Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 249 products of "Adenosine Receptor"
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Amp579 TFA
Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.Formula:C24H29ClF3N5O5SPurity:97.91%Color and Shape:SoildMolecular weight:592.03Pentoxifylline
CAS:Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.Formula:C13H18N4O3Purity:99.26% - 99.93%Color and Shape:SolidMolecular weight:278.31Adenosine 5'-monophosphate monohydrate
CAS:Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.
Formula:C10H14N5O7P·H2OPurity:97.68% - 98.49%Color and Shape:White PowderMolecular weight:365.24Ticlopidine hydrochloride
CAS:Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.Formula:C14H15Cl2NSPurity:99.85% - >99.99%Color and Shape:White PowderMolecular weight:300.25Aminophylline
CAS:Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.Formula:C7H8O2·C2H8N2Purity:99.31%Color and Shape:White Or Slightly Yellowish Granules Or Powder SolidMolecular weight:420.43AB928
CAS:AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].Formula:C23H22N8OPurity:98.09% - >99.99%Color and Shape:SolidMolecular weight:426.47Ref: TM-T14078
1mg52.00€5mg117.00€10mg187.00€25mg369.00€50mg437.00€100mg628.00€1mL*10mM (DMSO)127.00€YT 146
CAS:YT 146 is a biochemical.Formula:C18H25N5O4Purity:98.81% - 99.25%Color and Shape:SolidMolecular weight:375.42CGS 15943
CAS:CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.Formula:C13H8ClN5OPurity:97.4%Color and Shape:SolidMolecular weight:285.69Ref: TM-T14944
2mg34.00€5mg50.00€10mg82.00€25mg147.00€50mg222.00€100mg334.00€200mg494.00€1mL*10mM (DMSO)55.00€Doxofylline
CAS:Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Formula:C11H14N4O4Purity:99.958% - >99.99%Color and Shape:SolidMolecular weight:266.25Theophylline
CAS:Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and centralFormula:C7H8N4O2Purity:99.65% - 99.98%Color and Shape:White Solid PowderMolecular weight:180.16DPTN dihydrochloride
CAS:DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Formula:C22H20Cl2N4OSPurity:99.95%Color and Shape:SoildMolecular weight:459.39Quercetin-3'-o-phosphate TEA
Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.Formula:C21H26NO10PPurity:97.04%Color and Shape:SoildMolecular weight:483.41Adenosine A1 receptor activator T62
CAS:Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and alsoFormula:C15H14ClNOSPurity:97.83%Color and Shape:SolidMolecular weight:291.8Ref: TM-T14127
1mg64.00€5mg126.00€10mg180.00€25mg290.00€50mg396.00€100mg537.00€200mg712.00€1mL*10mM (DMSO)187.00€Theophylline monohydrate
CAS:Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calciumFormula:C7H8N4O2·H2OPurity:99.78%Color and Shape:SolidMolecular weight:198.18N6-Ethyladenosine
CAS:N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).Formula:C12H17N5O4Purity:99.96%Color and Shape:SolidMolecular weight:295.29Pamabrom
CAS:Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.Formula:C11H18BrN5O3Purity:99.84% - >99.99%Color and Shape:CoaMolecular weight:348.2N6-Cyclohexyladenosine
CAS:N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.Formula:C16H23N5O4Purity:99.92% - 99.98%Color and Shape:SolidMolecular weight:349.38Diphylline
CAS:Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.Formula:C10H14N4O4Purity:98.54%Color and Shape:Crystals From Alcohol SolidMolecular weight:254.24Acefylline
CAS:Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.Formula:C9H10N4O4Purity:99.57%Color and Shape:White Crystalline SolidMolecular weight:238.2A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effectiveFormula:C28H34N6O6Purity:98%Color and Shape:SolidMolecular weight:550.61Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Formula:C12H14ClN5O2SeColor and Shape:SolidMolecular weight:374.68A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.Formula:C34H34N6O6Purity:98%Color and Shape:SolidMolecular weight:622.67Xanthine amine congener dihydrochloride
CAS:XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.Formula:C21H30Cl2N6O4Color and Shape:SolidMolecular weight:501.41LUF6096
CAS:LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormula:C22H21Cl2N3OPurity:99.5%Color and Shape:SolidMolecular weight:414.33ABT-702
CAS:ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.Formula:C22H19BrN6OPurity:99.57%Color and Shape:SoildMolecular weight:463.33FSCPX
CAS:FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.Formula:C23H27FN4O6SPurity:99.4%Color and Shape:SolidMolecular weight:506.55Ref: TM-T39039
1mg82.00€5mg180.00€10mg271.00€25mg460.00€50mg617.00€100mg825.00€200mg1,108.00€1mL*10mM (DMSO)86.00€Norisoboldine hydrochloride
CAS:Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.Formula:C18H20ClNO4Color and Shape:SolidMolecular weight:349.818-Chloro caffeine
CAS:8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.Formula:C8H9ClN4O2Color and Shape:SolidMolecular weight:228.64hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Formula:C11H14ClN5O2SColor and Shape:SolidMolecular weight:315.78PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormula:C18H20N5O7S2·NH4·75H2OPurity:98%Color and Shape:SolidMolecular weight:532.09AR ligand 40
AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.Formula:C21H25N5Color and Shape:SolidMolecular weight:347.211PSB 0777 ammonium salt
CAS:adenosine A2A receptor full agonistFormula:C18H24N6O7S2Purity:98%Color and Shape:SolidMolecular weight:500.55MRS-1706
CAS:MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.Formula:C27H29N5O5Purity:99.00%Color and Shape:SolidMolecular weight:503.55Ref: TM-T16136
1mg34.00€5mg74.00€10mg113.00€25mg222.00€50mg356.00€100mg572.00€200mg803.00€1mL*10mM (DMSO)84.00€A3AR modulator 1
MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.Formula:C23H25IN4Color and Shape:SolidMolecular weight:484.38GW-328267
CAS:GW-328267 is an agonist of the adenosine A2 receptor.Formula:C21H26N10O4Color and Shape:SolidMolecular weight:482.5Xanthine amine congener trihydrochloride
CAS:Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formula:C21H29ClN6O4Purity:98.81%Color and Shape:SolidMolecular weight:464.95Danshenol B
Danshenol B is a natural product that can be used as a reference standard.Formula:C22H26O4Color and Shape:SolidMolecular weight:354.446A-286501
CAS:A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.Formula:C11H14BrN5O2Purity:98%Color and Shape:SolidMolecular weight:328.17Theophyllol
CAS:Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.Formula:C9H10N4Na2O4Color and Shape:SolidMolecular weight:284.18Adenosine receptor antagonist 1
CAS:A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.Formula:C22H15ClFN7OColor and Shape:SolidMolecular weight:447.863F6-9G5
3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.Purity:>95%Color and Shape:Odour LiquidMolecular weight:146.66 kDaN6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formula:C19H22N6O4Color and Shape:SolidMolecular weight:398.42Heterobivalent ligand-1
Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.Formula:C86H115FN16O21Color and Shape:SolidMolecular weight:1727.93LUF7690
CAS:LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection andFormula:C25H24FN5O6SColor and Shape:SolidMolecular weight:541.55Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.
Formula:C25H31F3N6O8Purity:98.08%Color and Shape:SoildMolecular weight:600.55A2A/A3 AR antagonist-1
A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).Formula:C56H71N15O12S2Color and Shape:SolidMolecular weight:1210.39GR79236
CAS:GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.Formula:C15H21N5O5Color and Shape:SolidMolecular weight:351.36(Rac)-Mirabegron-d5
CAS:(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.Formula:C21H24N4O2SPurity:98%Color and Shape:SolidMolecular weight:401.54LAS101057
CAS:LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.Formula:C18H14FN5OPurity:99.03% - >99.99%Color and Shape:SolidMolecular weight:335.34Theophylline-d6
CAS:Theophylline-d6, an internal standard for theophylline quantification in GC/LC-MS, relaxes bronchial muscles and treats asthma/COPD.Formula:C7H2D6N4O2Color and Shape:SolidMolecular weight:186.2
