Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 327 products of "Opioid Receptor"
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Deltorphin 2
CAS:Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of 1 nM.Formula:C38H54N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:782.88LY2795050
CAS:LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).Formula:C23H22ClN3O2Purity:97.77%Color and Shape:SolidMolecular weight:407.89Ref: TM-TQ0091
1mg50.00€2mg71.00€5mg110.00€10mg172.00€25mg281.00€50mgTo inquire1mL*10mM (DMSO)120.00€Gluten Exorphin C
CAS:Gluten exorphin C is an opioid peptide derived from wheat gluten.Formula:C29H45N5O8Purity:99.39%Color and Shape:SolidMolecular weight:591.7MCOPPB triHydrochloride
CAS:MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.Formula:C26H43Cl3N4Purity:99.89% - 99.91%Color and Shape:SolidMolecular weight:518.01Ref: TM-T2071
2mg33.00€5mg52.00€10mg82.00€25mg155.00€50mg241.00€100mg355.00€200mg507.00€1mL*10mM (DMSO)55.00€CTAP(TFA) (103429-32-9 free base)
CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM.Formula:C53H70F3N13O13S2Purity:99.62%Color and Shape:SolidMolecular weight:1218.33DPDPE TFA (88373-73-3 free base)
CAS:DPDPE TFA is selective δ-opioid receptor agonist peptide. DPDPE TFA has an analgesic effect and is antinociceptive in vivo.Formula:C32H40F3N5O9S2Purity:99.39%Color and Shape:SolidMolecular weight:759.81Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Formula:C22H19NO4Purity:99.45% - 99.78%Color and Shape:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderMolecular weight:361.39Dynorphin B (1-13) acetate(83335-41-5 free base)
Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.Formula:C76H119N21O19Purity:99.72%Color and Shape:SolidMolecular weight:1630.89BMS986188
CAS:BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.Formula:C30H31BrO4Purity:98.76%Color and Shape:SolidMolecular weight:535.47DAMGO
CAS:DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity in rodents.Formula:C26H35N5O6Purity:98.83% - 99.92%Color and Shape:SolidMolecular weight:513.59Ref: TM-T4351
1mg50.00€2mg60.00€5mg87.00€10mg140.00€25mg283.00€50mg423.00€100mg623.00€1mL*10mM (DMSO)88.00€PZM21
CAS:PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).Formula:C19H27N3O2SPurity:99.93% - >99.99%Color and Shape:SolidMolecular weight:361.5Ref: TM-T4386
1mg44.00€2mg57.00€5mg93.00€10mg120.00€25mg193.00€50mg281.00€100mg447.00€1mL*10mM (DMSO)92.00€Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).Formula:C50H72N15O15SPurity:>99.99%Color and Shape:SolidMolecular weight:1326.26[D-Ala2]leucine-enkephalin
CAS:[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta opioid receptors.Formula:C29H39N5O7Purity:98.06%Color and Shape:SolidMolecular weight:569.65Alvimopan monohydrate
CAS:Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.Formula:C25H34N2O5Purity:98%Color and Shape:SolidMolecular weight:442.55Naloxegol (NKTR-118)
CAS:Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].Formula:C34H53NO11Color and Shape:SolidMolecular weight:651.78Porcine dynorphin A(1-13) acetate
Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.Formula:C77H130N24O17Purity:99.14%Color and Shape:SolidMolecular weight:1664Difelikefalin acetate
CAS:Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist.Formula:C38H57N7O8Purity:99.55%Color and Shape:SolidMolecular weight:739.9(D-Ser2)-Leu-Enkephalin-Thr
(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.Formula:C33H46N6O10Purity:94.17%Color and Shape:SoildMolecular weight:686.75BAM 22P acetate
BAM 22P acetate is a potent opioid agonist.Formula:C132H188N38O33S2Purity:99.87%Color and Shape:SoildMolecular weight:2899.27Ref: TM-TP1211L
1mg100.00€5mg376.00€10mg565.00€25mg1,009.00€50mg1,359.00€100mg1,845.00€200mg2,485.00€Endomorphin 2
CAS:EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.Formula:C32H37N5O5Purity:99.64%Color and Shape:SolidMolecular weight:571.67LY2940094 tartrate
CAS:LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.Formula:C26H29ClF2N4O8SColor and Shape:SolidMolecular weight:631.04Dynorphin A acetate(80448-90-4 free base)
Dynorphin A acetate is an Endogenous kappa receptor agonist.Formula:C101H159N31O25Purity:99.69%Color and Shape:SolidMolecular weight:2207.58Salvinorin A
CAS:Salvinorin A is a non-nitrogenous κ-opioid selective agonist.Formula:C23H28O8Purity:99.06%Color and Shape:SolidMolecular weight:432.46Ref: TM-T23306
1mg259.00€5mg628.00€10mg897.00€25mg1,341.00€50mg1,791.00€100mg2,412.00€1mL*10mM (DMSO)695.00€AR-M 1000390 hydrochloride
CAS:ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.Formula:C23H29ClN2OPurity:98.66%Color and Shape:SolidMolecular weight:384.94Dermorphin TFA
CAS:Dermorphin TFA is a new class of opioids-like peptidesFormula:C42H51F3N8O12Purity:98% - >99.99%Color and Shape:SolidMolecular weight:916.89BW-180C
CAS:BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid receptor. Displays antinociceptive activity in vivo.Formula:C29H39N5O7Purity:>99.99%Color and Shape:SolidMolecular weight:569.65Ref: TM-TP1905
2mg39.00€5mg58.00€10mg93.00€25mg145.00€50mg260.00€100mg462.00€200mg655.00€1mL*10mM (DMSO)73.00€Sec-O-Glucosylhamaudol
CAS:Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.Formula:C21H26O10Purity:99.79%Color and Shape:SolidMolecular weight:438.43Sinomenine
CAS:Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.
Formula:C19H23NO4Purity:99.02% - 99.73%Color and Shape:White PowderMolecular weight:329.39N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formula:C17H17ClN4Purity:97.25% - 99.83%Color and Shape:Yellow Crystalline SolidMolecular weight:312.8Ref: TM-T5158
2mg34.00€5mg48.00€10mg79.00€25mg152.00€50mg235.00€100mg344.00€200mg490.00€1mL*10mM (DMSO)58.00€Nociceptin
CAS:Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.Formula:C79H129N27O22Purity:99.35%Color and Shape:SolidMolecular weight:1809.04Nociceptin (1-7) acetate
Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.Formula:C31H41N7O9Purity:98.92%Color and Shape:SoildMolecular weight:655.7Ref: TM-T23076L
1mg294.00€2mg439.00€5mg660.00€10mg999.00€25mg1,468.00€50mg1,998.00€100mg2,692.00€1mL*10mM (DMSO)897.00€[Leu5]-Enkephalin, amide acetate
[Leu5]-Enkephalin, amide acetate is a δ opioid receptor agonist.Formula:C30H42N6O8Purity:99.36%Color and Shape:SolidMolecular weight:614.69DAMGO TFA (78123-71-4(Free base))
DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and quality-assured.Formula:C28H36F3N5O8Purity:98.67% - 99.76%Color and Shape:SolidMolecular weight:627.6Corydaline
CAS:Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits CYP2C19 and CYP2C9.Formula:C22H27NO4Purity:98.97% - 99.86%Color and Shape:SolidMolecular weight:369.45BMS986187
CAS:BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.Formula:C31H34O4Purity:99.09%Color and Shape:SolidMolecular weight:470.6Dynorphin A 1-10 acetate(79994-24-4 free base)
Dynorphin A (1-10) acetate is an endogenous opioid neuropeptide, binds to extracellular loop 2 of the κ-opioid receptor.Formula:C59H95N19O14Purity:99.88%Color and Shape:SolidMolecular weight:1294.53Hemorphin-7 acetate(152685-85-3 free base)
Hemorphin-7 acetate is a hemorphin peptide, an endogenous opioid peptide derived from the β-chain of hemoglobin.Formula:C51H68N12O13Purity:99.66%Color and Shape:SolidMolecular weight:1057.16Aticaprant
CAS:Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective and quality-assured.Formula:C26H27FN2O2Purity:99.9% - 99.97%Color and Shape:SolidMolecular weight:418.5Ref: TM-TQ0082
1mg40.00€2mg52.00€5mg88.00€10mg126.00€25mg259.00€50mg406.00€100mg607.00€1mL*10mM (DMSO)87.00€EST73502 HCl
CAS:EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.Formula:C19H27ClF2N2O2Purity:99.96%Color and Shape:SolidMolecular weight:388.88Ref: TM-T39284
1mg96.00€5mg172.00€10mg244.00€25mg403.00€50mg567.00€100mg750.00€200mg1,018.00€1mL*10mM (DMSO)187.00€GR103545
CAS:GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can be used as in vivo imaging.Formula:C23H29Cl2N3O7Purity:99.75%Color and Shape:SolidMolecular weight:530.4Ref: TM-T9459
1mg93.00€2mg136.00€5mg178.00€10mg268.00€25mg482.00€50mg688.00€100mg964.00€1mL*10mM (DMSO)236.00€BRL 52537 hydrochloride
CAS:BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.Formula:C18H25Cl3N2OPurity:99.04%Color and Shape:SolidMolecular weight:391.76Ac-RYYRWK-NH2 acetate
Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.Formula:C51H73N15O11Purity:98.59%Color and Shape:SolidMolecular weight:1072.22JTC-801
CAS:JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.Formula:C26H25N3O2·HClPurity:99.27% - 99.59%Color and Shape:SolidMolecular weight:447.96Tyr-Gly-Gly-Phe-Met-OH
CAS:Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.
Formula:C27H35N5O7SPurity:≥95%Color and Shape:White Lyophilised SolidMolecular weight:573.66Deltorphin I
CAS:Deltorphin I is an agonist of δ-opioid receptor.Formula:C37H52N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:768.86Asimadoline hydrochloride
CAS:Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.Formula:C27H31ClN2O2Purity:98.94% - 99.32%Color and Shape:SolidMolecular weight:451.01Ref: TM-T4691
1mg35.00€5mg73.00€10mg111.00€25mg227.00€50mg338.00€100mg500.00€500mg1,074.00€1mL*10mM (DMSO)81.00€Endomorphin 1
CAS:Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays reasonable affinities for kappa3 binding sites (Ki: 20~30 nM).Formula:C34H38N6O5Purity:95.92%Color and Shape:Solid (Solid Powder )Molecular weight:610.7b-Casomorphin (1-3) Acetate
b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.Formula:C25H31N3O7Purity:98.99%Color and Shape:SolidMolecular weight:485.53Ref: TM-T21660L
5mg42.00€10mg57.00€25mg87.00€50mg131.00€100mg190.00€200mg285.00€1mL*10mM (DMSO)55.00€ADL-5747 (HCl)
CAS:ADL-5747, an opioid delta receptor agonist, is used potentially for the treatment of pain.Formula:C24H29ClN2O3Color and Shape:SolidMolecular weight:428.95N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Formula:C30H39N5O8Purity:>99.99%Color and Shape:SolidMolecular weight:597.66
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