Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
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MK-0249 FA
MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity …
Formula:
C24H26F3N3O4
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
477.48
Ref: TM-T12054L
| 1mg | 184.00 € | ||
| 5mg | 781.00 € | ||
| 10mg | 1,028.00 € | ||
| 25mg | 1,556.00 € | ||
| 50mg | 2,103.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Samelisant
CAS:1394808-82-2
Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.
Formula:
C21H31N3O3
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
373.49
Ref: TM-T9770
| 1mg | 111.00 € | ||
| 2mg | 163.00 € | ||
| 5mg | 275.00 € | ||
| 10mg | 440.00 € | ||
| 25mg | 724.00 € | ||
| 50mg | 1,015.00 € | ||
| 100mg | 1,357.00 € | ||
| 500mg | 2,683.00 € | ||
| 1mL*10mM (DMSO) | 282.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Tecastemizole
CAS:75970-99-9
Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of …
Formula:
C19H21FN4
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
324.4
Ref: TM-T26253
| 1mg | 56.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 297.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 603.00 € | ||
| 500mg | 1,201.00 € | ||
| 1mL*10mM (DMSO) | 138.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Sufotidine
CAS:80343-63-1
Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.
Formula:
C20H31N5O3S
Purity:
99% - 99.28%
Color and Shape:
Liquid
Molecular weight:
421.56
Ref: TM-T68146
| 1mg | 233.00 € | ||
| 5mg | 582.00 € | ||
| 10mg | 824.00 € | ||
| 25mg | 1,236.00 € | ||
| 50mg | 1,654.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
H4R antagonist 3
CAS:1003091-20-0
H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R …
Formula:
C19H21ClN4S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
372.92
Ref: TM-T77715
| 1mg | 183.00 € | ||
| 5mg | 452.00 € | ||
| 10mg | 648.00 € | ||
| 25mg | 1,011.00 € | ||
| 50mg | 1,394.00 € | ||
| 100mg | 1,843.00 € | ||
| 500mg | 3,676.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
BMY 25368 HCl
CAS:86134-36-3
BMY 25368 HCl is a competitive histamine H2 receptor antagonist that antagonizes gastric secretion stimulated …
Formula:
C19H26ClN3O3
Purity:
98.73% - 99.81%
Color and Shape:
Soild
Molecular weight:
379.88
Ref: TM-T23811L
| 1mg | 96.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 294.00 € | ||
| 25mg | 496.00 € | ||
| 50mg | 717.00 € | ||
| 100mg | 1,007.00 € | ||
| 500mg | 2,013.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Mifentidine
CAS:83184-43-4
Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric …
Formula:
C13H16N4
Purity:
100% - 99.20%
Color and Shape:
Liquid
Molecular weight:
228.29
Ref: TM-T68100
| 1mg | 182.00 € | ||
| 5mg | 451.00 € | ||
| 10mg | 646.00 € | ||
| 25mg | 1,007.00 € | ||
| 50mg | 1,390.00 € | ||
| 100mg | 1,837.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Donetidine
CAS:99248-32-5
Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
Formula:
C20H25N5O3S
Purity:
99.12%
Color and Shape:
Liquid
Molecular weight:
415.51
Ref: TM-T68056
| 1mg | 125.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 730.00 € | ||
| 50mg | 1,003.00 € | ||
| 100mg | 1,374.00 € | ||
| 500mg | 2,748.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Dalcotidine
CAS:120958-90-9
Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, …
Formula:
C18H29N3O2
Purity:
98.34%
Color and Shape:
Solid
Molecular weight:
319.44
Ref: TM-T31195
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,486.00 € | ||
| 500mg | 2,971.00 € | ||
| 1mL*10mM (DMSO) | 338.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
PF 03654746 FA
PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to …
Formula:
C19H26F2N2O3
Purity:
96.15%
Color and Shape:
Soild
Molecular weight:
368.42
Ref: TM-T12416L
| Undefined size | To inquire |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Oxmetidine
CAS:72830-39-8
Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular …
Formula:
C19H21N5O3S
Purity:
99.67%
Color and Shape:
Liquid
Molecular weight:
399.47
Ref: TM-T68122
| 1mg | 371.00 € | ||
| 5mg | 881.00 € | ||
| 10mg | 1,188.00 € | ||
| 25mg | 1,745.00 € | ||
| 50mg | 2,385.00 € | ||
| 100mg | 3,211.00 € | ||
| 500mg | 6,449.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Fenclozine Maleate
CAS:76823-82-0
Fenclozine Maleate (S 1429) is a potential histamine H1 receptor antagonist , which can be …
Formula:
C45H47ClN2O12
Purity:
98.47%
Color and Shape:
Soild
Molecular weight:
843.314
Ref: TM-T83975
| 1mg | 184.00 € | ||
| 5mg | 455.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 1,016.00 € | ||
| 50mg | 1,401.00 € | ||
| 100mg | 1,853.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
4-Methylhistamine
CAS:36507-31-0
4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for …
Formula:
C6H11N3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
125.17
Ref: TM-T80645
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Talastine
CAS:16188-61-7
Talastine is an antihistamine compound that can induce an allergic rash.
Formula:
C19H21N3O
Purity:
99.30% - 99.37%
Color and Shape:
Liquid
Molecular weight:
307.39
Ref: TM-T68150
| 1mg | 91.00 € | ||
| 5mg | 195.00 € | ||
| 10mg | 289.00 € | ||
| 25mg | 545.00 € | ||
| 50mg | 728.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,023.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Vapitadine
CAS:793655-64-8
Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.
Formula:
C17H20N4O
Purity:
100% - 100%
Color and Shape:
Soild
Molecular weight:
296.37
Ref: TM-T29096L
| 1mg | 182.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,926.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonist
Formula:
C7H13N3O2
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
171.2
Ref: TM-T23038L
| 1mg | 203.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 706.00 € | ||
| 25mg | 1,102.00 € | ||
| 50mg | 1,520.00 € | ||
| 100mg | 1,946.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Thioperamide maleate
CAS:148440-81-7
Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = …
Formula:
C19H28N4O4S
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
408.52
Ref: TM-T41247
| 1mg | 42.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 98.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Levocetirizine Dihydrochloride
CAS:130018-87-0
Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.
Formula:
C21H27Cl3N2O3
Purity:
99.75%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
461.81
Ref: TM-T22354
| 1g | 677.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 84.00 € | ||
| 50mg | 129.00 € | ||
| 100mg | 184.00 € | ||
| 200mg | 277.00 € | ||
| 500mg | 479.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Meclizine
CAS:569-65-3
Meclizine, also known as Meclozine, is a piperazine class H1 antagonist with antihistamine properties that …
Formula:
C25H27ClN2
Purity:
95.16%
Color and Shape:
Solid
Molecular weight:
390.95
Ref: TM-T40652
| 1mg | 182.00 € | ||
| 5mg | 419.00 € | ||
| 10mg | 612.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,291.00 € | ||
| 100mg | 1,757.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
Latrepirdine dihydrochloride
CAS:97657-92-6
Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.
Formula:
C21H25N3·2HCl
Purity:
98.45%
Color and Shape:
Solid
Molecular weight:
392.37
Ref: TM-T6562
| 2mg | 35.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 20 Dec 2024
