CymitQuimica logo
AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 574 products of "AChR"

Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Carbetapentane citrate
    Targetmol
    + Info

    Carbetapentane citrate

    CAS:
    <p>Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.</p>
    Formula:C20H31NO3·C6H8O7
    Purity:99.46%
    Color and Shape:White To Off-White Solid
    Molecular weight:525.59

    Ref: TM-T0464

  • Carbachol
    Targetmol
    + Info

    Carbachol

    CAS:
    <p>Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.</p>
    Formula:C6H15ClN2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:182.65

    Ref: TM-T0105

  • TAK-071
    Targetmol
    + Info

    TAK-071

    CAS:
    <p>TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).</p>
    Formula:C24H24FN3O3
    Purity:98.02%
    Color and Shape:Solid
    Molecular weight:421.46

    Ref: TM-T13066

  • Acetamiprid
    Targetmol
    + Info

    Acetamiprid

    CAS:
    <p>Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.</p>
    Formula:C10H11ClN4
    Purity:99.66%
    Color and Shape:White Powder
    Molecular weight:222.67

    Ref: TM-T14094

  • Rocuronium bromide
    Targetmol
    + Info

    Rocuronium bromide

    CAS:
    <p>Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.</p>
    Formula:C32H53BrN2O4
    Purity:99.77% - >99.99%
    Color and Shape:White Or Off-White Powder
    Molecular weight:609.68

    Ref: TM-T0156

  • Ipratropium bromide monohydrate
    Targetmol
    + Info

    Ipratropium bromide monohydrate

    CAS:
    <p>Ipratropium bromide, safer than atropine, treats bronchial disorders, rhinitis, and irregular heartbeat via inhalation.</p>
    Formula:C20H32BrNO4
    Purity:97.85%
    Color and Shape:Solid
    Molecular weight:430.38

    Ref: TM-T0098

  • Benzethonium chloride
    Targetmol
    + Info

    Benzethonium chloride

    CAS:
    <p>Benzethonium chloride (Quatrachlor) is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties.</p>
    Formula:C27H42ClNO2
    Purity:99.91%
    Color and Shape:White To Off-White Solid Solid Particulate/Powder
    Molecular weight:448.09

    Ref: TM-T0401

  • Navafenterol
    Targetmol
    + Info

    Navafenterol

    CAS:
    <p>AZD-8871, a potential COPD and asthma treatment, may work well with ICS.</p>
    Formula:C38H42N6O6S2
    Color and Shape:Solid
    Molecular weight:742.91

    Ref: TM-T30264

  • α-Conotoxin imi
    Targetmol
    + Info

    α-Conotoxin imi

    CAS:
    <p>alpha-Conotoxin imi is a nicotinic acetylcholine receptor ligand.</p>
    Formula:C52H78N20O15S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1351.56

    Ref: TM-T23707

  • M 8218
    Targetmol
    + Info

    M 8218

    CAS:
    <p>M 8218 is a bioactive chemical.</p>
    Formula:C20H29NO2
    Color and Shape:Solid
    Molecular weight:315.45

    Ref: TM-T33111

  • α-Conotoxin PIA
    Targetmol
    + Info

    α-Conotoxin PIA

    CAS:
    <p>Selective antagonist of α6-containing nicotinic receptors that discriminates between the closely related α6 and α3 subunits (IC50 values are 0.95 and 74.2 nM</p>
    Formula:C79H125N27O25S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1981.3

    Ref: TM-TP2065

  • Methylatropine (nitrate)
    Targetmol
    + Info

    Methylatropine (nitrate)

    CAS:
    <p>Methylatropine: Muscarinic antagonist, &lt;0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.</p>
    Formula:C18H26N2O6
    Color and Shape:Solid
    Molecular weight:366.414

    Ref: TM-T36204

  • Anabaseine
    Targetmol
    + Info

    Anabaseine

    CAS:
    <p>Anabaseine is a broad nicotinic agonist, favoring alpha-7 AChRs in muscle/brain, and weakly stimulates alpha-4 beta-2 nAChRs.</p>
    Formula:C10H12N2
    Color and Shape:Solid
    Molecular weight:160.22

    Ref: TM-T40431

  • N-Ethyl-N-(3-pyridylmethyl)amine
    Targetmol
    + Info

    N-Ethyl-N-(3-pyridylmethyl)amine

    CAS:
    <p>N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.</p>
    Formula:C8H12N2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:136.19

    Ref: TM-TN9660

  • Albanin A
    Targetmol
    + Info

    Albanin A

    <p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>
    Formula:C20H18O6
    Color and Shape:Solid
    Molecular weight:354.358

    Ref: TM-T124310

  • Doxacurium Chloride
    Targetmol
    + Info

    Doxacurium Chloride

    CAS:
    <p>Doxacurium Chloride is a muscarinic acetylcholine receptor M2 antagonist.</p>
    Formula:C56H78ClN2O16
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1070.69

    Ref: TM-T27199

  • α-Conotoxin EI
    Targetmol
    + Info

    α-Conotoxin EI

    CAS:
    <p>Selective antagonist of neuromuscular nicotinic receptors α1β1γδ</p>
    Formula:C83H125N27O27S5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2093.37

    Ref: TM-TP2218

  • Perindoprilat
    Targetmol
    + Info

    Perindoprilat

    CAS:
    <p>Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.</p>
    Formula:C17H28N2O5
    Purity:99.48%
    Color and Shape:Solid
    Molecular weight:340.41

    Ref: TM-T1484

  • β2AR/M-receptor agonist-1
    Targetmol
    + Info

    β2AR/M-receptor agonist-1

    CAS:
    <p>β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor and</p>
    Formula:C43H56BrN3O7
    Color and Shape:Solid
    Molecular weight:806.82

    Ref: TM-T74708

  • Br-PBTC
    Targetmol
    + Info

    Br-PBTC

    CAS:
    <p>Br-PBTC modulates nAChRs; targets α2/β2,4 subtypes; potent with 0.1-0.6 μM EC50; binds α subunit c-tail.</p>
    Formula:C14H15BrN2OS
    Color and Shape:Solid
    Molecular weight:339.25

    Ref: TM-T39286