Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
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CB1R/AMPK modulator 1
Compound 38-S is an orally active CB1R/AMPK modulator with a K i of 0.81 nM …
Formula:
C25H22Cl2N6O3S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
557.45
Ref: TM-T79649
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
CB2R agonist 3
CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value …
Purity:
98%
Ref: TM-T82769
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
NESS 0327
CAS:494844-07-4
NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is …
Formula:
C24H23Cl3N4O
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
489.82
Ref: TM-T22114
| 1mg | 123.00 € | ||
| 5mg | 300.00 € | ||
| 10mg | 429.00 € | ||
| 25mg | 643.00 € | ||
| 50mg | 867.00 € | ||
| 100mg | 1,156.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Taranabant racemate
CAS:701977-00-6
Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.
Formula:
C27H25ClF3N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
515.95
Ref: TM-T13081
| 2mg | 50.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Falcarinol
CAS:21852-80-2
Falcarinol, also known as Panaxynol, is a naturally occurring compound that acts as an orally …
Formula:
C17H24O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
244.37
Ref: TM-TN2360
| 20mg | 410.00 € | ||
| 1mL*10mM (DMSO) | 199.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
CB1/2 agonist 3
CAS:2772655-86-2
CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 …
Formula:
C25H41NO2
Color and Shape:
Liquid
Molecular weight:
387.6
Ref: TM-T61736
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 301.00 € | ||
| 100mg | 447.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
L-α-lysophosphatidylinositol sodium
CAS:796963-91-2
L-α-lysophosphatidylinositol sodium is an endogenous ligand of GPR55 and an endocannabinoid neurotransmitter.
Formula:
C25H48NaO12P
Color and Shape:
Liquid
Molecular weight:
594.6
Ref: TM-T77212
| 1mg | 429.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Virodhamine
CAS:287937-12-6
Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of …
Formula:
C22H37NO2
Purity:
98%
Color and Shape:
Soild
Molecular weight:
347.53
Ref: TM-T64371
| 2mg | 52.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Linoleoyl Ethanolamide
CAS:68171-52-8
Linoleoyl Ethanolamide is an endocannabinoid agent.
Formula:
C20H37NO2
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
323.51
Ref: TM-T8425
| 1mg | 36.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 162.00 € | ||
| 50mg | 236.00 € | ||
| 100mg | 343.00 € | ||
| 200mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
β-Caryophyllene
CAS:87-44-5
β-Caryophyllene ((-)-(E)-Caryophyllene) acts as an CB2 receptor agonist.
Formula:
C15H24
Purity:
95.43% - 99.11%
Color and Shape:
Turpentine (Ntp 1992)
Molecular weight:
204.35
Ref: TM-T9114
| 500mg | 48.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
AM281
CAS:202463-68-1
AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and …
Formula:
C21H19Cl2IN4O2
Purity:
100% - 99.2%
Color and Shape:
White To Off-White Solid
Molecular weight:
557.21
Ref: TM-T2264
| 1mg | 84.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 546.00 € | ||
| 50mg | 782.00 € | ||
| 100mg | 1,079.00 € | ||
| 500mg | 2,135.00 € | ||
| 1mL*10mM (DMSO) | 242.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
N-Oleoyl glycine
CAS:2601-90-3
N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of …
Formula:
C20H37NO3
Purity:
99.92%
Color and Shape:
Solid
Molecular weight:
339.51
Ref: TM-T13803
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 147.00 € | ||
| 100mg | 213.00 € | ||
| 200mg | 318.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
yangonin
CAS:500-62-9
Yangonin (Y100550) is a novel CB1 receptor ligand with affinity for human recombinant CB1 receptors.
Formula:
C15H14O4
Purity:
98.82% - 99.55%
Color and Shape:
Pale Yellow Powder
Molecular weight:
258.27
Ref: TM-T3S0738
| 1mg | 69.00 € | ||
| 5mg | 133.00 € | ||
| 10mg | 202.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 507.00 € | ||
| 100mg | 721.00 € | ||
| 1mL*10mM (DMSO) | 176.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
AM-2232
CAS:335161-19-8
AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.
Formula:
C24H20N2O
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
352.43
Ref: TM-T21450
| 1mL*10mM (DMSO) | 220.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
JD-5037
CAS:1392116-14-1
JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
Formula:
C27H27Cl2N5O3S
Purity:
98.14% - 98.87%
Color and Shape:
Solid
Molecular weight:
572.51
Ref: TM-T4453
| 1mg | 43.00 € | ||
| 2mg | 57.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 538.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
Org 27569
CAS:868273-06-7
Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state …
Formula:
C24H28ClN3O
Purity:
100% - ≥95%
Color and Shape:
Solid
Molecular weight:
409.95
Ref: TM-T2635
| 2mg | 36.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 153.00 € | ||
| 50mg | 276.00 € | ||
| 100mg | 412.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
Olivetol
CAS:500-66-3
Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.
Formula:
C11H16O2
Purity:
99.74%
Color and Shape:
(Melting Point 102-106°F) (Ntp 1992)
Molecular weight:
180.24
Ref: TM-T3736
| 500mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
RTICBM-189
CAS:551909-15-0
RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a …
Formula:
C15H14Cl2N2O
Purity:
98.32%
Color and Shape:
Solid
Molecular weight:
309.19
Ref: TM-T9466
| 5mg | 49.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 375.00 € | ||
| 200mg | 530.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
GW842166X
CAS:666260-75-9
GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.
Formula:
C18H17Cl2F3N4O2
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
449.25
Ref: TM-T6527
| 1mg | 35.00 € | ||
| 2mg | 50.00 € | ||
| 5mg | 76.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 221.00 € | ||
| 50mg | 327.00 € | ||
| 100mg | 486.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
PSB-SB-487
CAS:1399049-81-0
PSB-SB-487 is antagonist of GPR55.
Formula:
C26H32O4
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
408.53
Ref: TM-T8975
| 1mg | 37.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 352.00 € | ||
| 100mg | 489.00 € | ||
| 200mg | 673.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Friday 21 Feb 2025
