AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 643 products of "AChR"
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Encenicline
CAS:Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Formula:C16H17ClN2OSPurity:99.20%Color and Shape:SolidMolecular weight:320.84Ref: TM-T7193
1mg70.00€5mg133.00€10mg207.00€25mg349.00€50mg495.00€100mg675.00€200mg888.00€1mL*10mM (DMSO)144.00€GNF-7
CAS:GNF-7 is Bcr-Abl WT and Bcr-Abl T315I inhibitor with IC50 of 133 nM and 61 nM, respectively.Formula:C28H24F3N7O2Purity:97.05% - 99.7%Color and Shape:SolidMolecular weight:547.53Fmoc-Val-Ala-PAB-OH
CAS:Fmoc-Val-Ala-PAB-OH is a linker for ADCs and lysosomally cleavable RGD-paclitaxel conjugates.Formula:C30H33N3O5Purity:98.45% - 98.94%Color and Shape:SolidMolecular weight:515.6α-Conotoxin PIA acetate
α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.Purity:98%Color and Shape:LiquidMolecular weight:N/AIsopropamide Iodide
CAS:Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.
Formula:C23H33IN2OPurity:99.67%Color and Shape:SolidMolecular weight:480.43ML380
CAS:ML380 is a highly potent and the first CNS penetrant M5 positive allosteric modulator (PAM).Formula:C23H25F3N4O3SPurity:99.69%Color and Shape:SolidMolecular weight:494.53Ref: TM-T28069
2mg47.00€5mg71.00€10mg113.00€25mg178.00€50mg334.00€100mg500.00€500mg1,099.00€1mL*10mM (DMSO)78.00€Irsogladine
CAS:Irsogladine (Dicloguamine) is an anti-ulcer agent that promotes gap junction intercellular communication via M1 muscarinic acetylcholine receptor binding.Formula:C9H7Cl2N5Purity:99.74% - 99.91%Color and Shape:White Or Colorless Crystal Or Crystalline Powder Odorless Slightly BitterMolecular weight:256.09VU0152100
CAS:VU0152100 is an effective and selective allosteric potentiator of M4 mAChR (EC50: 380 ± 93 nM).Formula:C18H19N3O2SPurity:99.56%Color and Shape:SolidMolecular weight:341.43Ref: TM-T17238
2mg39.00€5mg58.00€10mg92.00€25mg195.00€50mg325.00€100mg522.00€200mg743.00€1mL*10mM (DMSO)64.00€VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Formula:C15H10BrNO2Purity:97.56%Color and Shape:SolidMolecular weight:316.15VU10010
CAS:VU10010 (VU 10010) is allosteric potentiator of M4 acetylcholine receptors.
Formula:C17H16ClN3OSPurity:99.36%Color and Shape:SolidMolecular weight:345.85Brompheniramine
CAS:Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.Formula:C16H19BrN2Color and Shape:SolidMolecular weight:319.24α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Formula:C69H107N23O24S4Purity:94.82% - 97.79%Color and Shape:SolidMolecular weight:1770.99Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Formula:C19H29N5O3·2(C2H4O2)Purity:99.60%Color and Shape:SolidMolecular weight:495.58Oxotremorine sesquifumarate
CAS:Oxotremorine sesquifumarate is a muscarinic agonist.
Formula:C12H18N2OC4H4O4Purity:97.94%Color and Shape:SolidMolecular weight:380.39TQS
CAS:TQS (4-Naphthalen-1-yl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide) is a positive allosteric modulator of α7 nACh receptors.Formula:C22H20N2O2SPurity:98.56%Color and Shape:SolidMolecular weight:376.47Ref: TM-T23469
5mg35.00€10mg52.00€25mg103.00€50mg167.00€100mg236.00€200mg338.00€1mL*10mM (DMSO)38.00€Tosedostat
CAS:Tosedostat (CHR-2797), an oral M1 aminopeptidase inhibitor, turns into CHR-79888, blocks tumor cell proteins, causing cell death.Formula:C21H30N2O6Purity:98.14% - 99.84%Color and Shape:SolidMolecular weight:406.47Clothianidin
CAS:Clothianidin (TI 435), an insecticide, stimulates nAChR as acetylcholine agonist, not AChE inhibitor.Formula:C6H8ClN5O2SPurity:99.71% - 99.87%Color and Shape:Solid PowderMolecular weight:249.68Propiverine hydrochloride
CAS:Propiverine is a widely used antimuscarinic drug with a mixed mode of action in the treatment of symptoms associated with overactive bladder (OAB).Formula:C23H30ClNO3Purity:99.93%Color and Shape:White Crystalling PowerMolecular weight:403.94PHA 568487
CAS:PHA 568487: α-7 nAChR agonist, rapid brain uptake, lessens oxidative stress & neuroinflammation.Formula:C20H24N2O7Color and Shape:SolidMolecular weight:404.419Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurity:99.76% - >99.99%Color and Shape:White SolidMolecular weight:203.75JHU37152
CAS:JHU37152 is a DREADD agonist; Ki: 1.8 nM at hM3Dq, 8.7 nM at hM4Di; EC50: 5 nM (hM3Dq), 0.5 nM (hM4Di) in HEK-293 cell assays.Formula:C19H20ClFN4Purity:99.72%Color and Shape:SolidMolecular weight:358.84Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Formula:C35H43N5O4Purity:98.12%Color and Shape:SolidMolecular weight:597.75Varenicline Tartrate
CAS:Varenicline Tartrate (CP 526555-18) is a benzazepine derivative that functions as an ALPHA4/BETA2 NICOTINIC RECEPTOR partial agonist.
Formula:C13H13N3·C4H6O6Purity:98.23% - 98.32%Color and Shape:Tan SolidMolecular weight:361.35Piperidolate
CAS:Piperidolate inhibits intestinal cramp induced by acetylcholineFormula:C21H25NO2Purity:98.45%Color and Shape:SolidMolecular weight:323.43PNU-282987 S enantiomer free base
CAS:PNU-282987 S enantiomer free base is an agonist of α7 nicotinic acetylcholine receptor (α7 nAChR).Formula:C14H17ClN2OPurity:99.74%Color and Shape:SolidMolecular weight:264.75Ref: TM-T7695
1mg71.00€5mg161.00€10mg219.00€25mg338.00€50mg460.00€100mg623.00€200mg837.00€1mL*10mM (DMSO)180.00€Simufilam dihydrochloride
CAS:Simufilam dihydrochloride is an oral, low-toxic FLNA activator for Alzheimer's research, restoring FLNA structure and function.Formula:C15H23Cl2N3OPurity:98.83%Color and Shape:SolidMolecular weight:332.3Ref: TM-T9172
1mg49.00€5mg95.00€10mg136.00€25mg279.00€50mg360.00€100mg470.00€200mg622.00€1mL*10mM (DMSO)96.00€Glycopyrrolate
CAS:Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.Formula:C19H28BrNO3Purity:99.41% - 99.64%Color and Shape:SolidMolecular weight:398.33Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Formula:C22H32BrNO5Purity:98.85%Color and Shape:SolidMolecular weight:470.4Ref: TM-T28827
1mg74.00€5mg160.00€10mg250.00€25mg452.00€50mg680.00€100mg1,008.00€200mg1,349.00€1mL*10mM (DMSO)165.00€Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formula:C7H14N4O3Purity:99.89%Color and Shape:White Crystalline PowderMolecular weight:202.21Pempidine
CAS:Pempidine (1,2,2,6,6-Pentamethylpiperidine) is a nicotinic antagonist, has been used as a ganglionic blocker in the treatment of hypertension.Formula:C10H21NPurity:98.18% - 99.28%Color and Shape:Colorless - Light Yellow Clear LiquidMolecular weight:155.28CCMI
CAS:CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.Formula:C19H15Cl2N3O2Purity:>99.99%Color and Shape:SolidMolecular weight:388.25Pozanicline dihydrochloride
CAS:Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)Formula:C11H18Cl2N2OPurity:98%Color and Shape:SolidMolecular weight:265.18W-84 dibromide
CAS:W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.Formula:C32H44Br2N4O4Purity:95.56%Color and Shape:SolidMolecular weight:708.52Dronedarone
CAS:Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Formula:C31H44N2O5SPurity:98.85% - 99.99%Color and Shape:SolidMolecular weight:556.76EB-3D
CAS:EB-3D is a potent and selective choline kinase alpha 1 (ChoKα1) inhibitor(IC50 : 1 μM).with anti-cancer activity.Formula:C30H36Br2N4O2Purity:99.48%Color and Shape:SolidMolecular weight:644.4Ref: TM-T7955
1mg87.00€2mg114.00€5mg177.00€10mg260.00€25mg447.00€50mg620.00€100mg875.00€200mg1,161.00€1mL*10mM (DMSO)263.00€Nor-benzetimide
CAS:Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.Formula:C16H20N2O2Purity:98.63%Color and Shape:SolidMolecular weight:272.34Ref: TM-T22380
1mg72.00€5mg136.00€10mg197.00€25mg324.00€50mg452.00€100mg607.00€200mg810.00€1mL*10mM (DMSO)135.00€Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Formula:C10H22ClNColor and Shape:SolidMolecular weight:191.74(S)-UFR2709
CAS:(S)-UFR2709, a nAChR competitive antagonist, favors α4β2 over α7, reduces anxiety and alcohol use in rats.Formula:C13H17NO2Color and Shape:SolidMolecular weight:219.284Adiphenine
CAS:Adiphenine is an inhibitor of nicotinic receptors.Formula:C20H25NO2Color and Shape:SolidMolecular weight:311.42Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Formula:C23H26N2O2Purity:99.87%Color and Shape:SolidMolecular weight:362.46VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Formula:C18H17N3O3SPurity:98.46%Color and Shape:SolidMolecular weight:355.41BQCA
CAS:BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.Formula:C18H15NO4Purity:97.22%Color and Shape:SolidMolecular weight:309.32VU0238441
CAS:VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.Formula:C16H9ClF3NO2Purity:100%Color and Shape:SolidMolecular weight:339.7Batefenterol Succinate
CAS:Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formula:C44H48ClN5O11Color and Shape:SolidMolecular weight:858.34Bestim
CAS:Bestim is an immunomodulatory dipeptide that is synthetic.Formula:C16H19N3O5Purity:99.76%Color and Shape:SolidMolecular weight:333.34Ref: TM-T25146
1mg84.00€5mg168.00€10mg245.00€25mg404.00€50mg567.00€100mg767.00€200mg1,018.00€1mL*10mM (DMSO)172.00€9-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purity:99.35% - 99.37%Color and Shape:SolidMolecular weight:163.18Oxyphenonium bromide
CAS:Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.
Formula:C21H34BrNO3Purity:98.96%Color and Shape:SolidMolecular weight:428.404Harman hydrochloride
CAS:Harman hydrochloride triggers CYP1A1 gene via AhR, potentially causing mutations and cancer.Formula:C12H11ClN2Purity:99.35%Color and Shape:SolidMolecular weight:218.68BNC210
CAS:BNC210 (IW-2143) is a α7 nAChR negative allosteric modulator. BNC210 has potent activity in animal models of anxiety and depression.Formula:C17H23N3O3Purity:97.05% - >99.99%Color and Shape:SolidMolecular weight:317.38NS9283
CAS:NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.
Formula:C14H8N4OPurity:99.12%Color and Shape:SolidMolecular weight:248.24ST034307
CAS:ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).Formula:C10H4Cl4O2Purity:99.28%Color and Shape:SolidMolecular weight:297.95Ref: TM-T16938
1mg38.00€2mg49.00€5mg81.00€10mg115.00€25mg235.00€50mg373.00€100mg597.00€200mg842.00€1mL*10mM (DMSO)88.00€TBPB
CAS:TBPB is an allosteric M1 mAChR agonist.
Formula:C25H32N4OPurity:97.87% - 99.9%Color and Shape:SolidMolecular weight:404.55Pipecuronium bromide
CAS:Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.Formula:C35H62Br2N4O4Purity:>99.99%Color and Shape:PowderMolecular weight:762.7Mepenzolate Bromide
CAS:Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.Formula:C21H26BrNO3Purity:95.73% - 99.21%Color and Shape:SolidMolecular weight:420.34AF-710B
CAS:AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.Formula:C20H27N3OSPurity:98.62% - 99.89%Color and Shape:SolidMolecular weight:357.51Xanomeline tartrate
CAS:Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂，具有抗精神病样活性，可改善认知，可用于研究精神分裂症和阿尔茨海默病。Formula:C18H29N3O7SPurity:99.19% - 99.99%Color and Shape:SolidMolecular weight:431.5Pentoxyverine
CAS:Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Formula:C20H31NO3Purity:97.11%Color and Shape:SolidMolecular weight:333.47Monepantel
CAS:Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.Formula:C20H13F6N3O2SPurity:99.83%Color and Shape:White PowderMolecular weight:473.39Ref: TM-T16126
1mg93.00€5mg236.00€10mg340.00€25mg670.00€50mg964.00€100mg1,378.00€1mL*10mM (DMSO)259.00€Velufenacin
CAS:Velufenacin is an antagonist of muscarinic receptor[1].Formula:C19H20ClFN2O2Purity:99.65%Color and Shape:SolidMolecular weight:362.83Ref: TM-T9771
1mg47.00€5mg96.00€10mg156.00€25mg270.00€50mg370.00€100mg522.00€200mg687.00€1mL*10mM (DMSO)105.00€Varenicline
CAS:Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.Formula:C13H13N3Purity:99.76%Color and Shape:SolidMolecular weight:211.26Ref: TM-T4246L
2mg34.00€5mg50.00€10mg75.00€25mg137.00€50mg200.00€100mg313.00€200mg464.00€1mL*10mM (DMSO)55.00€Flavoxate
CAS:Flavoxate is an anticholinergic with antimuscarinic effects.
Formula:C24H25NO4Color and Shape:SolidMolecular weight:391.46Atropine hydrobromide
CAS:Atropine hydrobromide is a biochemical.Formula:C17H24BrNO3Color and Shape:SolidMolecular weight:370.28Anatabine dicitrate
Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.Formula:C22H28N2O14Purity:98%Color and Shape:SolidMolecular weight:544.46Pyrantel
CAS:Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.Formula:C11H14N2SPurity:98%Color and Shape:Crystals From Methanol Yellowish Crystalline PowderMolecular weight:206.31(±)-Atropine-d3 (N-methyl-d3)
CAS:(±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.Formula:C17H20D3NO3Color and Shape:SolidMolecular weight:292.39Biperiden lactate
CAS:Biperiden lactate is a biochemical.
Formula:C24H35NO4Color and Shape:SolidMolecular weight:401.54Azacyclonol hydrochloride
CAS:Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.Formula:C18H22ClNOColor and Shape:Off White Crystalline PowderMolecular weight:303.83Oxantel
CAS:Oxantel is a fumarate reductase inhibitor with anthelmintic activity.Formula:C13H16N2OPurity:98%Color and Shape:SolidMolecular weight:216.28Diphenidol
CAS:Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.Formula:C21H27NOColor and Shape:Needles From Petroleum Ether SolidMolecular weight:309.45Catestatin
CAS:Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.Formula:C107H173N37O26SPurity:98%Color and Shape:SolidMolecular weight:2425.84VU0029767
CAS:VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.
Formula:C21H21N3O3Color and Shape:SolidMolecular weight:363.41Dianicline dihydrochloride
CAS:Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.Formula:C13H16N2OPurity:98%Color and Shape:SolidMolecular weight:216.28Phenglutarimide hydrochloride
CAS:Phenglutarimide hydrochloride is an anticholinergic. It is used as an antiparkinsonian agent.Formula:C17H25ClN2O2Color and Shape:SolidMolecular weight:324.85AN317
CAS:AN317 is a selective agonist for the nicotinic acetylcholine receptor (nAChR) containing α6β2, with dissociation constants (Ki) of 6.2 nM and 4.1 nM for the α6/α3β2β3 and α4β2 receptor subtypes, respectively. It induces dopamine release in rat striatal synaptosomes, enhances the activity of dopaminergic neurons in the substantia nigra, and exhibits protective effects against the dopaminergic neurotoxin MPP+ in rat neurons. AN317 also demonstrates favorable pharmacokinetic properties in rats and permeability across the blood-brain barrier (BB).Formula:C13H19N3Color and Shape:SolidMolecular weight:217.31Aprofene
CAS:Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.Formula:C21H27NO2Color and Shape:SolidMolecular weight:325.44N-Biotinyl p-aminophenyl arsenic acid
CAS:N-Biotinyl p-aminophenyl arsenic acid is a bifunctional reagent that binds to streptavidin and disulfide compounds. It diminishes the binding sites of rbungarotoxin on reduced nicotinic receptors with an IC50 ranging from 10-300 nM, thus shielding the receptors from irreversible alkylation by bromoacetylcholine.Formula:C16H22AsN3O4SColor and Shape:SolidMolecular weight:427.35Sulindac sulfide
CAS:Sulindac sulfide: NSAID targeting COX-1, inhibits Ras-Raf-1 and gamma-secretase (IC50: 20.2 μM), active sulinic acid metabolite.Formula:C20H17FO2SPurity:99.35%Color and Shape:SolidMolecular weight:340.41Pentolinium Tartrate
CAS:Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.Formula:C15H32N2·2C4H5O6Purity:98%Color and Shape:SolidMolecular weight:538.6AF-DX 384 free base
CAS:AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.Formula:C27H38N6O2Purity:98%Color and Shape:SolidMolecular weight:478.63Pozanicline
CAS:Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.Formula:C11H16N2OPurity:98%Color and Shape:SolidMolecular weight:192.26CB-6673567
CAS:CB-6673567 is a selective inhibitor of adenylyl cyclase.Formula:C19H14N4O3Color and Shape:SolidMolecular weight:346.34NGX-267
CAS:NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.Formula:C10H18N2OSColor and Shape:SolidMolecular weight:214.33Dac 5945
CAS:DAC 5945 is a more effective muscarinic antagonist in the airways than in the heart.Formula:C19H30ClN3OPurity:98%Color and Shape:SolidMolecular weight:351.91Hexocyclium metilsulfate
CAS:Hexocyclium metilsulfate has anti-gastric secretory effects in humans.Formula:C21H36N2O5SPurity:98%Color and Shape:SolidMolecular weight:428.59GS 283
CAS:GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.Formula:C17H17NO3Color and Shape:SolidMolecular weight:283.32(R)-VU 6008667
CAS:(R)-VU 6008667 is devoid of M5 NAM activity (IC50>10 μM).Formula:C24H17ClF2N2O2Color and Shape:SolidMolecular weight:438.85Anisodine hydrobromide
CAS:Anisodine hydrobromide is an inhibitor of adenosine kinase.Formula:C17H22BrNO5Color and Shape:White Crystals Or Crystalline PowderMolecular weight:400.27Btm 1042
CAS:Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.Formula:C21H26ClN3OSColor and Shape:SolidMolecular weight:403.97Hyoscyamine hydrobromide
CAS:Hyoscyamine hydrobromide is an agent of anticholinergic.Formula:C17H24BrNO3Purity:98%Color and Shape:SolidMolecular weight:370.28Sazetidine A dihydrochloride
CAS:α4β2 nicotinic acetylcholine receptor ligandFormula:C15H21ClN2O2Purity:98%Color and Shape:SolidMolecular weight:296.79FR 121196
CAS:FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.Formula:C12H16FN3O3SColor and Shape:SolidMolecular weight:301.34Prifuroline
CAS:Prifuroline is an agent of antiarrhythmic.Formula:C14H16N2OPurity:98%Color and Shape:SolidMolecular weight:228.29Epibatidine 2HCl
CAS:Epibatidine 2HCl is a potent nicotinic agonist.Formula:C11H15Cl3N2Purity:98%Color and Shape:SolidMolecular weight:281.61Flutropium Bromide
CAS:Flutropium Bromide is a competitive antagonist of acetylcholine. It is used to treat asthma and chronic obstructive pulmonary.Formula:C24H29BrFNO3Purity:98%Color and Shape:SolidMolecular weight:478.39Vesamicol
CAS:Vesamicol is an experimental drug. It acting presynaptically by inhibiting acetylcholine uptake into synaptic vesicles and reducing its release.Formula:C17H25NOPurity:98%Color and Shape:SolidMolecular weight:259.39Siltenzepine
CAS:Siltenzepine is an agent of anti-acid agent,and used in the treatment of peptic ulcers.Formula:C19H20ClN3O4Purity:98%Color and Shape:SolidMolecular weight:389.83Zamifenacin
CAS:Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.Formula:C27H29NO3Purity:98%Color and Shape:SolidMolecular weight:415.52ML381
CAS:ML381 is a M5-orthosteric antagonist with a high selectivity of muscarinic subtype.Formula:C21H21N3O4Color and Shape:SolidMolecular weight:379.41Neramexane Mesylate
CAS:Neramexane: NMDA & nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.Formula:C12H27NO3SPurity:98%Color and Shape:SolidMolecular weight:265.41BNC375
CAS:BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).Formula:C19H23ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:394.92
