Other Inhibitors
This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.
Found 37926 products of "Other Inhibitors"
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Vulolisib
CAS:<p>Vulolisib inhibits PI3K (α: IC50 0.2nM, β: 168nM, γ: 90nM, δ: 49nM), taken orally with anti-cancer properties.</p>Formula:C18H19F2N5O3SColor and Shape:SolidMolecular weight:423.44Terfluranol
CAS:<p>Terfluranol, a benzyl derivative, is utilized as an antitumor medication.</p>Formula:C17H17F3O2Color and Shape:SolidMolecular weight:310.31PRN694
CAS:<p>PRN694 is a potent, irreversible ITK/RLK inhibitor with IC50s: 0.3/1.4 nM; offers lasting effector cell suppression.</p>Formula:C28H35F2N5O2SPurity:98%Color and Shape:SolidMolecular weight:543.67AMG-315
CAS:<p>AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.</p>Formula:C24H41NO2Color and Shape:SolidMolecular weight:375.59SID 125240931
CAS:<p>SID 125240931 is a regulator of fluorine-activated proteins (FAPs). This compound disrupts the binding between fluoride and FAPs.</p>Formula:C19H24N4O3SColor and Shape:SolidMolecular weight:388.48BI-1388
CAS:<p>BI-1388 is a potent HCV NS3 protease inhibitor; halts replication across genotypes, including D168V/R155K mutants.</p>Formula:C41H53N7O9SColor and Shape:SolidMolecular weight:819.97HMGB1-IN-3
CAS:<p>HMGB1-IN-3 (compound E), a derivative of glycyrrhizic acid, exhibits potent inhibitory effects on HMGB1 (high mobility group protein 1). It is utilized in research related to intracerebral hemorrhage.</p>Formula:C31H46O4Color and Shape:SolidMolecular weight:482.69GNE-616
CAS:<p>GNE-616: a potent, stable, oral Nav1.7 inhibitor; Ki: 0.79 nM, Kd: 0.38 nM; for chronic pain.</p>Formula:C24H23F4N5O3SPurity:98%Color and Shape:SolidMolecular weight:537.53KY-02327 acetate
<p>KY-02327 acetate inhibits Dvl-CXXC5, stabilizes Wnt/β-catenin signaling, and enhances osteoblast differentiation.</p>Formula:C22H31N3O6Color and Shape:SolidMolecular weight:433.5Cenicriviroc Sulfone
CAS:<p>Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.</p>Formula:C41H52N4O5SColor and Shape:SolidMolecular weight:712.94Resolvin E4
CAS:<p>RvE4, a bioactive lipid from eicosapentaenoic acid and synthesized by 15-LO, is anti-inflammatory and boosts efferocytosis in human macrophages.</p>Formula:C20H30O4Color and Shape:SolidMolecular weight:334.45D6808
<p>D6808: selective c-Met inhibitor, IC50=2.9 nM, induces apoptosis and cell cycle arrest, for NSCLC/gastric cancer research.</p>Formula:C30H25F3N6O2Color and Shape:SolidMolecular weight:558.55AVE 0991
CAS:<p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>Formula:C29H32N4O5S2Purity:98.69%Color and Shape:SolidMolecular weight:580.72KFA1982
CAS:<p>KFA1982 is a novel and potent factor Xa inhibitor.</p>Formula:C28H34ClN3O9S2Color and Shape:SolidMolecular weight:656.17ONL-1204
CAS:<p>ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.</p>Formula:C71H100N18O16Color and Shape:SolidMolecular weight:1461.66ODN 21158
CAS:<p>ODN 21158 is a potent, non-cytotoxic inhibitor of G-modified TLR3 and TLR9. ODN 21158 dose-dependently inhibits IFN-α secretion.</p>Color and Shape:SolidGG-43
<p>GG-43 is a potent inhibitor of LIN28. The IC50 value of GG-43 against human LIN28A is 4 μM [1].</p>Formula:C21H21NO3Color and Shape:SolidMolecular weight:335.4Heme Oxygenase-2-IN-1
<p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>Formula:C19H17N3O2Color and Shape:SolidMolecular weight:319.36Balanol
CAS:<p>Balanol is an ATP-competitive Protein Kinase C and Protein Kinase A inhibitor.</p>Formula:C28H26N2O10Color and Shape:SolidMolecular weight:550.51EP4 receptor antagonist 2
CAS:<p>EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.</p>Formula:C27H29N3O5Color and Shape:SolidMolecular weight:475.54Croconic acid disodium
CAS:<p>Croconic acid (disodium) (Nacr) enhances gene expression related to lysine crotonylation (Kcr) modification, which promotes cell growth and proliferation. This compound also shows promise in boosting somatic cell nuclear transfer (SCNT) efficiency and optimizing research in cell culture conditions.</p>Formula:C5Na2O5Color and Shape:SolidMolecular weight:186.03ONO-AE1-259 lysine
CAS:<p>ONO-AE1-259 is a highly selective agonist of prostaglandin e2 receptor (ep2)</p>Formula:C28H49ClN2O6Color and Shape:SolidMolecular weight:545.15Hcyb1
<p>Hcyb1 specifically inhibits PDE2A with 0.57 μM IC50, over 250x selective, and has neuroprotective and antidepressant effects.</p>Formula:C24H20N4OColor and Shape:SolidMolecular weight:380.44Anticancer agent 27
<p>Anticancer agent 27 is a promising candidate for the treatment of cancer and deserves further development.</p>Formula:C28H31NO6Color and Shape:SolidMolecular weight:477.55DMP-728 free base
CAS:<p>DMP-728 free base is a highly potent and selective GPIIbDIIa antagonist</p>Formula:C25H36N8O7Color and Shape:SolidMolecular weight:560.60Azonafide-PEABA
CAS:<p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>Formula:C32H33N5O4Purity:98%Color and Shape:SolidMolecular weight:551.64Calphostin D
CAS:<p>Calphostins, PKC inhibitors from Cladosporium cladosporioides, include A, B, C, D, I; C is most potent.</p>Formula:C30H30O10Color and Shape:SolidMolecular weight:550.55Tonantzitlolone
CAS:<p>Tonantzitlolone activates TRPC1/4/5 channels, PKCα/θ, inhibits IRS1/PI3K/AKT, and triggers HSF1 to induce glucose dependence.</p>Formula:C26H40O7Color and Shape:SolidMolecular weight:464.592,3-dinor-11β-Prostaglandin F2α
CAS:<p>2,3-dinor-11β-Prostaglandin F2α (2,3-dinor-11β-PGF2α) was recovered from the urine of both normal monkeys and humans when infused with radiolabeled PGD2, where</p>Formula:C18H30O5Color and Shape:SolidMolecular weight:326.43PPO-IN-15
CAS:<p>PPO-IN-15 (compound (R)-I-5) serves as an inhibitor of protoporphyrinogen IX oxidase (PPO), offering efficacy against resistant weeds while maintaining safety for wheat and rice.</p>Formula:C17H18ClFN4O5SColor and Shape:SolidMolecular weight:444.87SHR902275
CAS:<p>SHR902275: potent RAF inhibitor, hits RAS mutations, oral use. cRAF IC50=1.6 nM, bRAFwt IC50=10 nM, bRAFV600E IC50=5.7 nM, hinders cell growth.</p>Formula:C26H23F3N4O4Color and Shape:SolidMolecular weight:512.48Tandutinib (MLN518) HCl
<p>Tandutinib antagonizes FLT3, PDGFR, and c-Kit with an IC50 of ~200 nM.</p>Formula:C31H43ClN6O4Purity:98%Color and Shape:SolidMolecular weight:599.16(S)-Dexfadrostat
CAS:<p>(S)-Dexfadrostat ((S)-Fadrozole), an aromatase inhibitor, exhibits an IC 50 of 4.6 nM in in vitro assays using human placental microsomes. It is applicable for research on estrogen-dependent breast cancer, gynecomastia, and systemic lupus erythematosus.</p>Formula:C14H13N3Color and Shape:SolidMolecular weight:223.27AVE-1330A free acid
CAS:<p>AVE-1330A free acid is a broad-spectrum non-beta-lactam beta-lactamase inhibitor.</p>Formula:C7H11N3O6SColor and Shape:SolidMolecular weight:265.24Esorubicin
CAS:<p>Esorubicin, a doxorubicin derivative, intercalates DNA, inhibits topoisomerase II, has less cardiotoxicity, but more myelosuppression.</p>Formula:C27H29NO10Color and Shape:SolidMolecular weight:527.52LPM4870108
<p>LPM4870108: Potent, oral pan-Trk inhibitor, selective over ALK, with anti-tumor effects. TrkC IC50=0.2nM, TrkA IC50=2.4nM.</p>Formula:C20H19FN6O3Color and Shape:SolidMolecular weight:410.4UNC7467
CAS:<p>UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.</p>Formula:C20H13NO3Purity:98.28% - 98.64%Color and Shape:SoildMolecular weight:315.325(S),6(R)-DiHETE
CAS:<p>5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.</p>Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47Isobetanin
CAS:<p>Isobetanin is a betacyanin that has been shown to enhance vitexin-2-O-xyloside mediated inhibition of proliferation of T24 bladder cancer cells.</p>Formula:C24H26N2O13Color and Shape:SolidMolecular weight:550.47OM-153
CAS:<p>OM-153 blocks tankyrase 1 (IC50: 13 nM) and 2 (IC50: 2 nM), stifling WNT signaling and COLO 320DM cell growth.</p>Formula:C28H24FN7O2Color and Shape:SolidMolecular weight:509.53CGS 22652
CAS:<p>CGS 22652 has thromboxane receptor antagonism combined with thromboxane synthase inhibition.</p>Formula:C22H29ClN2O4SColor and Shape:SolidMolecular weight:452.99P2X receptor-1
<p>P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.</p>Formula:C14H14ClN3O3S2Color and Shape:SolidMolecular weight:371.86BMS-554417
CAS:<p>BMS-554417 inhibits IGF-IR/insulin receptors, curbing cell proliferation and tumor growth, with IC50 values of 120 nm–>8.5 μmol/L.</p>Formula:C28H30ClN7O2Color and Shape:SolidMolecular weight:532.04Antibiotic MA 144M2
CAS:<p>Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.</p>Formula:C42H55NO16Color and Shape:SolidMolecular weight:829.88AFM-30a hydrochloride
<p>AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.</p>Formula:C24H28ClFN6O3Color and Shape:SolidMolecular weight:502.97Cofpropamine
CAS:<p>Cofpropamine, a caffeine derivative that inhibits polyadenylation, enhances the suppressive effects of Cyclophosphamide in animal models of rat adjuvant arthritis and mouse collagen-induced arthritis.</p>Formula:C13H21N5O3Color and Shape:SolidMolecular weight:295.34(6S)-CP-470711
CAS:<p>(6S)-CP-470711 (Compound 8) acts as an inhibitor of sorbitol dehydrogenase (SDH) in both humans and rats, exhibiting inhibitory concentrations (IC50) of 19 nM and 27 nM, respectively. Additionally, (6S)-CP-470711 has been shown to ameliorate diabetes in rats induced by Streptozotocin.</p>Formula:C18H26N6O2Color and Shape:SolidMolecular weight:358.44NB-216
CAS:<p>NB-216 is a macrocyclic peptidic BACE-1 inhibitor.</p>Formula:C35H45N3O4Color and Shape:SolidMolecular weight:571.75Anti-inflammatory agent 12
<p>Pentacyclic triterpene, anti-inflammatory agent 12, inhibits LPS inflammation (IC50: 2.22 μM). May benefit inflammatory disease studies.</p>Formula:C30H50O4Color and Shape:SolidMolecular weight:474.72Amrubicin HCl
CAS:<p>Amrubicin (SM-5887), an anthracycline, treats lung cancer by inhibiting DNA replication and topoisomerase II, with less cardiac toxicity.</p>Formula:C25H25NO9Color and Shape:SolidMolecular weight:483.47TA-316
CAS:<p>Agent induces megakaryocytes/platelets from stem cells to treat thrombopenia.</p>Formula:C28H25BrN4O5S2Purity:98%Color and Shape:SolidMolecular weight:641.56AZ-PFKFB3-67 quarterhydrate
<p>AZ-PFKFB3-67 quarterhydrate inhibits PFKFB3 (IC50: 11 nM), PFKFB2 (159 nM), and PFKFB1 (1130 nM).</p>Formula:C26H27N5O4Color and Shape:SolidMolecular weight:460.01XN methyl pyrazole
<p>XN methyl pyrazole exhibits beneficial effects on diet-induced obesity and enhances energy expenditure in mice fed with a high-fat diet [1].</p>Formula:C22H24N2O4Color and Shape:SolidMolecular weight:380.44Lp-PLA2-IN-6
CAS:<p>Lp-PLA2-IN-6: Potent tetracyclic inhibitor of rhLp-PLA2, with pIC50 of 10.0, and potential in neurodegenerative research.</p>Formula:C25H21F5N4O3Color and Shape:SolidMolecular weight:520.45Heparastatin
CAS:<p>Heparastatin is an inhibitor of heparanase.</p>Formula:C8H11F3N2O5Purity:98%Color and Shape:SolidMolecular weight:272.18ER272
CAS:<p>ER272 is a natural PKC activator, inducing hippocampal neurogenesis.</p>Formula:C24H34O6Color and Shape:SolidMolecular weight:418.52LX2761
CAS:<p>LX2761 is a stable inhibitor for SGLT1/2 with IC50s of 2.2/2.7 nM; it targets SGLT1 in the GI tract.</p>Formula:C32H47N3O6SPurity:98%Color and Shape:SolidMolecular weight:601.80Antibiotic MA 144M1
CAS:<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formula:C42H55NO15Color and Shape:SolidMolecular weight:813.88Ribocil-C R enantiomer
<p>Ribocil-C R enantiomer is the R enantiomer of Ribocil-C. Ribocil-C is a highly selective bacterial riboflavin riboswitches inhibitor.</p>Formula:C21H21N7OSPurity:98%Color and Shape:SolidMolecular weight:419.5Topoisomerase II inhibitor 6
<p>Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.</p>Formula:C19H18N4O2Color and Shape:SolidMolecular weight:334.37Diospyrin
CAS:<p>Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.</p>Formula:C22H14O6Color and Shape:SolidMolecular weight:374.34Thiomuscimol hydrobromide
CAS:<p>Thiomuscimol hydrobromide is an agonist of GABAA receptor.</p>Formula:C4H6N2OSPurity:98%Color and Shape:SolidMolecular weight:130.17Exicorilant
CAS:<p>Exicorilant is a selective oral GR antagonist (Ki: 7 nM) that may reduce obesity, glucose intolerance, & dyslipidemia.</p>Formula:C26H23F4N7O3SPurity:98%Color and Shape:SolidMolecular weight:589.56PDE4-IN-14
CAS:<p>PDE4-IN-14 (Compound 1) serves as an inhibitor of phosphodiesterase 4 (PDE4), applicable in research concerning diseases associated with PDE4, including</p>Formula:C19H20F2N4O3SColor and Shape:SolidMolecular weight:422.45Cilazapril HCl
CAS:<p>Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension.</p>Formula:C22H32ClN3O5Color and Shape:SolidMolecular weight:453.96BAY-091
CAS:<p>BAY-091 is a novel potent and highly selective PIP4K2A kinase inhibitor.</p>Formula:C26H21FN4O2Purity:97.66% - 99.23%Color and Shape:SoildMolecular weight:440.47FTO-IN-4
CAS:<p>FTO-IN-4 is a potent and selective inhibitor of adiposity and obesity-associated protein (FTO).</p>Formula:C22H16Cl2N6O6Color and Shape:SolidMolecular weight:531.31B-3852
CAS:<p>B-3852 is a Bradykinin inhibitor.</p>Formula:C55H74F3N15O11Color and Shape:SolidMolecular weight:1178.27rel-MDM2/4-p53-IN-3
<p>rel-MDM2/4-p53-IN-3 inhibits MDM2/4-p53 PPI, IC50: MDM2 18.5nM, MDM4 14.8nM, targets cancer research.</p>Formula:C25H24Cl2FN3O3Color and Shape:SolidMolecular weight:504.38LY3325656
CAS:<p>LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.</p>Formula:C21H23F3N6O2Color and Shape:SolidMolecular weight:448.44AD5075
CAS:<p>AD5075 is a bioactive chemical.</p>Formula:C22H20N2O5SColor and Shape:SolidMolecular weight:424.477(Z),11(Z)-Nonacosadiene
CAS:<p>7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.</p>Formula:C29H56Color and Shape:SolidMolecular weight:404.75Motuporin
CAS:<p>Motuporin is an inhibitor of type-1 and type-2A protein phosphatase catalytic subunits (PP-1c and PP-2Ac).</p>Formula:C40H57N5O10Color and Shape:SolidMolecular weight:767.91Ataprost
CAS:<p>Ataprost (ONO 41483), an oral Carboprostacyclin analogue, is 2.6x more potent in inhibiting ADP-induced platelet aggregation and can relieve coronary spasm.</p>Formula:C21H32O4Color and Shape:SolidMolecular weight:348.48Amdinocillin methylacetate
CAS:<p>Amdinocillin methylacetate is a Synthetic penicillin.</p>Formula:C18H27N3O4SColor and Shape:SolidMolecular weight:381.49ONO-DI-004
CAS:<p>ONO-DI-004 is a selective EP1 Prostanoid receptor agonist.</p>Formula:C24H38O6Color and Shape:SolidMolecular weight:422.55Oxeclosporin
CAS:<p>Oxeclosporin is a hydroxyethyl derivative of serine(8)-cyclosporine; inhibits proliferation and functions of lymphocytes.</p>Formula:C64H115N11O14Color and Shape:SolidMolecular weight:1262.66Griseorhodin G
CAS:<p>Griseorhodin G is a quinone antibiotic with antitumor activity.</p>Formula:C25H18O12Molecular weight:510.40Epoxyquinomicin B
CAS:<p>Epoxyquinomicin B is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus, with a minimum inhibitory concentration (MIC) of 6.25-12.5 µg/mL. It also shows cytotoxicity in cancer cells L1210, with an IC50 of 16.3 µg/mL. Additionally, Epoxyquinomicin B demonstrates anti-inflammatory effects on collagen-induced arthritis.</p>Formula:C14H11NO6Color and Shape:SolidMolecular weight:289.24Milbemycin α13
CAS:<p>Milbemycin α13 (Meilingmycin B) is an antibiotic that is effective against nematodes and mites.</p>Formula:C37H52O9Molecular weight:640.80Orvepitant
CAS:<p>Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.</p>Formula:C31H35F7N4O2Color and Shape:SolidMolecular weight:628.62Polyoxin K
CAS:<p>Polyoxin K is a nucleoside antifungal antibiotic that exhibits significant effectiveness against rice sheath blight.</p>Formula:C22H30N6O13Molecular weight:586.51ALK5-IN-7
CAS:<p>ALK5-IN-7 inhibits ALK5, useful in TGF-β disease research like cancer, fibrosis, and autoimmune disorders. See WO2021129621A1.</p>Formula:C26H28N4O3SColor and Shape:SolidMolecular weight:476.59Unoprostone isopropyl
CAS:<p>Unoprostone isopropyl, a prostanoid and synthetic docosanoid, is approved for the treatment of ocular hypertension and open-angle glaucoma.</p>Formula:C25H44O5Purity:98%Color and Shape:SolidMolecular weight:424.61Plm IV inhibitor-2
CAS:<p>"Plm IV inhibitor-2: Potent for Plm IV (IC50=24nM), affects Plm II/Plm I; malaria research compound."</p>Formula:C39H54N4O4Color and Shape:SolidMolecular weight:642.87Sovesudil hydrochloride
<p>Sovesudil (PHP-201) HCl: potent local ROCK inhibitor; targets ROCK I/II (IC50: 3.7/2.3 nM); lowers IOP, non-congesting.</p>Formula:C23H23ClFN3O3Color and Shape:SolidMolecular weight:443.9DD04107
CAS:<p>DD04107 inhibits α-CGRP release, targets Synaptotagmin 1 in sensory neurons.</p>Formula:C48H88N14O12SColor and Shape:SolidMolecular weight:1085.36eIF4A3-IN-4
<p>eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).</p>Formula:C24H20N2O5Color and Shape:SolidMolecular weight:416.43Amidinomycin
CAS:<p>Amidinomycin primarily acts against Gram-positive bacteria.</p>Formula:C9H18N4OMolecular weight:198.27Hexedine
CAS:<p>Hexedine is a biochemical.</p>Formula:C22H45N3Color and Shape:SolidMolecular weight:351.61PDE4B-IN-3
<p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>Formula:C30H35N3O4S2Color and Shape:SolidMolecular weight:565.75TEI-9063
CAS:<p>TEI-9063 is a stable and highly specific prostacyclin analogue of prostacyclin receptor in mast cell tumor p-815 cells.</p>Formula:C23H38O4Color and Shape:SolidMolecular weight:378.55GZN39838
CAS:<p>GZN39838, a natural Kv1.2 blocker, induces C-type inactivation without blocking the outer pore.</p>Formula:C22H30O6Color and Shape:SolidMolecular weight:390.47(1R,3S)-THCCA-Asn
<p>(1R,3S)-THCCA-Asn (4j) is a selective inhibitor of thrombin (IC50: 0.07-0.14 μM) with anti-thrombotic effects.</p>Formula:C24H24N4O6Color and Shape:SolidMolecular weight:464.47Griseolutein A
CAS:<p>Griseolutein A exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C17H14N2O6Color and Shape:SolidMolecular weight:342.303Retezorogant
CAS:<p>Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.</p>Formula:C23H33ClN2O3Color and Shape:SolidMolecular weight:420.97PGDM
CAS:<p>PGD2 is involved in allergy, asthma, sleep, temperature regulation, inhibits clotting, and relaxes blood vessels; PGDM, its metabolite, is a biomarker.</p>Formula:C16H24O7Color and Shape:SolidMolecular weight:328.366-Hydroxytetrangulol
CAS:<p>6-Hydroxytetrangulol is an inducer of CPP32 protease found in Streptomyces.</p>Formula:C19H12O5Color and Shape:SolidMolecular weight:320.30Cervicarcin
CAS:<p>Cervicarcin is an antitumor antibiotic (antibiotic) exhibiting strong inhibitory effects on sarcoma 180 and sarcoma NF, while showing weaker activity against sarcoma 37, Ehrlich ascites carcinoma, and Freund leukemia.</p>Formula:C19H20O9Color and Shape:SolidMolecular weight:392.357KOS-1584
CAS:<p>KOS-1584, a safer, more effective epothilone, inhibits cell division by stabilizing microtubules and evading P-gp.</p>Formula:C27H39NO5SColor and Shape:SolidMolecular weight:489.67Saframycin Mx2
CAS:<p>Saframycin Mx2 exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C29H38N4O8Color and Shape:SolidMolecular weight:570.634Arverapamil
CAS:<p>Arverapamil is a chiral metabolite of Verapamil.</p>Formula:C26H36N2O4Color and Shape:SolidMolecular weight:440.58Harziphilone
CAS:<p>Harziphilone exhibits mild activity against Gram-positive bacteria and possesses antitumor properties, showing inhibitory effects on lymphocytic leukemia L1210 and leukemia P388 with an IC50 of 0.26 μg/mL. Additionally, Harziphilone inhibits the binding of the Rev protein to [33P]-labeled Rev response element (RRE) RNA, with an IC50 of 2.0 μM.</p>Formula:C15H18O4Color and Shape:SolidMolecular weight:262.3013,4-Dimethoxytropolone
CAS:<p>3,4-Dimethoxytropolone can be isolated from the fermentation broth of Streptoverticillium hadanonense, and it shows activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C9H10O4Color and Shape:SolidMolecular weight:182.173PARP-1-IN-1
<p>PARP-1-IN-1: Selective, oral PARP-1 inhibitor with 0.96 nM IC50; well-tolerated and effective in single-dose MDA-MB-436 model.</p>Formula:C23H25FN4OColor and Shape:SolidMolecular weight:392.47PNU-140457
CAS:<p>PNU-140457 is a bio-active chemical.</p>Formula:C14H14FN5O3Color and Shape:SolidMolecular weight:319.29PPARγ agonist 2
<p>PPARγ agonist 2 is a highly effective compound that acts as a partial agonist for PPARγ.</p>Formula:C24H20O5Color and Shape:SolidMolecular weight:388.414α-PDD
CAS:<p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>Formula:C40H64O8Color and Shape:SolidMolecular weight:672.93Megovalicin G
CAS:<p>Megovalicin G is effective against Bacillus subtilis and Escherichia coli, and it also acts on Pseudomonas aeruginosa.</p>Formula:C35H61NO7Color and Shape:SolidMolecular weight:607.86Gusperimus
CAS:<p>Gusperimus was synthesized by chemical modification of spergualin and in combination with cyclosporine A to prevent diabetes in susceptible NOD mice.</p>Formula:C17H37N7O3Color and Shape:SolidMolecular weight:387.529-Hydroxycrisamicin
CAS:<p>9-Hydroxycrisamicin exhibits moderate activity against Gram-positive bacteria with a minimum inhibitory concentration (MIC) ranging from 6.25 to 25 μg/mL. Additionally, 9-Hydroxycrisamicin demonstrates significant growth inhibition towards various human tumor cell lines.</p>Formula:C32H22O13Color and Shape:SolidMolecular weight:614.51SARS-CoV-2 nsp14-IN-2
<p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>Formula:C21H21N5O5SColor and Shape:SolidMolecular weight:455.49Iroxanadine hydrobromide
CAS:<p>Iroxanadine hydrobromide is a MAPK p38 inhibitor potentially for the treatment of atherosclerosis.</p>Formula:C14H21BrN4OColor and Shape:SolidMolecular weight:341.25Flusoxolol
CAS:<p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>Formula:C22H30FNO4Color and Shape:SolidMolecular weight:391.48Mifepristone methochloride
CAS:<p>Mifepristone methochloride is a glucocorticoid antagonist. This product will be sold for research use only.</p>Formula:C30H38ClNO2Color and Shape:SolidMolecular weight:480.08Coriolin A
CAS:<p>Coriolin A exhibits activity against gram-positive bacteria, weakly against gram-negative bacteria, as well as yeasts and Trichomonas vaginalis. At a concentration of 5 μg/mL, it inhibits 61.6% of the growth of Yoshida sarcoma, but shows no inhibitory effect on Ehrlich ascites carcinoma in animals.</p>Formula:C15H20O5Color and Shape:SolidMolecular weight:280.316Griseolic acid C
CAS:<p>Griseolic acid C (Dihydrodeoxygriseolic acid) is an antibiotic found in the Streptomyces griseoaurantiacus SANK43894 strain. This compound is a potent inhibitor of cyclic adenosine monophosphate (cAMP) phosphodiesterase [EC 3.1.4.17], with an IC50 of 0.12 μM (enzyme sourced from rat brain tissue).</p>Formula:C14H15N5O7Color and Shape:SolidMolecular weight:365.2983'-O-Decarbamoylirumamycin
CAS:<p>3'-O-Decarbamoylirumamycin is a 20-membered macrolide antibiotic produced by Streptomyces subflavus subsp. irumaensis. It exhibits inhibitory effects against plant pathogenic fungi, such as Pyricularia oryzae and Sclerotinia.</p>Formula:C40H64O11Color and Shape:SolidMolecular weight:720.93Minnelide free acid
CAS:<p>Minnelide treats pancreatic cancer, hinders androgen-related prostate growth, shrinks tumors, and improves survival.</p>Formula:C21H27O10PColor and Shape:SolidMolecular weight:470.41Azicemicin A
CAS:<p>Azicemicin A exhibits mild antibacterial activity and shows no acute toxicity when administered via intraperitoneal injection to mice at a dosage of 150 mg/kg.</p>Formula:C23H25NO9Color and Shape:SolidMolecular weight:459.4468(S),15(S)-DiHETE
CAS:<p>8(S),15(S)-DiHETE, from 15(S)-HETE's oxidation by 15-LO, triggers eosinophil movement at 1.5 μM; it counteracts pain and LTB4 effects.</p>Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47AZD-3199 dihydrobromide
CAS:<p>AZD-3199 dihydrobromide is a β2 adrenergic receptor agonist potentially for the treatment of asthma and chronic obstructive.</p>Formula:C32H44Br2N4O4SColor and Shape:SolidMolecular weight:740.59SAR107375
CAS:<p>SAR107375 is a potent, orally active dual inhibitor of thrombin and factor Xa, with K_i values of 1 nM and 8 nM for factor Xa and thrombin, respectively [1].</p>Formula:C24H30ClN5O5S2Color and Shape:SolidMolecular weight:568.11Azirinomycin
CAS:<p>Azirinomycin exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C4H5NO2Color and Shape:SolidMolecular weight:99.088Gallinamide A
CAS:<p>Gallinamide A is a potent inhibitor of cathepsin L with an IC 50 value of 17.6 pM.</p>Formula:C31H52N4O7Color and Shape:SolidMolecular weight:592.77Cicaprost
CAS:<p>Cicaprost (ZK 96480) is an IP agonist with artery relaxing effects; EC50 is 5.8 nM.</p>Formula:C22H30O5Color and Shape:SolidMolecular weight:374.47Hymenidin
CAS:<p>Hymenidin, isolated from the Okinawan sponge Hymeniacidon sp., is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor.</p>Formula:C11H12BrN5OPurity:96.85% - 99.52%Color and Shape:SolidMolecular weight:310.15Aristoforin
CAS:<p>Aristoforin is a SIRT1 and SIRT2 inhibitor that induces cell cycle arrest, shows potent antitumor effects, and inhibits lymphangiogenesis in vivo.</p>Formula:C37H54O6Color and Shape:SolidMolecular weight:594.82Heme Oxygenase-1-IN-3
CAS:<p>Heme Oxygenase-1-IN-3 (compound 4) serves as a potent and selective inhibitor of heme oxygenase-1 (HO-1) with a dissociation constant (Kd) of 141 nM, making it suitable for use in cancer and neurodegenerative disease research.</p>Formula:C22H18BrFN4O2SColor and Shape:SolidMolecular weight:501.37CVS-1578
CAS:<p>CVS-1578 is a potent serine protease inhibitor, targeting the S2S3 thrombin and FXa subsites.</p>Formula:C20H30N6O5SColor and Shape:SolidMolecular weight:466.55MAP3K14-IN-173
CAS:<p>MAP3K14-IN-173 is a potent MAP3K14 kinase inhibitor.</p>Formula:C29H31N7O2Color and Shape:SolidMolecular weight:509.60Kaitocephalin
CAS:<p>Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.</p>Formula:C18H21Cl2N3O9Color and Shape:SolidMolecular weight:494.28Antitumor agent-75
<p>Antitumor agent-75 is a novel and potent antitumor agent.</p>Formula:C26H23FN6Color and Shape:SolidMolecular weight:438.5Sulprostone
CAS:<p>EP3 and EP1 receptor agonist</p>Formula:C23H31NO7SPurity:98%Color and Shape:White To Off-White SolidMolecular weight:465.56Zurletrectinib
CAS:<p>Zurletrectinib is a tyrosine kinase inhibitor with potential as an antineoplastic agent.</p>Formula:C19H19F2N7O2Color and Shape:SolidMolecular weight:415.4Gilvusmycin
CAS:<p>Gilvusmycin is an antibiotic with potent antitumor properties. It effectively inhibits the proliferation of P388, K562, A431, and MKN28 cells, with IC50 values (ng/mL) of 0.08, 0.86, 0.72, and 0.75, respectively.</p>Formula:C38H34N6O8Color and Shape:SolidMolecular weight:702.712SSTR5 antagonist 2 TFA
CAS:<p>Potent, oral SSTR5 antagonist 2 TFA may treat type 2 diabetes.</p>Formula:C34H36F4N2O7Purity:98%Color and Shape:SolidMolecular weight:660.65LY2934747
CAS:<p>LY2934747 is a novel, potent, and systemically bioavailable mGlu2/3 receptor agonist, exhibiting both antipsychotic and analgesic properties in vivo.</p>Formula:C10H13NO4Color and Shape:SolidMolecular weight:211.21Disorazol A
CAS:<p>Disorazol A1 is a tubulin inhibitor with antifungal properties. It functions by inhibiting tubulin polymerization and disrupting microtubule formation, thereby blocking mitosis and arresting the cell cycle at the G2/M phase, which induces apoptosis. Disorazol A1 also inhibits L929 mouse fibroblasts with an IC50 value of 3 pm and causes accumulation of p53 protein in the nucleus. Disorazol A1 holds potential for cancer research.</p>Formula:C43H54N2O10Color and Shape:SolidMolecular weight:758.896Encephalitic alphavirus-IN-1
<p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) & EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>Formula:C27H25FN6O2Color and Shape:SolidMolecular weight:484.52FCE-27262
CAS:<p>FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.</p>Formula:C23H31N3O3Color and Shape:SolidMolecular weight:397.51AMD-7049
CAS:<p>AMD-7049 is a biochemical.</p>Formula:C25H39N5Color and Shape:SolidMolecular weight:409.61(-)-15-Deoxyspergualin
CAS:<p>(-)-15-Deoxyspergualin is a potent antitumor agent that demonstrates significant inhibition against mouse leukemia L-1210.</p>Formula:C17H37N7O3Color and Shape:SolidMolecular weight:387.52Chrymutasin C
CAS:<p>Chrymutasin C is a glycoside antitumor antibiotic with cytotoxic properties.</p>Formula:C39H43NO17Color and Shape:SolidMolecular weight:797.755MDL-43291
CAS:<p>MDL-43291 is a leukotriene receptor antagonist.</p>Formula:C25H42O4SColor and Shape:SolidMolecular weight:438.66NCI-006
CAS:<p>NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.</p>Formula:C31H24F2N4O4S3Color and Shape:SolidMolecular weight:650.74Guraxetan
<p>Guraxetan can be used in the synthesis of the antitumour drug Lutetium (177Lu) zadavotide Guraxetan.</p>Formula:C20H34N4O9Color and Shape:SolidMolecular weight:474.51Glidobactin C
CAS:<p>Glidobactin C (GlbC) is an antitumor antibiotic with activity against pathogenic fungi and yeasts. It exhibits antifungal properties against Candida albicans and Aspergillus fumigatus, with a minimum inhibitory concentration (MIC) of 0.8 μg/mL. Additionally, Glidobactin C prolongs the survival time of mice inoculated with leukemia P388 cells.</p>Formula:C29H48N4O6Color and Shape:SolidMolecular weight:548.7152-Hydroxygentamicin C2
CAS:<p>2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C20H41N5O8Color and Shape:SolidMolecular weight:479.568YKL-05-093
CAS:<p>YKL-05-093 is a alt inducible kinase (SIK) inhibitor. YKL-05-093 increases bone formation and bone mass.</p>Formula:C35H40N6O4Color and Shape:SolidMolecular weight:608.73Pterulinic acid
CAS:<p>Pterulinic acid is an inhibitor of coenzyme I:coenzyme Q oxidoreductase. It demonstrates IC50 values (μg/mL) of 50 for the mammalian cell line L1210, 20 for HL60, 25 for HeLaS3, and 100 for BHK.</p>Formula:C15H11ClO4Color and Shape:SolidMolecular weight:290.70AN-12-H5
CAS:<p>AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.</p>Formula:C24H23N3O4S3Color and Shape:SolidMolecular weight:513.65Endophenazine A
CAS:<p>Endophenazine A exhibits activity against Gram-positive bacteria and filamentous fungi such as Mucor and Penicillium, but demonstrates limited herbicidal effect on Lemna.</p>Formula:C18H16N2O2Color and Shape:SolidMolecular weight:292.332CYP2C9/CYP2C19-IN-1
<p>CYP2C9/CYP2C19-IN-1 is a potent inhibitor of CYP2C9/CYP2C19 without liver toxicity or genotoxicity and can be used to study Zika virus (ZIKV) infection.</p>Formula:C27H28N2O6SColor and Shape:SolidMolecular weight:508.59DG013A
CAS:<p>DG013A inhibits ERAP1 & ERAP2 (IC50: 33 nM & 11 nM) to research autoimmune diseases & cancer.</p>Formula:C27H37N4O4PColor and Shape:SolidMolecular weight:512.58Antcin B
CAS:<p>Antcin B is an inhibitor of SARS-CoV-2 3-chymotrypsin-like protease (3CL Pro). It interacts with several crucial amino acid residues of 3CL Pro, including Leu141, Asn142, Glu166, and His163, through hydrogen bonding, salt bridges, and hydrophobic interactions, thereby inhibiting its activity. This inhibition blocks the cleavage of viral polyproteins and suppresses the replication of the SARS-CoV-2 virus within host cells. Antcin B shows potential for research in the context of COVID-19.</p>Formula:C29H40O5Color and Shape:SolidMolecular weight:468.625Nanaomycin B
CAS:<p>Nanaomycin B is an antibiotic with activity against Gram-positive bacteria, mycobacteria, mycoplasma, and fungi.</p>Formula:C16H16O7Color and Shape:SolidMolecular weight:320.294Sagopilone
CAS:<p>Sagopilone: synthetic epothilone, inhibits cell division and induces apoptosis, effective in MDR tumors, not P-gp substrate.</p>Formula:C30H41NO6SColor and Shape:SolidMolecular weight:543.71P2X7 receptor antagonist-1
<p>P2X7 receptor antagonist-1 is a purinergic P2X7 receptor antagonist with anti-neuroinflammatory effects.</p>Formula:C22H20F4N2O3Color and Shape:SolidMolecular weight:436.4LI-3948
CAS:<p>IP6K-IN-2 (compound 29c) is an IP6K inhibitor that demonstrates oral bioavailability and the ability to permeate the blood-brain barrier (IC 50 : 15.8 nM), making it suitable for research on central nervous system diseases.</p>Formula:C19H16Cl2FN3O3Color and Shape:SolidMolecular weight:424.25AZD2353
CAS:<p>AZD2353 is a potent inhibitor of diacylglycerol acetyl transferase 1 (DGAT1).</p>Formula:C22H19ClFN3O3Color and Shape:SolidMolecular weight:427.86Porothramycin B
CAS:<p>Porothramycin B is an antibiotic with activity against Gram-positive bacteria and anaerobes.</p>Formula:C19H23N3O4Color and Shape:SolidMolecular weight:357.404Dersimelagon phosphate
CAS:<p>Dersimelagon phosphate: MC1R agonist, boosts melanin, enhances light tolerance in EPP/XLP without sun.</p>Formula:C36H48F4N3O9PColor and Shape:SolidMolecular weight:773.75CJ-887
CAS:<p>CJ-887 is a STAT3 inhibitor.</p>Formula:C34H45N6O10PColor and Shape:SolidMolecular weight:728.73Faldaprevir sodium
CAS:<p>Faldaprevir sodium: HCV treatment, inhibits NS3/NS4A protease, P-glycoprotein, CYP3A4, UGT1A1.</p>Formula:C40H48BrN6NaO9SColor and Shape:SolidMolecular weight:891.81SGK1-IN-3
<p>SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.</p>Formula:C23H20Cl2N6O3SColor and Shape:SolidMolecular weight:531.412-Hydroxygentamicin B1
CAS:<p>2-Hydroxygentamicin B1 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C20H40N4O11Color and Shape:SolidMolecular weight:512.552Feudomycin B
CAS:<p>Feudomycin B is a macrolactam antibiotic that exhibits antitumor cell activity.</p>Formula:C28H31NO10Color and Shape:SolidMolecular weight:541.54615(R)-Lipoxin A4
CAS:<p>Lipid-derived lipoxins are produced at the site of vascular and mucosal inflammation where they down-regulate polymorphonuclear leukocyte recruitment and</p>Formula:C20H32O5Color and Shape:SolidMolecular weight:352.47BMS-520
CAS:<p>BMS-520: potent oral S1P1 agonist, effective in rat arthritis and mouse multiple sclerosis model.</p>Formula:C23H17F3N4O4Color and Shape:SolidMolecular weight:470.4Epiderstatin
CAS:<p>Epiderstatin is isolated from Streptomyces pulveraceus subsp. epiderstagenes; inhibits mitogenic activity of epidermal growth factor.</p>Formula:C15H20N2O4Color and Shape:SolidMolecular weight:292.33PDE4B/7A-IN-2
CAS:<p>5-HT1A/5-HT7 antagonist; 5-HT1A Ki=8 nM, 5-HT7 Ki=451 nM; PDE4B IC50=80.4 μM, PDE7A IC50=151.3 μM; stronger than escitalopram.</p>Formula:C25H35N3O2Color and Shape:SolidMolecular weight:409.56Granaticin B
CAS:<p>Granaticin B inhibits the initial phase of RNA biosynthesis and exhibits activity against Gram-positive bacteria, mycobacteria (weak), and Trichomonas vaginalis, along with the ability to suppress tumor cells.</p>Formula:C28H30O12Color and Shape:SolidMolecular weight:558.531PARP7-IN-12
CAS:<p>PARP7-IN-12, a potent inhibitor targeting PARP7, exhibits an IC50 of 7.836 nM. This compound is applicable in cancer research.</p>Formula:C23H27ClF3N5O5Color and Shape:SolidMolecular weight:545.94Antimalarial agent 2
<p>Antimalarial agent 2 is an orally active, novel antimalarial agent that exhibits rapid in vitro killing effects.</p>Formula:C27H25N3O5Color and Shape:SolidMolecular weight:471.5TRβ agonist 1
CAS:<p>TRβ Agonist 1, a selective and mutation-sensitive thyroid hormone receptor β (TRβ) agonist, demonstrates an EC50 value of 21 nM.</p>Formula:C29H25FN2O8Color and Shape:SolidMolecular weight:548.52Topoisomerase II inhibitor 5
<p>Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.</p>Formula:C26H27N5O4Color and Shape:SolidMolecular weight:473.52Nebramycin Ⅳ
CAS:<p>Nebramycin IV is an aminoglycoside antibiotic with a broad antimicrobial spectrum, demonstrating significant efficacy against Gram-positive bacteria, Gram-negative bacteria, and mycobacteria.</p>Formula:C19H38N6O11Color and Shape:SolidMolecular weight:526.539Antidepressant agent 2
<p>Antidepressant agent 2 showed significant antidepressant effects with a MED value of 0.1 mg/kg.</p>Formula:C21H22ClFN2O3SColor and Shape:SolidMolecular weight:436.93MEIS-IN-3
<p>MEIS-IN-3 is a potent inhibitor of MEIS.</p>Formula:C25H26N2O4Color and Shape:SolidMolecular weight:418.48CY208-243 Mandelate
CAS:<p>CY208-243 is a D1 agonist boosting memory in T-maze, enhances adenylate cyclase (EC50=125nM), and alters monkey electroretinogram.</p>Formula:C27H26N2O3Color and Shape:SolidMolecular weight:426.52Nnc 09-0026
CAS:<p>Nnc 09-0026 is a neuronal calcium channel blocker</p>Formula:C25H35Cl2F3N2OColor and Shape:SolidMolecular weight:507.46SENP2-IN-1
CAS:<p>SENP2-IN-1 selectively inhibits SENP2, SENP1, and SENP5 with low IC50 values; useful in cancer studies.</p>Formula:C32H29N3O5S2Color and Shape:SolidMolecular weight:599.72GS-9160
CAS:<p>GS-9160 is a novel and potent inhibitor of human immunodeficiency virus type 1 (HIV-1) integrase (IN) that specifically targets the process of strand transfer.</p>Formula:C20H18FN3O4SColor and Shape:SolidMolecular weight:415.44FK-906 HCl
CAS:<p>FK-906 HCl is a human renin inhibitor used for the long-term treatment of patients with essential hypertension.</p>Formula:C40H64ClN7O7Color and Shape:SolidMolecular weight:790.44RDN2150
CAS:<p>RDN2150 (Compound 25), a ZAP-70 inhibitor with an IC50 of 14.6 nM, covalently binds to the C346 residue of ZAP-70, suppressing the expression of CD25 and CD69</p>Formula:C28H29ClN8O4Color and Shape:SolidMolecular weight:577.03FMK-MEA
CAS:<p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>Formula:C21H26FN5O2Purity:98%Color and Shape:SolidMolecular weight:399.46Dinordrin
CAS:<p>Dinordrin is an implantation inhibitor and hormone.</p>Formula:C27H36O4Purity:98%Color and Shape:SolidMolecular weight:424.57KHK-IN-6
CAS:<p>KHK-IN-6 (compound 33) acts as a KHK inhibitor with an IC50 of 0.6nM.</p>Formula:C23H24F3N5O2SColor and Shape:SolidMolecular weight:491.53MRS4865
CAS:<p>MRS4865 (compound 7a) serves as a chimeric antagonist for the P2Y14 receptor and an agonist for UDP-glucose, offering protection against neuropathic pain.</p>Formula:C39H39F3N4O7Color and Shape:SolidMolecular weight:732.74SARS-CoV-2-IN-99
CAS:<p>SARS-CoV-2-IN-99 (compound 58) is an inhibitor of the main protease of SARS-CoV-2.</p>Formula:C20H16Br2NO4PColor and Shape:SolidMolecular weight:525.13AH22921
CAS:<p>AH22921 is an EP4 prostaglandin receptor antagonist with the ability to antagonize the activation of adenylyl cyclase by prostaglandins in CHO cells. It induces a rightward shift in the PGE? concentration-response curve in these cells, functioning as a non-competitive antagonist. AH22921 is selective for the EP4 receptor, inhibiting its activity in CHO cells without affecting the PGE? concentration-response curve in NPE cells that contain the EP2 receptor.</p>Formula:C29H35NO5Color and Shape:SolidMolecular weight:477.59Hynapene A
CAS:<p>Hynapene A exhibits an inhibitory minimum inhibitory concentration (MIC) of 123 μM against Eimeria tenella.</p>Formula:C18H28O5Color and Shape:SolidMolecular weight:324.412Hydroxyakalone
CAS:<p>Hydroxyakalone is an inhibitor of the enzyme xanthine oxidase (XOD, EC 1.2.3.2) and has an IC50 of 4.6 μM for XOD.</p>Formula:C5H5N5O2Color and Shape:SolidMolecular weight:167.126Ezomycin A1
CAS:<p>Ezomycin A1 is an antifungal antibiotic effective primarily against plant pathogens such as Sclerotinia and Botrytis. It is used to prevent and control diseases like Sclerotinia rot, gray mold, and candidiasis in crops.</p>Formula:C26H38N8O15SColor and Shape:SolidMolecular weight:734.69Bagremycin B
CAS:<p>Bagremycin B is produced by the bacterium Streptomyces strain Tu 4128. It exhibits weak activity against Gram-positive bacteria, Saccharomyces cerevisiae, and Candida albicans.</p>Formula:C17H15NO4Color and Shape:SolidMolecular weight:297.305Cytosaminomycin A
CAS:<p>Cytosaminomycin A is an antibiotic with anticoccidial and antibacterial properties.</p>Formula:C22H34N4O8SColor and Shape:SolidMolecular weight:514.592MEIS-IN-2
<p>MEIS-IN-2 is an inhibitor of MEIS1. MEIS-IN-2 can be used in studies of cardiac regeneration and haematopoietic stem cell (HSC) regulation.</p>Formula:C23H21ClN2O4Color and Shape:SolidMolecular weight:424.88EcGUS-IN-1
CAS:<p>EcGUS-IN-1 (Compound E-9) is a non-competitive inhibitor of β-glucuronidase, featuring an IC50 value of 2.68 μM and a Ki value of 1.64 μM. This compound effectively mitigates gastrointestinal adverse events (GIAE) associated with Escherichia coli infections by inhibiting the activity of E. coli β-glucuronidase.</p>Formula:C15H11F3N4SColor and Shape:SolidMolecular weight:336.33Ingenol 3-monobenzoate
CAS:<p>Ingenol 3-monobenzoate (Ingenol 3-benzoate) acts as an aversive inducing agent. It binds to and activates protein kinase C (PKC) with a Ki of 0.14 nM. This activation inhibits the gene expression of phosphoenolpyruvate carboxykinase, thereby suppressing gluconeogenesis and increasing blood cortisol levels, which results in food aversion.</p>Formula:C27H32O6Color and Shape:SolidMolecular weight:452.54
