Glucagon Receptor
Glucagon receptors are GPCRs that mediate the effects of glucagon, a hormone involved in regulating glucose homeostasis by promoting glycogen breakdown and glucose release from the liver. These receptors are critical in the management of blood sugar levels and are of particular interest in the study of diabetes and metabolic disorders. Glucagon receptor antagonists are being explored as potential treatments for hyperglycemia in type 2 diabetes. At CymitQuimica, we offer a variety of high-quality glucagon receptor modulators to support your research in endocrinology, diabetes, and metabolic regulation.
Found 164 products of "Glucagon Receptor"
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Anti-GCGR Antibody (7J909)
<p>Anti-GCGR Antibody (7J909) is an antibody targeting GCGR. Anti-GCGR Antibody (7J909) can be used in ELISA.</p>Color and Shape:Odour LiquidSCO-267
CAS:<p>SCO-267 is a full agonist of GPR40/FFAR1， stimulating insulin secretion and GLP-1 release in diabetic rats, improving glucose tolerance,type 2 diabetes.</p>Formula:C36H46N4O5Purity:99.89%Color and Shape:SolidMolecular weight:614.77GLP-1R modulator C5
CAS:<p>GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.</p>Formula:C24H21NO3Purity:99.59%Color and Shape:SolidMolecular weight:371.43Liraglutide
CAS:<p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>Formula:C172H265N43O51Purity:97.65% - 99.04%Color and Shape:SolidMolecular weight:3751.25PF-06882961 Tris
CAS:<p>PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>Formula:C35H41FN6O7Purity:98.74% - 99.79%Color and Shape:SolidMolecular weight:676.7GRA Ex-25
CAS:<p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>Formula:C29H36F3N3O5Purity:98.2% - 98.88%Color and Shape:SolidMolecular weight:563.61Shanzhiside methyl ester
CAS:<p>Shanzhiside methylester soothes neuropathic pain by triggering spinal GLP-1 receptors, boosting microglial β-endorphin through p38 MAPK.</p>Formula:C17H26O11Purity:98.998% - 99.32%Color and Shape:SolidMolecular weight:406.38Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Formula:C215H347N61O65S·6C2H4O2Purity:98% - 99.9%Color and Shape:SolidMolecular weight:5218.88BETP
CAS:<p>BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).</p>Formula:C20H17F3N2O2SPurity:98.51%Color and Shape:SolidMolecular weight:406.42HAEGTFTSDVSSYLE
<p>HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.</p>Formula:C71H103N17O28Purity:>99.99%Color and Shape:SolidMolecular weight:1642.71GLP-1(7-36), amide
CAS:<p>GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.</p>Formula:C149H226N40O45Purity:99.85%Color and Shape:White PowderMolecular weight:3297.63Exendin-4
CAS:<p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>Formula:C184H282N50O60SPurity:97.71% - 99.78%Color and Shape:SolidMolecular weight:4186.57Semaglutide
CAS:<p>Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).</p>Formula:C187H291N45O59Purity:96.92% - 99.78%Color and Shape:SolidMolecular weight:4114Exendin-4 acetate
CAS:<p>Exendin-4 acetate is a 39 amino acid peptide.Exendin-4 acetate is a long-acting GLP-1 receptor agonist(IC50 = 3.22 nM).</p>Formula:C186H286N50O62SPurity:98.48% - 99.78%Color and Shape:SolidMolecular weight:4247Oxyntomodulin acetate
<p>Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].</p>Purity:99.24%Color and Shape:LiquidMolecular weight:N/ABay 55-9837 acetate
<p>Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.</p>Purity:98.27%Color and Shape:LiquidMolecular weight:N/ASecretin (33-59), rat
CAS:<p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>Formula:C129H216N42O42Purity:98.12%Color and Shape:SolidMolecular weight:3027.35Glucagon (19-29), human acetate
<p>Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.</p>Formula:C63H93N15O20SPurity:98.11%Color and Shape:SolidMolecular weight:1412.57HAEGTFT acetate(926018-95-3 free base)
<p>HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Formula:C35H51N9O14Purity:>99.99%Color and Shape:SolidMolecular weight:821.84Tirzepatide Acetate(2023788-19-2 free base)
<p>Tirzepatide (LY3298176) Acetate (2023788-19-2 free base) is a new molecule that can control blood glucose levels.Cost-effective and quality-assured.</p>Formula:C227H352N48O70Purity:97.3% - 98.05%Color and Shape:SolidMolecular weight:4873.5Albiglutide TFA (782500-75-8 free base)
<p>Albiglutide TFA (782500-75-8 free base) (Albiglutide TFA) is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).</p>Formula:C150H225F3N40O47Purity:>99.99%Color and Shape:SolidMolecular weight:3397.63Teduglutide acetate
<p>Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy.</p>Formula:C166H256N44O56SPurity:97.39%Color and Shape:SoildMolecular weight:3812.13ML-SI3
CAS:<p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>Formula:C23H31N3O3SPurity:99.75%Color and Shape:SolidMolecular weight:429.58Exenatide
CAS:<p>Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.</p>Formula:C186H286N50O62SPurity:99.42%Color and Shape:SolidMolecular weight:4247Glucagon-like peptide 1 (1-37), human acetate
<p>Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.</p>Purity:98%Color and Shape:LiquidMolecular weight:N/ACotadutide acetate
<p>Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 pM and 10.2 pM.</p>Formula:C169H256N42O57Purity:98.28%Color and Shape:SolidMolecular weight:3788.14GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Formula:C151H228N40O47Purity:98.89%Color and Shape:SolidMolecular weight:3355.67Avexitide
CAS:<p>Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.</p>Formula:C149H234N40O47SPurity:98% - 99.65%Color and Shape:SolidMolecular weight:3369.76GLP-1 receptor agonist 9
CAS:<p>1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.</p>Formula:C32H31ClFN3O5Purity:98%Color and Shape:SolidMolecular weight:592.06PF-06291874
CAS:<p>PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.</p>Formula:C26H28F3N3O4Purity:99.12% - 99.27%Color and Shape:SolidMolecular weight:503.51NNC-0640
CAS:<p>NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.</p>Formula:C29H31N7O4SPurity:97.04%Color and Shape:SolidMolecular weight:573.67Glucagon receptor antagonists-5
CAS:<p>Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.</p>Formula:C30H29ClF3N3O3Purity:98%Color and Shape:SolidMolecular weight:572.02BAY-27-9955
CAS:<p>BAY-27-9955 is a glucagon receptor antagonist.</p>Formula:C23H31FOColor and Shape:SolidMolecular weight:342.49(R)-V-0219
<p>(R)-V-0219: GLP-1R PAM, orally active, triggers Ca++ flux in HEK-hGLP-1R cells.</p>Formula:C20H25F3N4O2Color and Shape:SolidMolecular weight:410.43GLP-1R agonist 1
CAS:<p>GLP-1R agonist 1, an imidazole derivative and potent GLP-1R activator, may aid diabetes research.</p>Formula:C32H29ClFN3O5Color and Shape:SolidMolecular weight:590.04Glucagon receptor antagonists-2
CAS:<p>Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist.</p>Formula:C22H30FNO2Purity:98%Color and Shape:SolidMolecular weight:359.48MS012
CAS:<p>MS012 is a Potent and Selective Inhibitors for G9a-Like Protein (GLP) Lysine Methyltransferase (Kd = 46 ± 15 nM).</p>Formula:C22H35N5O2Color and Shape:SolidMolecular weight:401.55(S)-V-0219
<p>(S)-V-0219: oral, GLP-1R PAM, boosts calcium in hGLP-1R HEK cells, lowers glucose, curbs hunger in mice.</p>Formula:C20H25F3N4O2Color and Shape:SolidMolecular weight:410.43GCGR antagonist 2
CAS:<p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>Formula:C28H26N4O2Color and Shape:SolidMolecular weight:450.53NNC 92-1687
CAS:<p>NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.</p>Formula:C15H12N2O3SPurity:98.70% - 99.70%Color and Shape:SolidMolecular weight:300.33L-168049
CAS:<p>L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM canine.</p>Formula:C24H20BrClN2OPurity:>99.99%Color and Shape:SolidMolecular weight:467.79GLP-1R agonist 9
CAS:<p>GLP-1R agonist 9 acts as a GLP-1R agonist, demonstrating efficacy with EC50 values of 1.1 nM and 11 nM against CHO GLP-1R Clone H6 and Clone C6, respectively.</p>Formula:C32H30ClF2N3O5Color and Shape:SolidMolecular weight:610.05GLP-1R agonist 17
CAS:<p>GLP-1R agonist 17 excels in stimulating GLP-1 receptors, useful for cardiovascular metabolic disease research.</p>Formula:C28H26ClFN4O4SColor and Shape:SolidMolecular weight:569.05Glucagon receptor antagonists-3
CAS:<p>Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist.</p>Formula:C22H30FNO2Purity:98%Color and Shape:SolidMolecular weight:359.48GLP-1 receptor agonist 3
CAS:<p>GLP-1 receptor agonist 3 is a GLP-1 receptor agonist,Example 4A-1, has EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively.</p>Formula:C31H30FN5O4Purity:98%Color and Shape:SolidMolecular weight:555.6GLP-1R agonist 12
CAS:<p>GLP-1R agonist 12 (Compound 123) 是一种 GLP-1R 激动剂，能够用于研究糖尿病。</p>Formula:C34H36N6O4Color and Shape:SolidMolecular weight:592.69LGD-6972 sodium
CAS:<p>LGD-6972 sodium is a glucagon receptor antagonist.</p>Formula:C43H46N2NaO5SPurity:98%Color and Shape:SolidMolecular weight:725.9Antitumor agent-101
CAS:<p>Antitumor agent-101 is a selective, covalent inhibitor targeting lysine methyltransferases G9a/GLP, demonstrating IC50 values of 8.5 nM for G9a and 5.5 nM for</p>Formula:C26H38N6O3Purity:98%Color and Shape:SolidMolecular weight:482.62MK 0893
CAS:<p>MK 0893 is a potent and selective Glucagon Receptor (GR) antagonist competitive, reversible cAMP activity, which attenuates blood glucose elevation.</p>Formula:C32H27Cl2N3O4Purity:98.79%Color and Shape:SolidMolecular weight:588.48MK3577
CAS:<p>MK3577 is a glucagon receptor antagonist.</p>Formula:C30H30ClFN2O3Color and Shape:SolidMolecular weight:521.02
