AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
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Glycopyrrolate
CAS:596-51-0
Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.
Formula:
C19H28BrNO3
Purity:
99.41% - 99.64%
Color and Shape:
Solid
Molecular weight:
398.33
Ref: TM-T2387
| 5mg | 38.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 64.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 128.00 € | ||
| 500mg | 303.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
CCMI
CAS:917837-54-8
CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.
Formula:
C19H15Cl2N3O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
388.25
Ref: TM-T7422
| 2mg | 39.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
W-84 dibromide
CAS:21093-51-6
W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.
Formula:
C32H44Br2N4O4
Purity:
95.56%
Color and Shape:
Solid
Molecular weight:
708.52
Ref: TM-T23524
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 245.00 € | ||
| 100mg | 364.00 € | ||
| 200mg | 517.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Nor-benzetimide
CAS:19315-71-0
Norbenzetimide, an organic compound, is prepared from benzetimide by catalytic transfer hydrogenolysis.
Formula:
C16H20N2O2
Purity:
98.63%
Color and Shape:
Solid
Molecular weight:
272.34
Ref: TM-T22380
| 1mg | 93.00 € | ||
| 2mg | 126.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 283.00 € | ||
| 25mg | 462.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 867.00 € | ||
| 200mg | 1,159.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
VU0152099
CAS:612514-42-8
VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).
Formula:
C18H17N3O3S
Purity:
98.46%
Color and Shape:
Solid
Molecular weight:
355.41
Ref: TM-T29123
| 5mg | 34.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 255.00 € | ||
| 200mg | 366.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
NS9283
CAS:913830-15-6
NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.
Formula:
C14H8N4O
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
248.24
Ref: TM-T28199
| 1mg | 46.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 298.00 € | ||
| 50mg | 469.00 € | ||
| 100mg | 687.00 € | ||
| 500mg | 1,444.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
TBPB
CAS:634616-95-8
TBPB is an allosteric M1 mAChR agonist.
Formula:
C25H32N4O
Purity:
97.87% - 99.9%
Color and Shape:
Solid
Molecular weight:
404.55
Ref: TM-T1760
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 116.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 350.00 € | ||
| 200mg | 522.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
9-Ethyladenine
CAS:2715-68-6
9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].
Formula:
C7H9N5
Purity:
99.35% - 99.41%
Color and Shape:
Solid
Molecular weight:
163.18
Ref: TM-T14065
| 50mg | 39.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 116.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Donepezil Hydrochloride
CAS:120011-70-3
Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 …
Formula:
C24H29NO3·HCl
Purity:
99.55% - 99.8%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
415.96
Ref: TM-T6478
| 25mg | 52.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 127.00 € | ||
| 500mg | 205.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
VU0467154
CAS:1451993-15-9
VU0467154 is a positive allosteric modulator of the M4 muscarinic acetylcholine receptor.
Formula:
C17H15F3N4O3S2
Purity:
98.05% - 98.28%
Color and Shape:
Solid
Molecular weight:
444.45
Ref: TM-T17244
| 2mg | 88.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 284.00 € | ||
| 50mg | 484.00 € | ||
| 100mg | 845.00 € | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Succinylcholine Chloride Dihydrate
CAS:6101-15-1
Succinylcholine Chloride Dihydrate (Succinyldicholine dichloride) is a nicotinic AChR agonist and also acts as a …
Formula:
C14H30N2O4·2Cl·2H2O
Purity:
99.87%
Color and Shape:
White Solid
Molecular weight:
397.34
Ref: TM-T6684
| 1g | 507.00 € | ||
| 10mg | 39.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 71.00 € | ||
| 100mg | 116.00 € | ||
| 200mg | 202.00 € | ||
| 500mg | 341.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Tacrine hydrochloride (hydrate)
CAS:206658-92-6
Tacrine hydrochloride hydrate (Tetrahydroaminacrine) is a cholinesterase inhibitor that crosses the blood-brain barrier.
Formula:
C13H14N2·XHCl·XH2O
Purity:
99.5% - 99.89%
Color and Shape:
Solid
Molecular weight:
234.72
Ref: TM-T2191
| 100mg | 51.00 € | ||
| 200mg | 74.00 € | ||
| 500mg | 107.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
NS3861
CAS:216853-59-7
NS3861 is a selective agonist for α3β4/α4β2 nAChRs, preferring β-subunits, with no effect on α4-based …
Formula:
C12H14BrNS
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
284.22
Ref: TM-T9542
| 5mg | 47.00 € | ||
| 10mg | 79.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 439.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Thiacloprid
CAS:111988-49-9
Thiacloprid: insecticide targeting insect nAChRs, IC50 - Drosophila: 2.7 nM, Mouse α4β2 nAChRs: 860 nM.
Formula:
C10H9ClN4S
Purity:
98.66%
Color and Shape:
Yellowish Crystalline Powder
Molecular weight:
252.72
Ref: TM-T38272
| 100mg | 44.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Isoxazole
CAS:288-14-2
Isoxazole (1,2-oxazole) is the inhibitor of acetylcholinesterase (AChE). The ligands of Isoxazole bind to and …
Formula:
C3H3NO
Purity:
99.34%
Color and Shape:
Colorless Liquid
Molecular weight:
69.06
Ref: TM-T7500
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Cyclopentolate Hydrochloride
CAS:5870-29-1
Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 …
Formula:
C17H26ClNO3
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
327.85
Ref: TM-T8383
| 10mg | 38.00 € | ||
| 25mg | 72.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 170.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
A-867744
CAS:1000279-69-5
A-867744 is an effective and selective type II positive allosteric modulator of the α7 nAChR …
Formula:
C20H19ClN2O3S
Purity:
95.66%
Color and Shape:
Solid
Molecular weight:
402.89
Ref: TM-TQ0117
| 2mg | 47.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 494.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Mivacurium dichloride
CAS:106861-44-3
Mivacurium dichloride: non-depolarizing, quick-acting muscle relaxant for minor surgeries and tracheal intubation.
Formula:
C58H80Cl2N2O14
Purity:
99.2% - 99.48%
Color and Shape:
Off-White Solid
Molecular weight:
1100.17
Ref: TM-T22371
| 2mg | 48.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 303.00 € | ||
| 200mg | 457.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
Fesoterodine
CAS:286930-02-7
Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.
Formula:
C26H37NO3
Purity:
96.27% - 97.1%
Color and Shape:
Solid
Molecular weight:
411.58
Ref: TM-T9419
| 5mg | 51.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 259.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
DMAB-anabaseine dihydrochloride
CAS:154149-38-9
DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containing
Formula:
C19H23Cl2N3
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
364.31
Ref: TM-T22735
| 1mg | 62.00 € | ||
| 2mg | 84.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 547.00 € | ||
| 200mg | 740.00 € |
Estimated delivery in United States, on Wednesday 7 May 2025
