AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Meseclazone
CAS:29053-27-8
Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP …
Formula:
C11H10ClNO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
239.65
Ref: TM-T16353
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Thonzylamine hydrochloride
CAS:63-56-9
Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.
Formula:
C16H23ClN4O
Purity:
99.84%
Color and Shape:
White Crystalline Powder
Molecular weight:
322.83
Ref: TM-T21014
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 273.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
GTS-21
CAS:148372-04-7
GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by …
Formula:
C19H20N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
308.37
Ref: TM-T19933
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
CP-810123
CAS:439608-12-5
CP-810123 is an α7 nAChR agonist used to treat cognitive deficits associated with psychiatric or …
Formula:
C14H18N4O
Purity:
98.63% - 99.23%
Color and Shape:
Solid
Molecular weight:
258.32
Ref: TM-T31079
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
TC-T 6000
CAS:949467-71-4
TC-T 6000 (hENT4-IN-1) is an ENT4 inhibitor with vasodilator activity that inhibits hENT1 and hENT2 …
Formula:
C26H48N8O2
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
504.71
Ref: TM-T34793
| 1mg | 73.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
PF-03635659
CAS:931409-24-4
PF-03635659: potent M3 antagonist, Ki=0.2 nM, long half-life, potential COPD treatment.
Formula:
C28H32N2O3
Purity:
98.05% - 99.83%
Color and Shape:
Solid
Molecular weight:
444.57
Ref: TM-T33941
| 1mg | 229.00 € | ||
| 5mg | 560.00 € | ||
| 10mg | 800.00 € | ||
| 25mg | 1,216.00 € | ||
| 50mg | 1,644.00 € | ||
| 100mg | 2,213.00 € | ||
| 500mg | 4,436.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Oxitropium Bromide
CAS:30286-75-0
Oxitropium bromide, a mAChR blocker, treats asthma and COPD as an anticholinergic bronchodilator.
Formula:
C19H26BrNO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
412.32
Ref: TM-T16417
| 25mg | 1,406.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Tarafenacin D-tartrate
CAS:1159101-48-0
Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold …
Formula:
C25H26F4N2O8
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
558.48
Ref: TM-T16989
| 2mg | 125.00 € | ||
| 5mg | 207.00 € | ||
| 25mg | 655.00 € | ||
| 50mg | 852.00 € | ||
| 100mg | 1,444.00 € | ||
| 1mL*10mM (DMSO) | 354.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
S16961
CAS:153874-14-7
S16961 (S169611) is an agonist of nicotinic receptor.
Formula:
C41H71NO6
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
674.01
Ref: TM-T12820
| 5mg | 50.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 137.00 € | ||
| 100mg | 188.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
SIB-1553A hydrochloride
CAS:191611-89-9
SIB-1553A hydrochloride is a nicotinic acetylcholine receptor agonist and a selective neuronal nAChR ligand
Formula:
C13H20ClNOS
Purity:
99.47% - 99.71%
Color and Shape:
Solid
Molecular weight:
273.82
Ref: TM-T16881
| 1mg | 92.00 € | ||
| 5mg | 224.00 € | ||
| 10mg | 359.00 € | ||
| 25mg | 595.00 € | ||
| 50mg | 838.00 € | ||
| 100mg | 1,130.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Afacifenacin
CAS:877606-63-8
Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.
Formula:
C27H26F3N3O2
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
481.51
Ref: TM-T29687
| 1mg | 333.00 € | ||
| 5mg | 787.00 € | ||
| 10mg | 1,074.00 € | ||
| 25mg | 1,510.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
GSK233705
CAS:850607-58-8
GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.
Formula:
C24H29BrN2
Purity:
99.67% - 99.76%
Color and Shape:
Solid
Molecular weight:
425.4
Ref: TM-T31207
| 1mg | 128.00 € | ||
| 5mg | 304.00 € | ||
| 10mg | 457.00 € | ||
| 25mg | 747.00 € | ||
| 50mg | 1,026.00 € | ||
| 100mg | 1,406.00 € | ||
| 500mg | 2,812.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
JNJ-39393406
CAS:953428-73-4
JNJ-39393406 is an α7 nicotinic acetylcholine receptor positive allosteric modulator for the study of tobacco …
Formula:
C19H18F2N6O3
Purity:
98.36%
Color and Shape:
Solid
Molecular weight:
416.38
Ref: TM-T27679
| 1mg | 96.00 € | ||
| 5mg | 200.00 € | ||
| 10mg | 303.00 € | ||
| 25mg | 490.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Phenserine
CAS:101246-66-6
Phenserine is a derivative of Physostigmine and is annoncompetitive, long-acting and selective inhibitor of AChE.
Formula:
C20H23N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
337.42
Ref: TM-T12446
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Iperoxo
CAS:247079-84-1
Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe …
Formula:
C10H17IN2O2
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
324.16
Ref: TM-T25538
| 1mg | 50.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 411.00 € | ||
| 50mg | 613.00 € | ||
| 100mg | 873.00 € | ||
| 500mg | 1,768.00 € | ||
| 1mL*10mM (DMSO) | 117.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Posatirelin
CAS:78664-73-0
Posatirelin, a synthetic peptide, modulates and nourishes brain systems, aiding in vascular dementia research.
Formula:
C17H28N4O4
Purity:
97.41% - 98.22%
Color and Shape:
Solid
Molecular weight:
352.43
Ref: TM-T34114
| 1mg | 128.00 € | ||
| 5mg | 304.00 € | ||
| 10mg | 457.00 € | ||
| 25mg | 747.00 € | ||
| 50mg | 1,026.00 € | ||
| 100mg | 1,406.00 € | ||
| 500mg | 2,812.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
CDD0102
CAS:146422-58-4
CDD0102 is a potent agonist of M1 Muscarinic receptor.
Formula:
C8H12N4O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
180.21
Ref: TM-T10731
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
SCH-900271
CAS:915210-50-3
SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.
Formula:
C14H16N2O4
Purity:
98.25% - 99%
Color and Shape:
Solid
Molecular weight:
276.29
Ref: TM-T34573
| 1mg | 118.00 € | ||
| 5mg | 275.00 € | ||
| 10mg | 419.00 € | ||
| 25mg | 692.00 € | ||
| 50mg | 938.00 € | ||
| 100mg | 1,320.00 € | ||
| 500mg | 2,632.00 € | ||
| 1mL*10mM (DMSO) | 263.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
UP202-56
CAS:163838-04-8
UP202-56 is an adenosinergic agonist and is an adenosine analog.
Formula:
C33H37N7O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
595.69
Ref: TM-T13256
| 25mg | 1,586.00 € | ||
| 50mg | 2,072.00 € | ||
| 100mg | 2,660.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
CB-7921220
CAS:115453-99-1
CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.
Formula:
C14H12N2O2
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
240.26
Ref: TM-T14880
| 2mg | 47.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 301.00 € | ||
| 50mg | 510.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
