AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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CHF5407
CAS:1004312-94-0
CHF5407(SVT-47060) is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic …
Formula:
C27H25BrF4N2O3S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
613.46
Ref: TM-T13992
| 1mg | 145.00 € | ||
| 5mg | 296.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
GP531
CAS:142344-87-4
GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.
Formula:
C16H21N5O4
Color and Shape:
Solid
Molecular weight:
347.37
Ref: TM-T13713
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
YM-46303
CAS:171722-81-9
YM-46303 is a selective and potent muscarinic receptor antagonist that exhibits high affinity for the …
Formula:
C20H23ClN2O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
358.86
Ref: TM-T13370
| 1mg | 665.00 € | ||
| 5mg | 1,710.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
mAChr-in-1
CAS:119391-56-9
mAChR-IN-1 is muscarinic cholinergic receptor(mAChR) antagonist (IC50=17 nM).
Formula:
C23H25IN2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
488.36
Ref: TM-T5476
| 25mg | 693.00 € | ||
| 1mL*10mM (DMSO) | 212.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Terodiline hydrochloride
CAS:7082-21-5
Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and …
Formula:
C20H28ClN
Purity:
98%
Color and Shape:
Solid
Molecular weight:
317.9
Ref: TM-T13129
| 25mg | 1,159.00 € | ||
| 50mg | 1,510.00 € | ||
| 100mg | 2,308.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Pozanicline
CAS:161417-03-4
Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing …
Formula:
C11H16N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
192.26
Ref: TM-T16563
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Sulfoxaflor
CAS:946578-00-3
Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. …
Formula:
C10H10F3N3OS
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
277.27
Ref: TM-T19940
| 1mg | 111.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 455.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 998.00 € | ||
| 100mg | 1,320.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
AF-DX 384 free base
CAS:118290-26-9
AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research …
Formula:
C27H38N6O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
478.63
Ref: TM-T22555
| 1mg | 128.00 € | ||
| 5mg | To inquire | ||
| 10mg | To inquire | ||
| 25mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Pentolinium Tartrate
CAS:52-62-0
Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking …
Formula:
C15H32N2·2C4H5O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
538.6
Ref: TM-T1236
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
(Rac)-VU 6008667
CAS:2092917-63-8
(Rac)-VU 6008667 is a selective M5 NAM with IC50 of 1.8 μM, high CNS penetration.
Formula:
C24H17ClF2N2O2
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
438.85
Ref: TM-T12679
| 1mg | 38.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 385.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
AQW051
CAS:669770-29-0
AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.
Formula:
C19H22N2O
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
294.39
Ref: TM-T26646
| 1mg | 35.00 € | ||
| 2mg | 48.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 464.00 € | ||
| 500mg | 1,008.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Oxotremorine M iodide
CAS:3854-04-4
Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.
Formula:
C11H19IN2O
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
322.19
Ref: TM-T12339
| 10mg | 50.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
ASM-024
CAS:1609534-88-4
ASM-024, a synthetic piperazine, activates nicotinic and β2-adrenergic receptors for potential asthma and bronchitis treatment …
Formula:
C15H25N2
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
233.37
Ref: TM-T26666
| 1mg | 245.00 € | ||
| 5mg | 610.00 € | ||
| 10mg | 868.00 € | ||
| 25mg | 1,301.00 € | ||
| 50mg | 1,758.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | 4,655.00 € | ||
| 1mL*10mM (DMSO) | 507.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
GAT107
CAS:1476807-74-5
GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.
Formula:
C18H17BrN2O2S
Purity:
98.76%
Color and Shape:
Solid
Molecular weight:
405.31
Ref: TM-T27404
| 1mg | 245.00 € | ||
| 5mg | 610.00 € | ||
| 10mg | 868.00 € | ||
| 25mg | 1,301.00 € | ||
| 50mg | 1,758.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | 4,655.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
N-0861 racemate
CAS:121241-87-0
N-0861 racemate is the racemate of N-0861.
Formula:
C13H17N5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
243.31
Ref: TM-T12136
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Xanomeline oxalate
CAS:141064-23-5
Xanomeline oxalate (LY246708), a potent SMRA, boosts phosphoinositide hydrolysis; key for Alzheimer's research.
Formula:
C16H25N3O5S
Purity:
98.22%
Color and Shape:
Solid
Molecular weight:
371.45
Ref: TM-T13353
| 5mg | 38.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 168.00 € | ||
| 100mg | 259.00 € | ||
| 200mg | 373.00 € | ||
| 1mL*10mM (DMSO) | 42.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
9-CP-Ade Mesylate
CAS:189639-09-6
9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate …
Formula:
C11H17N5O3S
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
299.35
Ref: TM-T23588
| 1mg | 66.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 216.00 € | ||
| 25mg | 399.00 € | ||
| 50mg | 588.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Aceclidine
CAS:827-61-2
Aceclidine (1-azabicyclo[2.2.2]octan-3-yl acetate) is a modulator of M3 mAChR and can be used in studies …
Formula:
C9H15NO2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
169.22
Ref: TM-T19870
| 1g | 172.00 € | ||
| 50mg | 42.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 116.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
MHP 133
CAS:147340-43-0
MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).
Formula:
C17H20ClN5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
377.83
Ref: TM-T13772
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
SCH 57790
CAS:221660-80-6
SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.
Formula:
C25H31N3O2S
Purity:
98.3% - 99.62%
Color and Shape:
Solid
Molecular weight:
437.6
Ref: TM-T28722
| 1mg | 245.00 € | ||
| 5mg | 610.00 € | ||
| 10mg | 868.00 € | ||
| 25mg | 1,301.00 € | ||
| 50mg | 1,758.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
