is a brain-permeable mGluR5 antagonist for the study of gastroesophageal reflux.
Formula:
C14H6F2N4O
Purity:
97.53%
Color and Shape:
Solid
Molecular weight:
284.22
Ref: TM-T14389
| 2mg | 42.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 447.00 € | ||
| 200mg | 627.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
BMT-145027
CAS:2018282-44-3
BMT-145027 is a positive allosteric modulator of mGluR5 without inherent agonist activity (EC50 = 47 …
Formula:
C23H14ClF3N4
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
438.83
Ref: TM-T10573
| 2mg | 39.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 270.00 € | ||
| 200mg | 375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
MFZ 10-7 hydrochloride
CAS:1779796-36-9
MFZ 10-7 hydrochloride is a highly potent and selective negative allosteric modulator of mGluR5 NAM
Formula:
C15H10ClFN2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
272.71
Ref: TM-T12025
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
NS 1209
CAS:205645-02-9
NS 1209 (SPD 502) is a AMPA receptor antagonist.
Formula:
C24H27N4NaO7S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
538.55
Ref: TM-T4009
| 25mg | 822.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
LY392098
CAS:211311-39-6
LY392098 (AMPA receptor modulator-3) is an allosteric modulator of AMPA receptor with EC50 of 4.4 …
Formula:
C18H22FNO2S
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
335.44
Ref: TM-T27951
| 1mg | 42.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 437.00 € | ||
| 200mg | 605.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
VU 0469650
CAS:1443748-47-7
VU 0469650 is a potent and selective negative allosteric modulator of mGluR1 (IC50 = 99 …
Formula:
C22H28N4O
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
364.48
Ref: TM-T29118
| 1mg | 66.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 550.00 € | ||
| 100mg | 815.00 € | ||
| 1mL*10mM (DMSO) | 142.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
(1R,2S)-VU0155041
CAS:1263273-14-8
(1R,2S)-VU0155041 is the cis regioisomer of VU0155041 and a partial agonist of mGluR4.
Formula:
C14H15Cl2NO3
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
316.18
Ref: TM-T13424
| 5mg | 38.00 € | ||
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Methoxy-PEPy
CAS:524924-76-3
Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 …
Formula:
C13H10N2O
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
210.23
Ref: TM-T12012
| 1mg | 35.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 492.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
LYPLAL1-IN-1
CAS:1966129-74-7
LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also …
Formula:
C29H29N7O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
539.59
Ref: TM-T15823
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
AZD6538
CAS:453566-30-8
AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such …
Formula:
C15H6FN5O
Purity:
98.68%
Color and Shape:
Solid
Molecular weight:
291.24
Ref: TM-T26719
| 1mg | 35.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 303.00 € | ||
| 100mg | 449.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
