AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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UB 165 fumarate
CAS:2454492-43-2
UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM …
Formula:
C17H19ClN2O4
Purity:
98.91%
Color and Shape:
Solid
Molecular weight:
350.8
Ref: TM-T13241
| 1mg | 333.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
YM-58790
CAS:168830-70-4
YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM …
Formula:
C27H31N3O2
Purity:
99%
Color and Shape:
Soild
Molecular weight:
429.55
Ref: TM-T72038
| 1mg | 144.00 € | ||
| 5mg | 306.00 € | ||
| 10mg | 490.00 € | ||
| 25mg | 940.00 € | ||
| 50mg | 1,596.00 € | ||
| 100mg | 2,563.00 € | ||
| 500mg | 3,591.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Metixene hydrochloride
CAS:1553-34-0
Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
Formula:
C20H24ClNS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.93
Ref: TM-T12020
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Sch412348
CAS:377727-26-9
Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.
Formula:
C22H21F2N9O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
465.46
Ref: TM-T12868
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Desformylflustrabromine hydrochloride
CAS:951322-11-5
Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 …
Formula:
C17H12INO5
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
437.19
Ref: TM-T11004
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 236.00 € | ||
| 100mg | 373.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Cimetropium Bromide
CAS:51598-60-8
Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.
Formula:
C21H28BrNO4
Color and Shape:
Solid
Molecular weight:
438.36
Ref: TM-T14966
| 2mg | 138.00 € | ||
| 25mg | 727.00 € | ||
| 50mg | 947.00 € | ||
| 100mg | 1,464.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
PHA 543613
CAS:478149-53-0
PHA 543613 is a specific agonist of α7 nAChR (Ki = 8.8 nM) and can …
Formula:
C15H17N3O2
Purity:
99% - 99.48%
Color and Shape:
Solid
Molecular weight:
271.31
Ref: TM-T23145
| 1mg | 50.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 945.00 € | ||
| 500mg | 2,052.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Propoxur
CAS:114-26-1
Propoxur: an insecticide causing temporary cholinergic effects in humans; chronic exposure leads to health issues; …
Formula:
C11H15NO3
Purity:
98.15% - 99.87%
Color and Shape:
Minute Crystals (Niosh 2016)
Molecular weight:
209.24
Ref: TM-T0976
| 1g | 94.00 € | ||
| 100mg | 34.00 € | ||
| 200mg | 47.00 € | ||
| 500mg | 71.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Darenzepine
CAS:84629-61-8
Darenzepine is a muscarinic receptor inhibitor.
Formula:
C21H21N3O2
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
347.41
Ref: TM-T10961
| 1mg | 215.00 € | ||
| 5mg | 426.00 € | ||
| 10mg | 598.00 € | ||
| 25mg | 889.00 € | ||
| 50mg | 1,188.00 € | ||
| 100mg | 1,605.00 € | ||
| 1mL*10mM (DMSO) | 472.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
PQCA
CAS:1144504-35-7
PQCA is a selective M1 receptor modulator with EC50s of 49 nM (monkey) and 135 …
Formula:
C22H20N4O3
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
388.42
Ref: TM-T12531
| 1mg | 51.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 192.00 € | ||
| 25mg | 304.00 € | ||
| 50mg | 420.00 € | ||
| 100mg | 560.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
hBChE-IN-2
CAS:2923366-36-1
hBChE-IN-2 is a BChE inhibitor and CB2R agonist with neuroprotective activity for the study of …
Formula:
C27H36N4O3
Purity:
99.69% - 99.86%
Color and Shape:
Soild
Molecular weight:
464.6
Ref: TM-T77509
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 1,872.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
3-Bromocytisine
CAS:207390-14-5
3-Bromocytisine ((-)-3-Bromocytisine) is an effective agonist of nAChR (IC50s: 0.28, 0.30 and 31.6 nM for …
Formula:
C11H13BrN2O
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
269.14
Ref: TM-T10108
| 1mg | 95.00 € | ||
| 5mg | 227.00 € | ||
| 10mg | 309.00 € | ||
| 25mg | 520.00 € | ||
| 50mg | 748.00 € | ||
| 100mg | 1,026.00 € | ||
| 1mL*10mM (DMSO) | 208.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
Timepidium bromide
CAS:35035-05-3
Timepidium bromide is an agent of anticholinergic.
Formula:
C17H22BrNOS2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
400.4
Ref: TM-T12825
| 25mg | 1,730.00 € | ||
| 50mg | 2,262.00 € | ||
| 100mg | 2,945.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
TZ3O
CAS:2218754-19-7
TZ3O is an anticholinergic compound with neuroprotective activity.TZ3O ameliorates memory impairment in Scopolamine-induced Alzheimer's type …
Formula:
C18H13NO4S
Purity:
99.84%
Color and Shape:
Liquid
Molecular weight:
339.37
Ref: TM-T77678
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 1,872.00 € | ||
| 500mg | 3,734.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
LY2033298
CAS:886047-13-8
LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.
Formula:
C13H14ClN3O2S
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
311.79
Ref: TM-T27931
| 1mg | 87.00 € | ||
| 5mg | 205.00 € | ||
| 10mg | 350.00 € | ||
| 25mg | 747.00 € | ||
| 50mg | 1,008.00 € | ||
| 100mg | 1,359.00 € | ||
| 200mg | 1,833.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
Tiotropium Bromide hydrate
CAS:411207-31-3
Tiotropium Bromide hydrate is a potent, long-lasting anticholinergic bronchodilator for COPD, with high affinity for …
Formula:
C19H24BrNO5S2
Purity:
98.44% - 99.41%
Color and Shape:
Solid
Molecular weight:
490.43
Ref: TM-T6707
| 25mg | 44.00 € | ||
| 50mg | 58.00 € | ||
| 100mg | 92.00 € | ||
| 200mg | 135.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
Tematropium
CAS:113932-41-5
Tematropium (CDDD3602) possesses anticholinergic effects and can be used in neurological studies.
Formula:
C21H31NO8S
Purity:
98.87%
Color and Shape:
Solid
Molecular weight:
457.54
Ref: TM-T10732
| 1mg | 212.00 € | ||
| 2mg | 284.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 615.00 € | ||
| 25mg | 929.00 € | ||
| 50mg | 1,244.00 € | ||
| 100mg | 1,691.00 € | ||
| 1mL*10mM (DMSO) | 507.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
ICL-CCIC-0019
CAS:936498-64-5
ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.
Formula:
C26H44Br2N4
Purity:
97.62%
Color and Shape:
Solid
Molecular weight:
572.46
Ref: TM-T27579
| 1mg | 185.00 € | ||
| 5mg | 415.00 € | ||
| 10mg | 613.00 € | ||
| 25mg | 938.00 € | ||
| 50mg | 1,311.00 € | ||
| 100mg | 1,768.00 € | ||
| 500mg | 3,535.00 € | ||
| 1mL*10mM (DMSO) | 545.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
VU 0255035
CAS:1135243-19-4
VU 0255035 is a highly selective, competitive and brain penetrant muscarinic M1 receptor antagonist with …
Formula:
C18H20N6O3S2
Purity:
96.53% - 98.26%
Color and Shape:
Solid
Molecular weight:
432.52
Ref: TM-T23508
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 533.00 € | ||
| 200mg | 743.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
Zamifenacin fumarate
CAS:127308-98-9
Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.
Formula:
C31H33NO7
Purity:
99.78%
Color and Shape:
Solid
Molecular weight:
531.6
Ref: TM-T13385
| 1mg | 40.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 533.00 € | ||
| 200mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Friday 11 Jul 2025
