AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Tribendimidine
CAS:115103-15-6
Tribendimidine: broad-spectrum oral anthelmintic, nAChR agonist, effective against A. lumbricoides and N. americanus.
Formula:
C28H32N6
Purity:
≥98%
Color and Shape:
Liquid
Molecular weight:
452.59
Ref: TM-T62769
| 5mg | 52.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 232.00 € | ||
| 100mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Xanomeline
CAS:131986-45-3
Xanomeline: orally active, M1/M4 selective activator for neurological disorders; promising in trials, crosses blood-brain barrier, …
Formula:
C14H23N3OS
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
281.42
Ref: TM-T36640
| 5mg | 54.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 162.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 454.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SCH 57790
CAS:221660-80-6
SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.
Formula:
C25H31N3O2S
Purity:
98.3% - 99.62%
Color and Shape:
Solid
Molecular weight:
437.6
Ref: TM-T28722
| 1mg | 240.00 € | ||
| 5mg | 596.00 € | ||
| 10mg | 848.00 € | ||
| 25mg | 1,272.00 € | ||
| 50mg | 1,717.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
ASM-024
CAS:1609534-88-4
ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment …
Formula:
C15H25N2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
233.37
Ref: TM-T26666
| 1mg | 240.00 € | ||
| 5mg | 597.00 € | ||
| 10mg | 852.00 € | ||
| 25mg | 1,273.00 € | ||
| 50mg | 1,719.00 € | ||
| 100mg | 2,331.00 € | ||
| 500mg | 4,564.00 € | ||
| 1mL*10mM (DMSO) | 503.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Xanomeline oxalate
CAS:141064-23-5
Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.
Formula:
C16H25N3O5S
Purity:
98.22%
Color and Shape:
Solid
Molecular weight:
371.45
Ref: TM-T13353
| 5mg | 37.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 249.00 € | ||
| 200mg | 359.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SIB-1553A hydrochloride
CAS:191611-89-9
SIB-1553A hydrochloride is a nicotinic acetylcholine receptor agonist and a selective neuronal nAChR ligand
Formula:
C13H20ClNOS
Purity:
99.47% - 99.71%
Color and Shape:
Solid
Molecular weight:
273.82
Ref: TM-T16881
| 1mg | 91.00 € | ||
| 5mg | 221.00 € | ||
| 10mg | 355.00 € | ||
| 25mg | 587.00 € | ||
| 50mg | 828.00 € | ||
| 100mg | 1,115.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Aceclidine
CAS:827-61-2
Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies …
Formula:
C9H15NO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
169.22
Ref: TM-T19870
| 1g | 166.00 € | ||
| 50mg | 41.00 € | ||
| 100mg | 51.00 € | ||
| 500mg | 112.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
PF-03635659
CAS:931409-24-4
PF-03635659: potent M3 antagonist, Ki=0.2 nM, long half-life, potential COPD treatment.
Formula:
C28H32N2O3
Purity:
98.05% - 99.83%
Color and Shape:
Solid
Molecular weight:
444.57
Ref: TM-T33941
| 1mg | 224.00 € | ||
| 5mg | 548.00 € | ||
| 10mg | 786.00 € | ||
| 25mg | 1,194.00 € | ||
| 50mg | 1,606.00 € | ||
| 100mg | 2,164.00 € | ||
| 500mg | 4,350.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
S16961
CAS:153874-14-7
S16961 (S169611) is an agonist of nicotinic receptor.
Formula:
C41H71NO6
Purity:
98.43%
Color and Shape:
Solid
Molecular weight:
674.01
Ref: TM-T12820
| 5mg | 50.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 134.00 € | ||
| 100mg | 184.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Afacifenacin
CAS:877606-63-8
Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.
Formula:
C27H26F3N3O2
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
481.51
Ref: TM-T29687
| 1mg | 326.00 € | ||
| 5mg | 772.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,322.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
GSK233705
CAS:850607-58-8
GSK233705, a muscarinic antagonist, is used to prevent/treat COPD and asthma.
Formula:
C24H29BrN2
Purity:
99.67% - 99.76%
Color and Shape:
Solid
Molecular weight:
425.4
Ref: TM-T31207
| 1mg | 125.00 € | ||
| 5mg | 298.00 € | ||
| 10mg | 446.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,374.00 € | ||
| 500mg | 2,765.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
TC-T 6000
CAS:949467-71-4
TC-T 6000 (hENT4-IN-1) is an ENT4 inhibitor with vasodilator activity that inhibits hENT1 and hENT2 …
Formula:
C26H48N8O2
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
504.71
Ref: TM-T34793
| 1mg | 72.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Iperoxo
CAS:247079-84-1
Iperoxo (Iperoxo iodide) is an agonist of Muscarinic AChR and can be used to probe …
Formula:
C10H17IN2O2
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
324.16
Ref: TM-T25538
| 1mg | 50.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 402.00 € | ||
| 50mg | 604.00 € | ||
| 100mg | 854.00 € | ||
| 500mg | 1,738.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Sulfoxaflor
CAS:946578-00-3
Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. …
Formula:
C10H10F3N3OS
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
277.27
Ref: TM-T19940
| 1mg | 109.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 444.00 € | ||
| 25mg | 712.00 € | ||
| 50mg | 974.00 € | ||
| 100mg | 1,289.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
UP202-56
CAS:163838-04-8
UP202-56 is an adenosinergic agonist and is an adenosine analog.
Formula:
C33H37N7O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
595.69
Ref: TM-T13256
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
CB-7921220
CAS:115453-99-1
CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.
Formula:
C14H12N2O2
Purity:
99.57%
Color and Shape:
Solid
Molecular weight:
240.26
Ref: TM-T14880
| 2mg | 46.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 295.00 € | ||
| 50mg | 501.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Cimetropium Bromide
CAS:51598-60-8
Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.
Formula:
C21H28BrNO4
Color and Shape:
Solid
Molecular weight:
438.36
Ref: TM-T14966
| 2mg | 134.00 € | ||
| 25mg | 711.00 € | ||
| 50mg | 933.00 € | ||
| 100mg | 1,442.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
mAChr-in-1
CAS:119391-56-9
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
Formula:
C23H25IN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
488.36
Ref: TM-T5476
| 25mg | 678.00 € | ||
| 1mL*10mM (DMSO) | 211.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
4-DAMP
CAS:1952-15-4
4-DAMP (4-DAMP methiodide) is a selective muscarinic M1 and M3 subtype receptor antagonist used in …
Formula:
C21H26INO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
451.34
Ref: TM-T22511
| 2mg | 49.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
hBChE-IN-2
CAS:2923366-36-1
hBChE-IN-2 is a BChE inhibitor and CB2R agonist with neuroprotective activity for the study of …
Formula:
C27H36N4O3
Purity:
99.69% - 99.86%
Color and Shape:
Soild
Molecular weight:
464.6
Ref: TM-T77509
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 646.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,390.00 € | ||
| 100mg | 1,837.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
