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Other Inhibitors

Other Inhibitors

This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.

Found 37926 products of "Other Inhibitors"

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  • VEGFR-2-IN-5 hydrochloride


    <p>VEGFR-2-IN-5 hydrochloride is an effective VEGFR2 inhibitor.</p>
    Formula:C19H25ClN8
    Color and Shape:Solid
    Molecular weight:400.91
  • Luffolide

    CAS:
    <p>Luffolide, a Luffariella sponge metabolite, shares manoalide's anti-inflammatory traits and fully inhibits PLA2's cleavage of phosphatidylcholine.</p>
    Formula:C27H40O6
    Color and Shape:Solid
    Molecular weight:460.60
  • Pinselin

    CAS:
    <p>Pinselin is a nitrogen-containing heterocyclic antibiotic with yeast-inhibiting properties.</p>
    Formula:C16H12O6
    Color and Shape:Solid
    Molecular weight:300.263
  • Echinocandin B nucleus

    CAS:
    <p>Echinocandin B nucleus (A-30912 A nucleus) is the reaction product catalyzed by Echinocandin B decarboxylase. It serves as an intermediate in the semisynthetic production of antifungal agents.</p>
    Formula:C34H51N7O15
    Color and Shape:Solid
    Molecular weight:797.807
  • NSC-217913

    CAS:
    <p>NSC-217913 acts as an inhibitor of WWP1, exhibiting an IC50 value of 158.3 μM.</p>
    Formula:C9H8Cl2N4O2S
    Color and Shape:Solid
    Molecular weight:307.16
  • PARP7-IN-12

    CAS:
    <p>PARP7-IN-12, a potent inhibitor targeting PARP7, exhibits an IC50 of 7.836 nM. This compound is applicable in cancer research.</p>
    Formula:C23H27ClF3N5O5
    Color and Shape:Solid
    Molecular weight:545.94
  • Glutaminyl cyclases-IN-1


    <p>Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.</p>
    Formula:C25H30N6O2S
    Color and Shape:Solid
    Molecular weight:478.61
  • PDE4B/7A-IN-2

    CAS:
    <p>5-HT1A/5-HT7 antagonist; 5-HT1A Ki=8 nM, 5-HT7 Ki=451 nM; PDE4B IC50=80.4 μM, PDE7A IC50=151.3 μM; stronger than escitalopram.</p>
    Formula:C25H35N3O2
    Color and Shape:Solid
    Molecular weight:409.56
  • Hydroxyethyl disulfide

    CAS:
    <p>Hydroxyethyl disulfide can counteract the inhibitory effects of showdomycin on methotrexate-resistant thymidylate synthase and is protected from deactivation by its substrate, deoxyuridine monophosphate, thus preserving the antibiotic's activity.</p>
    Formula:C4H10O2S2
    Color and Shape:Solid
    Molecular weight:154.25
  • NTPDase-IN-3

    CAS:
    <p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>
    Formula:C22H24ClN3OS2
    Color and Shape:Solid
    Molecular weight:446.03
  • Glidobactin B

    CAS:
    <p>Glidobactin B is an antitumor antibiotic. It is active against pathogenic fungi and yeasts and can prolong the survival time of mice inoculated with leukemia P388 cells.</p>
    Formula:C29H46N4O6
    Color and Shape:Solid
    Molecular weight:546.699
  • MK-7445

    CAS:
    <p>MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.</p>
    Formula:C21H13Cl2N7O
    Color and Shape:Solid
    Molecular weight:450.28
  • Melanocin A

    CAS:
    <p>Melanocin A is an inhibitor of melanin biosynthesis. It suppresses the synthesis of melanin and tyrosinase with an IC50 of 9.0 nM and MIC of 0.9 μM. Additionally, Melanocin A exhibits antioxidant properties.</p>
    Formula:C18H14N2O5
    Color and Shape:Solid
    Molecular weight:338.31
  • GSK1820795A

    CAS:
    <p>GSK1820795A: Telmisartan analog, selective hGPR132a antagonist, blocks yeast activation by N-acylamides, angiotensin II antagonist, partial PPARγ agonist.</p>
    Formula:C35H34N8
    Color and Shape:Solid
    Molecular weight:566.7
  • Chloronectrin

    CAS:
    <p>Chloronectrin exhibits activity against Gram-positive bacteria.</p>
    Formula:C25H33ClO6
    Color and Shape:Solid
    Molecular weight:464.979
  • Sagopilone

    CAS:
    <p>Sagopilone: synthetic epothilone, inhibits cell division and induces apoptosis, effective in MDR tumors, not P-gp substrate.</p>
    Formula:C30H41NO6S
    Color and Shape:Solid
    Molecular weight:543.71
  • GSK3527497 HCl

    CAS:
    <p>GSK3527497: potent TRPV4 inhibitor, IC50=12 nM, targets heart/respiratory issues, for oral/IV use, low-dose effective.</p>
    Formula:C17H17Cl2FN4O4S
    Color and Shape:Solid
    Molecular weight:463.3054
  • Barixibat

    CAS:
    <p>Barixibat is a bile acid transport inhibitor.</p>
    Formula:C42H55N5O8
    Color and Shape:Solid
    Molecular weight:757.91
  • Milbemycin α11

    CAS:
    <p>Milbemycin α11 (Meilingmycin A) is an antibiotic known for its ability to eliminate nematodes and mites.</p>
    Formula:C36H50O9
    Color and Shape:Solid
    Molecular weight:626.78
  • Griseochelin

    CAS:
    <p>Griseochelin exhibits activity against Gram-negative bacteria and inhibits Coccidioides.</p>
    Formula:C33H60O7
    Color and Shape:Solid
    Molecular weight:568.825
  • Ophiobolin D

    CAS:
    <p>Ophiobolin D is a terpene antibiotic with mild inhibitory effects on Staphylococcus aureus.</p>
    Formula:C25H36O4
    Color and Shape:Solid
    Molecular weight:400.55
  • Gilvocarcin E

    CAS:
    <p>Gilvocarcin E exhibits activity against Gram-positive bacteria and is capable of inhibiting Sarcoma 180 and P388 leukemia cells.</p>
    Formula:C27H28O9
    Color and Shape:Solid
    Molecular weight:496.506
  • SARS-CoV-2 nsp3-IN-1


    <p>Compound 15c selectively inhibits SARS-CoV-2 nsp3 Mac1 with IC50 of 6.1 μM.</p>
    Formula:C17H15N5O2
    Color and Shape:Solid
    Molecular weight:321.33
  • BMS-748730

    CAS:
    <p>BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.</p>
    Formula:C22H26ClN7O3S
    Color and Shape:Solid
    Molecular weight:504.01
  • UAWJ9-36-1

    CAS:
    <p>UAWJ9-36-1: potent broad-spectrum coronavirus Protease inhibitor; IC50 = 51 nM.</p>
    Formula:C23H29N3O5
    Color and Shape:Solid
    Molecular weight:427.49
  • PDE4B/7A-IN-1

    CAS:
    <p>5-HT1A antagonist; Ki=8nM, Kb=0.04nM. PDE4B IC50=80.4μM; PDE7A IC50=151.3μM. Good biofilm penetration, stable, anticognitive, antidepressant.</p>
    Formula:C25H35N3O3
    Color and Shape:Solid
    Molecular weight:425.56
  • (R)-ONO-2952


    <p>(R)-ONO-2952 is the R-enantiomer of ONO-2952. ONO-2952 is selective and oral effective TSPO antagonist, with Kis of 0.330-9.30 nM inhibiting rat and human TSPO.</p>
    Formula:C22H20ClFN2O2
    Color and Shape:Solid
    Molecular weight:398.86
  • CYP2C1/CYP2C19-IN-2


    <p>CYP2C1/CYP2C19-IN-2 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>
    Formula:C27H28N2O6S
    Color and Shape:Solid
    Molecular weight:508.59
  • ASB14780


    <p>ASB14780 is a 4-phenoxy derivative and an inhibitor of cytoplasmic phospholipase cPLA2α (IC50: 20 nM).</p>
    Color and Shape:Solid
  • MCTR1

    CAS:
    <p>MCTR1, a pro-resolving mediator derived from DHA, promotes tissue repair and reduces inflammation by enhancing phagocytosis and decreasing eicosanoids.</p>
    Formula:C32H47N3O9S
    Color and Shape:Solid
    Molecular weight:649.8
  • Oncopterin

    CAS:
    <p>Oncopterin is found in urine from patients with solid and blood cancers.</p>
    Formula:C12H18N6O3
    Color and Shape:Solid
    Molecular weight:294.31
  • Sucistil


    <p>Sucistil is an active biochemical. hemoglobin sucistil (bovine) is an oxygen carrier [1].</p>
    Formula:C9H15NO4S
    Color and Shape:Solid
    Molecular weight:233.28
  • Brostallicin HCl

    CAS:
    <p>Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.</p>
    Formula:C30H36BrClN12O5
    Color and Shape:Solid
    Molecular weight:760.04
  • GSK945237

    CAS:
    <p>GSK945237 is a type IIA topoisomerase inhibitor, effective on Gram-positive and negative bacteria, with favorable pharmacokinetics and in vivo efficacy.</p>
    Formula:C24H26FN5O3
    Color and Shape:Solid
    Molecular weight:451.49
  • Musettamycin

    CAS:
    <p>Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.</p>
    Formula:C36H45NO14
    Color and Shape:Solid
    Molecular weight:715.74
  • Haloquinone

    CAS:
    <p>Haloquinone is a quinone antibiotic that exhibits significant antibacterial activity against halophilic bacteria and is also effective against Gram-positive bacteria and mycoplasma.</p>
    Formula:C17H12O5
    Color and Shape:Solid
    Molecular weight:296.274
  • TP3011

    CAS:
    <p>TP3011 is a potent topoisomerase I inhibitor equipotent as SN38 and is an active metabolite of CH-0793076.</p>
    Formula:C26H26N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.51
  • Minnelide free acid

    CAS:
    <p>Minnelide treats pancreatic cancer, hinders androgen-related prostate growth, shrinks tumors, and improves survival.</p>
    Formula:C21H27O10P
    Color and Shape:Solid
    Molecular weight:470.41
  • Erabulenol A

    CAS:
    <p>Erabulenol A is a cholesterol ester transfer protein (CETP) inhibitor, extracted from Penicillumsp.</p>
    Formula:C20H20O6
    Color and Shape:Solid
    Molecular weight:356.369
  • Dermostatin B

    CAS:
    <p>Dermostatin B is a polyene antibiotic with antifungal properties, suitable for research on fungal infections.</p>
    Formula:C41H66O11
    Color and Shape:Solid
    Molecular weight:734.956
  • Schidigera-genin B

    CAS:
    <p>Schidigera-genin B is a steroidal saponin that can be isolated from Yucca glauca. It exhibits mild antifungal activity.</p>
    Formula:C27H40O4
    Color and Shape:Solid
    Molecular weight:428.604
  • CV 5975

    CAS:
    <p>CV 5975 is a nonsulfhydryl ACE inhibitor that was investigated for use in hypertension and heart failure.</p>
    Formula:C22H31N3O5S
    Color and Shape:Solid
    Molecular weight:449.56
  • GR-71251

    CAS:
    <p>GR-71251 is a Tachykinin receptor antagonist.</p>
    Formula:C74H105N19O13
    Color and Shape:Solid
    Molecular weight:1468.74
  • Sequoiaflavone

    CAS:
    <p>Sequoiaflavone is a biflavone isolated from Ginkgo biloba.</p>
    Formula:C31H20O10
    Color and Shape:Solid
    Molecular weight:552.48
  • OncoFAP

    CAS:
    <p>OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.</p>
    Formula:C21H19F2N5O5
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:459.40
  • Formadicin A

    CAS:
    <p>Formadicin A exhibits strong activity against various Pseudomonas, Proteus, and Alcaligenes bacteria.</p>
    Formula:C30H34N4O16
    Color and Shape:Solid
    Molecular weight:706.608
  • Diphenicillin

    CAS:
    <p>Diphenicillin (Ancillin (free acid); 2-Biphenylyl penicillin (free acid); SKF-12141 (free acid)) is a penicillin that resists Penicillinase and exhibits antibacterial activity. It shows effective activity against Gram-positive cocci. Diphenicillin is promising for research on infectious diseases caused by Gram-positive bacteria such as staphylococci, pneumococci, and group A streptococci.</p>
    Formula:C21H20N2O4S
    Color and Shape:Solid
    Molecular weight:396.459
  • DS88790512

    CAS:
    <p>DS88790512, IC50 at 11 nM, is an effective, selective, oral bioeffective TRPC6 inhibitor.</p>
    Formula:C22H29N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:367.48
  • ASP-8731

    CAS:
    <p>ASP8731 is a selective inhibitor of BACH1 that prevents inflammation and vascular occlusion, and induces fetal hemoglobin in sickle cell disease.</p>
    Formula:C20H21N5O4
    Color and Shape:Solid
    Molecular weight:395.41
  • TAK-024

    CAS:
    TAK-024 is an inhibitor of platelet(IC50s of 31, 79 and 51 nM in human, monkey and guinea pig, respectively).
    Formula:C27H34N10O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:594.62
  • Saframycin A

    CAS:
    <p>Saframycin A exhibits antibacterial activity against Gram-positive bacteria and shows weaker effects on Gram-negative bacteria and mycobacteria. Additionally, it inhibits mouse lymphocyte L-1210 cells, with an ID50 of 0.0056 μM.</p>
    Formula:C29H30N4O8
    Color and Shape:Solid
    Molecular weight:562.57
  • (1R,3S)-THCCA-Asn


    <p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>
    Formula:C24H24N4O6
    Color and Shape:Solid
    Molecular weight:464.47
  • 3'-O-Decarbamoylirumamycin

    CAS:
    <p>3'-O-Decarbamoylirumamycin is a 20-membered macrolide antibiotic produced by Streptomyces subflavus subsp. irumaensis. It exhibits inhibitory effects against plant pathogenic fungi, such as Pyricularia oryzae and Sclerotinia.</p>
    Formula:C40H64O11
    Color and Shape:Solid
    Molecular weight:720.93
  • BMS-554417

    CAS:
    <p>BMS-554417 inhibits IGF-IR/insulin receptors, curbing cell proliferation and tumor growth, with IC50 values of 120 nm–&gt;8.5 μmol/L.</p>
    Formula:C28H30ClN7O2
    Color and Shape:Solid
    Molecular weight:532.04
  • BI-207524

    CAS:
    <p>BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.</p>
    Formula:C35H36ClN5O5
    Color and Shape:Solid
    Molecular weight:642.14
  • Cytosaminomycin C

    CAS:
    <p>Cytosaminomycin C exhibits anti-Eimeria Tenella coccidial activity.</p>
    Formula:C23H36N4O8
    Color and Shape:Solid
    Molecular weight:496.554
  • Cytosaminomycin B

    CAS:
    <p>Cytosaminomycin B exhibits activity against Eimeria Tenella coccidia.</p>
    Formula:C26H37N5O8
    Color and Shape:Solid
    Molecular weight:547.601
  • Pluracidomycin B

    CAS:
    <p>Pluracidomycin B, a carbapenem antibiotic, exhibits activity against both Gram-positive and Gram-negative bacteria and also functions as an inhibitor of β-lactamase enzymes.</p>
    Formula:C11H13NO10S2
    Color and Shape:Solid
    Molecular weight:383.352
  • Unoprostone isopropyl

    CAS:
    <p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>
    Formula:C25H44O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:424.61
  • Topoisomerase II inhibitor 5


    <p>Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.</p>
    Formula:C26H27N5O4
    Color and Shape:Solid
    Molecular weight:473.52
  • Orvepitant

    CAS:
    <p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>
    Formula:C31H35F7N4O2
    Color and Shape:Solid
    Molecular weight:628.62
  • Ornoprostil

    CAS:
    <p>Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.</p>
    Formula:C23H38O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.54
  • Nafarelin acetate hydrate

    CAS:
    <p>Nafarelin: a GnRH agonist used to treat endometriosis, precocious puberty, and control IVF. Delivered as a nasal spray. Marketed as Synarel by Pfizer.</p>
    Formula:C66H83N17O13·xC2H4O2·xH2O
    Color and Shape:Solid
    Molecular weight:1400.563
  • Butaprost

    CAS:
    <p>Butaprost: EP2 receptor agonist, EC50=33 nM, Ki=2.4 μM (murine), reduces fibrosis via TGF-β/Smad2.</p>
    Formula:C24H40O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.57
  • ZK118182 isopropyl ester

    CAS:
    <p>ZK118182 isopropyl ester is a PG analog with potent DP-agonist activity (EC50 = 16.5 nM) and high affinity for the DP receptor (Ki = 74 nM).</p>
    Formula:C23H37ClO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:428.99
  • Antcin B

    CAS:
    <p>Antcin B is an inhibitor of SARS-CoV-2 3-chymotrypsin-like protease (3CL Pro). It interacts with several crucial amino acid residues of 3CL Pro, including Leu141, Asn142, Glu166, and His163, through hydrogen bonding, salt bridges, and hydrophobic interactions, thereby inhibiting its activity. This inhibition blocks the cleavage of viral polyproteins and suppresses the replication of the SARS-CoV-2 virus within host cells. Antcin B shows potential for research in the context of COVID-19.</p>
    Formula:C29H40O5
    Color and Shape:Solid
    Molecular weight:468.625
  • ONO-DI-004

    CAS:
    <p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>
    Formula:C24H38O6
    Color and Shape:Solid
    Molecular weight:422.55
  • TP-6076

    CAS:
    <p>TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A.</p>
    Formula:C28H32F3N3O7
    Color and Shape:Solid
    Molecular weight:579.56
  • FR 900452

    CAS:
    <p>FR 900452 is a platelet activating factor antagonist from fermentatiion products of Streptomyces phaeofaciens.</p>
    Formula:C22H25N3O3S
    Color and Shape:Solid
    Molecular weight:411.52
  • COTC

    CAS:
    <p>COTC is an anticancer bacterial metabolite; inhibits glyoxalase with GSH, halts HeLa cell growth, and fights tumor in Ehrlich murine model.</p>
    Formula:C11H14O6
    Color and Shape:Solid
    Molecular weight:242.23
  • MEN-10354

    CAS:
    <p>MEN-10354 is a less potent and less selective NK-2 tachykinin receptor antagonist compared to the linear analog, R 396.</p>
    Formula:C37H46N8O9
    Color and Shape:Solid
    Molecular weight:746.81
  • 3-IN-PP1

    CAS:
    <p>3-IN-PP1: PKD inhibitor (IC50: 94-108 nM for PKD1/2/3), broad anticancer agent for research.</p>
    Formula:C17H18N6
    Color and Shape:Solid
    Molecular weight:306.36
  • RS 2135

    CAS:
    <p>RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.</p>
    Formula:C18H21ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.83
  • Hydranthomycin

    CAS:
    <p>Hydranthomycin is an antibiotic with moderate antifungal activity, exhibiting a minimum inhibitory concentration (MIC) of 25 μg/mL against the rice blast fungus. Additionally, it inhibits the growth of Chlorella (tiny naked algae) and possesses herbicidal properties.</p>
    Formula:C20H20O5
    Color and Shape:Solid
    Molecular weight:340.37
  • Clavalanine

    CAS:
    <p>Clavalanine (Ro 22-5417) is capable of inhibiting various bacteria and fungi.</p>
    Formula:C8H12N2O4
    Color and Shape:Solid
    Molecular weight:200.192
  • Naltrindole

    CAS:
    <p>Naltrindole is a delta opioid receptor antagonist.</p>
    Formula:C26H26N2O3
    Color and Shape:Solid
    Molecular weight:414.5
  • PI4KIIIbeta-IN-11

    CAS:
    <p>PI4KIIIbeta-IN-11 is a PI4KIIIβ inhibitor (mean pIC50=9.1) that can be used to study diseases caused by RNA viruses and Plasmodium falciparum.</p>
    Formula:C33H39N7O3
    Color and Shape:Solid
    Molecular weight:581.71
  • FW 34569

    CAS:
    <p>FW 34569, an enkephalin analog, boosts growth hormones and prolactin, reduces cortisol and LH; FSH stable.</p>
    Formula:C30H43N5O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:617.76
  • Epithienamycin D

    CAS:
    <p>Epithienamycin D is a carbapenem antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Formula:C13H16N2O5S
    Color and Shape:Solid
    Molecular weight:312.342
  • NTPDase-IN-2

    CAS:
    <p>NTPDase-IN-2 inhibits h-NTPDase-2/-8 (IC50: 0.04, 2.27 µM), non-competitive for h-NTPDase-1/-2 (Km: 74 µM); useful in cancer, immune, bacterial research.</p>
    Formula:C24H20FN3OS2
    Color and Shape:Solid
    Molecular weight:449.56
  • IMR687

    CAS:
    <p>IMR687: a PDE9 inhibitor that could improve memory in Alzheimer's by slowing cGMP hydrolysis.</p>
    Formula:C21H26N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:394.47
  • AFM-30a hydrochloride


    <p>AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.</p>
    Formula:C24H28ClFN6O3
    Color and Shape:Solid
    Molecular weight:502.97
  • BSc5367

    CAS:
    <p>BSc5367 inhibits Nek1 kinase (IC50: 11.5 nM), key in cell cycle, DNA repair, impacting ALS, PKD, cancer.</p>
    Formula:C20H15N3O2
    Color and Shape:Soild
    Molecular weight:329.35
  • Anti-inflammatory agent 18


    <p>Anti-inflammatory agent 18: NO activity blocker (IC50: 15.94 μM), hampers HMGB1-induced inflammation, potential for COVID-19, sepsis study.</p>
    Formula:C30H50O6
    Color and Shape:Solid
    Molecular weight:506.71
  • Memnobotrin A

    CAS:
    <p>Memnobotrin A is an antibiotic with inhibitory effects on the NCI-460, MCF7, and SF-268 cell lines.</p>
    Formula:C25H33NO5
    Color and Shape:Solid
    Molecular weight:427.53
  • Retelliptine

    CAS:
    <p>Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.</p>
    Formula:C25H32N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:404.55
  • L 739749

    CAS:
    <p>L 739749 is a CAAX peptidomimetic. It is also an inhibitor of farnesyl-protein transferase.</p>
    Formula:C24H41N3O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.73
  • UNC9426

    CAS:
    <p>UNC9426 is an orally active, potent and selective TYRO3 inhibitor with an IC50 of 2.1 nM. UNC9426 reduces platelet aggregation without prolonging bleeding time.</p>
    Formula:C32H34F6N6O
    Purity:98.051%
    Color and Shape:Solid
    Molecular weight:632.642
  • Naltalimide

    CAS:
    <p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>
    Formula:C28H28N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.53
  • AL-GDa62


    <p>AL-GDa62, a gastric cancer treatment lead, has EC50 of 3.2 μM (MCF10A-WT) and 2 μM (MCF10A-CDH1 -/-).</p>
    Formula:C24H28FN3O
    Color and Shape:Solid
    Molecular weight:393.5
  • L 156903

    CAS:
    <p>L 156903 is a bioactive chemical. It also inhibits the binding of neurotensin to brain tissue.</p>
    Formula:C35H41N7O5S
    Color and Shape:Solid
    Molecular weight:671.81
  • Sulprostone

    CAS:
    <p>EP3 and EP1 receptor agonist</p>
    Formula:C23H31NO7S
    Purity:98%
    Color and Shape:White To Off-White Solid
    Molecular weight:465.56
  • Pamiparib maleate

    CAS:
    <p>Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.</p>
    Formula:C44H42F2N8O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:944.859
  • 4α-PDD

    CAS:
    <p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>
    Formula:C40H64O8
    Color and Shape:Solid
    Molecular weight:672.93
  • Ambelline

    CAS:
    <p>Ambelline has antitumor activity.</p>
    Formula:C18H21NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.36
  • STA-1474

    CAS:
    <p>STA-1474, a soluble prodrug of ganetespib (STA-9090), becomes a strong HSP90 inhibitor effective against canine tumors.</p>
    Formula:C20H21N4O6P
    Color and Shape:Solid
    Molecular weight:444.38
  • ZK159222

    CAS:
    <p>ZK159222 is an effective 1α,25-(OH)2D3 receptor (VDR) agonist. ZK159222 has a partial agonistic character.</p>
    Formula:C32H48O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:512.72
  • SHR902275

    CAS:
    <p>SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.</p>
    Formula:C26H23F3N4O4
    Color and Shape:Solid
    Molecular weight:512.48
  • Azirinomycin

    CAS:
    <p>Azirinomycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>
    Formula:C4H5NO2
    Color and Shape:Solid
    Molecular weight:99.088
  • Crotocin

    CAS:
    <p>Crotocin exhibits bactericidal activity against Cryptococcus neoformans, Candida albicans, and Saccharomyces cerevisiae (brewer’s yeast), but it can be inactivated by blood.</p>
    Formula:C19H24O5
    Color and Shape:Solid
    Molecular weight:332.391
  • Cremeomycin

    CAS:
    <p>Cremeomycin exhibits activity against Gram-positive bacteria, including methicillin-resistant Staphylococcus aureus (MRSA), with a minimum inhibitory concentration (MIC) of 0.2-0.39 μg/mL. It also demonstrates cytotoxic effects in vitro against mouse tumor cell lines P388, L1210, IMC, S180, B16, and SS3.</p>
    Formula:C8H6N2O4
    Color and Shape:Solid
    Molecular weight:194.144
  • L 668750

    CAS:
    <p>L 668750 is an inhibitor of platelet-activating factor.</p>
    Formula:C25H34O9S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:510.6
  • Indinavir monohydrate

    CAS:
    <p>Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.</p>
    Formula:C36H49N5O5
    Color and Shape:Solid
    Molecular weight:631.82
  • SBI-581


    <p>SBI-581: oral, potent TAO3 inhibitor, IC50=42nM, alters TKS5α at RAB11+ vesicles, blocks invadopodia, good mouse pharmacokinetics, anti-tumor.</p>
    Formula:C24H21N3O2
    Color and Shape:Solid
    Molecular weight:383.44
  • Deoxyradicinin

    CAS:
    <p>Deoxyradicinin is a biosynthetic precursor of Radicinin. It can inhibit Xylella fastidiosa and Liberibacter crescens, with a minimum inhibitory concentration (MIC) of 3.5 μg/mL against Liberibacter crescens. Deoxyradicinin is applicable for research on controlling plant diseases caused by these pathogens.</p>
    Formula:C12H12O4
    Color and Shape:Solid
    Molecular weight:220.221
  • GSK2578999A

    CAS:
    <p>GSK2578999A is a betulin derivative with antitumor activity.</p>
    Formula:C46H62ClNO7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:776.44
  • IACS-8779 disodium

    CAS:
    <p>IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.</p>
    Formula:C21H23N9Na2O10P2S2
    Color and Shape:Solid
    Molecular weight:733.52
  • Nolpitantium Free Base

    CAS:
    <p>Nolpitantium is a potent, selective NK1 receptor antagonist that inhibits substance P without affecting NK2/NK3 receptors.</p>
    Formula:C37H45Cl2N2O2
    Color and Shape:Solid
    Molecular weight:620.67
  • Domitroban

    CAS:
    <p>Domitroban, also known as S-145, is a thromboxane (Tx) A2-receptor antagonist with partial agonistic activity in vascular smooth muscle.</p>
    Formula:C20H27NO4S
    Color and Shape:Solid
    Molecular weight:377.5
  • Kynapcin-28

    CAS:
    <p>Kynapcin-28 is a non-competitive inhibitor of prolyl endopeptidase (PEP) with an IC50 of 76.80 μM and exhibits weak inhibitory effects on other serine proteases.</p>
    Formula:C19H12O10
    Color and Shape:Solid
    Molecular weight:400.293
  • NVP-CFC218

    CAS:
    <p>NVP-CFC218 is a novel potent and selective p53-HDM2 inhibitor.</p>
    Formula:C37H45ClN4O4
    Color and Shape:Solid
    Molecular weight:645.23
  • Coriolin B

    CAS:
    <p>Coriolin B exhibits activity against Gram-positive bacteria, weak activity against Gram-negative bacteria, yeast, and Trichomonas vaginalis. At a concentration of 5 μg/mL, Coriolin B inhibits 61.6% of Yoshida sarcoma growth but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>
    Formula:C23H36O6
    Color and Shape:Solid
    Molecular weight:408.528
  • Antileishmanial agent-5


    <p>Antileishmanial agent-4, a ribonucleoside analogue, targets L.infantum and T.cruzi with EC50s of 0.68 μM and 0.83 μM.</p>
    Formula:C17H17ClN4O4
    Color and Shape:Solid
    Molecular weight:376.79
  • Chitinase-IN-5


    <p>Chitinase-IN-5 (8i) blocks OfChi-h (IC50: 0.051 μM), has insecticidal qualities, useful for eco-friendly pest control.</p>
    Formula:C20H21ClFN7
    Color and Shape:Solid
    Molecular weight:413.88
  • Coriolin A

    CAS:
    <p>Coriolin A exhibits activity against gram-positive bacteria, weakly against gram-negative bacteria, as well as yeasts and Trichomonas vaginalis. At a concentration of 5 μg/mL, it inhibits 61.6% of the growth of Yoshida sarcoma, but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>
    Formula:C15H20O5
    Color and Shape:Solid
    Molecular weight:280.316
  • Trypanothione synthetase-IN-4


    <p>Trypanothione synthetase-IN-4, an L. infantum inhibitor, has potent anti-leishmanicidal properties (EC50: 0.6 μM).</p>
    Formula:C29H52INO2
    Color and Shape:Solid
    Molecular weight:573.63
  • Lunacalcipol

    CAS:
    <p>Lunacalcipol is used for the treatment of Secondary Hyperparathyroidism.</p>
    Formula:C28H42O4S
    Color and Shape:Solid
    Molecular weight:474.7
  • Foroxymithine

    CAS:
    <p>Foroxymithine is an inhibitor of angiotensin-converting enzyme.</p>
    Formula:C22H37N7O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:575.57
  • Flurdihydroergotamine

    CAS:
    <p>Flurdihydroergotamine, a serotonin 5HT1 receptor agonist, is used as an antimigraine drug.</p>
    Formula:C34H36F3N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:651.68
  • SMP-797 HCl

    CAS:
    <p>SMP-797 HCl, an ACAT (acyl-CoA-cholesterol acyltransferase) inhibitor, is used potentially for the treatment of Hyperlipidemia.</p>
    Formula:C34H44ClN5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:622.20
  • Antileishmanial agent-4


    <p>Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].</p>
    Formula:C17H18N4O4
    Color and Shape:Solid
    Molecular weight:342.35
  • Antimalarial agent 2


    <p>Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.</p>
    Formula:C27H25N3O5
    Color and Shape:Solid
    Molecular weight:471.5
  • Carbacyclin

    CAS:
    <p>Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.</p>
    Formula:C21H34O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.49
  • FR 901537

    CAS:
    <p>FR 901537 is a new aromatase inhibitor with antitumor effects.</p>
    Formula:C23H29N3O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:507.62
  • Lorajmine

    CAS:
    <p>Lorajmine, a monochloroacetyl derivative of ajmaline, is a class Ia antiarrhythmic agent that is rapidly hydrolyzed to ajmaline by plasma and tissue esterases.</p>
    Formula:C22H27ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.91
  • KY-02327 acetate


    <p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>
    Formula:C22H31N3O6
    Color and Shape:Solid
    Molecular weight:433.5
  • Dinordrin I diacetate

    CAS:
    <p>Dinordrin I diacetate is an implantation inhibitor and hormone.</p>
    Formula:C25H32O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.52
  • Alentemol hydrobromide

    CAS:
    <p>Alentemol hydrobromide is a Dopamine agonist.</p>
    Formula:C19H26BrNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:364.32
  • LIT-001 free base

    CAS:
    <p>LIT-001, a nonpeptide OT-R agonist, enhances mouse autism-like behavior, with EC50=55 nM and Ki=226 nM.</p>
    Formula:C28H33N7O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:531.67
  • Citreamicin β

    CAS:
    <p>Citreamicin β exhibits activity against aerobic and anaerobic Gram-positive bacteria.</p>
    Formula:C35H29NO12
    Color and Shape:Solid
    Molecular weight:655.604
  • Mycinamicin Ⅵ

    CAS:
    <p>Mycinamicin VI is a macrolide antibiotic with antibacterial activity against Gram-positive bacteria.</p>
    Formula:C35H57NO11
    Color and Shape:Solid
    Molecular weight:667.83
  • Fleephilone

    CAS:
    <p>Fleephilone is a fungal metabolite isolated from Trichoderma harzianum. It acts as an HIV REV/RRE binding inhibitor, hindering the interaction between REV protein and RRE RNA with an IC50 of 7.6 μM.</p>
    Formula:C24H27NO7
    Color and Shape:Solid
    Molecular weight:441.474
  • Rimegepant sulfate hydrate

    CAS:
    <p>Rimegepant (BMS-927711/BHV-3000): oral CGRP blocker for migraines, effective without vasoconstriction, beats placebo, well-tolerated.</p>
    Formula:C56H64F4N12O13S
    Color and Shape:Solid
    Molecular weight:1221.2526
  • AZ0108

    CAS:
    <p>AZ0108, an oral PARP1,2,6 inhibitor, selectively blocks centrosome clustering, is viable for in vivo studies, and doesn't inhibit PARP3/TNKS1.</p>
    Formula:C24H20F4N6O2
    Color and Shape:Solid
    Molecular weight:500.45
  • Macquarimicin A

    CAS:
    <p>Macquarimicin A is an antibiotic.</p>
    Formula:C19H22O5
    Color and Shape:Solid
    Molecular weight:330.375
  • 2-PPA

    CAS:
    2-PPA serves as a selective TMEM175 inhibitor (IC 50 =32 μM), primarily influencing lysosomal activity. Through acute inhibition of TMEM175, 2-PPA enhances lysosomal macromolecular catabolism, which in turn boosts macrophage activity and other digestive processes. This compound holds significance in Parkinson's disease research.
    Formula:C11H10N2
    Color and Shape:Solid
    Molecular weight:170.21
  • GW311616 hydrochloride

    CAS:
    <p>GW-311616 hydrochloride is a long duration, orally bioavailable, and selective human neutrophil elastase (HNE) inhibitor (IC50: 22 nM; Ki: 0.31 nM).</p>
    Formula:C19H32ClN3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.99
  • HMGB1-IN-3

    CAS:
    <p>HMGB1-IN-3 (compound E), a derivative of glycyrrhizic acid, exhibits potent inhibitory effects on HMGB1 (high mobility group protein 1). It is utilized in research related to intracerebral hemorrhage.</p>
    Formula:C31H46O4
    Color and Shape:Solid
    Molecular weight:482.69
  • Kirrothricin

    CAS:
    <p>Kirrothricin exhibits antibacterial properties, but it is inactive against Bacillus subtilis, Escherichia coli, and fungi.</p>
    Formula:C44H64N2O10
    Color and Shape:Solid
    Molecular weight:780.986
  • 7β,16α-Dihydroxybufalin

    CAS:
    <p>7β,16α-Dihydroxybufalin, a dihydroxylated derivative of bufalin, demonstrates cytotoxic properties against various cancer cell lines.</p>
    Formula:C24H34O6
    Color and Shape:Solid
    Molecular weight:418.52
  • ETH 157

    CAS:
    <p>ETH 157 is a synthetic neutral carrier-based Na+ selective microelectrode, with sufficient selectivity against K+, Ca2+, and Mg2+ for extracellular measurement of Na+ activity.</p>
    Formula:C36H32N2O4
    Color and Shape:Solid
    Molecular weight:556.65
  • S24-14

    CAS:
    <p>S24-14 serves as an effective anti-osteoporosis agent by inhibiting osteoclastogenesis, promoting osteoblast differentiation, and reducing bone resorption.</p>
    Formula:C19H12N2O3S
    Color and Shape:Solid
    Molecular weight:348.38
  • SGK1-IN-3


    <p>SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.</p>
    Formula:C23H20Cl2N6O3S
    Color and Shape:Solid
    Molecular weight:531.41
  • NPR-C activator 1

    CAS:
    <p>NPR-C activator 1 is an activator of the natriuretic peptide receptor C (NPR-C), which can be used to study cardiovascular diseases.</p>
    Formula:C18H24N6O3
    Purity:98.74%
    Color and Shape:Solid
    Molecular weight:372.42
  • MRS2279

    CAS:
    <p>Selective, high affinity competitive antagonist of the P2Y1 receptor</p>
    Formula:C13H18ClN5O8P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.71
  • Ro-51

    CAS:
    <p>dual P2X3 and P2X2/3 antagonist</p>
    Formula:C17H23IN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:474.29
  • LK-732

    CAS:
    <p>LK-732 is a thrombin inhibitor with antithrombotic activity. It exhibits dose-dependent inhibition in models of hypercoagulability, with an IC50 value of 1.3 mg/kg. LK-732 is used in cardiovascular and cerebrovascular research.</p>
    Formula:C25H29N5O3S
    Color and Shape:Solid
    Molecular weight:479.59
  • Erizepine

    CAS:
    <p>Erizepine, an octopamine receptor 3 (OAR3) antagonist, exhibits a Ki value of 474 nM. This compound is utilized in insect research.</p>
    Formula:C20H22N2
    Color and Shape:Solid
    Molecular weight:290.4
  • BE-10988

    CAS:
    <p>BE-10988 is a DNA topoisomerase (DNAtopoisomerase) inhibitor. It suppresses the growth of P388 murine leukemia cell lines that are resistant to Doxorubicin and Vinblastine by promoting the formation of DNA topoisomerase complexes.</p>
    Formula:C13H10N4O3S
    Color and Shape:Solid
    Molecular weight:302.31
  • KF-19418

    CAS:
    <p>KF-19418 is a follicle stimulant that directly activates follicles in vitro and promotes hair growth in vivo.</p>
    Formula:C21H14N4O
    Color and Shape:Solid
    Molecular weight:338.36
  • SORT1-IN-1

    CAS:
    <p>SORT1-IN-1 (compound 2) is a SORT1 inhibitor.</p>
    Formula:C17H13F3N2O4
    Color and Shape:Solid
    Molecular weight:366.29
  • BM635 mesylate (1493762-74-5 free base)


    <p>BM635 mesylate is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).</p>
    Formula:C26H33FN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.61
  • DJT06001

    CAS:
    <p>DJT06001 is a selective Factor Xa inhibitor, reducing thrombus formation with low risk of bleeding.</p>
    Formula:C21H20ClN3O5S
    Color and Shape:Solid
    Molecular weight:461.92
  • Anticancer agent 28


    <p>Anticancer agent 28 is 50x more potent than Oridonin, IC50 of 0.09 μM against K562; effective in H22 mouse tumors.</p>
    Formula:C28H33NO6
    Color and Shape:Solid
    Molecular weight:479.56
  • Hcyb1


    <p>Hcyb1 specifically inhibits PDE2A with 0.57 μM IC50, over 250x selective, and has neuroprotective and antidepressant effects.</p>
    Formula:C24H20N4O
    Color and Shape:Solid
    Molecular weight:380.44
  • NB-216

    CAS:
    <p>NB-216 is a macrocyclic peptidic BACE-1 inhibitor.</p>
    Formula:C35H45N3O4
    Color and Shape:Solid
    Molecular weight:571.75
  • 6-Hydroxytetrangulol

    CAS:
    <p>6-Hydroxytetrangulol is an inducer of CPP32 protease found in Streptomyces.</p>
    Formula:C19H12O5
    Color and Shape:Solid
    Molecular weight:320.30
  • Lycopodine

    CAS:
    <p>Lycopodine, a bioactive compound derived from Lycopodium clavatum spores, effectively inhibits the proliferation of HeLa cells through the induction of</p>
    Formula:C16H25NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:247.38
  • H-Glu(4MβNA)-OH

    CAS:
    <p>H-Glu(4MβNA)-OH serves as a substrate for aminopeptidases (APs).</p>
    Formula:C16H18N2O4
    Color and Shape:Solid
    Molecular weight:302.33
  • Axl-IN-3


    <p>Axl-IN-3 is a selective, potent and orally active inhibitor of AXL kinase (IC50: 41.5 nM) and has a low inhibitory effect on other kinases.</p>
    Formula:C24H25ClN6O2
    Color and Shape:Solid
    Molecular weight:464.95
  • Hesperidin dihydrochalcone

    CAS:
    Hesperidin dihydrochalcone, a non-toxic sweetener with high sweetness and low calories, exhibits multiple biological activities including anti-oxidation, liver and kidney protection, bacteriostasis, and enhancement of gastrointestinal health.
    Formula:C28H36O15
    Color and Shape:Solid
    Molecular weight:612.58
  • XR8-89

    CAS:
    <p>XR8-89, a potent PLpro inhibitor (IC50=0.1μM), blocks SARS-CoV-2 replication; useful for research.</p>
    Formula:C29H36N4O2S
    Color and Shape:Solid
    Molecular weight:504.69
  • Epicochlioquinone A

    CAS:
    <p>Epicochlioquinone A inhibits rat liver microsomal ACAT with an IC50 of 1.7 μM and inhibits plasma lecithin-cholesterol acyltransferase (LCAT) with an IC50 of 15.8 μM. At a dosage of 75 mg/kg, it can reduce cholesterol absorption in rats by 50%.</p>
    Formula:C30H44O8
    Color and Shape:Solid
    Molecular weight:532.666
  • Papyracon D

    CAS:
    <p>Papyracon D exhibits moderate inhibitory effects on L1210 and HL60 cells and shows mild inhibition against nematodes. It also has a slight inhibitory effect on Gram-positive bacteria.</p>
    Formula:C14H18O5
    Molecular weight:266.29
  • Antitrypanosomal agent 6


    <p>Compound 18a: potent vs. T. brucei (IC50: 0.47 μM), &gt;2x efficacy compared to Nifurtimox, good ADME, binds AT-rich DNA.</p>
    Formula:C22H29Cl2N5O
    Color and Shape:Solid
    Molecular weight:450.4
  • Dihydropergillin

    CAS:
    <p>Dihydropergillin is produced by the Aspergillus terreus strain (ATCC 38849) and has the ability to inhibit plant growth.</p>
    Formula:C15H18O4
    Molecular weight:262.30
  • PEN-866

    CAS:
    <p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>
    Formula:C49H49N7O9
    Color and Shape:Solid
    Molecular weight:879.95
  • hTrkA-IN-2


    <p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>
    Formula:C24H22F3N5O3
    Color and Shape:Solid
    Molecular weight:485.46
  • Oral antiplatelet agent 1

    CAS:
    <p>Oral antiplatelet agent 1 is a potent antiplatelet agent with an IC50 of 2.94 μM in vitro.</p>
    Formula:C23H24N4O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:468.53
  • BMS-751324

    CAS:
    <p>BMS-751324: p38α MAPK inhibitor with carbamyl-methyl, esters, phosphate from HPA. Reduces rat arthritis swelling and TNFα.</p>
    Formula:C32H35N6O10P
    Color and Shape:Solid
    Molecular weight:694.63
  • HbF inducer-1


    <p>HbF inducer-1 is a fetal hemoglobin inducer which is orally bioavailable.</p>
    Formula:C18H19N3O3
    Color and Shape:Solid
    Molecular weight:325.36
  • PDE4B-IN-3


    <p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>
    Formula:C30H35N3O4S2
    Color and Shape:Solid
    Molecular weight:565.75
  • Fipronil desulfinyl

    CAS:
    <p>Fipronil desulfinyl, a photodegradation product of the insecticide Fipronil, exhibits similar in vivo toxicity to Fipronil and possesses higher environmental toxicity.</p>
    Formula:C12H4Cl2F6N4
    Color and Shape:Solid
    Molecular weight:389.08
  • Kalafungin

    CAS:
    <p>Kalafungin inhibits various fungi, yeasts, protozoa, and gram-positive bacteria, less so for gram-negative bacteria.</p>
    Formula:C16H12O6
    Color and Shape:Solid
    Molecular weight:300.26
  • CI 922

    CAS:
    <p>CI 922 is an anaphylaxis mediator release inhibitor. It inhibits the activation of human neutrophils.</p>
    Formula:C26H30N10O6
    Color and Shape:Solid
    Molecular weight:578.58
  • FPR2 agonist 2


    <p>Potent FPR2 agonist, crosses blood-brain barrier, EC50: 0.13 nM; reduces inflammation and mitochondrial dysfunction, inhibits caspase-3.</p>
    Formula:C25H20F2N4O2
    Color and Shape:Solid
    Molecular weight:446.45
  • DSP-6952

    CAS:
    <p>DSP-6952 is a 5-HT4 receptor partial agonist, inhibiting visceral hypersensitivity and ameliorating gastrointestinal dysfunction.</p>
    Formula:C21H32BrClN4O5
    Color and Shape:Solid
    Molecular weight:535.86
  • Iroxanadine hydrobromide

    CAS:
    <p>Iroxanadine hydrobromide is a MAPK p38 inhibitor potentially for the treatment of atherosclerosis.</p>
    Formula:C14H21BrN4O
    Color and Shape:Solid
    Molecular weight:341.25
  • Flusoxolol

    CAS:
    <p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>
    Formula:C22H30FNO4
    Color and Shape:Solid
    Molecular weight:391.48
  • LY 178210

    CAS:
    <p>LY 178210 is a 5-hydroxytryptamine receptor agonist.</p>
    Formula:C18H25N3O
    Color and Shape:Solid
    Molecular weight:299.41
  • MB-7133

    CAS:
    <p>MB-7133 is an inhibitor of DNA synthesis.</p>
    Formula:C17H21N4O8P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.34
  • Antiviral agent 15


    <p>Compound 15f, a Clofazimine derivative, inhibits rabies (EC50: 1.45 μM) and SARS-CoV-2 (EC50: 14.6 μM).</p>
    Formula:C27H24FN5O
    Color and Shape:Solid
    Molecular weight:453.51
  • MSX-3 free acid

    CAS:
    <p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>
    Formula:C21H23N4O7P
    Color and Shape:Solid
    Molecular weight:474.40
  • ETP-47037

    CAS:
    <p>ETP-47037: strong PI3Kα inhibitor (IC50: 0.99 nM), also targets PI3Kβ, δ, γ; may protect telomeres.</p>
    Formula:C20H27N9O3S
    Color and Shape:Solid
    Molecular weight:473.55
  • VEGFR-2-IN-26

    CAS:
    <p>VEGFR-2-IN-26 inhibits VEGFR-2 (IC50: 15.5 nM), combating various cancers' cell growth.</p>
    Formula:C24H19F3N6O2
    Color and Shape:Solid
    Molecular weight:480.44
  • P-gp modulator 1

    CAS:
    <p>P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulator</p>
    Formula:C41H72N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:689.02
  • WM382

    CAS:
    <p>WM382, a potent dual PMIX/X inhibitor, has IC50s of 1.4 nM/0.03 nM and effective against various malaria stages.</p>
    Formula:C29H36N4O4
    Color and Shape:Solid
    Molecular weight:504.62
  • MDL-43291

    CAS:
    <p>MDL-43291 is a leukotriene receptor antagonist.</p>
    Formula:C25H42O4S
    Color and Shape:Solid
    Molecular weight:438.66
  • SARS-CoV-2-IN-8


    <p>SARS-CoV-2-IN-8 is a major protease inhibitor of SARS-CoV-2 (IC50: 0.75 μM).</p>
    Formula:C35H38N6O3
    Color and Shape:Solid
    Molecular weight:590.71
  • MV061194

    CAS:
    <p>MV061194 is a potent and selective cathepsin K (Cat K) inhibitor.</p>
    Formula:C28H37N5O4S
    Color and Shape:Solid
    Molecular weight:539.69
  • Sargachromanol E

    CAS:
    <p>Sargachromanol E is a compound isolated from the marine brown alga, Sargassum horneri. It has been studied for its inhibitory effect on skin ageing.</p>
    Formula:C27H40O4
    Color and Shape:Solid
    Molecular weight:428.6
  • 5,6-Dihydro-4-methoxy-2H-pyran-2-one

    CAS:
    <p>5,6-Dihydro-4-methoxy-2H-pyran-2-one is produced by the Penicillium italicum strain MRC 1360.</p>
    Formula:C6H8O3
    Molecular weight:128.13
  • Monorden diacetate

    CAS:
    <p>Monorden diacetate a Hsp90 Inhibitor. Monorden diacetate is a Promising Lead Compound for the Development of Novel Fungicides.</p>
    Formula:C22H21ClO8
    Color and Shape:Solid
    Molecular weight:448.85
  • Quorum Sensing-IN-1


    <p>Quorum Sensing-IN-1 is a small-molecule inhibitor of quorum sensing.</p>
    Formula:C13H10N2O2S2
    Color and Shape:Solid
    Molecular weight:290.36
  • Piperazinomycin

    CAS:
    <p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>
    Formula:C18H20N2O2
    Color and Shape:Solid
    Molecular weight:296.36
  • 18-Deoxyherboxidiene

    CAS:
    <p>18-Deoxyherboxidiene (RQN-18690A) inhibits angiogenesis, targeting SF3b in U2 snRNP spliceosome, affects HUVEC, useful for cancer research.</p>
    Formula:C25H42O5
    Color and Shape:Solid
    Molecular weight:422.6
  • PLAP-IN-1

    CAS:
    <p>PLAP-IN-1: Potent, selective inhibitor of PLAP, IC50 of 32 nM; doesn't notably inhibit TNAP.</p>
    Formula:C25H21Cl2N3O5
    Color and Shape:Soild
    Molecular weight:514.36
  • MDL-27210

    CAS:
    <p>MDL-27210 is the ethyl ester prodrug of a potent angiotensin-converting enzyme inhibitor, MDL-27088.</p>
    Formula:C27H32N2O5
    Color and Shape:Solid
    Molecular weight:464.55
  • KNI 10033

    CAS:
    <p>KNI 10033 is a potent inhibitor of HIV protease</p>
    Formula:C40H45N5O7S2
    Color and Shape:Solid
    Molecular weight:771.95
  • GK241

    CAS:
    <p>GK241 (compound 31a-c), a 2-oxoamide-based compound, exhibits inhibitory activity against group IIA secretory phospholipase A2 (GIIA sPLA2) in humans and mice, with IC50 values of 143 nM and 68 nM, respectively. The mechanism of inhibition has been explored through molecular dynamics simulations.</p>
    Formula:C21H39NO4
    Color and Shape:Solid
    Molecular weight:369.54