AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 645 products of "AChR"
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TMPH
CAS:TMPH is an inhibitor of nAChR and inhibits nAChRs lacking α5, α6, or β3 subunits. TMPH can be used in studies about nAChR dysfunction or neurological disorders.Formula:C16H31NO2Purity:99.78%Color and Shape:SoildMolecular weight:269.42Ref: TM-T60080
2mg35.00€5mg55.00€10mg84.00€25mg133.00€50mg205.00€100mg301.00€200mg425.00€1mL*10mM (DMSO)54.00€Anabaseine
CAS:Anabaseine is a broad nicotinic agonist, favoring alpha-7 AChRs in muscle/brain, and weakly stimulates alpha-4 beta-2 nAChRs.Formula:C10H12N2Color and Shape:SolidMolecular weight:160.22Fesoterodine L-mandelate
CAS:Fesoterodine L-mandelate is a efficacious antimuscarinic agent for the overactive bladder (OAB).Formula:C34H45NO6Color and Shape:SolidMolecular weight:563.735(S)-(+)-Dimethindene maleate
CAS:(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptorsFormula:C24H28N2O4Purity:99.94%Color and Shape:SolidMolecular weight:408.49NKH477
CAS:NKH477 (Colforsin dapropate hydrochloride) is a derivative of forskolin with antidepressant activity.Formula:C27H44ClNO8Purity:98% - 98%Color and Shape:SolidMolecular weight:546.09Metixene hydrochloride hydrate
CAS:Metixene HCl hydrate is a potential anticholinergic for Parkinson's with IC50 of 55 nM and Ki of 15 nM against muscarine receptors.Formula:C20H26ClNOSPurity:99.99%Color and Shape:SolidMolecular weight:363.95Fipexide hydrochloride
CAS:Fipexide (hydrochloride) is a kind of psychoactive drug of the piperazine class.Formula:C20H22Cl2N2O4Color and Shape:SolidMolecular weight:425.31Tolterodine
CAS:Tolterodine ((R)-(+)-Tolterodine) is an mACh antagonist used in the treatment of detrusor instability and overactive bladder syndrome.Formula:C22H31NOPurity:99.71%Color and Shape:White Like Or Light Brown Crystalline PowderMolecular weight:325.49YM-58790 hydrochloride
CAS:YM-58790 is a potent M3 muscarinic receptor antagonist(Ki of 15 nM).Formula:C27H32ClN3O2Purity:98%Color and Shape:SolidMolecular weight:466.02Palmatine hydroxide
CAS:Palmatine hydroxide: oral IDO-1 inhibitor (IC50: 3-157μM), targets WNV protease, has anti-cancer/viral and neuroprotective properties.Formula:C21H23NO5Color and Shape:SolidMolecular weight:369.41β2AR/M-receptor agonist-2
CAS:β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).Formula:C36H49ClN4O7SColor and Shape:SolidMolecular weight:717.31ABT-107
CAS:ABT-107: α7 neuronal receptor agonist; protects rats' brains from 6-OHDA-induced damage.Formula:C19H20N4OColor and Shape:SolidMolecular weight:320.396NSC 23766
CAS:NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.Formula:C24H35N7Purity:99.49%Color and Shape:SolidMolecular weight:421.58Dexetimide
CAS:Dexetimide, a muscarinic receptor antagonist, treats neuroleptic-induced parkinsonism.Formula:C23H26N2O2Color and Shape:SolidMolecular weight:362.46Varenicline Hydrochloride
CAS:Varenicline Hydrochloride (CP 526555) is an orally active partial agonist of the α4β2 nicotinic acetylcholine receptor (α4β2 nAChR, IC50 = 250 nM).Formula:C13H14ClN3Purity:99.854%Color and Shape:SolidMolecular weight:247.72Ref: TM-T23502
1mg37.00€5mg77.00€10mg99.00€25mg182.00€50mg282.00€100mg419.00€200mg612.00€1mL*10mM (DMSO)83.00€Glycerophosphoinositol choline
CAS:Glycerophosphoinositol choline is the salt of choline and glycerophosphoinositol.Formula:C14H32NO12PColor and Shape:SolidMolecular weight:437.38Cevimeline hydrochloride
CAS:Cevimeline HCl is a muscarinic agonist enhancing salivary and sweat gland secretion.Formula:C10H18ClOSColor and Shape:SolidMolecular weight:235.77Dibucaine hydrochloride
CAS:Dibucaine hydrochloride (Cinchocaine hydrochloride), a long-acting local amide anestheticsis, is usually used for surface anesthesia.Formula:C20H30ClN3O2Purity:99.66%Color and Shape:White PowderMolecular weight:379.92Cevimeline
CAS:Cevimeline: muscarinic agonist, treats dry mouth & Sjögren's, boosts saliva post-cancer radiotherapy.Formula:C10H17NOSColor and Shape:Off-White SolidMolecular weight:199.31(±)-Darifenacin
CAS:(±)-Darifenacin is the racemate of Darifenacin. Darifenacin is a selective antagonist of M3 muscarinic receptor.Formula:C28H30N2O2Color and Shape:SolidMolecular weight:426.55
