Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 296 products of "Opioid Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Nociceptin
CAS:<p>Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide dynorphin A.</p>Formula:C79H129N27O22Purity:99.35%Color and Shape:SolidMolecular weight:1809.04LY2940094 tartrate
CAS:<p>LY-2940094, a nociceptin receptor antagonist, is used potentially for the treatment of major depressive disorder and alcoholism.</p>Formula:C26H29ClF2N4O8SColor and Shape:SolidMolecular weight:631.04b-Casomorphin (1-3) Acetate
<p>b-Casomorphin (1-3) Acetate is a tri-peptide with an opioid effect.</p>Formula:C25H31N3O7Purity:98.99%Color and Shape:SolidMolecular weight:485.53BMS986187
CAS:<p>BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.</p>Formula:C31H34O4Purity:99.09%Color and Shape:SolidMolecular weight:470.6Salvinorin A
CAS:<p>Salvinorin A is a non-nitrogenous κ-opioid selective agonist.</p>Formula:C23H28O8Purity:99.06%Color and Shape:SolidMolecular weight:432.46Naloxegol oxalate
CAS:<p>Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.</p>Formula:C36H55NO15Purity:99.67% - >99.99%Color and Shape:SolidMolecular weight:741.83MCOPPB triHydrochloride
CAS:<p>MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.</p>Formula:C26H43Cl3N4Purity:99.89% - 99.91%Color and Shape:SolidMolecular weight:518.01BAM 22P acetate
<p>BAM 22P acetate is a potent opioid agonist.</p>Formula:C132H188N38O33S2Purity:99.87%Color and Shape:SoildMolecular weight:2899.27Nalmefene hydrochloride
CAS:<p>Nalmefene antagonizes the effects of opioids by competing for the opioid receptors in the CNS.</p>Formula:C21H26ClNO3Purity:98% - 99.85%Color and Shape:SolidMolecular weight:375.89AR-M 1000390 hydrochloride
CAS:<p>ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from SNC 80.</p>Formula:C23H29ClN2OPurity:98.66%Color and Shape:SolidMolecular weight:384.94Tyr-Gly-Gly-Phe-Met-OH
CAS:<p>Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding to the opioid receptor.</p>Formula:C27H35N5O7SPurity:≥95%Color and Shape:White Lyophilised SolidMolecular weight:573.66N-terminally acetylated Leu-enkephalin
<p>Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.</p>Formula:C30H39N5O8Purity:>99.99%Color and Shape:SolidMolecular weight:597.66Endomorphin 2
CAS:<p>EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles via presynaptic/postsynaptic mechanisms.</p>Formula:C32H37N5O5Purity:99.64%Color and Shape:SolidMolecular weight:571.67Methylnaltrexone bromide
CAS:<p>Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.</p>Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35EST73502 HCl
CAS:<p>EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.</p>Formula:C19H27ClF2N2O2Purity:99.96%Color and Shape:SolidMolecular weight:388.88JTC-801
CAS:<p>JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly inhibits receptors δ, κ, and μ.</p>Formula:C26H25N3O2·HClPurity:99.27% - 99.59%Color and Shape:SolidMolecular weight:447.96Orphanin FQ(1-11) acetate(178249-41-7 free base)
<p>Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.</p>Formula:C51H79N15O16Purity:95.54%Color and Shape:SolidMolecular weight:1158.26Dermorphin TFA
CAS:<p>Dermorphin TFA is a new class of opioids-like peptides</p>Formula:C42H51F3N8O12Purity:98% - >99.99%Color and Shape:SolidMolecular weight:916.89Deltorphin I
CAS:<p>Deltorphin I is an agonist of δ-opioid receptor.</p>Formula:C37H52N8O10Purity:>99.99%Color and Shape:SolidMolecular weight:768.86BMS-986122
CAS:<p>BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1</p>Formula:C16H15BrClNO3S2Purity:98.42%Color and Shape:SolidMolecular weight:448.78Dynorphin A acetate(80448-90-4 free base)
<p>Dynorphin A acetate is an Endogenous kappa receptor agonist.</p>Formula:C101H159N31O25Purity:99.69%Color and Shape:SolidMolecular weight:2207.58ADL-5859
CAS:<p>ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for the</p>Formula:C24H28N2O3·HClPurity:98.78% - 99.11%Color and Shape:SolidMolecular weight:428.95Sec-O-Glucosylhamaudol
CAS:<p>Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.</p>Formula:C21H26O10Purity:99.79%Color and Shape:SolidMolecular weight:438.43BRL 52537 hydrochloride
CAS:<p>BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke and heart attack research.</p>Formula:C18H25Cl3N2OPurity:99.04%Color and Shape:SolidMolecular weight:391.76Nociceptin (1-7) acetate
<p>Nociceptin (1-7) acetate is a potent agonist of opioid receptor-like 1 (ORL1) receptor.</p>Formula:C31H41N7O9Purity:98.92%Color and Shape:SoildMolecular weight:655.7(D-Ser2)-Leu-Enkephalin-Thr
<p>(D-Ser2)-Leu-Enkephalin-Thr is a delta selective agent of opioid receptor and shows analgesic effects.</p>Formula:C33H46N6O10Purity:94.17%Color and Shape:SoildMolecular weight:686.75Porcine dynorphin A(1-13) acetate
<p>Porcine dynorphin A(1-13) acetate is a potent κ-opioid agonist with antinociceptive properties, increasing [Ca2+]i like NMDA.</p>Formula:C77H130N24O17Purity:99.14%Color and Shape:SolidMolecular weight:1664Ac-RYYRWK-NH2 acetate
<p>Ac-RYYRWK-NH2 acetate is a potent partial agonist of the nociceptin receptor(NOP), which is the endogenous ORL1 receptor agonist.</p>Formula:C51H73N15O11Purity:98.59%Color and Shape:SolidMolecular weight:1072.22Naloxegol (NKTR-118)
CAS:<p>Naloxegol (NKTR-118; AZ-13337019) is an opioid-receptor antagonist[1].</p>Formula:C34H53NO11Color and Shape:SolidMolecular weight:651.78Sinomenine
CAS:<p>Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the treatment of rheumatism and arthritis.</p>Formula:C19H23NO4Purity:99.02% - 99.73%Color and Shape:White PowderMolecular weight:329.39Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Formula:C76H119N21O19Purity:99.72%Color and Shape:SolidMolecular weight:1630.89Bisacodyl
CAS:<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Formula:C22H19NO4Purity:99.45% - 99.78%Color and Shape:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderMolecular weight:361.39LY2795050
CAS:<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Formula:C23H22ClN3O2Purity:97.77%Color and Shape:SolidMolecular weight:407.89Alvimopan monohydrate
CAS:<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Formula:C25H34N2O5Purity:98%Color and Shape:SolidMolecular weight:442.55[Met5]-Enkephalin, amide TFA
<p>[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.</p>Formula:C29H37F3N6O8SPurity:99.81%Color and Shape:SolidMolecular weight:686.7GRT2932Q
CAS:<p>GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].</p>Formula:C25H26ClN3OColor and Shape:SolidMolecular weight:419.95LY2048978
CAS:<p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:312.41ML138
CAS:<p>ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.</p>Formula:C19H14Cl2N4OSColor and Shape:SolidMolecular weight:417.31SCH 221510
CAS:<p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>Formula:C28H31NOPurity:99.54%Color and Shape:SolidMolecular weight:397.55μ opioid receptor agonist 2
CAS:<p>μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.</p>Formula:C25H34N4OColor and Shape:SolidMolecular weight:406.56TIPP
CAS:<p>TIPP is an agent of delta opioid antagonist.</p>Formula:C37H38N4O6Purity:98%Color and Shape:SolidMolecular weight:634.72Opioid receptor modulator 1
CAS:<p>Opioid receptor modulator 1 is a modulator of opioid receptor.</p>Formula:C18H23NO2Purity:98%Color and Shape:SolidMolecular weight:285.38LY2444296
CAS:<p>LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).</p>Formula:C24H22F2N2O2Purity:99.18%Color and Shape:SolidMolecular weight:408.44BW 373U86
CAS:<p>BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [</p>Formula:C27H37N3O2Color and Shape:SolidMolecular weight:435.6ML 190
CAS:<p>ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.</p>Formula:C27H32N6O3Purity:99.88%Color and Shape:SolidMolecular weight:488.58GSK1521498 free base (hydrochloride)
CAS:<p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>Formula:C24H21ClF2N4Purity:98%Color and Shape:SolidMolecular weight:438.9ADL-5859 HCl
CAS:<p>ADL-5859 is a delta-opioid receptor agonist.</p>Formula:C24H28N2O3Purity:98%Color and Shape:SolidMolecular weight:392.49DIPPA hydrochloride
CAS:<p>κ receptor antagonist</p>Formula:C22H24Cl3N3OSPurity:98%Color and Shape:SolidMolecular weight:484.87PF-4455242 HCl
CAS:<p>PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.</p>Formula:C21H29ClN2O2SPurity:99.59%Color and Shape:SolidMolecular weight:408.99CP-866087
CAS:<p>CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.</p>Formula:C24H28N2O2Purity:99.56% - >99.99%Color and Shape:SoildMolecular weight:376.49
![[Met5]-Enkephalin, amide TFA](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1254.webp&w=3840&q=75)
