GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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Foliglurax
CAS:1883329-51-8
Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) …
Formula:
C23H23N3O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
421.51
Ref: TM-T11311L
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
VU6001376
CAS:1968546-34-0
VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 …
Formula:
C18H14F2N6OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
400.41
Ref: TM-T17248
| 25mg | 1,586.00 € | ||
| 50mg | 2,072.00 € | ||
| 100mg | 2,660.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Ro 67-4853
CAS:302841-89-0
Ro 67-4853 is a positive allosteric modulator of mGluR1, selectively enhancing the response to the …
Formula:
C19H19NO4
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
325.36
Ref: TM-T23248
| 1mg | 70.00 € | ||
| 5mg | 151.00 € | ||
| 10mg | 214.00 € | ||
| 25mg | 367.00 € | ||
| 50mg | 533.00 € | ||
| 100mg | 758.00 € | ||
| 200mg | 999.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
VU0155041 sodium
CAS:1259372-69-4
VU0155041 sodium is a positive allosteric modulator of mGluR4 that promotes extinction in male rats.
Formula:
C14H14Cl2NNaO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
338.16
Ref: TM-T23507
| 5mg | 154.00 € | ||
| 10mg | 273.00 € | ||
| 50mg | 782.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
HexylHIBO
CAS:334887-43-3
HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values …
Formula:
C12H20N2O4
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
256.3
Ref: TM-T22840
| 1mg | 85.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 565.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Dasolampanel
CAS:503294-13-1
Dasolampanel (NGX-426) is an ionotropic glutamate receptor AMPA and Kainate receptor antagonist for the study …
Formula:
C17H20ClN5O3
Purity:
99%
Color and Shape:
Solid
Molecular weight:
377.83
Ref: TM-T31208
| 1mg | 723.00 € | ||
| 5mg | 1,510.00 € | ||
| 25mg | 2,745.00 € | ||
| 50mg | 3,591.00 € | ||
| 100mg | 4,940.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
(S)-MCPG
CAS:150145-89-4
(S)-MCPG is the active isomer of (RS)-MCPG, non-selective group I/group II metabotropic glutamate receptor antagonist.
Formula:
C10H11NO4
Purity:
98.72%
Color and Shape:
Solid
Molecular weight:
209.20
Ref: TM-T13452
| 1mg | 35.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
DMeOB
CAS:40252-74-2
DMeOB (3,3'-Dimethoxybenzaldazine) is a negative regulator with mGluR5 agonist activity and is used in the …
Formula:
C16H16N2O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
268.31
Ref: TM-T22736
| 1mg | 35.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 311.00 € | ||
| 100mg | 472.00 € | ||
| 500mg | 1,017.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Dipraglurant
CAS:872363-17-2
Dipraglurant: a blood-brain permeable mGluR5 NAM, orally active, selective, IC50 = 21 nM, treats PD-LID.
Formula:
C16H12FN3
Purity:
98.7%
Color and Shape:
Solid
Molecular weight:
265.29
Ref: TM-T15134
| 1mg | 97.00 € | ||
| 5mg | 227.00 € | ||
| 10mg | 329.00 € | ||
| 25mg | 723.00 € | ||
| 50mg | 1,064.00 € | ||
| 100mg | 1,415.00 € | ||
| 1mL*10mM (DMSO) | 274.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
A-794282
CAS:869802-44-8
A-794282 is a selective antagonist of mGluR1.
Formula:
C19H18N4OS
Purity:
≥98%
Color and Shape:
Solid
Molecular weight:
350.44
Ref: TM-T26486
| 1mg | 279.00 € | ||
| 2mg | 414.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Biphenylindanone A
CAS:866823-73-6
Biphenylindanone A is a selective potentiator of human mGluR2 (hmGluR2),and for the treatment of neurological …
Formula:
C30H30O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
454.56
Ref: TM-T14615
| 5mg | 364.00 € | ||
| 10mg | 633.00 € | ||
| 25mg | 1,454.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
MFZ 10-7
CAS:1224431-15-5
MFZ 10-7 is anegative allosteric modulator of the mGluR5.
Formula:
C15H9FN2
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
236.24
Ref: TM-T22976
| 1mg | 40.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 545.00 € | ||
| 200mg | 740.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
Philanthotoxin 74 dihydrochloride
CAS:1227301-51-0
Philanthotoxin 74 dihydrochloride is an antagonist of AMPAR with IC50s of 263 and 296 nM …
Formula:
C24H44Cl2N4O3
Purity:
98.6%
Color and Shape:
Solid
Molecular weight:
507.54
Ref: TM-T16524
| 1mg | 51.00 € | ||
| 5mg | 146.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 190.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
FPTQ
CAS:864863-72-9
FPTQ is a highly effective antagonist of mGluR 1, displaying IC50 values of 6 nM …
Formula:
C17H12FN5
Purity:
99.68% - 99.88%
Color and Shape:
Solid
Molecular weight:
305.31
Ref: TM-T5509
| 1mg | 50.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 310.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 557.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
cis-PDA
CAS:46026-75-9
cis-PDA (cis PDA) is a general ionotropic receptor antagonist. cis-PDA acts by blocking NMDA, AMPA, …
Formula:
C7H11NO4
Purity:
≥98%
Color and Shape:
White Solid
Molecular weight:
173.17
Ref: TM-T20571
| 10mg | 34.00 € | ||
| 25mg | 49.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 11 Jul 2025
Pomaglumetad methionil hydrochloride
CAS:635318-26-2
LY2140023 hydrochloride: oral methionine prodrug of LY404039, a selective mGlu2/3 agonist, studied for schizophrenia.
Formula:
C12H19ClN2O7S2
Purity:
99.01%
Color and Shape:
Solid
Molecular weight:
402.87
Ref: TM-T61972
| 1mg | 202.00 € | ||
| 5mg | 512.00 € | ||
| 10mg | 740.00 € | ||
| 25mg | 1,121.00 € | ||
| 50mg | 1,539.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
VU0360172
CAS:1310012-12-4
VU0360172 is a positive allosteric modulator of mGlu5 receptors (EC50 = 16 nM; Ki = …
Formula:
C18H15FN2O
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
294.32
Ref: TM-T29126
| 1mg | 57.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 376.00 € | ||
| 50mg | 588.00 € | ||
| 100mg | 833.00 € | ||
| 1mL*10mM (DMSO) | 115.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
VU6004909
CAS:1860797-76-7
VU6004909 is an mGlu5 receptor orthosteric modulator that reverses MK801-induced increased cortical activity and cognitive …
Formula:
C21H15FN2O4
Purity:
96.68% - 98.44%
Color and Shape:
Liquid
Molecular weight:
378.35
Ref: TM-T79784
| 1mg | 47.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 256.00 € | ||
| 50mg | 410.00 € | ||
| 100mg | 647.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
VU6005649
CAS:2137047-43-7
VU6005649 is an agonist of CNS penetrant mGlu7/8 receptor (EC50s: 0.65 μM and 2.6 μM …
Formula:
C16H12F5N3O
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
357.28
Ref: TM-T13321
| 5mg | 40.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 170.00 € | ||
| 100mg | 259.00 € | ||
| 200mg | 369.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
L-AP4
CAS:23052-81-5
L-APB is an effective and specific agonist for the group III mGluRs (EC50s: 0.13, 0.29, …
Formula:
C4H10NO5P
Purity:
98%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
183.1
Ref: TM-T15692
| 1mg | To inquire | ||
| 5mg | To inquire | ||
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 11 Jul 2025
