Melatonin Receptor
Los receptores de ácido lisofosfatídico (LPA) son un grupo de GPCR que responden al LPA, un lípido bioactivo involucrado en la proliferación, migración y supervivencia celular. La señalización de LPA juega un papel crucial en varios procesos fisiológicos, incluyendo la cicatrización de heridas, el desarrollo vascular y la metástasis del cáncer. La modulación de la actividad de los receptores de LPA se está explorando para aplicaciones terapéuticas en el cáncer, la fibrosis y las enfermedades inflamatorias. En CymitQuimica, ofrecemos una gama de moduladores de receptores de LPA de alta calidad para apoyar su investigación en señalización celular, oncología y trastornos inflamatorios.
Found 27 products for "Melatonin Receptor".
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Luzindole
CAS:Luzindole (N-0774) is a selective melatonin receptor antagonist.Formula:C19H20N2OPurity:98.53%Color and Shape:SolidMolecular weight:292.37Agomelatine
CAS:Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.Formula:C15H17NO2Purity:99.92%Color and Shape:White SolidMolecular weight:243.301Ramelteon
CAS:Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.Formula:C16H21NO2Purity:97.21% - 99.92%Color and Shape:SolidMolecular weight:259.3434Melatonin-Tamoxifen Conjugate
Melatonin-Tamoxifen Conjugate (compound 16c) is an anticancer drug conjugate made of Melatonin and Tamoxifen, serving as an effective antagonist of ERα (IC50 = 863 nM). In cells expressing the hMT1 receptor, it binds to MLT receptors (Ki = 3.1 nM) and exhibits the ability to promote β-arrestin activation (EC50 = 914 nM) and ERK activation (EC50 = 98 nM). The IC50 values for Melatonin-Tamoxifen Conjugate in MCF-7, MDA-MB-231, and HT-1080 cell lines are 6.8 μM, 6.4 μM, and 1.7 μM, respectively.Formula:C47H58N4O4Color and Shape:SolidMolecular weight:742.99Histamine & Melatonin Receptor-Targeted Compound Library
A unique collection of xnum compounds targeting histaminergic receptor and melatonin receptor for high throughput screening (HTS) and high content screening (HCSColor and Shape:Odour Solid4-P-PDOT
CAS:4-P-PDOT (4-phenyl-2- propionamidotetralin) is a potent, selective and affinity Melatonin receptor (MT2) antagonist.Formula:C19H21NOPurity:99.91%Color and Shape:White SolidMolecular weight:279.38UCM1400
UCM1400 is a melatonin receptor (MT) subtype-selective modulator. It acts as an agonist on MT1 with a pKi value of 7.94 and as an antagonist on MT2 with a pKi value of 8.11. UCM1400 inhibits MT2 receptor-mediated reduction of cyclic adenosine monophosphate (cAMP) with a pIC50 value of 7.87. It exhibits antiproliferative activity on human glioma cells and inhibits tumor growth, making it a potential candidate for cancer research, including studies on gliomas.Ramelteon-D5
CAS:Ramelteon-d5 is a deuterated compound of Ramelteon.Formula:C16H16D5NO2Color and Shape:SolidMolecular weight:264.37N-ACETYLTRYPTAMINE
CAS:N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.Formula:C12H14N2OPurity:98.79%Color and Shape:SolidMolecular weight:202.2524Tasimelteon
CAS:Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Formula:C15H19NO2Purity:98.93% - 99.93%Color and Shape:SolidMolecular weight:245.3169S26131
CAS:S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki ofFormula:C31H34N2O4Purity:99.77%Color and Shape:White SolidMolecular weight:498.6127Melatonin
CAS:Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.Formula:C13H16N2O2Purity:98% - 99.89%Color and Shape:Pale Yellow Leaflets From Benzene SolidMolecular weight:232.2783ACH-000143
CAS:ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formula:C13H16ClN3O3Purity:98.15%Color and Shape:White SolidMolecular weight:297.737UCM 608
CAS:UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.Formula:C19H20N2O2Purity:99.47%Color and Shape:Yellow SolidMolecular weight:308.37S20928
CAS:S20928 is an antagonist of melatonin receptor.Formula:C17H19NOColor and Shape:SolidMolecular weight:253.34DH97
CAS:MT2 melatonin receptor antagonistFormula:C22H26N2OPurity:98%Color and Shape:SolidMolecular weight:334.458-M-PDOT
CAS:8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.Formula:C14H19NO2Purity:99.54% - 99.54%Color and Shape:White SolidMolecular weight:233.31GR 128107
CAS:GR 128107 is an antagonist of melatonin receptor.Formula:C16H20N2O2Color and Shape:SolidMolecular weight:272.34S-22153
CAS:S22153 is an antagonist of melatonin receptor.Formula:C14H17NOSColor and Shape:SolidMolecular weight:247.36Melatonin receptor agonist 1
CAS:Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].Formula:C15H19N3O2Color and Shape:SolidMolecular weight:273.33
