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Cannabinoid Receptor

Cannabinoid Receptor

Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.

Found 196 products of "Cannabinoid Receptor"

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  • CB2R/FAAH modulator-3

    CAS:
    <p>CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.</p>
    Formula:C22H31NO2
    Purity:99.81%
    Color and Shape:Soild
    Molecular weight:341.49
  • Afubiata

    CAS:
    <p>ADB-FUBIATA is a synthetic cannabinoid studied for its metabolic profile, along with AFUBIATA, CH-FUBIATA, and CH-PIATA. This in vitro analysis by Watanabe S, et al., examines these compounds, as published in "Arch Toxicol," 2023 Dec;97(12):3085-3094.</p>
    Formula:C27H29FN2O
    Color and Shape:Solid
    Molecular weight:416.53
  • TRPV1/CB2 agonist 1


    <p>TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.</p>
    Color and Shape:Odour Solid
  • CB1R agonist 1


    <p>CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.</p>
    Formula:C20H18F3N3O3S
    Color and Shape:Solid
    Molecular weight:437.435
  • VIP36


    <p>VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.</p>
    Formula:C27H35FN6O4
    Color and Shape:Solid
    Molecular weight:526.603
  • Virodhamine

    CAS:
    <p>Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.</p>
    Formula:C22H37NO2
    Purity:98%
    Color and Shape:Soild
    Molecular weight:347.53
  • Taranabant racemate

    CAS:
    <p>Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.</p>
    Formula:C27H25ClF3N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.95
  • AM251

    CAS:
    <p>AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).</p>
    Formula:C22H21Cl2IN4O
    Purity:97.43% - 98.79%
    Color and Shape:A Crystalline Solid
    Molecular weight:555.24
  • yangonin

    CAS:
    <p>Yangonin (Y100550) is a novel CB1 receptor ligand with affinity for human recombinant CB1 receptors.</p>
    Formula:C15H14O4
    Purity:98.82% - 99.55%
    Color and Shape:Pale Yellow Powder
    Molecular weight:258.27
  • N-Oleoyl glycine

    CAS:
    <p>N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of CB1 receptor and the enhancement of insulin-mediated Akt</p>
    Formula:C20H37NO3
    Purity:97.43%
    Color and Shape:Solid
    Molecular weight:339.51
  • Hemopressin (rat) acetate(568588-77-2 free base)


    <p>Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.</p>
    Formula:C5H81N13O14
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:1148.31
  • PSB-SB-487

    CAS:
    <p>PSB-SB-487 is antagonist of GPR55.</p>
    Formula:C26H32O4
    Purity:98.53%
    Color and Shape:Solid
    Molecular weight:408.53
  • RVD-Hpα acetate(1193362-76-3 free base)


    <p>RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>
    Formula:C67H109N19O19
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:1484.71
  • ML-191

    CAS:
    <p>ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.</p>
    Formula:C24H25N3O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:403.47
  • Linoleoyl Ethanolamide

    CAS:
    <p>Linoleoyl Ethanolamide is an endocannabinoid agent.</p>
    Formula:C20H37NO2
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:323.51
  • ML-184

    CAS:
    <p>ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.</p>
    Formula:C25H34N4O3S
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:470.63
  • Otenabant

    CAS:
    <p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>
    Formula:C25H25Cl2N7O
    Purity:99.43%
    Color and Shape:Solid
    Molecular weight:510.42
  • AM281

    CAS:
    <p>AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.</p>
    Formula:C21H19Cl2IN4O2
    Purity:98.6% - >99.99%
    Color and Shape:White To Off-White Solid
    Molecular weight:557.21
  • CB1-IN-1

    CAS:
    <p>CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.</p>
    Formula:C33H31Cl2F3N6O3S2
    Purity:99.08% - 99.76%
    Color and Shape:Solid
    Molecular weight:751.67
  • JD-5037

    CAS:
    <p>JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.</p>
    Formula:C27H27Cl2N5O3S
    Purity:99.54% - 99.84%
    Color and Shape:Solid
    Molecular weight:572.51