Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
Found 218 products for "Cannabinoid Receptor".
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Nervonoyl ethanolamide
CAS:Nervonoyl ethanolamide (NEA), an endogenous cannabinoid, functions as both a presynaptic and postsynaptic neuromodulator. Additionally, it is utilized in inflammation research [1].Formula:C26H51NO2Color and Shape:SolidMolecular weight:409.69Hemopressin (human, mouse)
CAS:Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.Formula:C50H79N13O12Purity:98%Color and Shape:SolidMolecular weight:1054.26Drinabant
CAS:Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.Formula:C23H20Cl2F2N2O2SPurity:99.8%Color and Shape:SolidMolecular weight:497.38Δ8-THC-C8
CAS:Δ8-THC-C8 is a semi-synthetic cannabinoid. It acts as an agonist for the cannabinoid receptor 1 (CB1) with an EC50 value of 13.8 nM.Formula:C24H36O2Color and Shape:SolidMolecular weight:356.54UVI3502
UVI3502 is a cannabinoid receptor 1 (CB1) antagonist with an IC50 value of 4641 nM for CB1 and approximately 16200 nM for CB2. It can inhibit Gi/o protein coupling induced by the agonist CP55,940. UVI3502 shows potential for research into diseases related to the endocannabinoid system in the central nervous system, such as cognitive impairments and neurodegenerative disorders.Afubiata
CAS:ADB-FUBIATA is a synthetic cannabinoid studied for its metabolic profile, along with AFUBIATA, CH-FUBIATA, and CH-PIATA. This in vitro analysis by Watanabe S, et al., examines these compounds, as published in "Arch Toxicol," 2023 Dec;97(12):3085-3094.Formula:C27H29FN2OColor and Shape:SolidMolecular weight:416.53CB2 receptor agonist 9
CAS:CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.Formula:C16H23N3O2SColor and Shape:SolidMolecular weight:321.44CB2R/FAAH modulator-3
CAS:CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formula:C22H31NO2Purity:99.81%Color and Shape:SoildMolecular weight:341.49CB1R agonist 1
CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.Formula:C20H18F3N3O3SColor and Shape:SolidMolecular weight:437.435Virodhamine
CAS:Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.Formula:C22H37NO2Purity:98.20%Color and Shape:Brown LiquidMolecular weight:347.53Taranabant racemate
CAS:Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.Formula:C27H25ClF3N3O2Purity:98%Color and Shape:SolidMolecular weight:515.95Parecoxib sodium
CAS:Parecoxib sodium is a prodrug of Valdecoxib and a selective COX-2 inhibitor prodrug and CB1 agonist (EC50=2.4 µM), alleviate pain and inflammation.Formula:C19H17N2NaO4SPurity:98%Color and Shape:White SolidMolecular weight:392.4Olivetol
CAS:Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.Formula:C11H16O2Purity:99.98%Color and Shape:(Melting Point 102-106°F) (Ntp 1992)Molecular weight:180.24Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Formula:C20H37NO2Purity:99.97%Color and Shape:SolidMolecular weight:323.51Ref: TM-T8425
1mg34.00€5mg64.00€1mL*10mM (DMSO)80.00€10mg95.00€25mg156.00€50mg225.00€100mg329.00€200mg495.00€Otenabant
CAS:Otenabant (CP-945598) has been investigated for the treatment of Obesity.Formula:C25H25Cl2N7OPurity:99.43%Color and Shape:SolidMolecular weight:510.42ARN272
CAS:ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).Formula:C27H20N4O2Purity:98.23%Color and Shape:SolidMolecular weight:432.47(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formula:C23H20Cl2N4O2SPurity:99.28% - 99.83%Color and Shape:SolidMolecular weight:487.4Bay 59-3074
CAS:Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).Formula:C18H13F6NO4SPurity:97.68% - 99.69%Color and Shape:SolidMolecular weight:453.36ML-191
CAS:ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Formula:C24H25N3O3Purity:99.58%Color and Shape:SolidMolecular weight:403.47Otenabant hydrochloride
CAS:Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).Formula:C25H26Cl3N7OPurity:99.79% - ≥95%Color and Shape:SolidMolecular weight:546.88
