Glucagon Receptor
Glucagon receptors are GPCRs that mediate the effects of glucagon, a hormone involved in regulating glucose homeostasis by promoting glycogen breakdown and glucose release from the liver. These receptors are critical in the management of blood sugar levels and are of particular interest in the study of diabetes and metabolic disorders. Glucagon receptor antagonists are being explored as potential treatments for hyperglycemia in type 2 diabetes. At CymitQuimica, we offer a variety of high-quality glucagon receptor modulators to support your research in endocrinology, diabetes, and metabolic regulation.
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Glucagon (1-29), bovine, human, porcine hydrochloride
CAS:28270-04-4
Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon …
Formula:
C153H225N43O49S·ClH
Purity:
95.65% - 98.03%
Color and Shape:
Solid
Molecular weight:
3519.21
Ref: TM-T15389L
| 1mg | 86.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 466.00 € | ||
| 50mg | 677.00 € | ||
| 100mg | 915.00 € | ||
| 500mg | 1,841.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
PF-06882961
CAS:2230198-02-2
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:
C31H30FN5O4
Purity:
95.1% - 99.54%
Color and Shape:
Solid
Molecular weight:
555.6
Ref: TM-T12431
| 1mg | 50.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 153.00 € | ||
| 25mg | 195.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | 427.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
GLP-1 (9-36) amide
CAS:161748-29-4
GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.
Formula:
C140H214N36O43
Purity:
97%
Color and Shape:
Solid
Molecular weight:
3089.41
Ref: TM-TP2252
| 1mg | 88.00 € | ||
| 5mg | 238.00 € | ||
| 10mg | 353.00 € | ||
| 25mg | 584.00 € | ||
| 50mg | 823.00 € | ||
| 100mg | 1,109.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
(S, R)-LSN 3318839
CAS:2765539-92-0
(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.
Formula:
C26H23Cl2N3O2
Purity:
99.57%
Color and Shape:
Soild
Molecular weight:
480.39
Ref: TM-T63166L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,699.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
GLP-1R Antagonist 1
CAS:488097-06-9
GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor …
Formula:
C16H11ClF6N4O2
Purity:
90%
Color and Shape:
Solid
Molecular weight:
440.73
Ref: TM-T15387
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 423.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
GLP-1 receptor agonist 9 citrate
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
Formula:
C38H39ClFN3O12
Purity:
95%
Color and Shape:
Liquid
Molecular weight:
784.18
Ref: TM-T9579L
| 1mg | 181.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,287.00 € | ||
| 100mg | 1,738.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Semaglutide TFA (910463-68-2 free base)
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 …
Formula:
NA
Purity:
98%
Color and Shape:
Solid
Molecular weight:
4210.63
Ref: TM-T12878
| 1mg | 219.00 € | ||
| 5mg | 758.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Orforglipron
CAS:2212020-52-3
Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist …
Formula:
C48H48F2N10O5
Purity:
99.15% - 99.61%
Color and Shape:
Solid
Molecular weight:
882.96
Ref: TM-T11408
| 1mg | 239.00 € | ||
| 5mg | 587.00 € | ||
| 10mg | 922.00 € | ||
| 25mg | 1,848.00 € | ||
| 50mg | 2,499.00 € | ||
| 100mg | 3,378.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
V-0219 hydrochloride
V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.
Formula:
C20H26ClF3N4O2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
446.89
Ref: TM-T60047L
| 1mg | 65.00 € | ||
| 5mg | 133.00 € | ||
| 10mg | 206.00 € | ||
| 25mg | 393.00 € | ||
| 50mg | 586.00 € | ||
| 100mg | 834.00 € | ||
| 500mg | 1,658.00 € | ||
| 1mL*10mM (DMSO) | 171.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
GLP-1R Agonist DMB
CAS:281209-71-0
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 …
Formula:
C13H15Cl2N3O2S
Purity:
99.52%
Color and Shape:
Liquid
Molecular weight:
348.25
Ref: TM-T36579
| 1mg | 51.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 233.00 € | ||
| 25mg | 397.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
GLP-1R modulator C16
CAS:875005-43-9
GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.
Formula:
C21H26ClFN2O3
Purity:
99.6% - 99.6%
Color and Shape:
Liquid
Molecular weight:
408.89
Ref: TM-T40997
| 1mg | 98.00 € | ||
| 2mg | 140.00 € | ||
| 5mg | 222.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
V-0219
CAS:878453-71-5
V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about …
Formula:
C20H25F3N4O2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
410.43
Ref: TM-T60047
| 2mg | 108.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GLP-1R modulator C5
CAS:421578-93-0
GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane …
Formula:
C24H21NO3
Purity:
99.59%
Color and Shape:
Liquid
Molecular weight:
371.43
Ref: TM-T61483
| 1mg | 42.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Exendin-4 acetate
CAS:914454-01-6
Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 …
Formula:
C186H286N50O62S
Purity:
98.65%
Color and Shape:
Solid
Molecular weight:
4247
Ref: TM-T8748
| 1mg | 67.00 € | ||
| 5mg | 135.00 € | ||
| 10mg | 193.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 412.00 € | ||
| 100mg | 607.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PF-06882961 Tris
CAS:2230198-03-3
PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Formula:
C35H41FN6O7
Purity:
98.11% - 99.52%
Color and Shape:
Solid
Molecular weight:
676.7
Ref: TM-T8876
| 1mg | 129.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 694.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,318.00 € | ||
| 500mg | 2,626.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
GRA Ex-25
CAS:307983-31-9
GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.
Formula:
C29H36F3N3O5
Purity:
98.2% - 98.88%
Color and Shape:
Solid
Molecular weight:
563.61
Ref: TM-T3422
| 1mg | 62.00 € | ||
| 2mg | 88.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 203.00 € | ||
| 25mg | 414.00 € | ||
| 50mg | 609.00 € | ||
| 100mg | 869.00 € | ||
| 1mL*10mM (DMSO) | 184.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Shanzhiside methyl ester
CAS:64421-28-9
Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 …
Formula:
C17H26O11
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
406.38
Ref: TM-T3896
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 134.00 € | ||
| 50mg | 185.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Lixisenatide acetate (320367-13-3 free base)
CAS:1997361-87-1
Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of …
Formula:
C215H347N61O65S·6C2H4O2
Purity:
98% - 99.9%
Color and Shape:
Solid
Molecular weight:
5218.88
Ref: TM-TP1469
| 1mg | 62.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 179.00 € | ||
| 25mg | 299.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 582.00 € | ||
| 200mg | 784.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BETP
CAS:1371569-69-5
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and …
Formula:
C20H17F3N2O2S
Purity:
97.92%
Color and Shape:
Solid
Molecular weight:
406.42
Ref: TM-TQ0124
| 1mg | 47.00 € | ||
| 5mg | 91.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 414.00 € | ||
| 100mg | 661.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
GLP-1(7-36), amide
CAS:107444-51-9
GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the …
Formula:
C149H226N40O45
Purity:
99.85%
Color and Shape:
White Powder
Molecular weight:
3297.63
Ref: TM-T3984
| 1mg | 173.00 € | ||
| 2mg | 306.00 € | ||
| 5mg | 516.00 € | ||
| 10mg | 741.00 € | ||
| 25mg | 1,152.00 € | ||
| 50mg | 1,539.00 € | ||
| 100mg | 2,095.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
