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GNRH Receptor

GNRH Receptor

Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.

Found 69 products of "GNRH Receptor"

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  • LGnRH-III, lamprey acetate(147859-97-0 free base)
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    LGnRH-III, lamprey acetate(147859-97-0 free base)

    <p>LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion</p>
    Formula:C61H78N18O16
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:1319.38

    Ref: TM-TP1700L

  • Cetrorelix Acetate
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    Cetrorelix Acetate

    CAS:
    <p>Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.</p>
    Formula:C70H92ClN17O14·xC2H4O2
    Purity:97.96%
    Color and Shape:Solid
    Molecular weight:1491.11

    Ref: TM-T5520

  • NBI-42902
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    NBI-42902

    CAS:
    <p>NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.</p>
    Formula:C27H24F3N3O3
    Color and Shape:Solid
    Molecular weight:495.49

    Ref: TM-T69383

  • BAY 1214784
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    BAY 1214784

    CAS:
    <p>BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.</p>
    Formula:C29H26ClF4N3O5S2
    Color and Shape:Solid
    Molecular weight:672.11

    Ref: TM-T72990

  • Argtide
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    Argtide

    CAS:
    <p>Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.</p>
    Formula:C80H104ClN21O14
    Color and Shape:Solid
    Molecular weight:1619.27

    Ref: TM-T70819

  • Opigolix
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    Opigolix

    CAS:
    <p>Opigolix is a Gonadotropin-releasing hormone receptor antagonist.</p>
    Formula:C25H19F3N4O5S
    Purity:98.60% - 98.97%
    Color and Shape:Solid
    Molecular weight:544.5

    Ref: TM-T17301

  • BAY-298
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    BAY-298

    CAS:
    <p>BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.</p>
    Formula:C27H21ClFN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.93

    Ref: TM-T10469

  • CymitQuimica logo
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    [D-Ala6]-LH-RH

    CAS:
    <p>[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].</p>
    Formula:C56H77N17O13
    Color and Shape:Solid
    Molecular weight:1196.32

    Ref: TM-T76351

  • T 98475
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    T 98475

    CAS:
    <p>gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active</p>
    Formula:C37H37F2N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:657.77

    Ref: TM-T23412

  • BAY-784
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    BAY-784

    CAS:
    <p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>
    Formula:C29H26ClF4N3O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:672.11

    Ref: TM-T10475

  • DCOIT
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    DCOIT

    CAS:
    <p>DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].</p>
    Formula:C11H17Cl2NOS
    Color and Shape:Solid
    Molecular weight:282.22

    Ref: TM-T84706

  • Abarelix acetate
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    Abarelix acetate

    CAS:
    <p>Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.</p>
    Formula:C72H95ClN14O14·xC2H4O2
    Color and Shape:Solid
    Molecular weight:1476.14

    Ref: TM-T68701

  • BAY-899
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    BAY-899

    CAS:
    <p>BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.</p>
    Formula:C25H19F2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.45

    Ref: TM-T10476

  • Acyline
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    Acyline

    CAS:
    <p>Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.</p>
    Formula:C80H102ClN15O14
    Color and Shape:Solid
    Molecular weight:1533.21

    Ref: TM-T70266

  • Merigolix
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    Merigolix

    CAS:
    <p>Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .</p>
    Formula:C36H35F7N4O6
    Color and Shape:Solid
    Molecular weight:752.68

    Ref: TM-T73327

  • GnRH-R antagonist 1
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    GnRH-R antagonist 1

    CAS:
    <p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>
    Formula:C31H28F5N7O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:721.65

    Ref: TM-T72492

  • GnRH antagonist 2
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    GnRH antagonist 2

    CAS:
    <p>GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.</p>
    Formula:C28H27F2N9O5
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:607.57

    Ref: TM-T37003

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    (R)-BAY-899

    <p>(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.</p>
    Formula:C25H19F2N5O2
    Color and Shape:Solid
    Molecular weight:459.45

    Ref: TM-T62881

  • Dimethandrolone Undecanoate
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    Dimethandrolone Undecanoate

    CAS:
    <p>Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.</p>
    Formula:C31H50O3
    Purity:99.65% - >99.99%
    Color and Shape:Solid
    Molecular weight:470.73

    Ref: TM-T27176

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