GNRH Receptor
Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.
Found 69 products of "GNRH Receptor"
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Degarelix acetate(214766-78-6 free base)
CAS:<p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>Formula:C84H107ClN18O18Purity:98.66%Color and Shape:SolidMolecular weight:1692.34Abarelix
CAS:<p>Abarelix (PPI 149) is a potent gonadotrophin-releasing hormone (GnRH) antagonist, which is used for prostate cancer treatment.</p>Formula:C72H95ClN14O14Purity:>99.99%Color and Shape:SolidMolecular weight:1416.06Alarelin Acetate
CAS:<p>Alarelin Acetate is a synthetic GnRH agonist which can directly inhibit proliferation and DNA synthesis of rat GSMC through GnRH receptors.</p>Formula:C56H78N16O12Purity:99.81% - >99.99%Color and Shape:White PowderMolecular weight:1167.34(R)-Elagolix
CAS:<p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>Formula:C32H30F5N3O5Purity:99.08%Color and Shape:SolidMolecular weight:631.59Kisspeptin-54(human)
CAS:<p>Endogenous ligand for KISS1 receptor; Ki values: rat 1.80 nM, human 1.45 nM. Inhibits tumor spread, stimulates gonadotropin release.</p>Formula:C258H401N79O78Purity:98%Color and Shape:SolidMolecular weight:5857.49Phoenixin-14
CAS:<p>Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/</p>Formula:C75H110N18O20Purity:98%Color and Shape:SolidMolecular weight:1583.78Phoenixin-14 TFA
<p>Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.</p>Formula:C75H110N18O20·xC2HF3O2Purity:99.11%Color and Shape:SolidMolecular weight:1583.78 (free base)Linzagolix choline
CAS:<p>Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.</p>Formula:C27H28F3N3O8SPurity:99.64%Color and Shape:SolidMolecular weight:611.59Surfagon
CAS:<p>Surfagon is an effective LHRH agonist.</p>Formula:C56H78N16O12Purity:98%Color and Shape:SolidMolecular weight:1167.34LGnRH-III, lamprey
CAS:<p>GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.</p>Formula:C59H74N18O14Purity:98%Color and Shape:SolidMolecular weight:1259.33MI 1544
CAS:<p>MI 1544 is a LHRH antagonist.</p>Formula:C71H94ClN17O13Color and Shape:SolidMolecular weight:1429.09Luteinizing Hormone Releasing Hormone (LH-RH), salmon
CAS:<p>LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.</p>Formula:C60H73N15O13Purity:98%Color and Shape:SolidMolecular weight:1212.31Goserelin acetate(65807-02-5 Free base)
<p>Goserelin acetate （ICI-118630 acetate） is a naturally occurring decapeptide, a GnRH (gonadotropin releasing hormone) agonist that reduces the production of sex hormones (testosterone and estrogen) for the treatment of prostate cancer, breast cancer and endometriosis.</p>Purity:99.77%Color and Shape:Odour SolidBim 21009
CAS:<p>Bim 21009 is an inhibitor of gonadorelin.</p>Formula:C74H92ClN17O13Purity:98%Color and Shape:SolidMolecular weight:1463.08Prolactin Releasing Peptide (1-31), human
CAS:<p>Human Prolactin Releasing Peptide (1-31) is a potent GPR10 agonist; Ki values are 1.03 nM (human) and 0.33 nM (rat).</p>Formula:C160H252N56O42SPurity:98%Color and Shape:SolidMolecular weight:3664.15[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:<p>[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.</p>Formula:C67H84N16O13Color and Shape:SolidMolecular weight:1321.48Fsh receptor-binding inhibitor fragment(bi-10)
CAS:<p>FSH antagonist bi-10 suppresses ovulation, induces follicular atresia, and may help in ovarian cancer by downregulating FSHR/ERβ.</p>Formula:C42H67N13O19Color and Shape:SolidMolecular weight:1058.06Zebrafish Kisspeptin-1
CAS:<p>Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.</p>Formula:C58H84N16O15Color and Shape:SolidMolecular weight:1245.39GnRH Associated Peptide (1-24), human
CAS:<p>GnRH Associated Peptide (GAP) (1-24), human, is the 1-24 fragment of hGAP linked to LH-RH via a 3 amino acid site.</p>Formula:C117H190N32O43Color and Shape:SolidMolecular weight:2732.95LH-RH (7-10)
CAS:<p>LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.</p>Formula:C19H36N8O4Color and Shape:SolidMolecular weight:440.54(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:<p>Analog of LHRH, stimulates LH and FSH release, controls reproduction.</p>Formula:C59H84N18O14Color and Shape:SolidMolecular weight:1269.41Kisspeptin-54(human) TFA
<p>Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.</p>Formula:C258H401N79O78·C2HF3O2Color and Shape:SolidMolecular weight:5971.45sGnRH-A
CAS:<p>sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.</p>Formula:C64H83N17O12Color and Shape:SolidMolecular weight:1282.45Kisspeptin 13
CAS:<p>Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.</p>Formula:C78H107N21O18Color and Shape:SolidMolecular weight:1626.81Azaline B
CAS:<p>Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.</p>Formula:C80H102ClN23O12Color and Shape:SolidMolecular weight:1613.27A 76154
CAS:<p>A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).</p>Formula:C70H93FN12O12Color and Shape:SolidMolecular weight:1313.584Wy 43657
CAS:<p>Wy 43657 is a gonadorelin antagonist.</p>Formula:C71H86N14O13Purity:98%Color and Shape:SolidMolecular weight:1343.554APTAA-LHRH
CAS:<p>APTAA-LHRH is a gonadorelin antagonist.</p>Formula:C69H91Cl2N17O14Purity:98%Color and Shape:SolidMolecular weight:1453.47RS 18286
CAS:<p>RS 18286 is a LHRH antagonist.</p>Formula:C74H101Cl2N17O14Color and Shape:SolidMolecular weight:1523.6Azaline
CAS:<p>Azaline is a gonadorelin antagonist.</p>Formula:C74H106ClN23O12Purity:98%Color and Shape:SolidMolecular weight:1545.26LHRH, Ala(6)-
CAS:<p>LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.</p>Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32Avorelin
CAS:<p>Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.</p>Formula:C65H85N17O12Purity:98%Color and Shape:SolidMolecular weight:1296.48LHRH
CAS:<p>Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and has</p>Formula:C55H74N16O14Purity:98%Color and Shape:SolidMolecular weight:1183.27AG 045572
CAS:<p>AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 is</p>Formula:C30H37NO5Purity:99.96%Color and Shape:SolidMolecular weight:491.62Lecirelin
CAS:<p>Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.</p>Formula:C59H84N16O12Color and Shape:SolidMolecular weight:1209.4Deslorelin acetate(57773-65-6 free base)
<p>Deslorelin acetate(57773-65-6 free base) is a gonadotropin releasing hormone super-agonist (GnRH agonist)</p>Formula:C66H87N17O14Purity:99.84%Color and Shape:SolidMolecular weight:1342.5Buserelin Acetate (57982-77-1 free base)
CAS:<p>Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).</p>Formula:C62H90N16O15Purity:99.31% - 99.78%Color and Shape:SolidMolecular weight:1299.48Triptorelin acetate(57773-63-4 free base)
CAS:<p>Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.</p>Formula:C66H86N18O15Purity:99.90%Color and Shape:White PowderMolecular weight:1371.53Cetrorelix diacetate
CAS:<p>Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.</p>Formula:C74H100ClN17O18Purity:98.38%Color and Shape:SolidMolecular weight:1551.17Lecirelin acetate(61012-19-9 free base)
<p>Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts</p>Formula:C61H88N16O14Purity:98.1%Color and Shape:SolidMolecular weight:1269.45Nafarelin acetate(76932-56-4 free base)
CAS:<p>Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.</p>Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55Elagolix sodium
CAS:<p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>Formula:C32H29F5N3NaO5Purity:99.71%Color and Shape:SolidMolecular weight:653.57Histrelin acetate
CAS:<p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>Formula:C68H90N18O14Purity:99.92%Color and Shape:SolidMolecular weight:1383.55Relugolix
CAS:<p>Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with</p>Formula:C29H27F2N7O5SPurity:98.64% - 99.97%Color and Shape:SolidMolecular weight:623.63Linzagolix
CAS:<p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>Formula:C22H15F3N2O7SPurity:99.33%Color and Shape:SolidMolecular weight:508.42Fluorogestone acetate
CAS:<p>FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.</p>Formula:C23H31FO5Purity:99.47%Color and Shape:CoaMolecular weight:406.49Goserelin acetate
CAS:<p>Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.</p>Formula:C61H88N18O16Purity:99.77% - >99.99%Color and Shape:White Crystalline PowderMolecular weight:1329.46Fertirelin
CAS:<p>Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).</p>Formula:C55H76N16O12Purity:>99.99%Color and Shape:SolidMolecular weight:1153.29Ganirelix Acetate
CAS:<p>Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist</p>Formula:C82H117ClN18O15Purity:96.05%Color and Shape:SolidMolecular weight:1630.4Sufugolix
CAS:<p>Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.</p>Formula:C36H31F2N5O4SPurity:97.78%Color and Shape:SolidMolecular weight:667.72LGnRH-III, lamprey acetate(147859-97-0 free base)
<p>LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion</p>Formula:C61H78N18O16Purity:99.66%Color and Shape:SolidMolecular weight:1319.38Cetrorelix Acetate
CAS:<p>Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.</p>Formula:C70H92ClN17O14·xC2H4O2Purity:97.96%Color and Shape:SolidMolecular weight:1491.11NBI-42902
CAS:<p>NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.</p>Formula:C27H24F3N3O3Color and Shape:SolidMolecular weight:495.49BAY 1214784
CAS:<p>BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.</p>Formula:C29H26ClF4N3O5S2Color and Shape:SolidMolecular weight:672.11Argtide
CAS:<p>Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.</p>Formula:C80H104ClN21O14Color and Shape:SolidMolecular weight:1619.27Opigolix
CAS:<p>Opigolix is a Gonadotropin-releasing hormone receptor antagonist.</p>Formula:C25H19F3N4O5SPurity:98.60% - 98.97%Color and Shape:SolidMolecular weight:544.5BAY-298
CAS:<p>BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.</p>Formula:C27H21ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:473.93[D-Ala6]-LH-RH
CAS:<p>[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].</p>Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32T 98475
CAS:<p>gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active</p>Formula:C37H37F2N3O4SPurity:98%Color and Shape:SolidMolecular weight:657.77BAY-784
CAS:<p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>Formula:C29H26ClF4N3O5S2Purity:98%Color and Shape:SolidMolecular weight:672.11DCOIT
CAS:<p>DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].</p>Formula:C11H17Cl2NOSColor and Shape:SolidMolecular weight:282.22Abarelix acetate
CAS:<p>Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.</p>Formula:C72H95ClN14O14·xC2H4O2Color and Shape:SolidMolecular weight:1476.14BAY-899
CAS:<p>BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.</p>Formula:C25H19F2N5O2Purity:98%Color and Shape:SolidMolecular weight:459.45Acyline
CAS:<p>Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.</p>Formula:C80H102ClN15O14Color and Shape:SolidMolecular weight:1533.21Merigolix
CAS:<p>Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .</p>Formula:C36H35F7N4O6Color and Shape:SolidMolecular weight:752.68GnRH-R antagonist 1
CAS:<p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>Formula:C31H28F5N7O6SPurity:98%Color and Shape:SolidMolecular weight:721.65GnRH antagonist 2
CAS:<p>GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.</p>Formula:C28H27F2N9O5Purity:98.08%Color and Shape:SolidMolecular weight:607.57(R)-BAY-899
<p>(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.</p>Formula:C25H19F2N5O2Color and Shape:SolidMolecular weight:459.45Dimethandrolone Undecanoate
CAS:<p>Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.</p>Formula:C31H50O3Purity:99.65% - >99.99%Color and Shape:SolidMolecular weight:470.73Ref: TM-T27176
Discontinued product
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