Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 249 products of "Adenosine Receptor"
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KFM19
CAS:KFM19 is a potent and selective adenosine receptor (A1-receptor) antagonist (IC50 : 50 nM) for the study of neurological disorders.Formula:C16H22N4O3Purity:98.62%Color and Shape:SolidMolecular weight:318.37MRS3558
CAS:MRS3558 is an agonist of A3 adenosine receptors.Formula:C20H20Cl2N6O3Color and Shape:SolidMolecular weight:463.32GP3269
CAS:GP3269 is a selective, potent, orally active human adenosine kinase (AK) inhibitor (IC50: 11 nM) with anticonvulsant effects in rats.Formula:C23H21FN4O3Color and Shape:SolidMolecular weight:420.44Sulmazole
CAS:Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.Formula:C14H13N3O2SPurity:99.94%Color and Shape:SolidMolecular weight:287.34Xanthine amine congener
CAS:Xanthine amine congener is an Adenosine receptor antagonist.Formula:C21H28N6O4Purity:99.7%Color and Shape:SolidMolecular weight:428.48PSB-10 hydrochloride
CAS:PSB-10 hydrochloride is a human adenosine A3 receptor antagonist.Formula:C16H15Cl4N5OPurity:98%Color and Shape:SolidMolecular weight:435.14MSX-2
CAS:MSX-2 is an A2A adenosine receptor antagonist.Formula:C21H22N4O4Purity:98%Color and Shape:SolidMolecular weight:394.42MNI-444
CAS:MNI-444 is a PET radiotracer for adenosine 2A receptors.Formula:C24H26FN9O2Color and Shape:SolidMolecular weight:491.52KF21213
CAS:KF21213 shows a high affinity for the adenosine A2A receptors (Ki=3.0 nM). KF21213 is a highly selective ligand for mapping CNS adenosine A2A receptors.Formula:C19H22N4O3Purity:98%Color and Shape:SolidMolecular weight:354.4ATL802
CAS:ATL802 is an adenosine A2B Receptor antagonist.Formula:C24H22F3N7O3Purity:98%Color and Shape:SolidMolecular weight:513.47MRS5698
CAS:MRS5698, an A3 adenosine receptor agonist with Ki ~3 nM, blocks chronic pain, highly selective (>1000-fold over A1/A2A).Formula:C28H23ClF2N6O3Purity:98%Color and Shape:SolidMolecular weight:564.97ST4206
CAS:ST4206 is an antagonist of adenosine A2A. For adenosine A2A receptor and adenosine A1 receptor, the Kis values are 12 nM and 197 nM , respectively.Formula:C12H14N8OPurity:98%Color and Shape:SolidMolecular weight:286.29A1/A3 AR antagonist 3
CAS:A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful inFormula:C22H19N5O3Purity:98%Color and Shape:SolidMolecular weight:401.42PF-02575799
CAS:PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).Formula:C42H37FN4O4Purity:98%Color and Shape:SolidMolecular weight:680.77PSB 0788
CAS:adenosine A2B receptor antagonistFormula:C25H27ClN6O4SPurity:98%Color and Shape:SolidMolecular weight:543.04CGS 21680
CAS:CGS 21680 is a chemical compound that acts as a selective agonist for both adenosine and its A2A receptor, demonstrating a binding affinity (K i) of 27 nM.Formula:C23H29N7O6Color and Shape:SolidMolecular weight:499.52Dansyl-NECA
CAS:Dansyl-NECA is a selective agonist of fluorescent adenosine A1 receptor.Formula:C30H40N8O6SColor and Shape:SolidMolecular weight:640.75PSB-1901 free base
CAS:PSB-1901: potent A2B Adenosine Receptor Antagonist; Ki=0.0835 nM; >10,000x selective; effective in mice for preclinical studies.Formula:C24H25BrN6O4SColor and Shape:SolidMolecular weight:573.46CV1808
CAS:CV-1808 is a coronary vasodilator, antihypertensive, and antipsychotic following systemic administration in vivo. CV-1808 is an adenosine A2 receptor agonist.Formula:C16H18N6O4Color and Shape:Off-White To Pale Yellow SolidMolecular weight:358.35GS-6201
CAS:GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.Formula:C21H21F3N6O2Purity:99.78% - 99.94%Color and Shape:SolidMolecular weight:446.43Ref: TM-T15418
1mg34.00€5mg71.00€10mg114.00€25mg235.00€50mg380.00€100mg572.00€200mg805.00€1mL*10mM (DMSO)78.00€MRS 1754
CAS:MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
Formula:C26H26N6O4Purity:97.57% - 99.3%Color and Shape:SolidMolecular weight:486.52ABT-702 hydrochloride
CAS:ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].Formula:C22H20BrClN6OColor and Shape:SolidMolecular weight:499.79PSB-1115 potassium salt
CAS:PSB-1115 potassium salt, a selective A2B Adenosine Receptor antagonist, inhibits the 2,4,6-trinitrobenzenesulfonic acid (TNBS)-induced contraction inhibition of acetylcholine (ACh) [1].Formula:C14H13KN4O5SColor and Shape:SolidMolecular weight:388.44A2B receptor antagonist 1
CAS:A2B receptor antagonist 1 (EXAMPLE 9B) is a potent A2B adenosine receptor antagonist.Formula:C21H24N6O2Purity:99.53%Color and Shape:SolidMolecular weight:392.45Ref: TM-T10058
1mg349.00€5mg697.00€10mg888.00€25mg1,395.00€50mg1,783.00€100mg2,530.00€1mL*10mM (DMSO)800.00€PSB-603
CAS:PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.
Formula:C24H25ClN6O4SPurity:97.13%Color and Shape:SolidMolecular weight:529.01PSB 1115
CAS:PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.Formula:C14H14N4O5SPurity:98.69% - >99.99%Color and Shape:SolidMolecular weight:350.35LJ-4517
LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.Formula:C19H21N5O3SColor and Shape:SolidMolecular weight:399.47Zaladenant
CAS:Zaladenant is an adenosine receptor antagonist with antitumor properties.Formula:C19H15F3N6OColor and Shape:SolidMolecular weight:400.357M1069
M1069 is an oral A2A/A2B receptor antagonist, 100x more selective over A1/A3, with antitumor properties by blocking adenosine's immunosuppressive effects.Formula:C25H30N4O8SColor and Shape:SolidMolecular weight:546.59CVT-5440
CAS:CVT-5440 is a selective, high-affinity (2B) adenosine receptor antagonist with good selectivity.Formula:C27H28N6O5Color and Shape:SolidMolecular weight:516.55A1AR antagonist 1
Compound 18g, a potent A1AR blocker with Ki: 2.08 nM (hA1), 6.91 nM (hA2A), 31.2 nM (hA2B).Formula:C18H14N4OColor and Shape:SolidMolecular weight:302.33DMPX
CAS:DMPX (3,7-Dimethyl-1-propargylxanthine) is a caffeine-like compound capable of crossing the blood-brain barrier. It serves as an A2-selective adenosine receptor (AR) antagonist, effectively and selectively blocking the hypothermia and behavioral inhibition induced by A2 adenosine receptor agonists, such as NECA. DMPX is utilized in research on diseases like Parkinson's disease.Formula:C10H10N4O2Color and Shape:SolidMolecular weight:218.212A3AR antagonist 5
CAS:A3AR antagonist 5 (Compound 16) acts as a selective antagonist for the human adenosine A3 receptor (human adenosine A3 receptor), with an affinity expressed as a pC value of 4.542 μM.Formula:C18H16N2O2SColor and Shape:SolidMolecular weight:324.40ADORA2A/PDE4D-IN-1
CAS:ADORA2A/PDE4D-IN-1 (Compound 9) is a dual inhibitor of the adenosine A2a receptor (ADORA2A) and phosphodiesterase 4D (PDE4D). This compound is applicable for research in bronchial asthma.Formula:C14H11N5Color and Shape:SolidMolecular weight:249.271UK-432097
CAS:UK 432097 is an adenosine A2A agonist.Formula:C40H47N11O6Color and Shape:SolidMolecular weight:777.87MSX-3
CAS:MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2.Formula:C21H23N4Na2O7PPurity:98%Color and Shape:SolidMolecular weight:520.389YGZ-331
CAS:YGZ-331, a sedative hypnotic, acts by elevating GABA levels as a derivative of the adenosine nucleoside NGBA. It functions through activating A1R and A2aR, and inhibiting the phosphorylation of CaMKII (pCaMKII), thereby exerting its calming effects. Additionally, YGZ-331 reduces spontaneous motor activity in mice.Formula:C19H23N5O4Color and Shape:SolidMolecular weight:385.42CP-608039
CAS:CP-608039 is a selective adenosine A3 receptor agonist for both human A3 and human A1 receptors.Formula:C23H25ClN8O5Color and Shape:SolidMolecular weight:528.95Tonapofylline
CAS:Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Formula:C22H32N4O4Purity:98.57%Color and Shape:SolidMolecular weight:416.51MRS7799
CAS:MRS7799 is a selective A3 Adenosine Receptor antagonist with Kd values of 0.55 nM for humans, 3.74 nM for mice, and 2.80 nM for rats. MRS7799 can be utilized in research related to neurodegenerative diseases, cancer, cardiac and cerebral ischemia, and autoimmune inflammatory diseases.Formula:C22H18N4OSColor and Shape:SolidMolecular weight:386.47hA3AR agonist 1
hA3AR agonist 1 is a potent human A 3 adenosine receptor (hA 3 AR) agonist (Ki = 2.40 nM) .Formula:C10H14N6OSColor and Shape:SolidMolecular weight:266.32A1/A3 AR antagonist 1
Compound 10 is a potent dual A1/A3 AR antagonist, with Ki values of 37.6 nM (hA1), 25.4 nM (hA3), and 1.47 nM (rA1), studied in renal, lung, and Alzheimer's.
Formula:C24H18N2O3SColor and Shape:SolidMolecular weight:414.48PSB 36
CAS:A1 adenosine receptor antagonistFormula:C21H30N4O3Purity:98%Color and Shape:SolidMolecular weight:386.49L-97-1
CAS:L-97-1 is an antagonist of the adenosine A1 receptor.Formula:C29H38N6O3Purity:98%Color and Shape:SolidMolecular weight:518.65KF26777
CAS:KF26777 is a potent and selective antagonist of adenosine A3 receptor.Formula:C16H16BrN5OPurity:98%Color and Shape:SolidMolecular weight:374.23Neladenoson
CAS:Neladenoson is an effective and selective agonist of the Adenosine A1 Receptor (A1R). EGFR-IN-162 shows potential for research in heart failure.Formula:C29H24ClN5O2S2Color and Shape:SolidMolecular weight:574.12Inupadenant HCl
CAS:Inupadenant (EOS-850) is a selective A2a receptor antagonist, targeting immunosuppression in tumors.Formula:C25H27ClF2N8O4S2Color and Shape:SolidMolecular weight:641.11ATL444
CAS:ATL444 is an adenosine receptor antagonist with affinity (Ki values) for rA1AR, rA2AAR, rA2BAR, and rA3AR of 7.0, 2.5, 61.8, and >1000 nM, respectively.Formula:C17H19N5OColor and Shape:SolidMolecular weight:309.37A2A receptor antagonist 2
A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).Formula:C25H28FN7O3Color and Shape:SolidMolecular weight:493.53
