AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 643 products of "AChR"
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N-Ethyl-N-(3-pyridylmethyl)amine
CAS:N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.Formula:C8H12N2Purity:99.65%Color and Shape:SolidMolecular weight:136.19Dibucaine hydrochloride
CAS:Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.Formula:C20H30ClN3O2Purity:99.66%Color and Shape:White PowderMolecular weight:379.92Metixene hydrochloride hydrate
CAS:Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and Ki of 15 nM against muscarine receptors.Formula:C20H26ClNOSPurity:99.99%Color and Shape:SolidMolecular weight:363.95Telenzepine dihydrochloride
CAS:muscarinic M1 receptor antagonistFormula:C19H23ClN4O2SPurity:98%Color and Shape:SolidMolecular weight:406.93Solifenacin D5 hydrochloride
CAS:Solifenacin D5 HCl: deuterium-labeled M1, M2, M3 muscarinic receptor antagonist with pKi 7.6, 6.9, 8.0.Formula:C23H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:403.96Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Formula:C20H22Cl2N2O4Color and Shape:SolidMolecular weight:425.31N6-Methyladenosine 5'-monophosphate disodium salt
CAS:N6-Methyladenosine 5'-monophosphate disodium salt is a glycogen phosphorylase b activator and an inhibitor of adenylate kinase II.Formula:C11H14N5Na2O7PPurity:99.36% - 99.36%Color and Shape:SolidMolecular weight:405.21Cevimeline
CAS:Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.Formula:C10H17NOSColor and Shape:Off-White SolidMolecular weight:199.31Fesoterodine L-mandelate
CAS:Fesoterodine L-mandelate is a efficacious antimuscarinic agent for the overactive bladder (OAB).Formula:C34H45NO6Color and Shape:SolidMolecular weight:563.735YM-58790 hydrochloride
CAS:YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).Formula:C27H32ClN3O2Purity:98%Color and Shape:SolidMolecular weight:466.02Palmatine hydroxide
CAS:Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.Formula:C21H23NO5Color and Shape:SolidMolecular weight:369.41β2AR/M-receptor agonist-2
CAS:β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).Formula:C36H49ClN4O7SColor and Shape:SolidMolecular weight:717.31Dexetimide
CAS:Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.Formula:C23H26N2O2Color and Shape:SolidMolecular weight:362.46Varenicline Hydrochloride
CAS:Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).Formula:C13H14ClN3Purity:99.854%Color and Shape:SolidMolecular weight:247.72Ref: TM-T23502
1mg37.00€5mg77.00€10mg99.00€25mg182.00€50mg282.00€100mg419.00€200mg612.00€1mL*10mM (DMSO)83.00€Glycerophosphoinositol choline
CAS:Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.Formula:C14H32NO12PColor and Shape:SolidMolecular weight:437.38Cevimeline hydrochloride
CAS:Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.Formula:C10H18ClOSColor and Shape:SolidMolecular weight:235.77(±)-Darifenacin
CAS:(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.Formula:C28H30N2O2Color and Shape:SolidMolecular weight:426.55VU0467485
CAS:VU0467485 boosts ACh at M4 receptors (EC50: 26.6 nM rat, 78.8 nM human), selective for M4 over M1/2/3/5.Formula:C17H17FN4O2SPurity:98%Color and Shape:SolidMolecular weight:360.41SSR180711 hydrochloride
CAS:SSR180711 hydrochloride (SSR-180711A HCl) is an Alpha7 nicotinic acetylcholine partial agonist that can be used to study neurolysis.Formula:C14H18BrClN2O2Purity:99.22%Color and Shape:SolidMolecular weight:361.66Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formula:C11H16ClNOPurity:98.9%Color and Shape:SolidMolecular weight:213.7NBTGR
CAS:NBTGR is a potent nucleoside transport inhibitor(adenosine uptake ,Ki of 70 nM).Formula:C17H18N6O6SPurity:98%Color and Shape:SolidMolecular weight:434.43Biperiden
CAS:Biperiden is a muscarinic antagonist for Parkinson's and drug-induced extrapyramidal symptoms.Formula:C21H29NOPurity:99.65%Color and Shape:Crystals SolidMolecular weight:311.46Ispronicline
CAS:Ispronicline (TC-1734) An orally active, selective, and potent α4β2 nAChR partial agonist with antidepressant, neuroprotective, and long-lasting cognitiveFormula:C14H22N2OPurity:97.70% - 99.16%Color and Shape:SolidMolecular weight:234.34Pirmenol hydrochloride
CAS:Pirmenol hydrochloride functions by inhibiting I_K.ACh through the blockade of muscarinic receptors, demonstrating a potent effect with an IC_50 value of 0.1 μMFormula:C22H31ClN2OColor and Shape:SolidMolecular weight:374.95Tebanicline dihydrochloride
CAS:Tebanicline dihydrochloride: oral analgesic, nAChR modulator, Ki=37 pM at α4β2 receptors, inhibits cytisine binding.Formula:C9H13Cl3N2OColor and Shape:SolidMolecular weight:271.57(S)-(+)-Dimethindene maleate
CAS:(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptorsFormula:C24H28N2O4Purity:99.94%Color and Shape:SolidMolecular weight:408.49Sabcomeline hydrochloride
CAS:Sabcomeline is a selective M1 receptor partial agonist.Formula:C10H16ClN3OColor and Shape:SolidMolecular weight:229.71Tolterodine
CAS:Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.Formula:C22H31NOPurity:99.71%Color and Shape:White Like Or Light Brown Crystalline PowderMolecular weight:325.49NS3861 fumarate
CAS:NS3861 fumarate, a partial α3β4 nAChR agonist, binds α3β2, α4β4, α4β2 with Ki values of 0.62, 25, 7.8, 55 nM.Formula:C16H18BrNO4SColor and Shape:SolidMolecular weight:400.29ABT-107
CAS:ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.Formula:C19H20N4OColor and Shape:SolidMolecular weight:320.396NSC 23766
CAS:NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.Formula:C24H35N7Purity:99.49%Color and Shape:SolidMolecular weight:421.58DL-Cystine
CAS:DL-Cystine is a cysteine derivative that inhibits endothelial cell proliferation by regulating TGFβ1. a GPR inhibitor and nAChR agonist .Formula:C6H12N2O4S2Color and Shape:SolidMolecular weight:240.3NKH477
CAS:NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.Formula:C27H44ClNO8Purity:98% - 98%Color and Shape:SolidMolecular weight:546.09α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Formula:C69H107N23O24S4Purity:94.82% - 97.79%Color and Shape:SolidMolecular weight:1770.99Succinylcholine Chloride Dihydrate
CAS:Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a depolarizing neuromuscular blocker.
Formula:C14H30N2O4·2Cl·2H2OPurity:99.87%Color and Shape:White SolidMolecular weight:397.34Tebanicline hydrochloride
CAS:Tebanicline hydrochloride (Ebanicline hydrochloride) , is an effective synthetic nicotinic (non-opioid) analgesic drug.Formula:C9H12Cl2N2OPurity:91.74% - 98.78%Color and Shape:SolidMolecular weight:235.11Piperidolate hydrochloride
CAS:Piperidolate hydrochloride, an antimuscarinic, reduces acetylcholine-induced intestinal spasms in rats and dogs.Formula:C21H26ClNO2Purity:99.5%Color and Shape:SolidMolecular weight:359.89Clothianidin
CAS:Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.Formula:C6H8ClN5O2SPurity:99.71% - 99.87%Color and Shape:Solid PowderMolecular weight:249.68VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Formula:C15H10BrNO2Purity:97.56%Color and Shape:SolidMolecular weight:316.15Tosedostat
CAS:Tosedostat (CHR-2797), an oral M1 aminopeptidase inhibitor, turns into CHR-79888, blocks tumor cell proteins, causing cell death.Formula:C21H30N2O6Purity:98.14% - 99.84%Color and Shape:SolidMolecular weight:406.47VU0152100
CAS:VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).Formula:C18H19N3O2SPurity:99.56%Color and Shape:SolidMolecular weight:341.43Ref: TM-T17238
2mg39.00€5mg58.00€10mg92.00€25mg195.00€50mg325.00€100mg522.00€200mg743.00€1mL*10mM (DMSO)64.00€Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41VU0467154
CAS:VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.Formula:C17H15F3N4O3S2Purity:99.51% - 99.53%Color and Shape:SolidMolecular weight:444.45Ref: TM-T17244
1mg47.00€2mg63.00€5mg92.00€10mg126.00€25mg236.00€50mg400.00€100mg695.00€200mg945.00€1mL*10mM (DMSO)101.00€NS9283
CAS:NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.
Formula:C14H8N4OPurity:99.12%Color and Shape:SolidMolecular weight:248.24Varenicline Tartrate
CAS:Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.
Formula:C13H13N3·C4H6O6Purity:98.23% - 98.32%Color and Shape:Tan SolidMolecular weight:361.35Propiverine hydrochloride
CAS:Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).Formula:C23H30ClNO3Purity:99.93%Color and Shape:White Crystalling PowerMolecular weight:403.94ML380
CAS:ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).Formula:C23H25F3N4O3SPurity:99.69%Color and Shape:SolidMolecular weight:494.53Ref: TM-T28069
2mg47.00€5mg71.00€10mg113.00€25mg178.00€50mg334.00€100mg500.00€500mg1,099.00€1mL*10mM (DMSO)78.00€Isopropamide Iodide
CAS:Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.
Formula:C23H33IN2OPurity:99.67%Color and Shape:SolidMolecular weight:480.43JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Formula:C19H20ClFN4Purity:99.72%Color and Shape:SolidMolecular weight:358.84Mc-Val-Ala-PAB
CAS:Mc-Val-Ala-PAB, an effective linker, is utilized in antibody-drug-conjugate (ADC).Formula:C25H34N4O6Purity:98.34% - 99.24%Color and Shape:SolidMolecular weight:486.56Nitenpyram
CAS:Nitenpyram (Capstar) is a nicotinic acetylcholine receptor (AchR) agonist, used as veterinary medicine to treat parasites of livestock and pets.Formula:C11H15ClN4O2Purity:99.03%Color and Shape:Light-Yellow CrystalMolecular weight:270.72Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurity:99.76% - >99.99%Color and Shape:White SolidMolecular weight:203.75Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Formula:C19H29N5O3·2(C2H4O2)Purity:99.60%Color and Shape:SolidMolecular weight:495.58Procyclidine hydrochloride
CAS:Procyclidine hydrochloride ((±)-Procyclidine hydrochlorid) is a potent anticholinergic agent and also have NMDA antagonist properties.Formula:C19H30ClNOPurity:99.24% - 99.88%Color and Shape:Crystals From Petroleum Ether White PowderMolecular weight:323.9KH7
CAS:KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Formula:C17H15BrN4O2SPurity:98.43%Color and Shape:SolidMolecular weight:419.3Batefenterol
CAS:Batefenterol (GSK961081) is a muscarinic antagonist and β2-agonist with high affinity (Ki: 1.4/1.3/3.7 nM).Formula:C40H42ClN5O7Purity:97.94% - 98.4%Color and Shape:SolidMolecular weight:740.24Solifenacin hydrochloride
CAS:Solifenacin Hcl is a muscarinic receptor antagonist.Formula:C23H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:398.93Encenicline
CAS:Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Formula:C16H17ClN2OSPurity:99.20%Color and Shape:SolidMolecular weight:320.84Ref: TM-T7193
1mg70.00€5mg133.00€10mg207.00€25mg349.00€50mg495.00€100mg675.00€200mg888.00€1mL*10mM (DMSO)144.00€Mecamylamine
CAS:Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Formula:C11H21NColor and Shape:SolidMolecular weight:167.29Oxyphencyclimine Hydrochloride
CAS:Oxyphencyclimine Hydrochloride (Ulcociclinina) is a synthetic tertiary amine and antimuscarinic agent with antispasmodic and antisecretory activities.Formula:C20H29ClN2O3Purity:99.55%Color and Shape:SolidMolecular weight:380.91Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formula:C7H14N4O3Purity:99.89%Color and Shape:White Crystalline PowderMolecular weight:202.21Propiverine
CAS:Propiverine reduces muscle spasms by limiting calcium influx, targeting bladder smooth muscles, aiding OAB research.Formula:C23H29NO3Color and Shape:SolidMolecular weight:367.48NS 1738
CAS:NS 1738 (NSC-213859) is a positive allosteric modulator of the α7-containing neuronal nicotinic acetylcholine receptors (nAChRs)Formula:C14H9Cl2F3N2O2Purity:99.11%Color and Shape:SolidMolecular weight:365.13Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Formula:C22H32BrNO5Purity:98.85%Color and Shape:SolidMolecular weight:470.4Ref: TM-T28827
1mg74.00€5mg160.00€10mg250.00€25mg452.00€50mg680.00€100mg1,008.00€200mg1,349.00€1mL*10mM (DMSO)165.00€ZSET1446
CAS:ZSET1446 (ST-101) is a T-type calcium channel activator potentially for the treatment of learning deficits in various types of Alzheimer disease (AD) models.Formula:C15H12N2OPurity:99.32%Color and Shape:SolidMolecular weight:236.27Ref: TM-T8448
1mg50.00€5mg103.00€10mg144.00€25mg281.00€50mg409.00€100mg572.00€200mg772.00€1mL*10mM (DMSO)119.00€EB-3D
CAS:EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.Formula:C30H36Br2N4O2Purity:99.48%Color and Shape:SolidMolecular weight:644.4Ref: TM-T7955
1mg87.00€2mg114.00€5mg177.00€10mg260.00€25mg447.00€50mg620.00€100mg875.00€200mg1,161.00€1mL*10mM (DMSO)263.00€Dronedarone
CAS:Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Formula:C31H44N2O5SPurity:98.85% - 99.99%Color and Shape:SolidMolecular weight:556.76Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Formula:C10H21NPurity:98.18% - 99.28%Color and Shape:Colorless - Light Yellow Clear LiquidMolecular weight:155.28Oxyphenonium bromide
CAS:Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.
Formula:C21H34BrNO3Purity:98.96%Color and Shape:SolidMolecular weight:428.404MC-Val-Cit-PABC-PNP
CAS:MC-Val-Cit-PABC-PNP, also known as Mc-Val-Cit-PABC-PNP, is a cathepsin cleavable ADC peptide linker.Formula:C35H43N7O11Purity:97.2% - 98.055%Color and Shape:SolidMolecular weight:737.76Propantheline
CAS:Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.Formula:C23H30NO3Color and Shape:SolidMolecular weight:368.49Simufilam dihydrochloride
CAS:Simufilam dihydrochloride is an oral, low-toxic FLNA activator for Alzheimer's research, restoring FLNA structure and function.Formula:C15H23Cl2N3OPurity:98.83%Color and Shape:SolidMolecular weight:332.3Ref: TM-T9172
1mg49.00€5mg95.00€10mg136.00€25mg279.00€50mg360.00€100mg470.00€200mg622.00€1mL*10mM (DMSO)96.00€VU0357017 hydrochloride
CAS:VU0357017 hydrochloride (ML071 hydrochloride) is highly selective M1 agonists act at an allosteric site to activate the receptor (EC50: 477 ± 172 nM; Pec50: 6.Formula:C18H28ClN3O3Purity:99% - 99.97%Color and Shape:SolidMolecular weight:369.89Iptakalim Hydrochloride
CAS:Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholineFormula:C9H22ClNPurity:98%Color and Shape:SolidMolecular weight:179.731Bestim
CAS:Bestim is an immunomodulatory dipeptide that is synthetic.Formula:C16H19N3O5Purity:99.76%Color and Shape:SolidMolecular weight:333.34Ref: TM-T25146
1mg84.00€5mg168.00€10mg245.00€25mg404.00€50mg567.00€100mg767.00€200mg1,018.00€1mL*10mM (DMSO)172.00€VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Formula:C18H17N3O3SPurity:98.46%Color and Shape:SolidMolecular weight:355.41Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Formula:C10H22ClNColor and Shape:SolidMolecular weight:191.74Rivanicline hemioxalate
Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.Formula:C12H16N2O4Purity:98%Color and Shape:SolidMolecular weight:207.23suvn-911
CAS:suvn-911 is a potent and selective antagonist of neuronal nicotinic acetylcholine α4β2 receptor (Ki = 1.5 nM) with antidepressant activity.Formula:C11H14Cl2N2OPurity:98.88%Color and Shape:SolidMolecular weight:261.15Ref: TM-T9787
1mg67.00€5mg133.00€10mg205.00€25mg339.00€50mg482.00€100mg658.00€200mg888.00€1mL*10mM (DMSO)172.00€Coluracetam
CAS:Coluracetam (MKC-231)(MKC-231) is a Choline Uptake Enhancer.Formula:C19H23N3O3Purity:99.96%Color and Shape:SolidMolecular weight:341.4Aclidinium bromide
CAS:Aclidinium bromide (LAS-W 330) is a synthetic anticholinergic agent that is used as an inhalant for treatment of acute bronchospasm due to chronic bronchitis.
Formula:C26H30NO4S2·BrPurity:99.53% - 99.69%Color and Shape:SolidMolecular weight:564.55Encenicline hydrochloride
CAS:Encenicline hydrochloride (EVP-6124 hydrochloride) is a new-type partial agonist of α7 neuronal nicotinic acetylcholine receptors (nAChRs).Formula:C16H17ClN2OS·HClPurity:98.34% - 99.85%Color and Shape:SolidMolecular weight:357.3Adiphenine
CAS:Adiphenine is an inhibitor of nicotinic receptors.Formula:C20H25NO2Color and Shape:SolidMolecular weight:311.42Irsogladine
CAS:Irsogladine (Dicloguamine) is an anti-ulcer agent that promotes gap junction intercellular communication via M1 muscarinic acetylcholine receptor binding.Formula:C9H7Cl2N5Purity:99.74% - 99.91%Color and Shape:White Or Colorless Crystal Or Crystalline Powder Odorless Slightly BitterMolecular weight:256.09VU0238441
CAS:VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.Formula:C16H9ClF3NO2Purity:100%Color and Shape:SolidMolecular weight:339.7Benzetimide hydrochloride
CAS:Benzetimide hydrochloride (R4929) is an antagonist of muscarinic acetylcholine receptor.treatment neuroleptic-induced parkinsonism.Formula:C23H27ClN2O2Purity:99.32%Color and Shape:Off-White PowderMolecular weight:398.93Oxyphencyclimine
CAS:Oxyphencyclimine is a muscarinic receptor antagonist (MRA) anticholinergic drug used to treat peptic ulcers.Formula:C20H28N2O3Color and Shape:SolidMolecular weight:344.45(S)-UFR2709
CAS:(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.Formula:C13H17NO2Color and Shape:SolidMolecular weight:219.284mAChR-IN-1 hydrochloride
CAS:mAChR-IN-1 hydrochloride is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 Nm.Formula:C23H26ClIN2O2Purity:99.87%Color and Shape:SolidMolecular weight:524.82Ref: TM-T5655
1mg38.00€5mg86.00€10mg126.00€25mg215.00€50mg298.00€100mg371.00€200mg494.00€1mL*10mM (DMSO)89.00€Batefenterol Succinate
CAS:Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formula:C44H48ClN5O11Color and Shape:SolidMolecular weight:858.34Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Formula:C23H26N2O2Purity:99.87%Color and Shape:SolidMolecular weight:362.46LY2119620
CAS:LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.Formula:C19H24ClN5O3SPurity:99.7%Color and Shape:SolidMolecular weight:437.94Pirmenol
CAS:Pirmenol is a new antiarrhythmic drugFormula:C22H30N2OPurity:97.24%Color and Shape:SolidMolecular weight:338.49GNF-7
CAS:GNF-7 is Bcr-Abl WT and Bcr-Abl T315I inhibitor with IC50 of 133 nM and 61 nM, respectively.Formula:C28H24F3N7O2Purity:97.05% - 99.7%Color and Shape:SolidMolecular weight:547.53Darifenacin
CAS:Darifenacin (UK-88525) is a muscarinic receptor M3 antagonist with anticonvulsant activity and can be used to study urinary incontinence and overactive bladder.Formula:C28H30N2O2Purity:99.78%Color and Shape:SolidMolecular weight:426.55Ref: TM-T62320
2mg39.00€5mg58.00€10mg93.00€25mg152.00€50mg236.00€100mg356.00€200mg522.00€1mL*10mM (DMSO)64.00€Harman hydrochloride
CAS:Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.Formula:C12H11ClN2Purity:99.35%Color and Shape:SolidMolecular weight:218.68Ilmetropium iodide
CAS:Ilmetropium iodide is a bronchodilator.Formula:C20H30INO3Purity:98.45%Color and Shape:SolidMolecular weight:459.36Brompheniramine
CAS:Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.Formula:C16H19BrN2Color and Shape:SolidMolecular weight:319.24Ursulcholic acid
CAS:Ursulcholic acid (Ursulcholic) is a water-soluble anticholinergic compound.Formula:C24H40O10S2Purity:98%Color and Shape:SolidMolecular weight:552.7Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Formula:C16H20N2O2Purity:98.63%Color and Shape:SolidMolecular weight:272.34Ref: TM-T22380
1mg72.00€5mg136.00€10mg197.00€25mg324.00€50mg452.00€100mg607.00€200mg810.00€1mL*10mM (DMSO)135.00€
