Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 397 products for "Histamine Receptor".
Filter by
Purity percentage
0
100
|
0
|
50
|
90
|
95
|
100
- Lower prices
- Higher prices
- Lower purities
- Higher purities
- Faster estimated delivery
GSK-1004723
CAS:GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.Formula:C39H49ClN4O2Color and Shape:SolidMolecular weight:641.28Phenindamine
CAS:Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].Formula:C19H19NColor and Shape:SolidMolecular weight:261.36ST-1006
CAS:ST-1006: histamine H4 agonist, pKi 7.94, anti-inflammatory, anti-pruritic, promotes basophil migration.Formula:C16H20Cl2N6Purity:99.96% - 99.98%Color and Shape:SolidMolecular weight:367.28Ref: TM-T34709
1mg86.00€1mL*10mM (DMSO)187.00€5mg188.00€10mg299.00€25mg487.00€50mg600.00€100mg743.00€200mg990.00€Enerisant
CAS:Enerisant (TS-091) is a histamine H3 receptor antagonist that promotes pro-cognitive effects and reverses scopolamine-induced cognitive deficits.Formula:C22H30N4O3Purity:99.97%Color and Shape:SolidMolecular weight:398.50Ref: TM-T67828
1mg49.00€2mg67.00€5mg102.00€1mL*10mM (DMSO)111.00€10mg166.00€25mg339.00€50mg439.00€100mg610.00€200mg827.00€Histamine H3 antagonist-1
CAS:Compound 10o, a histamine H3 antagonist-1, functions as both a histamine H3 antagonist and a serotonin reuptake inhibitor, making it useful for research in depression [1].Formula:C24H28F3N3O2Color and Shape:SolidMolecular weight:447.49KF-17625
CAS:KF-17625 is an orally active bronchodilator. It inhibits bronchoconstriction induced by Carbachol, Histamine, or Leukotriene D4. Additionally, KF-17625 suppresses phosphodiesterase (PDE) IV in canine trachea with an IC50 of 12 μM and reduces histamine release from rat mast cells induced by Concanavalin-A at a 10 μM concentration with a 44% inhibition rate. This compound is applicable in research related to immunology and inflammation.Formula:C15H10N4OMolecular weight:262.27Dimephosphon
CAS:Dimephosphon is an anti-inflammatory agent exhibiting both antihistamine and antiserotonin activities. It aids in maintaining spinal cord conduction function and reduces the excitability of motor neurons around lesion areas. Additionally, Dimephosphon directly stimulates lymph vessel movement, enhancing lymph circulation. This compound is useful for studying inflammatory edema, acute spinal cord injuries, and lymphatic circulation disorders.Formula:C8H17O4PColor and Shape:SolidMolecular weight:208.19Nedocromil sodium
CAS:Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.Formula:C19H17NNaO7Purity:98%Color and Shape:SolidMolecular weight:394.335H1R ligand-1
CAS:H1R ligand-1 (Compound fragment 1) is a high-affinity ligand for the human histamine H1 receptor (H1R). It can serve as a scaffold for synthesizing a series of derivatives to investigate H1R binding kinetics.Formula:C19H23NOColor and Shape:SolidMolecular weight:281.392H3R antagonist 5
CAS:H3R antagonist 5 (Compound 1b) is a selective inverse agonist of the histamine H3 receptor that can penetrate the blood-brain barrier, with an IC50 of 0.54 nM. It is applicable for research related to the central nervous system.Formula:C23H32N2O4Color and Shape:SolidMolecular weight:400.511JNJ 40279486
CAS:JNJ 40279486 is an innovative and highly selective antagonist of the histamine H4 receptor (histamine H4receptor), with a Ki of 9 nM. It is a potential candidate for research in immune-driven inflammatory diseases.Formula:C14H15ClN6OMolecular weight:318.77CI-624
CAS:CI-624 reduces the secretion and output of hydrogen ions, sodium ions, potassium ions, and pepsin. This compound may be utilized in research focusing on cancer and autoimmune diseases.Formula:C8H8N2SColor and Shape:SolidMolecular weight:164.228Sitamaquine hydrochloride
CAS:Sitamaquine hydrochloride (WR 6026) is an orally active 8-aminoquinoline analog with antileishmanial activity. This compound inhibits mitochondrial complex II (succinate dehydrogenase) and is characterized by its lipophilic weak base properties. It rapidly accumulates in the acidic compartments of Leishmania parasites, predominantly localizing within the acidocalcisomes.Formula:C21H35Cl2N3OColor and Shape:SolidMolecular weight:416.43Arpromidine
CAS:Arpromidine (BU-E-50) acts as an agonist for the histamine H2 receptor and an antagonist for the histamine H1 receptor. It demonstrates positive inotropic effects with a lower risk of inducing arrhythmias. Arpromidine can be utilized in studies related to congestive heart failure.Formula:C21H25FN6Color and Shape:SolidMolecular weight:380.462Tixanox sodium
CAS:Tixanox sodium effectively blocks histamine release in the lungs triggered by anti-IgE. It has also been demonstrated that when administered orally, Tixanox sodium can successfully counteract exercise-induced asthma.Formula:C15H9NaO5SColor and Shape:SolidMolecular weight:324.28H3R antagonist 1
CAS:H3R-IN-1 is an effective inverse agonist of the histamine receptor 3 (H3R).Formula:C19H23N3O3Color and Shape:SolidMolecular weight:341.4ONO-8809
CAS:ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.Formula:C30H46BrNO4SPurity:98%Color and Shape:SolidMolecular weight:596.66
