AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Read more
Asoxime dichloride
CAS:34433-31-3
Asoxime dichloride (HI-6) blocks AChRs, including α7 nAChR, and boosts vaccination in the nervous system.
Formula:
C14H16Cl2N4O3
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
359.21
Ref: TM-T14333
| 5mg | 57.00 € | ||
| 10mg | 91.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Meseclazone
CAS:29053-27-8
Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP …
Formula:
C11H10ClNO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
239.65
Ref: TM-T16353
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
AQW051
CAS:669770-29-0
AQW051 (VQW-765) is an oral α7-nAChR activator for cognitive impairments, used in anxiety disorder studies.
Formula:
C19H22N2O
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
294.39
Ref: TM-T26646
| 1mg | 36.00 € | ||
| 2mg | 48.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 461.00 € | ||
| 500mg | 1,000.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Pentolinium Tartrate
CAS:52-62-0
Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking …
Formula:
C15H32N2·2C4H5O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
538.6
Ref: TM-T1236
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Pozanicline
CAS:161417-03-4
Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing …
Formula:
C11H16N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
192.26
Ref: TM-T16563
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Terodiline hydrochloride
CAS:7082-21-5
Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and …
Formula:
C20H28ClN
Purity:
98%
Color and Shape:
Solid
Molecular weight:
317.9
Ref: TM-T13129
| 25mg | 1,132.00 € | ||
| 50mg | 1,476.00 € | ||
| 100mg | 2,270.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
GTS-21
CAS:148372-04-7
GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by …
Formula:
C19H20N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
308.37
Ref: TM-T19933
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
YM-46303
CAS:171722-81-9
YM-46303 is a selective and potent muscarinic receptor antagonist that exhibits high affinity for the …
Formula:
C20H23ClN2O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
358.86
Ref: TM-T13370
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
CHF5407
CAS:1004312-94-0
CHF5407(SVT-47060) is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic …
Formula:
C27H25BrF4N2O3S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
613.46
Ref: TM-T13992
| 1mg | 650.00 € | ||
| 5mg | 1,678.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Desformylflustrabromine hydrochloride
CAS:951322-11-5
Desformylflustrabromine hydrochloride (dFBr hydrochloride) is a selective agonist of nicotinic acetylcholine receptor (nAChR) in α4β2 …
Formula:
C17H12INO5
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
437.19
Ref: TM-T11004
| 2mg | 36.00 € | ||
| 5mg | 53.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 370.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
YM-58790
CAS:168830-70-4
YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM …
Formula:
C27H31N3O2
Purity:
99%
Color and Shape:
Soild
Molecular weight:
429.55
Ref: TM-T72038
| 1mg | 142.00 € | ||
| 5mg | 300.00 € | ||
| 10mg | 480.00 € | ||
| 25mg | 919.00 € | ||
| 50mg | 1,560.00 € | ||
| 100mg | 2,505.00 € | ||
| 500mg | 3,508.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Metixene hydrochloride
CAS:1553-34-0
Metixene hydrochloride is an anticholinergic antiparkinsonian agent.
Formula:
C20H24ClNS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.93
Ref: TM-T12020
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Oxitropium Bromide
CAS:30286-75-0
Oxitropium bromide, a mAChR blocker, treats asthma and COPD as an anticholinergic bronchodilator.
Formula:
C19H26BrNO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
412.32
Ref: TM-T16417
| 25mg | 1,406.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Tarafenacin D-tartrate
CAS:1159101-48-0
Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold …
Formula:
C25H26F4N2O8
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
558.48
Ref: TM-T16989
| 2mg | 122.00 € | ||
| 5mg | 204.00 € | ||
| 25mg | 640.00 € | ||
| 50mg | 859.00 € | ||
| 100mg | 1,405.00 € | ||
| 1mL*10mM (DMSO) | 352.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
GAT107
CAS:1476807-74-5
GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.
Formula:
C18H17BrN2O2S
Purity:
98.76%
Color and Shape:
Solid
Molecular weight:
405.31
Ref: TM-T27404
| 1mg | 240.00 € | ||
| 5mg | 596.00 € | ||
| 10mg | 852.00 € | ||
| 25mg | 1,272.00 € | ||
| 50mg | 1,717.00 € | ||
| 100mg | 2,336.00 € | ||
| 500mg | 4,568.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
SCH-900271
CAS:915210-50-3
SCH-900271 treats dyslipidemia by targeting nicotinic acid receptors, addressing hyperlipidaemia.
Formula:
C14H16N2O4
Purity:
98.25% - 99%
Color and Shape:
Solid
Molecular weight:
276.29
Ref: TM-T34573
| 1mg | 116.00 € | ||
| 5mg | 271.00 € | ||
| 10mg | 409.00 € | ||
| 25mg | 677.00 € | ||
| 50mg | 920.00 € | ||
| 100mg | 1,296.00 € | ||
| 500mg | 2,582.00 € | ||
| 1mL*10mM (DMSO) | 261.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
S 24795
CAS:304679-75-2
S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.
Formula:
C14H13BrINO
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
418.07
Ref: TM-T23286
| 1mg | 35.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 368.00 € | ||
| 100mg | 580.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Oxotremorine M iodide
CAS:3854-04-4
Oxotremorine M iodide (Oxotremorine methiodide) is an agonist of mAChR and potentiates NMDA receptors.
Formula:
C11H19IN2O
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
322.19
Ref: TM-T12339
| 10mg | 50.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Sch412348
CAS:377727-26-9
Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.
Formula:
C22H21F2N9O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
465.46
Ref: TM-T12868
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
McN-A 343
CAS:55-45-8
McN-A 343: Selective M1 muscarinic agonist; reduces inflammation in colitis models.
Formula:
C14H18Cl2N2O2
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
317.21
Ref: TM-T22963
| 25mg | 53.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 21 Jan 2025
