Adenosine Receptor
Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.
Found 249 products of "Adenosine Receptor"
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Inupadenant
CAS:Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].Formula:C25H26F2N8O4S2Color and Shape:SolidMolecular weight:604.65CAY10680
CAS:CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.Formula:C18H16N2O2SColor and Shape:SolidMolecular weight:324.4FR-194921
CAS:FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.Formula:C23H23N5OColor and Shape:SolidMolecular weight:385.46CVT-2759
CAS:CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.Formula:C17H24N6O6Color and Shape:SolidMolecular weight:408.41Adenosine receptor inhibitor 2
CAS:Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.Formula:C17H20BrN5O2Color and Shape:SolidMolecular weight:406.28Acefylline piperazine
CAS:Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.Formula:C9H10N4O4·xC4H10N2Color and Shape:SolidMolecular weight:562.54JNJ-40255293
CAS:JNJ-40255293 is an antagonist of adenosine A2A/A1.Formula:C23H22N4O3Purity:98%Color and Shape:SolidMolecular weight:402.45AK-IN-1
CAS:AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.Formula:C22H21N3O4Color and Shape:SolidMolecular weight:391.42ATL-801
CAS:ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.Formula:C24H25N7O3Color and Shape:SolidMolecular weight:459.5Kira8 Hydrochloride
CAS:Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.Formula:C31H30Cl2N6O3SPurity:98%Color and Shape:SolidMolecular weight:637.58A2AAR/HDAC-IN-2
CAS:A2AAR/HDAC-IN-2: potent dual A2AAR/HDAC inhib., Ki 10.3 nM, IC50 18.5 nM, anti-tumor potential.Formula:C23H26N6O4Color and Shape:SolidMolecular weight:450.49Theophylline sodium glycinate
CAS:Theophylline sodium glycinate inhibits PDE3, treats asthma/COPD, blocks adenosine receptors, activates HDAC, reduces inflammation and induces apoptosis.Formula:C9H12N5NaO4Color and Shape:SolidMolecular weight:277.216hA2AAR antagonist 1
CAS:Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.Formula:C15H15N5OColor and Shape:SolidMolecular weight:281.31LUF5831
CAS:LUF5831 is an agonist of adenosine A1 receptor.Formula:C15H12N4O2SColor and Shape:SolidMolecular weight:312.35Draflazine
CAS:Draflazine: ENT1 inhibitor, reverses hypersensitivity in CFA and carrageenan-induced hyperalgesia.Formula:C30H33Cl2F2N5O2Purity:98%Color and Shape:SolidMolecular weight:604.52LUF5981
CAS:LUF5981 is a selective agonist of human adenosine A1 receptor.Formula:C24H23N3Color and Shape:SolidMolecular weight:353.46Cirazoline hydrochloride
CAS:Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.Formula:C13H17ClN2OPurity:99.863%Color and Shape:SolidMolecular weight:252.74Bamifylline Hydrochloride
CAS:Bamifylline Hydrochloride, an adenosine A1 receptor antagonist, is uesd to treat bronchiectasis and chronic obstructive pulmonary disease.Formula:C20H28ClN5O3Color and Shape:SolidMolecular weight:421.92MRS1067
CAS:MRS1067 is an antagonist of A3 adenosine receptor.Formula:C19H16Cl2O3Color and Shape:SolidMolecular weight:363.23VUF8504
CAS:VUF8504 is a novel ligand of adenosine A3 receptor.Formula:C22H17N3O2Color and Shape:SolidMolecular weight:355.39WRC-0571
CAS:WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.Formula:C17H26N6OPurity:98%Color and Shape:SolidMolecular weight:330.43Naxifylline
CAS:Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.Formula:C18H24N4O3Color and Shape:SolidMolecular weight:344.41CP 66713
CAS:CP-66713 is an adenosine A2 receptor antagonist.Formula:C15H10ClN5Color and Shape:SolidMolecular weight:295.73A2AAR antagonist 1
CAS:Compound 21a, A2AAR antagonist with 20 nM Ki, useful in neurodegenerative disease study.Formula:C12H8BrN3OColor and Shape:SolidMolecular weight:290.12MRE3008F20
CAS:MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.Formula:C21H20N8O3Purity:97.29%Color and Shape:SolidMolecular weight:432.44A2AR-antagonist-1
CAS:Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.Formula:C27H25N5O2Purity:98%Color and Shape:SolidMolecular weight:451.52VUF 5574
CAS:VUF 5574 is a selective antagonist of adenosine A3 receptor with a Ki of 4.03 nM for the recombinant human receptor.Formula:C21H17N5O2Purity:99.53%Color and Shape:SolidMolecular weight:371.39ST3932
CAS:ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Formula:C12H16N8OPurity:98%Color and Shape:SolidMolecular weight:288.31N6-Cyclopentyladenosine
CAS:N6-Cyclopentyladenosine (CPA) is a selective agonist of the adenosine A1 receptor and can be used to mimic the action of the adenosine A1 receptor, with Ki's ofFormula:C15H21N5O4Purity:99.95%Color and Shape:SolidMolecular weight:335.36N-[(4-Aminophenyl)methyl]adenosine
CAS:N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Formula:C17H20N6O4Purity:98.75%Color and Shape:SolidMolecular weight:372.38Ref: TM-T16166
1mg52.00€5mg111.00€10mg166.00€25mg318.00€50mg504.00€100mg803.00€1mL*10mM (DMSO)141.00€Sonedenoson
CAS:Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.Formula:C18H20ClN5O5Purity:99.79%Color and Shape:SolidMolecular weight:421.84KI-7
CAS:KI-7 is an adenosine A2B receptor positive allosteric modulator.Formula:C23H18N2O2Purity:98.33%Color and Shape:SolidMolecular weight:354.4Ref: TM-T9238
2mg35.00€5mg55.00€10mg95.00€25mg172.00€50mg264.00€100mg399.00€200mg560.00€1mL*10mM (DMSO)62.00€Adenosine antagonist-1
CAS:Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
Formula:C18H13N7SPurity:99.28% - 99.95%Color and Shape:SolidMolecular weight:359.41BAY 60-6583
CAS:BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3Formula:C19H17N5O2SPurity:98.46% - 99.8%Color and Shape:SolidMolecular weight:379.44Ref: TM-T14506
1mg39.00€2mg50.00€5mg84.00€10mg116.00€25mg233.00€50mg376.00€100mg567.00€200mg797.00€1mL*10mM (DMSO)101.00€GW-493838
CAS:GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgiaFormula:C21H21ClFN7O4Purity:99.11% - 99.58%Color and Shape:SolidMolecular weight:489.89Ref: TM-T27509
1mg143.00€5mg346.00€10mg492.00€25mg740.00€50mg999.00€100mg1,350.00€500mg2,647.00€1mL*10mM (DMSO)399.00€ST-1535
CAS:ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.Formula:C12H16N8Purity:99.64% - 99.69%Color and Shape:SolidMolecular weight:272.31N6-(2-Phenylethyl)adenosine
CAS:N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM forFormula:C18H21N5O4Purity:99.83%Color and Shape:SolidMolecular weight:371.39A2A receptor antagonist 1
CAS:A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.Formula:C16H12FN5OPurity:99.52% - 99.93%Color and Shape:SolidMolecular weight:309.3Ref: TM-T37792
2mgTo inquire5mg62.00€10mg87.00€25mg183.00€50mg280.00€100mg416.00€200mgTo inquire1mL*10mM (DMSO)47.00€N 0861
CAS:N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formula:C13H17N5Purity:98.78%Color and Shape:SolidMolecular weight:243.31Ref: TM-T70722
1mg164.00€2mg234.00€5mg389.00€10mg532.00€25mg820.00€50mg1,063.00€100mg1,423.00€200mg1,945.00€ANR 94
CAS:ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.Formula:C9H13N5OPurity:98.9%Color and Shape:SolidMolecular weight:207.23Ref: TM-T22031
5mg46.00€10mg71.00€25mg130.00€50mg219.00€100mg309.00€200mg434.00€1mL*10mM (DMSO)46.00€ISAM-140
CAS:ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.Formula:C19H19N3O3Purity:99.51%Color and Shape:SolidMolecular weight:337.37GS-9667
CAS:GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia viaFormula:C21H24FN5O4SPurity:99.77% - 99.96%Color and Shape:SolidMolecular weight:461.51APNEA
CAS:APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Formula:C18H22N6O4Purity:99.88%Color and Shape:SolidMolecular weight:386.41LAS38096
CAS:LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .Formula:C17H12N6OPurity:99.18% - 99.95%Color and Shape:SolidMolecular weight:316.32Evodenoson
CAS:Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.Formula:C23H29N7O6Purity:99.75% - 99.83%Color and Shape:SolidMolecular weight:499.52MRS1220
CAS:MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeuticFormula:C21H14ClN5O2Purity:98.43%Color and Shape:SolidMolecular weight:403.822'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formula:C16H22ClN5O4Purity:99.93%Color and Shape:SolidMolecular weight:383.83FK-453
CAS:FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.Formula:C23H25N3O2Purity:99.44%Color and Shape:SolidMolecular weight:375.46Selodenoson
CAS:Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.Formula:C17H24N6O4Purity:99.39%Color and Shape:SolidMolecular weight:376.41Neladenoson dalanate
CAS:Neladenoson dalanate (BAY-1067197), an oral Adenosine A1 receptor partial agonist, is safe with good pharmacokinetics for chronic heart disease.Formula:C35H34ClN7O4S2Color and Shape:SolidMolecular weight:716.27
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