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GNRH Receptor

GNRH Receptor

Gonadotropin-releasing hormone (GnRH) receptors are GPCRs that bind to GnRH, a hormone responsible for regulating the release of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland. These receptors are crucial for reproductive function and are targeted in therapies for conditions such as prostate cancer, endometriosis, and infertility. GnRH receptor agonists and antagonists are also used in assisted reproductive technologies. At CymitQuimica, we provide a comprehensive range of high-quality GnRH receptor modulators to support your research in reproductive health, endocrinology, and hormone therapy.

Found 69 products of "GNRH Receptor"

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  • Nafarelin acetate(76932-56-4 free base)

    CAS:
    <p>Nafarelin acetate (76932-56-4) is a GnRH analog that reduces LH and FSH release, used for estrogen-related treatments.</p>
    Formula:C68H87N17O15
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:1382.55
  • Elagolix sodium

    CAS:
    <p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>
    Formula:C32H29F5N3NaO5
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:653.57
  • Histrelin acetate

    CAS:
    <p>Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.</p>
    Formula:C68H90N18O14
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:1383.55
  • Relugolix

    CAS:
    <p>Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with</p>
    Formula:C29H27F2N7O5S
    Purity:98.64% - 99.97%
    Color and Shape:Solid
    Molecular weight:623.63
  • Linzagolix

    CAS:
    <p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>
    Formula:C22H15F3N2O7S
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:508.42
  • Fluorogestone acetate

    CAS:
    <p>FGA (Fluorogestone Acetate, SC9880) is 20-25x more potent than progesterone with high potency and short activity duration.</p>
    Formula:C23H31FO5
    Purity:99.47%
    Color and Shape:Coa
    Molecular weight:406.49
  • Goserelin acetate

    CAS:
    <p>Goserelin acetate (Fertilan) is a synthetic long-acting agonist of gonadotropin-releasing hormone, used in treatments of cancer.</p>
    Formula:C61H88N18O16
    Purity:99.77% - >99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:1329.46
  • Fertirelin

    CAS:
    <p>Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).</p>
    Formula:C55H76N16O12
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1153.29
  • Ganirelix Acetate

    CAS:
    <p>Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonist</p>
    Formula:C82H117ClN18O15
    Purity:96.05%
    Color and Shape:Solid
    Molecular weight:1630.4
  • Sufugolix

    CAS:
    <p>Sufugolix (TAK-013) is a potent and orally available luteinizing hormone-releasing hormone LHRH receptor.</p>
    Formula:C36H31F2N5O4S
    Purity:97.78%
    Color and Shape:Solid
    Molecular weight:667.72
  • LGnRH-III, lamprey acetate(147859-97-0 free base)


    <p>LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretion</p>
    Formula:C61H78N18O16
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:1319.38
  • Cetrorelix Acetate

    CAS:
    <p>Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.</p>
    Formula:C70H92ClN17O14·xC2H4O2
    Purity:97.96%
    Color and Shape:Solid
    Molecular weight:1491.11
  • NBI-42902

    CAS:
    <p>NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.</p>
    Formula:C27H24F3N3O3
    Color and Shape:Solid
    Molecular weight:495.49
  • BAY 1214784

    CAS:
    <p>BAY 1214784: potent, oral hGnRH-R antagonist, reduces LH levels, low variability, good tolerance, may research uterine fibroids.</p>
    Formula:C29H26ClF4N3O5S2
    Color and Shape:Solid
    Molecular weight:672.11
  • Argtide

    CAS:
    <p>Argtide is an luteinizing hormone releasing hormone (LHRH) antagonist.</p>
    Formula:C80H104ClN21O14
    Color and Shape:Solid
    Molecular weight:1619.27
  • Opigolix

    CAS:
    <p>Opigolix is a Gonadotropin-releasing hormone receptor antagonist.</p>
    Formula:C25H19F3N4O5S
    Purity:98.60% - 98.97%
    Color and Shape:Solid
    Molecular weight:544.5
  • BAY-298

    CAS:
    <p>BAY-298: oral LH-R antagonist; IC50: 96nM (hLH), 23nM (rLH), 78nM (cLH); first to lower sex hormones in vivo.</p>
    Formula:C27H21ClFN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:473.93
  • [D-Ala6]-LH-RH

    CAS:
    <p>[D-Ala6]-LH-RH, a Luteinizing-hormone-releasing hormone (LHRH) analogue, functions as a gonadotropin-releasing hormone (GnRH) receptor agonist [1].</p>
    Formula:C56H77N17O13
    Color and Shape:Solid
    Molecular weight:1196.32
  • T 98475

    CAS:
    <p>gonadotropin-releasing hormone (GnRH, LHRH) receptor antagonist,orally active</p>
    Formula:C37H37F2N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:657.77
  • BAY-784

    CAS:
    <p>BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).</p>
    Formula:C29H26ClF4N3O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:672.11