Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 381 products of "Histamine Receptor"
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VUF 8430 dihydrobromide
CAS:histamine H4 receptor full agonistFormula:C4H12BrN5SPurity:98%Color and Shape:SolidMolecular weight:242.14Seliforant
CAS:Seliforant is a histamine H4 receptor antagonist.Formula:C12H21N5Purity:98%Color and Shape:SolidMolecular weight:235.33Adriforant hydrochloride
CAS:<p>Adriforant hydrochloride is an antagonist of histamine H4 receptor.</p>Formula:C13H25Cl3N6Purity:98%Color and Shape:SolidMolecular weight:371.74UK-9040
CAS:UK-9040 inhibits gastric secretory.Formula:C23H31NSPurity:98%Color and Shape:SolidMolecular weight:353.56VUF 8430
CAS:VUF 8430 is a selective agonist for the H4 receptor.Formula:C4H11N5SPurity:98%Color and Shape:SolidMolecular weight:161.23VUF 5681 dihydrobromide
CAS:<p>histamine H3 receptor silent antagonist</p>Formula:C11H21Br2N3Purity:98%Color and Shape:SolidMolecular weight:355.11Thioperamide
CAS:histamine H3 and H4 antagonist/inverse agonistFormula:C15H24N4SPurity:98%Color and Shape:White SolidMolecular weight:292.44A331440
CAS:A331440 is an modulator of L-histidine and histamine H3 receptor.Formula:C22H27N3OColor and Shape:SolidMolecular weight:349.47MK-0249
CAS:<p>MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).</p>Formula:C23H24F3N3O2Purity:99.90%Color and Shape:SolidMolecular weight:431.45Loratadine N-oxide
CAS:Loratadine N-oxide is a metabolite of the histamine H1 receptor inverse agonist loratadine.Formula:C22H23ClN2O3Color and Shape:SolidMolecular weight:398.88GSK 189254 HCl
CAS:GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.Formula:C21H26ClN3O2Purity:98%Color and Shape:SolidMolecular weight:387.9Repirinast
CAS:Repirinast is a mediator release inhibitor. It is used to treat asthma.Formula:C20H21NO5Color and Shape:SolidMolecular weight:355.38Immepip
CAS:Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.Formula:C9H15N3Color and Shape:SolidMolecular weight:165.24Phenyltoloxamine
CAS:Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).Formula:C17H21NOColor and Shape:SolidMolecular weight:255.35Mizolastine dihydrochloride
CAS:Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).Formula:C24H27Cl2FN6OPurity:98%Color and Shape:SolidMolecular weight:505.42GSK334429
CAS:GSK334429 is an antagonist of histamine H3 receptor.Formula:C20H29F3N4OColor and Shape:SolidMolecular weight:398.47Sequifenadine
CAS:Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].Formula:C22H27NOColor and Shape:SolidMolecular weight:321.46A-940894
CAS:A-940894: Potent H4 receptor antagonist, anti-inflammatory, binds well to human/rat H4, low affinity for H1/H2/H3, good pharmacokinetics.Formula:C17H21N5Color and Shape:SolidMolecular weight:295.38N-Acetylhistamine
CAS:N-Acetylhistamine (N-Omega-acetylhistamine) is a metabolite of histamine.Formula:C7H11N3OPurity:99.51%Color and Shape:SolidMolecular weight:153.18Izuforant
CAS:Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).Formula:C12H12BrN7Color and Shape:SolidMolecular weight:334.17
