Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 242 products of "Adenosine Receptor"
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Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Formula:C24H29ClF3N5O5SPurity:96.56%Color and Shape:SoildMolecular weight:592.03Pamabrom
CAS:<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Formula:C11H18BrN5O3Purity:99.84% - >99.99%Color and Shape:CoaMolecular weight:348.2Adenosine 5'-monophosphate monohydrate
CAS:<p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>Formula:C10H14N5O7P·H2OPurity:97.68% - 98.49%Color and Shape:White PowderMolecular weight:365.24Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Formula:C14H15Cl2NSPurity:99.85% - >99.99%Color and Shape:White PowderMolecular weight:300.25Quercetin-3'-o-phosphate TEA
<p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>Formula:C21H26NO10PPurity:95.63%Color and Shape:SoildMolecular weight:483.41AB928
CAS:<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Formula:C23H22N8OPurity:98.09% - >99.99%Color and Shape:SolidMolecular weight:426.47Pentoxifylline
CAS:<p>Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.</p>Formula:C13H18N4O3Purity:99.26% - 99.93%Color and Shape:SolidMolecular weight:278.31Diphylline
CAS:<p>Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.</p>Formula:C10H14N4O4Purity:98.54%Color and Shape:Crystals From Alcohol SolidMolecular weight:254.24Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formula:C11H14N4O4Purity:99.958% - >99.99%Color and Shape:SolidMolecular weight:266.25Theophylline
CAS:<p>Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central</p>Formula:C7H8N4O2Purity:99.65% - 99.98%Color and Shape:White Solid PowderMolecular weight:180.16DPTN dihydrochloride
CAS:<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Formula:C22H20Cl2N4OSPurity:99.95%Color and Shape:SoildMolecular weight:459.39Adenosine A1 receptor activator T62
CAS:<p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>Formula:C15H14ClNOSPurity:97.83%Color and Shape:SolidMolecular weight:291.8YT 146
CAS:<p>YT 146 is a biochemical.</p>Formula:C18H25N5O4Purity:98.81% - 99.25%Color and Shape:SolidMolecular weight:375.42Theophylline monohydrate
CAS:<p>Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium</p>Formula:C7H8N4O2·H2OPurity:99.78%Color and Shape:SolidMolecular weight:198.18Aminophylline
CAS:<p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>Formula:C7H8O2·C2H8N2Purity:99.31%Color and Shape:White Or Slightly Yellowish Granules Or Powder SolidMolecular weight:420.43N6-Ethyladenosine
CAS:<p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>Formula:C12H17N5O4Purity:99.96%Color and Shape:SolidMolecular weight:295.29Acefylline
CAS:<p>Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.</p>Formula:C9H10N4O4Purity:99.57%Color and Shape:White Crystalline SolidMolecular weight:238.2CGS 15943
CAS:<p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>Formula:C13H8ClN5OPurity:97.4%Color and Shape:SolidMolecular weight:285.69N6-Cyclohexyladenosine
CAS:<p>N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.</p>Formula:C16H23N5O4Purity:99.84% - 99.98%Color and Shape:SolidMolecular weight:349.38A3AR agonist 2
<p>Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.</p>Formula:C34H34N6O6Purity:98%Color and Shape:SolidMolecular weight:622.67Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Formula:C12H14ClN5O2SeColor and Shape:SolidMolecular weight:374.68hA3AR agonist 2
<p>hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.</p>Formula:C11H14ClN5O2SColor and Shape:SolidMolecular weight:315.78Xanthine amine congener dihydrochloride
CAS:<p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>Formula:C21H30Cl2N6O4Color and Shape:SolidMolecular weight:501.41Heterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Formula:C86H115FN16O21Color and Shape:SolidMolecular weight:1727.93LUF6096
CAS:<p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>Formula:C22H21Cl2N3OPurity:99.5%Color and Shape:SolidMolecular weight:414.33ABT-702
CAS:<p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>Formula:C22H19BrN6OPurity:99.57%Color and Shape:SoildMolecular weight:463.33Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Formula:C25H31F3N6O8Purity:98.08%Color and Shape:SoildMolecular weight:600.558-Chloro caffeine
CAS:<p>8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.</p>Formula:C8H9ClN4O2Color and Shape:SolidMolecular weight:228.64PSB 0777 ammonium hydrate
<p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>Formula:C18H20N5O7S2·NH4·75H2OPurity:98%Color and Shape:SolidMolecular weight:532.09A3AR agonist 1
<p>A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective</p>Formula:C28H34N6O6Purity:98%Color and Shape:SolidMolecular weight:550.61AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Formula:C21H25N5Color and Shape:SolidMolecular weight:347.211PSB 0777 ammonium salt
CAS:<p>adenosine A2A receptor full agonist</p>Formula:C18H24N6O7S2Purity:98%Color and Shape:SolidMolecular weight:500.55MRS-1706
CAS:<p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>Formula:C27H29N5O5Purity:99.00%Color and Shape:SolidMolecular weight:503.55N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:<p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>Formula:C19H22N6O4Color and Shape:SolidMolecular weight:398.42Norisoboldine hydrochloride
CAS:<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Formula:C18H20ClNO4Color and Shape:SolidMolecular weight:349.81FSCPX
CAS:<p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>Formula:C23H27FN4O6SPurity:98%Color and Shape:SolidMolecular weight:506.55Xanthine amine congener trihydrochloride
CAS:<p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>Formula:C21H29ClN6O4Purity:98.81%Color and Shape:SolidMolecular weight:464.95Danshenol B
<p>Danshenol B is a natural product that can be used as a reference standard.</p>Formula:C22H26O4Color and Shape:SolidMolecular weight:354.4463F6-9G5
<p>3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.</p>Purity:>95%Color and Shape:Odour LiquidTheophyllol
CAS:<p>Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.</p>Formula:C9H10N4Na2O4Color and Shape:SolidMolecular weight:284.18Adenosine receptor antagonist 1
CAS:<p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>Formula:C22H15ClFN7OColor and Shape:SolidMolecular weight:447.86LUF7690
CAS:<p>LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and</p>Formula:C25H24FN5O6SColor and Shape:SolidMolecular weight:541.55A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Formula:C23H25IN4Color and Shape:SolidMolecular weight:484.38A-286501
CAS:<p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>Formula:C11H14BrN5O2Purity:98%Color and Shape:SolidMolecular weight:328.17GW-328267
CAS:<p>GW-328267 is an agonist of the adenosine A2 receptor.</p>Formula:C21H26N10O4Color and Shape:SolidMolecular weight:482.5A2A/A3 AR antagonist-1
<p>A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).</p>Formula:C56H71N15O12S2Color and Shape:SolidMolecular weight:1210.39LAS101057
CAS:<p>LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.</p>Formula:C18H14FN5OPurity:99.03% - >99.99%Color and Shape:SolidMolecular weight:335.34(Rac)-Mirabegron-d5
CAS:<p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>Formula:C21H24N4O2SPurity:98%Color and Shape:SolidMolecular weight:401.54GR79236
CAS:<p>GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.</p>Formula:C15H21N5O5Color and Shape:SolidMolecular weight:351.36MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Formula:C17H19N5OC2H2O4Purity:97.10%Color and Shape:SolidMolecular weight:354.39
