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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 574 products of "AChR"

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  • ANQ-9040
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    ANQ-9040

    CAS:
    <p>ANQ-9040 is a nondepolarizing neuromuscular relaxant of the steroid class.</p>
    Formula:C36H58N2O5S
    Color and Shape:Solid
    Molecular weight:630.92

    Ref: TM-T30079

  • G-Protein antagonist peptide
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    G-Protein antagonist peptide

    CAS:
    <p>Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.</p>
    Formula:C57H64N12O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1093.27

    Ref: TM-TP1902

  • Bencycloquidium Bromide
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    Bencycloquidium Bromide

    CAS:
    <p>Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.</p>
    Formula:C21H32BrNO2
    Color and Shape:Solid
    Molecular weight:410.39

    Ref: TM-T26770

  • nAChR modulator-2
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    nAChR modulator-2

    CAS:
    <p>nAChR modulator-2, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>
    Formula:C12H8ClN3O2
    Color and Shape:Solid
    Molecular weight:261.66

    Ref: TM-T74397

  • trans-Cevimeline hydrochloride
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    trans-Cevimeline hydrochloride

    CAS:
    <p>AF 102A hydrochloride is a biochemical.</p>
    Formula:C10H18ClNOS
    Color and Shape:Solid
    Molecular weight:235.77

    Ref: TM-T29681

  • CymitQuimica logo
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    Irsogladine maleate

    CAS:
    <p>Compound PDK0375, with CAS No. 84504-69-8, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0375 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>
    Formula:C9H7Cl2N5
    Color and Shape:Solid
    Molecular weight:256.09

    Ref: TM-PDK0375

  • Octamylamine
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    Octamylamine

    CAS:
    <p>Octamylamine is a bioactive chemical.</p>
    Formula:C13H29N
    Color and Shape:Solid
    Molecular weight:199.3761

    Ref: TM-T33778

  • nAChR agonist 2
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    nAChR agonist 2

    CAS:
    <p>Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,</p>
    Formula:C11H16N2
    Color and Shape:Solid
    Molecular weight:176.263

    Ref: TM-T40177

  • Fentonium bromide
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    Fentonium bromide

    CAS:
    <p>Fentonium bromide is a biochemical.</p>
    Formula:C31H34BrNO4
    Color and Shape:Solid
    Molecular weight:564.51

    Ref: TM-T31781

  • Mant-GTPγS
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    Mant-GTPγS

    CAS:
    <p>Mant-GTPγS, an effective GTP analog, displays strong competitive inhibition of adenylyl cyclase (AC). Additionally, it acts as a potent inhibitor of YdeH.</p>
    Formula:C18H23N6O14P3S
    Color and Shape:Solid
    Molecular weight:672.39

    Ref: TM-T38782

  • M4 mAChR agonist-1 
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    M4 mAChR agonist-1 

    CAS:
    <p>M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 &gt;10 μM).</p>
    Formula:C14H18N4OS
    Purity:99.14%
    Color and Shape:Solid
    Molecular weight:290.38

    Ref: TM-T9889

  • α-Conotoxin EI
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    α-Conotoxin EI

    CAS:
    <p>Selective antagonist of neuromuscular nicotinic receptors α1β1γδ</p>
    Formula:C83H125N27O27S5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2093.37

    Ref: TM-TP2218

  • VU6028418
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    VU6028418

    CAS:
    <p>VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).</p>
    Color and Shape:Solid

    Ref: TM-T71675

  • 5-AMAM-2-CP
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    5-AMAM-2-CP

    CAS:
    <p>5-AMAM-2-CP, a significant metabolite of Acetamiprid, serves as a global insecticide within the neonicotinoid class and acts as an nAChR agonist [1] [2].</p>
    Formula:C9H11ClN2O
    Color and Shape:Solid
    Molecular weight:198.65

    Ref: TM-T74086

  • Anabaseine
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    Anabaseine

    CAS:
    <p>Anabaseine is a broad nicotinic agonist, favoring alpha-7 AChRs in muscle/brain, and weakly stimulates alpha-4 beta-2 nAChRs.</p>
    Formula:C10H12N2
    Color and Shape:Solid
    Molecular weight:160.22

    Ref: TM-T40431

  • Epiboxidine hydrochloride
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    Epiboxidine hydrochloride

    CAS:
    <p>Epiboxidine HCl: potent α4β2 nAChR agonist; Ki 0.46 nM (rat), 1.2 nM (human); Epibatidine analog.</p>
    Formula:C10H15ClN2O
    Color and Shape:Solid
    Molecular weight:214.69

    Ref: TM-T74131

  • Angiopeptin
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    Angiopeptin

    CAS:
    <p>Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.</p>
    Formula:C54H71N11O10S2
    Color and Shape:Solid
    Molecular weight:1098.34

    Ref: TM-T25087

  • PF-06827443
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    PF-06827443

    <p>PF-06827443 is a orally bioavailable, CNS-penetrant M1-selective PAM with minimal agonist activity.</p>
    Formula:C24H24N2O4
    Color and Shape:Solid
    Molecular weight:404.47

    Ref: TM-T28377

  • Soclenicant
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    Soclenicant

    CAS:
    <p>Soclenicant is a negative-altering modulator of α 7 -nAChR for anxiety, depression, and PTSD, due to its high selectivity, oral availability</p>
    Formula:C24H26N4O3
    Purity:99.57%
    Color and Shape:Soild
    Molecular weight:418.49

    Ref: TM-T203814

  • Destomycin A
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    Destomycin A

    CAS:
    <p>Destomycin A, an aminoglycoside antibiotic, exhibits activity against bacterial (Gram-positive and Gram-negative), antifungal, and anthelmintic agents. It inhibits peptide synthesis in Escherichia coli cells and stimulates adenylate cyclase in animal tissues.</p>
    Formula:C20H37N3O13
    Color and Shape:Solid
    Molecular weight:527.52

    Ref: TM-TN8311