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Adenosine Receptor

Adenosine Receptor

Adenosine receptors are a class of GPCRs that respond to the endogenous nucleoside adenosine. These receptors are involved in regulating various physiological processes, including cardiovascular function, sleep-wake cycles, and immune responses. Adenosine receptor modulators have therapeutic potential in treating conditions such as cardiac arrhythmias, inflammation, and neurodegenerative diseases. At CymitQuimica, we provide a selection of high-quality adenosine receptor modulators to support your research in cardiovascular biology, neuroscience, and immunology.

Found 242 products of "Adenosine Receptor"

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  • L-97-1
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    L-97-1

    CAS:
    <p>L-97-1 is an antagonist of the adenosine A1 receptor.</p>
    Formula:C29H38N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.65

    Ref: TM-T24384

  • CVT-5440
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    CVT-5440

    CAS:
    <p>CVT-5440 is a selective, high-affinity (2B) adenosine receptor antagonist with good selectivity.</p>
    Formula:C27H28N6O5
    Color and Shape:Solid
    Molecular weight:516.55

    Ref: TM-T31122

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    A1AR antagonist 1

    <p>Compound 18g, a potent A1AR blocker with Ki: 2.08 nM (hA1), 6.91 nM (hA2A), 31.2 nM (hA2B).</p>
    Formula:C18H14N4O
    Color and Shape:Solid
    Molecular weight:302.33

    Ref: TM-T60687

  • DMPX
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    DMPX

    CAS:
    <p>DMPX (3,7-Dimethyl-1-propargylxanthine) is a caffeine-like compound capable of crossing the blood-brain barrier. It serves as an A2-selective adenosine receptor (AR) antagonist, effectively and selectively blocking the hypothermia and behavioral inhibition induced by A2 adenosine receptor agonists, such as NECA. DMPX is utilized in research on diseases like Parkinson's disease.</p>
    Formula:C10H10N4O2
    Color and Shape:Solid
    Molecular weight:218.212

    Ref: TM-T204595

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    A2A receptor antagonist 2

    <p>A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).</p>
    Formula:C25H28FN7O3
    Color and Shape:Solid
    Molecular weight:493.53

    Ref: TM-T63326

  • ADORA2A/PDE4D-IN-1
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    ADORA2A/PDE4D-IN-1

    CAS:
    <p>ADORA2A/PDE4D-IN-1 (Compound 9) is a dual inhibitor of the adenosine A2a receptor (ADORA2A) and phosphodiesterase 4D (PDE4D). This compound is applicable for research in bronchial asthma.</p>
    Formula:C14H11N5
    Color and Shape:Solid
    Molecular weight:249.271

    Ref: TM-T204528

  • PSB 36
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    PSB 36

    CAS:
    <p>A1 adenosine receptor antagonist</p>
    Formula:C21H30N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.49

    Ref: TM-T23202

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    LJ-4517

    <p>LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.</p>
    Formula:C19H21N5O3S
    Color and Shape:Solid
    Molecular weight:399.47

    Ref: TM-T61914

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    M1069

    <p>M1069 is an oral A2A/A2B receptor antagonist, 100x more selective over A1/A3, with antitumor properties by blocking adenosine's immunosuppressive effects.</p>
    Formula:C25H30N4O8S
    Color and Shape:Solid
    Molecular weight:546.59

    Ref: TM-T63856

  • UK-432097
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    UK-432097

    CAS:
    <p>UK 432097 is an adenosine A2A agonist.</p>
    Formula:C40H47N11O6
    Color and Shape:Solid
    Molecular weight:777.87

    Ref: TM-T29049

  • YGZ-331
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    YGZ-331

    CAS:
    <p>YGZ-331, a sedative hypnotic, acts by elevating GABA levels as a derivative of the adenosine nucleoside NGBA. It functions through activating A1R and A2aR, and inhibiting the phosphorylation of CaMKII (pCaMKII), thereby exerting its calming effects. Additionally, YGZ-331 reduces spontaneous motor activity in mice.</p>
    Formula:C19H23N5O4
    Color and Shape:Solid
    Molecular weight:385.42

    Ref: TM-T200016

  • CP-608039
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    CP-608039

    CAS:
    <p>CP-608039 is a selective adenosine A3 receptor agonist for both human A3 and human A1 receptors.</p>
    Formula:C23H25ClN8O5
    Color and Shape:Solid
    Molecular weight:528.95

    Ref: TM-T31068

  • Neladenoson
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    Neladenoson

    CAS:
    <p>Neladenoson is an effective and selective agonist of the Adenosine A1 Receptor (A1R). EGFR-IN-162 shows potential for research in heart failure.</p>
    Formula:C29H24ClN5O2S2
    Color and Shape:Solid
    Molecular weight:574.12

    Ref: TM-T207262

  • MRS7799
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    MRS7799

    CAS:
    <p>MRS7799 is a selective A3 Adenosine Receptor antagonist with Kd values of 0.55 nM for humans, 3.74 nM for mice, and 2.80 nM for rats. MRS7799 can be utilized in research related to neurodegenerative diseases, cancer, cardiac and cerebral ischemia, and autoimmune inflammatory diseases.</p>
    Formula:C22H18N4OS
    Color and Shape:Solid
    Molecular weight:386.47

    Ref: TM-T206672

  • Tonapofylline
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    Tonapofylline

    CAS:
    <p>Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.</p>
    Formula:C22H32N4O4
    Purity:98.57%
    Color and Shape:Solid
    Molecular weight:416.51

    Ref: TM-T17117

  • A3AR antagonist 5
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    A3AR antagonist 5

    CAS:
    <p>A3AR antagonist 5 (Compound 16) acts as a selective antagonist for the human adenosine A3 receptor (human adenosine A3 receptor), with an affinity expressed as a pC value of 4.542 μM.</p>
    Formula:C18H16N2O2S
    Color and Shape:Solid
    Molecular weight:324.40

    Ref: TM-T200493

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    hA3AR agonist 1

    <p>hA3AR agonist 1 is a potent human A 3 adenosine receptor (hA 3 AR) agonist (Ki = 2.40 nM) .</p>
    Formula:C10H14N6OS
    Color and Shape:Solid
    Molecular weight:266.32

    Ref: TM-T60444

  • KF26777
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    KF26777

    CAS:
    <p>KF26777 is a potent and selective antagonist of adenosine A3 receptor.</p>
    Formula:C16H16BrN5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.23

    Ref: TM-T27729

  • MSX-3
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    MSX-3

    CAS:
    <p>MSX-3 is an antagonist of the A2A adenosine receptor and a prodrug of MSX-2.</p>
    Formula:C21H23N4Na2O7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:520.389

    Ref: TM-T25841

  • Inupadenant HCl
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    Inupadenant HCl

    CAS:
    <p>Inupadenant (EOS-850) is a selective A2a receptor antagonist, targeting immunosuppression in tumors.</p>
    Formula:C25H27ClF2N8O4S2
    Color and Shape:Solid
    Molecular weight:641.11

    Ref: TM-T69648