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GNRH Receptor

GNRH Receptor

Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.

Found 69 products of "GNRH Receptor"

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  • DCOIT
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    DCOIT

    CAS:
    <p>DCOIT, an isothiazolinone derivative, stimulates the synthesis of follicle-stimulating hormone and luteinizing hormone in the brain by activating the gonadotropin-releasing hormone receptor (GnRHR). Additionally, it interferes with G protein-coupled receptors, MAPK, and Ca 2+ signaling pathways [1].</p>
    Formula:C11H17Cl2NOS
    Color and Shape:Solid
    Molecular weight:282.22

    Ref: TM-T84706

  • Abarelix acetate
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    Abarelix acetate

    CAS:
    <p>Abarelix acetate: synthetic GnRHR antagonist, spikes histamine, lowers LH and testosterone temporarily, used in advanced prostate cancer.</p>
    Formula:C72H95ClN14O14·xC2H4O2
    Color and Shape:Solid
    Molecular weight:1476.14

    Ref: TM-T68701

  • BAY-899
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    BAY-899

    CAS:
    <p>BAY-899, oral LH-R antagonist, IC50: 185 nM (hLH), 46 nM (rLH), lowers sex hormones in vivo.</p>
    Formula:C25H19F2N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.45

    Ref: TM-T10476

  • Acyline
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    Acyline

    CAS:
    <p>Acyline, a GnRH antagonist, suppresses gonadotropins and testosterone in animals and maintains the effect for 2 weeks in men with one dose.</p>
    Formula:C80H102ClN15O14
    Color and Shape:Solid
    Molecular weight:1533.21

    Ref: TM-T70266

  • Merigolix
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    Merigolix

    CAS:
    <p>Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .</p>
    Formula:C36H35F7N4O6
    Color and Shape:Solid
    Molecular weight:752.68

    Ref: TM-T73327

  • GnRH-R antagonist 1
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    GnRH-R antagonist 1

    CAS:
    <p>Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.</p>
    Formula:C31H28F5N7O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:721.65

    Ref: TM-T72492

  • GnRH antagonist 2
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    GnRH antagonist 2

    CAS:
    <p>GnRH antagonist 2 is a GnRH receptor antagonist, useful for studying endocrine diseases.</p>
    Formula:C28H27F2N9O5
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:607.57

    Ref: TM-T37003

  • CymitQuimica logo
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    (R)-BAY-899

    <p>(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.</p>
    Formula:C25H19F2N5O2
    Color and Shape:Solid
    Molecular weight:459.45

    Ref: TM-T62881

  • Dimethandrolone Undecanoate
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    Dimethandrolone Undecanoate

    CAS:
    <p>Dimethandrolone Undecanoate (DMAU) is a novel orally available androgen with progestational activity and is a potential male contraceptive compound.</p>
    Formula:C31H50O3
    Purity:99.65% - >99.99%
    Color and Shape:Solid
    Molecular weight:470.73

    Ref: TM-T27176

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