GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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A-794282
CAS:869802-44-8
A-794282 is a selective antagonist of mGluR1.
Formula:
C19H18N4OS
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
350.44
Ref: TM-T26486
| 1mg | 279.00 € | ||
| 2mg | 414.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
JNJ-55511118
CAS:2036081-86-2
JNJ-55511118 is a TARP γ8 allosteric modulator with anticonvulsant activity, which can be used in …
Formula:
C14H8ClF3N2O2
Color and Shape:
Solid
Molecular weight:
328.67
Ref: TM-T25558
| 1mg | 93.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 435.00 € | ||
| 25mg | 965.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
DCB
CAS:6971-97-7
DCB is an mGluR5 allosteric ligand that blocks mGluR modulation, countering DMeOB and DFB effects.
Formula:
C14H10Cl2N2
Purity:
99.12% - 99.9%
Color and Shape:
Solid
Molecular weight:
277.15
Ref: TM-T22711
| 5mg | 39.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 170.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 378.00 € | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
(E/Z)-SIB-1893
CAS:6266-99-5
(E/Z)-SIB-1893 (SIB 1893) is the racemate of (E)-SIB-1893 and (Z)-SIB-1893.
Formula:
C14H13N
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
195.26
Ref: TM-T23353
| 5mg | 73.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 562.00 € | ||
| 500mg | 1,216.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
ABP688
CAS:924298-51-1
ABP688 is a non-competitive and selective mGluR5 antagonist(Ki = 1.7 nM). ABP688 can be used …
Formula:
C15H16N2O
Purity:
97.85%
Color and Shape:
Solid
Molecular weight:
240.3
Ref: TM-T26520
| 5mg | 38.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 110.00 € | ||
| 50mg | 168.00 € | ||
| 100mg | 251.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
VU 0469650
CAS:1443748-47-7
VU 0469650 is a potent and selective negative allosteric modulator of mGluR1 (IC50 = 99 …
Formula:
C22H28N4O
Purity:
97.27%
Color and Shape:
Solid
Molecular weight:
364.48
Ref: TM-T29118
| 1mg | 66.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 369.00 € | ||
| 50mg | 550.00 € | ||
| 100mg | 815.00 € | ||
| 1mL*10mM (DMSO) | 142.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
Foliglurax
CAS:1883329-51-8
Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) …
Formula:
C23H23N3O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
421.51
Ref: TM-T11311L
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
BMT-145027
CAS:2018282-44-3
BMT-145027 is a positive allosteric modulator of mGluR5 without inherent agonist activity (EC50 = 47 …
Formula:
C23H14ClF3N4
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
438.83
Ref: TM-T10573
| 2mg | 39.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 270.00 € | ||
| 200mg | 375.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
ML337
CAS:1443118-44-2
ML337 is a negative allosteric modulator of mGlu3 with an IC50 of 593 nM.
Formula:
C21H20FNO3
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
353.39
Ref: TM-T23003
| 1mg | 35.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 309.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
LY382884
CAS:211566-75-5
LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade …
Formula:
C18H23NO4
Purity:
98.06% - 98.71%
Color and Shape:
Solid
Molecular weight:
317.38
Ref: TM-T27949
| 1mg | 710.00 € | ||
| 5mg | 1,491.00 € | ||
| 10mg | 1,882.00 € | ||
| 25mg | 2,452.00 € | ||
| 50mg | 3,022.00 € | ||
| 100mg | 4,085.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
LY392098
CAS:211311-39-6
LY392098 (AMPA receptor modulator-3) is an allosteric modulator of AMPA receptor with EC50 of 4.4 …
Formula:
C18H22FNO2S
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
335.44
Ref: TM-T27951
| 1mg | 42.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 437.00 € | ||
| 200mg | 605.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
NS 1209
CAS:205645-02-9
NS 1209 (SPD 502) is a AMPA receptor antagonist.
Formula:
C24H27N4NaO7S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
538.55
Ref: TM-T4009
| 25mg | 822.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
AZD6538
CAS:453566-30-8
AZD6538 is an mGluR5 negative allosteric modulator used in the study of CNS-related diseases such …
Formula:
C15H6FN5O
Purity:
98.68%
Color and Shape:
Solid
Molecular weight:
291.24
Ref: TM-T26719
| 1mg | 35.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 303.00 € | ||
| 100mg | 449.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
HexylHIBO
CAS:334887-43-3
HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values …
Formula:
C12H20N2O4
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
256.3
Ref: TM-T22840
| 1mg | 85.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 565.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 15 May 2025
Dasolampanel
CAS:503294-13-1
Dasolampanel (NGX-426) is an ionotropic glutamate receptor AMPA and Kainate receptor antagonist for the study …
Formula:
C17H20ClN5O3
Purity:
99%
Color and Shape:
Solid
Molecular weight:
377.83
Ref: TM-T31208
| 1mg | 723.00 € | ||
| 5mg | 1,510.00 € | ||
| 25mg | 2,745.00 € | ||
| 50mg | 3,591.00 € | ||
| 100mg | 4,940.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
(S)-MCPG
CAS:150145-89-4
(S)-MCPG is the active isomer of (RS)-MCPG, non-selective group I/group II metabotropic glutamate receptor antagonist.
Formula:
C10H11NO4
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
209.20
Ref: TM-T13452
| 1mg | 35.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Thursday 15 May 2025
CBiPES hydrochloride
CAS:856702-40-4
CBiPES hydrochloride (CBiPES HCl) is an orthosteric modulator of the mGlu2 receptor and is used …
Formula:
C21H20ClN3O2S
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
413.92
Ref: TM-T22638
| 1mg | 170.00 € | ||
| 5mg | 416.00 € | ||
| 10mg | 603.00 € | ||
| 25mg | 935.00 € | ||
| 50mg | 1,254.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,410.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
CPCCOEt
CAS:179067-99-3
CPCCOEt is a low affinity, selective, non-competitive and reversible antagonist of mGluR1b
Formula:
C13H13NO4
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
247.25
Ref: TM-T22692
| 5mg | 52.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 134.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 313.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
S 18986
CAS:175340-20-2
S 18986 is a selective, orally active, brain penetrant positive allosteric modulator of AMPA-type receptors, …
Formula:
C10H12N2O2S
Purity:
99.25%
Color and Shape:
Solid
Molecular weight:
224.28
Ref: TM-T16816
| 1mg | 35.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 15 May 2025
VU 0285683
CAS:327056-22-4
VU 0285683 is a specific negative allosteric modulator of mGluR5 with a high affinity for …
Formula:
C14H7FN4O
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
266.23
Ref: TM-T23509
| 1mg | 42.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 335.00 € | ||
| 200mg | 455.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
