Melatonin Receptor
Los receptores de ácido lisofosfatídico (LPA) son un grupo de GPCR que responden al LPA, un lípido bioactivo involucrado en la proliferación, migración y supervivencia celular. La señalización de LPA juega un papel crucial en varios procesos fisiológicos, incluyendo la cicatrización de heridas, el desarrollo vascular y la metástasis del cáncer. La modulación de la actividad de los receptores de LPA se está explorando para aplicaciones terapéuticas en el cáncer, la fibrosis y las enfermedades inflamatorias. En CymitQuimica, ofrecemos una gama de moduladores de receptores de LPA de alta calidad para apoyar su investigación en señalización celular, oncología y trastornos inflamatorios.
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Agomelatine
CAS:138112-76-2
Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.
Formula:
C15H17NO2
Purity:
99.92%
Color and Shape:
White Solid
Molecular weight:
243.3
Ref: TM-T1445
| 5mg | 67.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 237.00 € | ||
| 100mg | 306.00 € | ||
| 500mg | 732.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Luzindole
CAS:117946-91-5
Luzindole (N-0774) is a selective melatonin receptor antagonist.
Formula:
C19H20N2O
Purity:
98.53%
Color and Shape:
Off-White Amorphous Solid
Molecular weight:
292.37
Ref: TM-T15795
| 1mg | 51.00 € | ||
| 5mg | 143.00 € | ||
| 10mg | 233.00 € | ||
| 25mg | 389.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 812.00 € | ||
| 500mg | 1,625.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Ramelteon
CAS:196597-26-9
Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as …
Formula:
C16H21NO2
Purity:
97.21% - 99.92%
Color and Shape:
Crystalline Solid
Molecular weight:
259.34
Ref: TM-T1463
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 133.00 € | ||
| 50mg | 198.00 € | ||
| 100mg | 319.00 € | ||
| 500mg | 503.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
4-P-PDOT
CAS:134865-74-0
4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.
Formula:
C19H21NO
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
279.38
Ref: TM-T14042
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 210.00 € | ||
| 50mg | 388.00 € | ||
| 100mg | 580.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
UCM 608
CAS:151889-03-1
UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces …
Formula:
C19H20N2O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
308.37
Ref: TM-T22499
| 2mg | 51.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 98.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 238.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
N-ACETYLTRYPTAMINE
CAS:1016-47-3
N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination …
Formula:
C12H14N2O
Purity:
98.79%
Color and Shape:
Powder
Molecular weight:
202.25
Ref: TM-T8600
| 10mg | 43.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 107.00 € | ||
| 100mg | 164.00 € | ||
| 200mg | 235.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Tasimelteon
CAS:609799-22-6
Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 …
Formula:
C15H19NO2
Purity:
98.08% - 99.93%
Color and Shape:
Solid
Molecular weight:
245.32
Ref: TM-T3495
| 10mg | 44.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 109.00 € | ||
| 100mg | 175.00 € | ||
| 500mg | 438.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
S26131
CAS:296280-56-3
S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of
Formula:
C31H34N2O4
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
498.61
Ref: TM-T16834
| 5mg | 42.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 171.00 € | ||
| 100mg | 245.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Melatonin
CAS:73-31-4
Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. …
Formula:
C13H16N2O2
Purity:
98% - 99.79%
Color and Shape:
Pale Yellow Leaflets From Benzene Solid
Molecular weight:
232.28
Ref: TM-T1659
| 1g | 37.00 € | ||
| 5g | 69.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
ACH-000143
CAS:2225836-30-4
ACH-000143 have been identified as a novel agonist of the melatonin receptors MT1 and MT2.
Formula:
C13H16ClN3O3
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
297.74
Ref: TM-T9193
| 1mg | 51.00 € | ||
| 5mg | 112.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 307.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 590.00 € | ||
| 200mg | 795.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
2-Iodomelatonin
CAS:93515-00-5
2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map …
Formula:
C13H15IN2O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
358.17
Ref: TM-T10073
| 10mg | 45.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 123.00 € | ||
| 100mg | 185.00 € | ||
| 200mg | 277.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
6-Chloromelatonin
CAS:63762-74-3
6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.
Formula:
C13H15ClN2O2
Purity:
97.90% - 99.36%
Color and Shape:
Solid
Molecular weight:
266.72
Ref: TM-T22530
| 1mg | 325.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,551.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
