GNRH Receptor
Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.
Found 84 products of "GNRH Receptor"
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Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurity:99.33%Color and Shape:SolidMolecular weight:508.42Goserelin acetate
CAS:Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.
Formula:C61H88N18O16Purity:99.77% - >99.99%Color and Shape:White Crystalline PowderMolecular weight:1329.46Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Formula:C70H92ClN17O14·xC2H4O2Purity:97.96%Color and Shape:SolidMolecular weight:1491.11Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Formula:C55H74N16O13Color and Shape:SolidMolecular weight:1167.29Argtide
CAS:Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.Formula:C80H104ClN21O14Color and Shape:SolidMolecular weight:1619.27NBI-42902
CAS:NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.Formula:C27H24F3N3O3Color and Shape:SolidMolecular weight:495.49EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Formula:C15H27N5O6Color and Shape:SolidMolecular weight:373.4BAY 1214784
CAS:BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.Formula:C29H26ClF4N3O5S2Purity:100% - 99.77%Color and Shape:SolidMolecular weight:672.11Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurity:98.60% - 98.97%Color and Shape:SolidMolecular weight:544.5BAY-784
CAS:BAY-784 is a potent GnRH receptor antagonist with nanomolar activity in human and rat receptors, widely used in endocrine and reproductive research.Formula:C29H26ClF4N3O5S2Purity:99.22% - 99.75%Color and Shape:SolidMolecular weight:672.115α-Pregnane-3α,20α-diol
CAS:5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one fromFormula:C21H36O2Color and Shape:SolidMolecular weight:320.51T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFormula:C37H37F2N3O4SPurity:98%Color and Shape:SolidMolecular weight:657.77BAY-298
CAS:BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.Formula:C27H21ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:473.93DCOIT
CAS:DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].Formula:C11H17Cl2NOSColor and Shape:SolidMolecular weight:282.22[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32Abarelix acetate
CAS:Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.Formula:C72H95ClN14O14·xC2H4O2Color and Shape:SolidMolecular weight:1476.14BAY-899
CAS:BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.Formula:C25H19F2N5O2Purity:98%Color and Shape:SolidMolecular weight:459.45(R)-BAY-899
(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.Formula:C25H19F2N5O2Color and Shape:SolidMolecular weight:459.45GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Formula:C31H28F5N7O6SPurity:98%Color and Shape:SolidMolecular weight:721.65GnRH antagonist 2
CAS:GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.Formula:C28H27F2N9O5Purity:98.08%Color and Shape:SolidMolecular weight:607.57
