GNRH Receptor
Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.
Found 85 products for "GNRH Receptor".
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Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Formula:C66H86N18O15Purity:99.59% - 99.90%Color and Shape:White SolidMolecular weight:1371.53Ref: TM-T21410
5mg52.00€10mg78.00€1mL*10mM (DMSO)116.00€25mg119.00€50mg172.00€100mg259.00€200mg388.00€Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formula:C32H29F5N3NaO5Purity:99.71%Color and Shape:White SolidMolecular weight:653.57Ref: TM-T5031
2mg34.00€5mg50.00€1mL*10mM (DMSO)71.00€10mg75.00€25mg137.00€50mg215.00€100mg340.00€200mg504.00€Nafarelin acetate(76932-56-4 free base)
CAS:Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.Formula:C68H87N17O15Purity:99.98%Color and Shape:SolidMolecular weight:1382.55Linzagolix
CAS:Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormula:C22H15F3N2O7SPurity:99.33% - 99.95%Color and Shape:White SolidMolecular weight:508.42Goserelin acetate
CAS:Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.Formula:C61H88N18O16Purity:99.77% - >99.99%Color and Shape:SolidMolecular weight:1329.46EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Formula:C15H27N5O6Color and Shape:SolidMolecular weight:373.4Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Formula:C55H74N16O13Color and Shape:SolidMolecular weight:1167.29Cetrorelix Acetate
CAS:Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Formula:C70H92ClN17O14·xC2H4O2Purity:99.97%Color and Shape:SolidMolecular weight:1491.11Argtide
CAS:Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.Formula:C80H104ClN21O14Color and Shape:SolidMolecular weight:1619.27BAY 1214784
CAS:BAY 1214784 is a selective and orally active human GnRH-R antagonist, which can effectively reduce plasma luteinizing hormone levels by up to 49%.Formula:C29H26ClF4N3O5S2Purity:100% - 99.77%Color and Shape:White SolidMolecular weight:672.11NBI-42902
CAS:NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.Formula:C27H24F3N3O3Color and Shape:SolidMolecular weight:495.49Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurity:98.60% - 98.97%Color and Shape:SolidMolecular weight:544.55α-Pregnane-3α,20α-diol
CAS:5α-Pregnane-3α,20α-diol, an active metabolite of progesterone, is synthesized through intermediates 5α-pregnane-20α-ol-3-one and 5α-pregnane-3α-ol-20-one fromFormula:C21H36O2Color and Shape:SolidMolecular weight:320.51DCOIT
CAS:DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].Formula:C11H17Cl2NOSColor and Shape:SolidMolecular weight:282.22BAY-784
CAS:BAY-784 is a potent GnRH receptor antagonist with nanomolar activity in human and rat receptors, widely used in endocrine and reproductive research.Formula:C29H26ClF4N3O5S2Purity:99.22% - 99.75%Color and Shape:White SolidMolecular weight:672.11BAY-298
CAS:BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.Formula:C27H21ClFN3O2Purity:98%Color and Shape:SolidMolecular weight:473.93T 98475
CAS:gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally activeFormula:C37H37F2N3O4SPurity:98%Color and Shape:SolidMolecular weight:657.77[D-Ala6]-LH-RH
CAS:[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32Acyline
CAS:Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.Formula:C80H102ClN15O14Color and Shape:SolidMolecular weight:1533.21Merigolix
CAS:Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .Formula:C36H35F7N4O6Color and Shape:SolidMolecular weight:752.68
